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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 124 / 282
Etripamil DB12605
small molecule | CAS: 1593673-23-4

Etripamil has been used in trials studying the treatment of Paroxysmal Supraventricular Tachycardia (PSVT).

Kategori:
Acids, CarbocyclicAntiarrhythmic agentsBenzene Derivatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etrolizumab DB12189
biotech | CAS: 1044758-60-2

Inflammatory bowel disease (IBD), including ulcerative colitis and Crohn's disease, is typified by a chronic gastrointestinal inflammatory microenvironment, driven in part by the excessive infiltration and retention of intestinal-homing lymphocytes.[A244564, …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Integrin beta-7
Waktu ParuhEtrolizumab adminis…
Vol. DistribusiModelling of etroli…
KlirensEtrolizumab has a m…
Genetik -
Etrumadenant DB17506
small molecule | CAS: 2239273-34-6

Deskripsi belum tersedia.

Target Protein:
Adenosine receptor A2aAdenosine receptor A2b
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etryptamine DB01546
small molecule | CAS: 2235-90-7

In the 1960's, alpha-ethyltryptamine (?ET), a non hydrazine reversible monoamine oxidase inhibitor, was developed in the United States by the Upjohn chemical company for use as an antidepressant. ?ET was an FDA approved antidepressant under the name Monase. H…

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etybenzatropine DB13468
small molecule | CAS: 524-83-4

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlkaloidsAnti-Parkinson Drugs +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etynodiol DB13866
small molecule | CAS: 1231-93-2

Etynodiol (INN), or ethynodiol (BAN) is a steroidal progestin related to norethisterone which was never marketed. While etynodiol is sometimes used as a synonym for etynodiol diacetate, it usually refers to etynodiol diacetate (see [DB00823]), not etynodiol.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EU204 DB17438
biotech

EU204 (EBViNT) is an Epstein-Barr virus (EBV)-positive T-cell therapy currently undergoing phase 1 and 2a clinical trials in Korea for patients with EBV-positive lymphoma and solid cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eucalyptol DB03852
small molecule | CAS: 470-82-6

Eucalyptol is naturally produced cyclic ether and monoterpenoid. Eucalyptol is an ingredient in many brands of mouthwash and cough suppressant. It controls airway mucus hypersecretion and asthma via anti-inflammatory cytokine inhibition. Eucalyptol is an effe…

Kategori:
AgrochemicalsAlcoholsAnti-Infective Agents +29
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eucalyptus globulus leaf Approved DB14320
biotech

Eucalyptus globulus leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eucalyptus gum Approved DB15537
biotech | CAS: 9000-20-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Eucommia ulmoides bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Euflavine DB13326
small molecule | CAS: 86-40-8

Deskripsi belum tersedia.

Kategori:
Acridine DerivativesAcridinesAntiseptics and Disinfectants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eupatilin DB16885
small molecule | CAS: 22368-21-4

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesDrugs, Chinese Herbal +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
European pilchard Approved DB10622
biotech

European pilchard allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eurotium amstelodami Approved DB15526
biotech

Eurotium amstelodami allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Eutrema japonicum whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evacetrapib DB11655
small molecule | CAS: 1186486-62-3

Evacetrapib has been used in trials studying the basic science and treatment of Dyslipidemia, Hyperlipidemia, Hypercholesterolemia, Hepatic Insufficiency, and Cardiovascular Disease.

Kategori:
Anticholesteremic AgentsBenzazepinesCholesterol Ester Transfer Proteins, antagonists & inhibitors +3
Target Protein:
Cholesteryl ester transfer protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evalstotug DB19410
biotech | CAS: 2460399-39-5

Evalstotug is under investigation in clinical trial NCT05271604 (A Phase 2 Open Label Study of BA3021 in Patients With Recurrent or Metastatic Squamous Cell Carcinoma of the Head and Neck).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evatanepag DB12022
small molecule | CAS: 223488-57-1

Evatanepag has been used in trials studying the treatment of Tibial Fractures.

