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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 124 / 134
Tigecycline Approved DB00560
small molecule | CAS: 220620-09-7

Tigecycline is a glycylcycline antibiotic developed and marketed by Wyeth under the brand name Tygacil. It was developed in response to the growing prevalence of antibiotic resistance in bacteria such as Staphylococcus aureus. It was granted fast-track approv…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
16S ribosomal RNA30S ribosomal protein S930S ribosomal protein S12 +3
Waktu Paruh27-43 hours
Vol. Distribusi-
Klirens-
Genetik -
Tigulixostat DB18799
small molecule | CAS: 1287766-55-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilarginine Approved DB11815
small molecule | CAS: 17035-90-4

Tilarginine has been investigated for the basic science, treatment, and diagnostic of Obesity, Type 2 Diabetes, Ocular Physiology, and Regional Blood Flow.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +4
Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilbroquinol Approved DB13222
small molecule | CAS: 7175-09-9

Tilbroquinol was approved in France, Morocco, and Saudi Arabia but it has been withdrawn in France and Saudi Arabia markets mainly due to its hepatotoxicity risk outweighing the drug benefit [L5467]. In Morocco, the drug has been limited to use in the treatme…

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tildrakizumab Approved DB14004
biotech | CAS: 1326244-10-3

Tildrakizumab is a high-affinity, humanized, IgG1 ? antibody targeting interleukin 23 p19 that shows promise in the evolution of treatment strategy in chronic plaque psoriasis [A32255]. The Food and Drug Administration (FDA) approved ILUMYA (tildrakizumab-…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-23
Waktu ParuhThe half-life is ap…
Vol. DistribusiThe geometric mean …
KlirensThe mean (CV%) syst…
Genetik -
Tiletamine DB11549
small molecule | CAS: 14176-49-9

This drug is a dissociative anesthetic agent that falls under the drug category of _NMDA receptor antagonists_. Tiletamine is chemically similar to another dissociative anesthetic, ketamine. Tiletamine hydrochloride, the salt form, exists as odorless white cr…

Kategori:
AnestheticsAnesthetics, DissociativeAnesthetics, General +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilletia caries Approved DB10705
biotech

Tilletia caries allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tilmicosin DB11471
small molecule | CAS: 108050-54-0

Tilmicosin is a macrolide antibiotic. It is used in veterinary medicine for the treatment of bovine respiratory disease and ovine respiratory disease associated with _Mannheimia haemolytica_.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsLactones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiludronic acid Approved DB01133
small molecule | CAS: 89987-06-4

Tiludronate, or (4-chlorophenyl)thio-methylene-1,1-bisphosphonate, is a first generation bisphosphonate similar to [etidronic acid] and [clodronic acid].[A1923,A203111] These drugs were developed to mimic the action of pyrophosphate, a regulator of calcificat…

Kategori:
BisphosphonatesBone Density Conservation AgentsDrugs Affecting Bone Structure and Mineralization +6
Target Protein:
HydroxylapatiteAdenosine triphosphate (ATP)Tyrosine-protein phosphatase non-receptor type 12 +3
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe volume of distr…
KlirensTiludronic acid has…
Genetik -
Timcodar DB12761
small molecule | CAS: 179033-51-3

Timcodar has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timdarpacept DB17544
biotech | CAS: 2749520-17-8

IMM01 is a recombinant human signal regulatory protein ? (SIRP?) IgG 1 fusion protein.[A257261] IMM01 is under investigation in clinical trial NCT05140811 (A Study of IMM01 Combined With Azacitidine in Patients With Acute Myeloid Leukemia and Myelodysplastic …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timolumab DB18597
biotech | CAS: 1073538-99-4

Timolumab is a recombinant, fully-human, IgG4 immunoglobulin with antigen-binding specificity for human vascular adhesion protein-1 (VAP-1).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Timonacic DB12856
small molecule | CAS: 444-27-9

Timonacic has been used in trials studying the treatment of HIV Infections.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tinzaparin Approved DB06822
small molecule | CAS: 9041-08-1

Tinzaparin is a low molecular weight heparin (LMWH), produced by enzymatic depolymerization of unfractionated heparin from porcine intestinal mucosa. It is a heterogeneous mixture of with an average molecular weight between 5500 and 7500 daltons. Tinzaparin i…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Target Protein:
Antithrombin-IIIIntegrin alpha-4Stromal cell-derived factor 1
Waktu ParuhAnti-Xa activity is…
Vol. DistribusiAnti-Xa activity is…
KlirensClearance is dose-d…
Genetik -
Tioconazole Approved DB01007
small molecule | CAS: 65899-73-2

