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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Halaman 124 / 315
Elbasvir Approved DB11574
small molecule | CAS: 1370468-36-2

Elbasvir is a direct-acting antiviral medication used as part of combination therapy to treat chronic hepatitis C, an infectious liver disease caused by infection with hepatitis C virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine d…

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +18
Target Protein:
Nonstructural protein 5A
Waktu ParuhThe geometric mean …
Vol. DistribusiElbasvir has an est…
KlirensThe clearance of el…
Genetik -
Elcatonin DB13742
small molecule | CAS: 60731-46-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Parathyroid AgentsBone Density Conservation Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eldecalcitol DB05295
small molecule | CAS: 104121-92-8

Eldecalcitol (ED-71), a vitamin D analog, is a more potent inhibitor of bone resorption than alfacalcidol in an estrogen-deficient rat model of osteoporosis. Eldecalcitol, effectively and safely increased lumbar and hip bone mineral density (BMD) in osteopor…

Kategori:
Bone Density Conservation AgentsFused-Ring CompoundsSecosteroids +4
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eldelumab DB06116
biotech | CAS: 946414-98-8

MDX-1100, a fully human antibody that targets IP10 (also known as CXCL10), a chemokine expressed in association with multiple inflammatory disease indications, such as rheumatoid arthritis, inflammatory bowel disease and multiple sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
C-X-C motif chemokine 10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elebsiran DB19018
biotech | CAS: 2648009-64-5

Elebsiran is under investigation in clinical trial NCT05461170 (SOLSTICE: Combination Therapy for the Treatment of Chronic Hepatitis D Infection.).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eleclazine DB12394
small molecule | CAS: 1443211-72-0

Eleclazine has been used in trials studying the treatment of LQT2 Syndrome, Long QT Syndrome, Ischemic Heart Disease, Ventricular Arrhythmia, and Long QT Syndrome Type 3, among others.

Kategori:
Azepines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elenbecestat DB15391
small molecule | CAS: 1388651-30-6

Elenbecestat is under investigation in clinical trial NCT02956486 (A 24-Month Study to Evaluate the Efficacy and Safety of Elenbecestat (E2609) in Subjects With Early Alzheimer's Disease).

Target Protein:
Beta-secretase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elenestinib DB18489
small molecule | CAS: 2505078-08-8

Elenestinib is a selective KIT inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elesclomol DB05719
small molecule | CAS: 488832-69-5

Elesclomol is a novel, injectable, drug candidate that kills cancer cells by elevating oxidative stress levels beyond a breaking point, triggering programmed cell death. In preclinical models elesclomol showed potent killing of a broad range of cancer cell ty…

Kategori:
AmidesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eletriptan Approved DB00216
small molecule | CAS: 143322-58-1

Eletriptan is a second generation triptan drug developed by Pfizer Inc for the treatment of migraine headaches.

Kategori:
Agents that produce hypertensionAminesAnalgesics +30
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1F +1
Gen Terkait:
GNB3
Waktu ParuhThe terminal elimin…
Vol. Distribusi* 138 L
Klirens* Renal cl=3.9 L/h
Genetik 1 Varian
Eleuthero Approved DB14303
biotech

Eleuthero is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAraliaceaeBiological Products +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elexacaftor Approved DB15444
small molecule | CAS: 2216712-66-0

Elexacaftor (previously VX-445) is a small molecule, next-generation corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) protein.[A187361] It received FDA approval in October 2019 in combination with [tezacaftor] and [ivacaftor] as the…

Kategori:
Cystic Fibrosis Transmembrane Conductance Regulator CorrectorsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +24
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Elezanumab DB15240
biotech | CAS: 1791416-49-3

Elezanumab is under investigation in clinical trial NCT03737812 (A Study to Assess the Safety and Efficacy of Elezanumab When Added to Standard of Care in Progressive Forms of Multiple Sclerosis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elgemtumab DB15430
biotech | CAS: 1512559-37-3