Target Protein:
Prostaglandin E2 receptor EP2 subtype
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evenamide DB18775
small molecule | CAS: 1092977-61-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 308064-97-3

Evening primrose oil comes from the extraction from _Oenothera biennis_ seeds and it is commonly used as an alternative source for omega-6 essential fatty acids. In its composition it presents some fatty acids such as [DB00132] and [DB13854].[A33131] Evening …

Kategori:
Agents that reduce seizure thresholdAngiospermsAnti-Inflammatory Agents +26
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Evernia prunastri Approved DB14172
biotech

Evernia prunastri allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseStandardized Chemical Allergen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Everolimus Approved DB01590
small molecule | CAS: 159351-69-6

Everolimus is a derivative of Rapamycin (sirolimus), and works similarly to Rapamycin as an mTOR (mammalian target of rapamycin) inhibitor. It is currently used as an immunosuppressant to prevent rejection of organ transplants. In a similar fashion to other m…

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +32
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh~30 hours.
Vol. DistribusiThe blood-to-plasma…
KlirensFollowing a 3 mg ra…
Genetik -
Evexomostat DB19140
small molecule | CAS: 2416263-67-5

Evexomostat is under investigation in clinical trial NCT05570253 (A Study of SDX-7320 in Combination With Eribulin for People With Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evinacumab Approved DB15354
biotech | CAS: 1446419-85-7

Evinacumab is a recombinant human IgG4 monoclonal antibody targeted against angiopoietin-like protein 3 (ANGPTL3) and the first drug of its kind. The ANGPTL family of proteins serve a number of physiologic functions - including involvement in the regulation o…

Kategori:
Amino Acids, Peptides, and ProteinsAngiopoietin-like 3 InhibitorAngiopoietin-like 3 Inhibitors +8
Target Protein:
Angiopoietin-related protein 3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Evobrutinib DB15170
small molecule | CAS: 1415823-73-2

Evobrutinib is under investigation in clinical trial NCT03934502 (Effect of Meal Composition and Timing on Evobrutinib Bioavailability).

Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evocalcet DB12388
small molecule | CAS: 870964-67-3

Evocalcet has been used in trials studying the treatment of Hyperparathyroidism and Secondary Hyperparathyroidism.

Kategori:
Anti-Parathyroid AgentsCalcium HomeostasisSystemic Hormonal Preparations, Excl. Sex Hormones and Insulins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evodenoson DB12295
small molecule | CAS: 844873-47-8

Evodenoson has been used in trials studying the treatment of Open-angle Glaucoma and Ocular Hypertension.

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evofosfamide DB06091
small molecule | CAS: 918633-87-1

TH-302 is a novel cancer therapeutic specifically activated under the low oxygen or "hypoxic" conditions typical of solid tumor cancer cells. TH-302 is a nitroimidazole-linked prodrug of a brominated derivative of an isophosphoramide mustard previously used i…

Kategori:
Hydrocarbons, HalogenatedImidazolesMustard Compounds +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evogliptin DB12625
small molecule | CAS: 1222102-29-5

Evogliptin has been used in trials studying the treatment and screening of Osteoporosis, Renal Impairment, Type 2 Diabetes Mellitus, Diabetes Mellitis Type 2, and Diabetes Mellitus, Type 2.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +4
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evolocumab Approved DB09303
biotech | CAS: 1256937-27-5

Evolocumab is a monoclonal antibody designed for the treatment of hyperlipidemia by Amgen. It is a subcutaneous injection approved by the FDA for individuals on maximum statin therapy who still require additional LDL-cholesterol lowering. It is approved for b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu Paruh-
Vol. Distribusi-
KlirensEvolocumab showed n…
Genetik -
Evorpacept DB17573
biotech | CAS: 2484949-51-9

evorpacept is under investigation in clinical trial NCT04755244 (A Study of Evorpacept (ALX148) With Venetoclax and Azacitidine for Acute Myeloid Leukemia (ASPEN-05)).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EVT 201 DB05721
small molecule | CAS: 308239-86-3