Tioconazole is an imidazole antifungal used to treat fungal and yeast infections. Topical formulations are used for ringworm, jock itch, athlete's foot, and tinea versicolor or "sun fungus". Tioconazole interacts with 14-alpha demethylase, a cytochrome P-450 …

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +21
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiopronin Approved DB06823
small molecule | CAS: 1953-02-2

Tiopronin is a prescription thiol drug used primarily in the treatment of severe homozygous cystinuria. Patients with cystinuria excrete high levels of cystine in their urine and are at risk for kidney stone formation. Tiopronin is used as a second-line thera…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +7
Waktu ParuhTiopronin has a lon…
Vol. DistribusiThe volume of distr…
KlirensTotal renal clearan…
Genetik -
Tiotropium Approved DB01409
small molecule | CAS: 186691-13-4

Tiotropium is a long-acting, antimuscarinic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD) and asthma.[A180163,L7084,L7087,L7090,L7093] Tiotropium acts mainly on M3 muscarinic receptors located in the airways to produce …

Kategori:
Adrenergics, InhalantsAgents producing tachycardiaAgents to Treat Airway Disease +22
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe terminal half l…
Vol. DistribusiThe volume of distr…
KlirensThe total clearance…
Genetik -
biotech | CAS: 1052105-48-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiphenamil DB19367
small molecule | CAS: 82-99-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicPhenylacetates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tipiracil Approved DB09343
small molecule | CAS: 183204-74-2

Tipiracil is a thymidine phosphorylase inhibitor. It is used in combination with trifluridine, in a ratio of 1:0.5, to form TAS-102. The main function of Tipiracil in TAS-102 is to increase trifluridine bioavailability by inhibiting its catabolism.[A31255] TA…

Kategori:
MATE 1 SubstratesMATE 1 Substrates with a Narrow Therapeutic IndexMATE substrates +6
Target Protein:
Thymidine phosphorylase
Waktu ParuhAfter administratio…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Tiprelestat DB18368
biotech | CAS: 820211-82-3

Deskripsi belum tersedia.

Target Protein:
MyeloblastinNeutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiracizine DB13635
small molecule | CAS: 83275-56-3

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCardiac TherapyCardiovascular Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiragolumab DB16409
biotech | CAS: 1918185-84-8

Tiragolumab is under investigation in clinical trial NCT04513925 (A Study of Atezolizumab and Tiragolumab Compared With Durvalumab in Participants With Locally Advanced, Unresectable Stage III Non-small Cell Lung Cancer (NSCLC)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tiratricol DB03604
small molecule | CAS: 51-24-1

A metabolite of T3 and T4 thyroid hormones; promoted for hyperlipidemia, localized lipodystrophy, and obesity. Tiratricol has been used in trials studying the treatment of Allan-Herndon-Dudley Syndrome.

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +9
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tirbanibulin Approved DB06137
small molecule | CAS: 897016-82-9

Tirbanibulin (KX-O1 or KX2–391) is a dual inhibitor of Src Kinase and tubulin.[A225726] On December 14, 2020, tirbanibulin was approved by the FDA for the topical treatment of actinic keratosis on the face or scalp. It is marketed under the brand name Klisyri…

Kategori:
AcetatesAcids, AcyclicAmides +39
Target Protein:
Tubulin beta chainProto-oncogene tyrosine-protein kinase Src
Waktu ParuhThe half-life is ab…
Vol. DistribusiThere is limited in…
KlirensThere is limited in…
Genetik -
Tirofiban Approved DB00775
small molecule | CAS: 144494-65-5

Tirofiban prevents the blood from clotting during episodes of chest pain or a heart attack, or while the patient is undergoing a procedure to treat a blocked coronary artery. It is a non-peptide reversible antagonist of the platelet glycoprotein (GP) IIb/IIIa…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +9
Target Protein:
Integrin alpha-IIbIntegrin beta-3
Waktu Paruh2 hours
Vol. Distribusi* 22 to 42 L
Klirens* 213 - 314 mL/min …
Genetik -
Tirzepatide Approved DB15171
biotech | CAS: 2023788-19-2

Tirzepatide is a novel dual glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor agonist. Dual GIP/GLP-1 agonists gained increasing attention as new therapeutic agents for glycemic and weight control as they demonstr…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +17
Target Protein:
Glucagon-like peptide 1 receptorGastric inhibitory polypeptide receptor
Waktu ParuhThe half-life is ap…
Vol. DistribusiFollowing subcutane…
KlirensThe apparent popula…
Genetik -
Tisagenlecleucel Approved DB13881
biotech | CAS: 1823078-37-0