Elgemtumab is under investigation in clinical trial NCT02167854 (Open-Label Study Evaluating the Safety and Tolerability of LJM716, BYL719 and Trastuzumab in Patients With Metastatic HER2+ Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eliglustat Approved DB09039
small molecule | CAS: 491833-29-5

Eliglustat is a glucosylceramide synthase inhibitor used for the long-term treatment of type 1 Gaucher disease.[A3752,L41404] Gaucher disease is a rare genetic disorder characterized by the deficiency of acid ?-glucosidase, an enzyme that converts glucosylcer…

Kategori:
Alimentary Tract and MetabolismCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +15
Target Protein:
Ceramide glucosyltransferase
Waktu ParuhEliglustat has a te…
Vol. DistribusiIn CYP2D6 extensive…
KlirensIn healthy CYP2D6 e…
Genetik -
Elimusertib DB19041
small molecule | CAS: 1876467-74-1

Elimusertib is under investigation in clinical trial NCT05071209 (Elimusertib for the Treatment of Relapsed or Refractory Solid Tumors).

Target Protein:
Serine/threonine-protein kinase ATR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elinogrel DB06350
small molecule | CAS: 936500-94-6

A P2Y12 inhibitor and platelet aggregation inhibitor.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingQuinazolines +2
Target Protein:
P2Y purinoceptor 12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elinzanetant DB18968
small molecule | CAS: 929046-33-3

Elinzanetant is under investigation in clinical trial NCT05099159 (A Study to Learn More About How Well Elinzanetant Works and How Safe It Is for the Treatment of Vasomotor Symptoms (Hot Flashes) That Are Caused by Hormonal Changes Over 26 Weeks in Women Who …

Target Protein:
Neuromedin-K receptorSubstance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eliprodil DB12869
small molecule | CAS: 119431-25-3

Eliprodil has been used in trials studying the treatment of Parkinson Disease and Movement Disorders.

Kategori:
Central Nervous System AgentsCompounds used in a research, industrial, or household settingExcitatory Amino Acid Agents +5
Target Protein:
Glutamate receptor ionotropic, NMDA 2BGlutamate receptor ionotropic, NMDA 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elismetrep DB15287
small molecule | CAS: 1400699-64-0

Elismetrep is under investigation in clinical trial NCT02429102 (A Study to Investigate the Safety, Tolerability and Pharmacokinetics of MT-8554 in Healthy Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elivaldogene autotemcel Approved DB16746
biotech

Elivaldogene autotemcel is a gene therapy consisting of genetically modified autologous cells. It is used to provide functional copies of human adrenoleukodystrophy protein (ALDP) in patients with adrenoleukodystrophy,[L39491] an X-linked genetic disorder cha…

Kategori:
Alimentary Tract and MetabolismCellular and Gene TherapyVarious Alimentary Tract and Metabolism Products
Waktu ParuhAs elivaldogene aut…
Vol. DistribusiAs elivaldogene aut…
KlirensAs elivaldogene aut…
Genetik -
biotech | CAS: 1905397-73-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ellagic acid DB08846
small molecule | CAS: 476-66-4

Ellagic acid is present in several fruits such as cranberries, strawberries, raspberries, and pomegranates. In pomegranates, there are several therapeutic compounds but ellagic acid is the most active and abundant. Ellagic acid is also present in vegetables. …

Kategori:
BenzopyransCytochrome P-450 CYP2E1 InhibitorsCytochrome P-450 CYP2E1 Inhibitors (strength unknown) +6
Target Protein:
Heat shock 70 kDa protein 1AHeat shock 70 kDa protein 1BGlycogen synthase kinase-3 beta +17
Waktu Paruh-
Vol. Distribusi-
KlirensEllagic acid is eli…
Genetik -
Ellipticine DB17026
small molecule | CAS: 519-23-3

Ellipticine is a potent antineoplastic agent.[A252992]

Kategori:
AlkaloidsAntineoplastic AgentsCarbazoles +8
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elm Approved DB14258
biotech

Elm is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elobixibat DB12486
small molecule | CAS: 439087-18-0

Elobixibat has been used in trials studying the treatment and basic science of Dyslipidemia, Constipation, Chronic Constipation, Functional Constipation, and Chronic Idiopathic Constipation.