EVT 201 is a novel partial positive allosteric modulator of the GABAA receptor complex which is being developed as a treatment for insomnia. It is being developed by Evotec Inc.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EVT 302 DB06057
small molecule

EVT 302 is an orally active, potent, highly selective and reversible inhibitor of MAO-B. It is in the development for smoking cessation, and potential for disease modification in Alzheimer's disease.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EVT-101 DB05956
small molecule | CAS: 1189088-41-2

Deskripsi belum tersedia.

Target Protein:
Glutamate receptor ionotropic, NMDA 2BRetinoic acid receptor RXR-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EW-A-401 DB05525
biotech

EW-A-401 is a circle of genetic material (plasmid DNA) that instructs the body to produce a genetically-engineered transcription factor, a protein that regulates expression of genes. This specific transcription factor has been shown in animal studies to incre…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exagamglogene autotemcel Approved DB15572
biotech

Sickle cell disease (SCD) is a genetic disorder characterized by the production of abnormal sickle-shaped red blood cells (called hemoglobin S, HbS) that initiate a pathophysiology resulting in severe pain, progressive multi-organ damage, and premature death.…

Kategori:
Autologous Cultured CellBlood and Blood Forming Organs
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exarafenib DB17582
small molecule | CAS: 2639957-39-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exatecan DB12185
small molecule | CAS: 171335-80-1

Exatecan has been used in trials studying the treatment of Sarcoma, Leukemia, Lymphoma, Lung Cancer, and Liver Cancer, among others.

Kategori:
AlkaloidsAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exbivirumab DB17747
biotech | CAS: 569658-80-6

Exbivirumab is an investigational monoclonal antibody. It is one of the active ingredients in HepeX-B, a drug product containing two human monoclonal antibodies to the hepatitis B virus (HBV) surface antigen.[A259202]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exebacase DB16161
biotech | CAS: 1404122-92-4

Exebacase is under investigation in clinical trial NCT03163446 (Safety, Efficacy and Pharmacokinetics of CF-301 vs. Placebo in Addition to Antibacterial Therapy for Treatment of S. Aureus Bacteremia).

Kategori:
EnzymesEnzymes and CoenzymesHydrolases +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exenatide Approved DB01276
biotech | CAS: 141758-74-9

Exenatide is a glucagon-like peptide-1 (GLP-1) analog[L42690]. It activates the GLP-1 receptor and increases insulin secretion, decreases glucagon secretion, and slows gastric emptying to improve glycemic control[L42690]. Exenatide was given FDA approval on A…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnti-Obesity Agents +16
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh2.4 hours[Label]
Vol. Distribusi28.3L[Label].
Klirens9.1 L/hour[Label].
Genetik -
Exicorilant DB16162
small molecule | CAS: 1781244-77-6

Exicorilant is under investigation in clinical trial NCT03437941 (Study to Evaluate CORT125281 in Combination With Enzalutamide in Patients With Mcrpc).

Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exidavnemab DB19452
biotech | CAS: 2438229-02-6

Exidavnemab is under investigation in clinical trial NCT06671938 (Safety, Tolerability, and Pharmacokinetics of Exidavnemab in Patients With Parkinson's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exisulind DB06246
small molecule | CAS: 59973-80-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +10
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseGlutathione S-transferase PAldo-keto reductase family 1 member B1 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exlinkibart DB17474
biotech | CAS: 2642171-64-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EXOB-001 DB18257
biotech

EXOB-001 consists of extracellular vesicles derived from cultured human umbilical cord mesenchymal stromal cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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EXT608 DB18453
biotech

EXT608 is a long-acting PTH derivative under investigation for the treatment of hyperparathyroidism.[L48270]

Waktu Paruh-
Vol. Distribusi-
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Ezabenlimab DB17483
biotech | CAS: 2249882-54-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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