Tisagenlecleucel is a CD19-directed genetically modified autologous T cell immunotherapy, or a CAR-T cell therapy for B-cell acute lymphoblastic leukemia. It was granted approval by FDA in August 2017 under the market name Kymriah. Tisagenlecleucel is an immu…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Immunological +10
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe mean half life …
Vol. DistribusiThe drug is found t…
Klirens-
Genetik -
Tisotumab vedotin Approved DB16732
biotech | CAS: 1418731-10-8

Tisotumab vedotin is a tissue factor-directed antibody-drug conjugate (ADC) comprised of an anti-tissue factor (TF) human IgG1-kappa antibody conjugated to monomethyl auristatin E (MMAE), a microtubule-disrupting agent, via a protease-cleavable valine-citrull…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Tissue factor
Waktu ParuhThe median terminal…
Vol. DistribusiThe tisotumab vedot…
KlirensThe linear clearanc…
Genetik -
Titanium dioxide Approved DB09536
small molecule | CAS: 13463-67-7

Titanium dioxide, also known as titanium(IV) oxide or titania, is the naturally occurring oxide of titanium. It is used as a pigment under the names titanium white, Pigment White 6 (PW6), or CI 77891. It is typically extracted from ilmenite, rutile and anatas…

Kategori:
Astringents and DeodorantsBiocompatible MaterialsColoring Agents +13
Target Protein:
Macrophage receptor MARCO
Waktu ParuhThe kinetics of TiO…
Vol. DistribusiSix hours after tit…
KlirensThe clearance of ti…
Genetik -
Tivozanib Approved DB11800
small molecule | CAS: 475108-18-0

Renal cell carcinoma (RCC) is responsible for 3% of cancer cases[A231314] and is one of the 10 most common cancers in adults. The average age of diagnosis is between age 65 to 74.[L32529] Tivozanib, also known as FOTIVDA, is a kinase inhibitor developed to t…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +13
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +8
Waktu ParuhThe half-life of ti…
Vol. DistribusiTivozanib has an ap…
KlirensThe apparent cleara…
Genetik -
Tixagevimab Approved DB16394
biotech | CAS: 2420564-02-7

SARS-CoV-2, the causative agent of COVID-19, enters cells via the interaction between the trimeric spike (S) glycoprotein and host cell angiotensin-converting enzyme 2 (ACE2). Blocking the interaction between the receptor-binding domain (RBD) of the S1 subuni…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Spike glycoprotein
Waktu ParuhTixagevimab has a h…
Vol. DistribusiTixagevimab has an …
KlirensTixagevimab has an …
Genetik -
Tixocortol Approved DB09091
small molecule | CAS: 61951-99-3

Tixocortol is a 21-thiol derivative of hydrocortisone classified as a class A corticosteroid. It is a synthetic steroid with topical anti-inflammatory properties without the systemic glucocorticoid and mineralocorticoid activities and toxicity.[L1078]

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +20
Target Protein:
Glucocorticoid receptorHistone deacetylase 2
Waktu ParuhTixocortol presents…
Vol. DistribusiStudies have shown …
KlirensStudies have shown …
Genetik -
Tizanidine Approved DB00697
small molecule | CAS: 51322-75-9

Tizanidine is a fast-acting drug used for the management of muscle spasm, which may result from the effects of multiple sclerosis, stroke, an acquired brain injury, or a spinal cord injury [T574]. It may also be caused by musculoskeletal injury [A177583]. R…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +24
Target Protein:
Alpha-1 adrenergic receptorsAlpha-2 adrenergic receptorsNischarin
Waktu ParuhApproximately 2.5 h…
Vol. DistribusiExtensively distrib…
Klirens**A note on renal i…
Genetik -
TL-895 DB16471
small molecule | CAS: 1415823-49-2

TL-895 is a potent, orally active, ATP-competitive, and highly selective irreversible BTK inhibitor with an IC50 and a Ki of 1.5 nM and 11.9 nM, respectively. TL-895 is under investigation in several clinical trials for its safety and efficacy in various cond…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TLY-012 DB18336
biotech

TLY-012 is a PEGylated recombinant human tumor necrosis factor-related apoptosis-inducing ligand (PEGylated TRAIL).[L48166]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TM5614 DB16516
small molecule