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAzepines +5
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elocalcitol DB06194
small molecule | CAS: 199798-84-0

Elocalcitol is a calcitriol analog for inhibition of prostate cell growth; in phase II clinical trial in patients with benign prostate hyperplasia (4/2004).

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elosulfase alfa Approved DB09051
biotech | CAS: 9025-60-9

Elosulfase alfa is a synthetic version of the enzyme N-acetylgalactosamine-6-sulfatase. It was approved by the FDA in 2014 for the treatment of Morquio syndrome. Elosulfase alfa was developed by BioMarin Pharmaceutical Inc. and is marketed under the brand Vim…

Kategori:
Alimentary Tract and MetabolismCarbon-Oxygen LyasesChondroitinases and Chondroitin Lyases +9
Waktu Paruhweek 0: 7.52 min w…
Vol. Distribusi396 mL/kg, standard…
Klirens10.0 mL/min/kg. (…
Genetik -
Elotuzumab Approved DB06317
biotech | CAS: 915296-00-3

Elotuzumab is a humanized IgG1 (Immunoglobulin G) monoclonal antibody indicated in combination with lenalidomide and dexamethasone for the treatment of patients with multiple myeloma who have received one to three prior therapies. Elotuzumab targets SLAMF7, a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
SLAM family member 7
Waktu Paruh-
Vol. Distribusi-
KlirensThe clearance of el…
Genetik -
Elraglusib DB16047
small molecule | CAS: 1034895-42-5

Elraglusib is under investigation in clinical trial NCT04218071 (Actuate 1901: 9-ING-41 in Myelofibrosis).

Target Protein:
Glycogen synthase kinase-3 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elranatamab Approved DB15395
biotech | CAS: 2408850-14-4

Elranatamab is a bispecific B-cell maturation antigen (BCMA)-directed CD3 T-cell engager. It is a humanized immunoglobulin 2-alanine kappa antibody derived from two monoclonal antibodies (mAbs), an anti-BCMA mAb and an anti-CD3 mAb,[A261060] each of which con…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalBispecific B-cell maturation antigen (BCMA)-directed CD3 T-cell engager +5
Target Protein:
Tumor necrosis factor receptor superfamily member 17T-cell surface glycoprotein CD3
Waktu ParuhThe mean (CV%) half…
Vol. DistribusiThe mean (CV%) stea…
KlirensThe mean (CV%) clea…
Genetik -
Elsamitrucin DB05129
small molecule | CAS: 97068-30-9

The cytostatic agent Elsamitrucin is a new fermentation product active in a variety of in vivo tumor models of murine and human origin. (PMID: 8150873)

Kategori:
Antibiotics, AntineoplasticAntineoplastic AgentsCarbohydrates +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA +1
Waktu Paruh36–60 h
Vol. Distribusi-
Klirens-
Genetik -
Elsiglutide DB06336
small molecule | CAS: 914009-84-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elsubrutinib DB18850
small molecule | CAS: 1643570-24-4

Elsubrutinib is under investigation in clinical trial NCT04451772 (A Study of the Safety of Oral Elsubrutinib Capsules and Oral Upadacitinib Tablets Given Alone or in Combination (ABBV-599) for Adult Participants With Moderately to Severely Active Systemic Lu…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elsulfavirine DB14929
small molecule | CAS: 868046-19-9

Elsulfavirine is under investigation in clinical trial NCT03706898 (Study to Evaluate the Safety and PK of Elpida® in Healthy Subjects and Patients With Hepatic Impairment and to Assess the Impact of Food Intake and Drug-Drug Interactions With Other Antiviral…

Kategori:
AmidesAminesAniline Compounds +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltanexor DB16153
small molecule | CAS: 1642300-52-4

Eltanexor is under investigation in clinical trial NCT02649790 (Study of the Safety, Tolerability and Efficacy of KPT-8602 in Patients With Relapsed/refractory Cancer Indications).