TM5614 is a novel, orally active, plasminogen activator inhibitor 1 (PAI-1) inhibitor[A228788,A228793,]. PAI-1 is a marker of obesity, type 2 diabetes, and metabolic syndrome[L31673,A228793,A228798], and current studies are exploring downstream effects of its…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Plasminogen activator inhibitor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMC-649128 DB15152
small molecule | CAS: 1019639-33-8

TMC-649128 is under investigation in clinical trial NCT01391117 (TMC649128HPC1002 - a Trial inGenotype 1 Hepatitis C Virus (HCV) - Infected Participants to Determine the Safety, Tolerability, Pharmacokinetics and Antiviral Activity of TMC649128, Alone and Com…

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMP DB04243
small molecule

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleotidesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Target Protein:
Single-stranded DNA-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TMV-083 DB16430
biotech

TMV-083 is an attenuated live virus COVID-19 vaccine candidate which employs the measles vaccine as a vector[L30433]. It expresses a spike protein antigen from SARS-CoV-2[L30433].

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TN-201 DB18700
biotech

TN-201 is a gene therapy comprising a native AAV9 capsid with a genomic cassette containing a cardiomyocyte-specific promoter and the wild-type human MYBPC3 gene.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TN-401 DB18140
biotech

TN-401 is a native AAV9 capsid with a genomic cassette containing a cardiomyocyte-specific promoter and the wild-type human PKP2 gene.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TNB-383B DB17268
biotech

TNB-383B is a CD3 and B-cell maturation antigen T-cell engaging bispecific antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TNB-486 DB19420
biotech

TNB-486 is under investigation in clinical trial NCT06564038 (A Study of AZD0486 Monotherapy or in Combination With Other Anti-cancer Agents for Mature B-cell Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tobemstomig DB18987
biotech | CAS: 2648839-43-2

Tobemstomig is under investigation in clinical trial NCT05908786 (A Study Evaluating the Efficacy and Safety of Neoadjuvant Immunotherapy Combinations in Patients With Surgically Resectable Hepatocellular Carcinoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tobevibart DB18986
biotech | CAS: 2645440-65-7

Tobevibart is under investigation in clinical trial NCT05612581 (A Platform Study to Evaluate Investigational Therapies in Chronic Hepatitis B Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tobramycin Approved DB00684
small molecule | CAS: 32986-56-4

Aminoglycosides, many of which are derived directly from _Streptomyces_ spp., are concentration-dependent bactericidal antibiotics with a broad spectrum of activity against Gram-positive and Gram-negative organisms.[A232294] Inhaled tobramycin is notable for …

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +13
Target Protein:
16S ribosomal RNA23S ribosomal RNABacterial outer membrane +1
Waktu ParuhTobramycin has an a…
Vol. DistribusiInhalation tobramyc…
KlirensInhaled tobramycin …
Genetik -
Tocilizumab Approved DB06273
biotech | CAS: 375823-41-9

Tocilizumab is a recombinant humanized monoclonal antibody IL-6 receptor inhibitor used to treat inflammatory and autoimmune conditions.[L12789] It was first described in the literature in 2003 when Chugai, a subsidiary of Roche began developing IL-6 inhibiti…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +21
Target Protein:
Interleukin-6 receptor subunit alpha
Waktu ParuhThe half life of to…
Vol. DistribusiIn rheumatoid arthr…
KlirensThe linear clearanc…
Genetik -
Tocofersolan Approved DB11635
small molecule | CAS: 9002-96-4

D-Alpha-tocopheryl polyethylene glycol 1000 succinate (Tocofersolan, Vedrop), has been developed in Europe as an orally bioavailable source of vitamin E in children suffering from cholestasis [L2371]. Cholestasis is the reduction or stoppage of bile flow, eit…

Kategori:
Alimentary Tract and MetabolismBenzopyransCompounds used in a research, industrial, or household setting +9
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh29.7 h [L2371]
Vol. DistribusiLocated principally…
Klirens-
Genetik -
Tocopherol Approved DB11251
small molecule | CAS: 1406-66-2

Tocopherol exists in four different forms designated as ?, ?, ?, and ?. They present strong antioxidant activities, and it is determined as the major form of vitamin E. Tocopherol, as a group, is composed of soluble phenolic compounds that consist of a chroma…

Kategori:
Alimentary Tract and MetabolismAntioxidantsBenzopyrans +16
Target Protein:
Free radicals
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensClearance ranged fr…
Genetik -
Menampilkan 6151–6200 dari 6694
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