Target Protein:
Exportin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltanolone DB12308
small molecule | CAS: 128-20-1

Eltanolone is under investigation in clinical trial NCT02603926 (Treatment of Fragile-X Associated Tremor/Ataxia Syndrome (FXTAS) With Allopregnanolone).

Kategori:
AnestheticsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit gamma-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltoprazine DB12883
small molecule | CAS: 98224-03-4

Eltoprazine has been used in trials studying the treatment of Schizophrenia and Cognitive Impairment.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNeurotransmitter Agents +6
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltrekibart DB19017
biotech | CAS: 2484883-56-7

Eltrekibart is under investigation in clinical trial NCT06046729 (A Study of Eltrekibart (LY3041658) in Adult Participants With Moderate to Severe Hidradenitis Suppurativa).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eltrombopag Approved DB06210
small molecule | CAS: 496775-61-2

Eltrombopag is used to treat low blood platelet counts in adults with chronic immune (idiopathic) thrombocytopenia (ITP), when certain other medicines, or surgery to remove the spleen, have not worked well enough. ITP is a condition that may cause unusual bru…

Kategori:
Acids, CarbocyclicBCRP/ABCG2 InhibitorsBenzene Derivatives +25
Target Protein:
Thrombopoietin receptor
Gen Terkait:
F5 SERPINC1
Waktu ParuhAbout 21-32 hours i…
Vol. DistribusiBased on a radiolab…
Klirens-
Genetik 2 Varian
Elubrixin DB12135
small molecule | CAS: 688763-64-6

Elubrixin has been used in trials studying the treatment of Cystic Fibrosis, Colitis, Ulcerative, and Chronic Obstructive Pulmonary Disease (COPD).

Kategori:
AmidesBenzene DerivativesReceptors, Interleukin-8B, antagonists & inhibitors +2
Target Protein:
C-X-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eluforsen DB16154
biotech | CAS: 2101868-82-8

Eluforsen is under investigation in clinical trial NCT02532764 (Dose Escalation Study of QR-010 in Homozygous ?F508 Cystic Fibrosis Patients).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eluvixtamab DB17252
biotech | CAS: 1679391-73-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eluxadoline Approved DB09272
small molecule | CAS: 864821-90-9

Eluxadoline is a mixed mu-opioid receptor agonist, kappa-opioid receptor agonist, and a-delta opioid receptor antagonist indicated for use in diarrhea-predominant irritable bowel syndrome (IBS-D). The mu-, kappa-, and delta-opioid receptors mediate endogenous…

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Aromatic +15
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhThe mean plasma eli…
Vol. Distribusi-
Klirens-
Genetik -
Elvitegravir Approved DB09101
small molecule | CAS: 697761-98-1

Elvitegravir is a human immunodeficiency virus type 1 (HIV-1) integrase strand transfer inhibitor (INSTI) used for the treatment of HIV-1 infection in antiretroviral treatment-experienced adults. Because integrase is necessary for viral replication, inhibitio…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +22
Target Protein:
IntegraseGag-Pol polyprotein
Waktu ParuhThe median terminal…
Vol. Distribusi-
Klirens-
Genetik -
Elvucitabine DB06236
small molecule | CAS: 181785-84-2

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +13
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ELX-02 DB15080
small molecule | CAS: 1375073-95-2

ELX-02 is under investigation in clinical trial NCT03309605 (Phase 1 Study of ELX-02 in Healthy Adult Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elymus repens pollen Approved DB10489
biotech

Elymus repens pollen is the pollen of the Elymus repens plant. Elymus repens pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elzasonan DB18969
small molecule | CAS: 361343-19-3

Elzasonan is under investigation in clinical trial NCT00275197 (A Research Study to Compare the Treatments of a Combination of Elzasonan With Zoloft, to Zoloft Alone, or Placebo in People With Major Depressive Disorder (MDD)).

Kategori:
Oxazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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