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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 123 / 272
Fidarestat DB02021
small molecule | CAS: 136087-85-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsImidazoles
Target Protein:
Aldo-keto reductase family 1 member B1Aldo-keto reductase family 1 member B10
Waktu Paruh-
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Fidaxomicin Approved DB08874
small molecule | CAS: 873857-62-6

Fidaxomicin is a novel macrolide antibiotic used in the treatment of diarrhea caused by _Clostridioides_ (formerly _Clostridium_) _difficile_ in adult and pediatric patients over the age of 6 months.[L11575] Fidaxomicin is a naturally-occurring 18-member macr…

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
RNA polymerase sigma factor SigA
Waktu ParuhFollowing oral admi…
Vol. DistribusiFidaxomicin is main…
KlirensThere is limited in…
Genetik -
Fidrisertib DB18064
small molecule | CAS: 2141955-96-4

Deskripsi belum tersedia.

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Fig Approved DB10633
biotech

Fig allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
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Figitumumab DB11685
biotech | CAS: 943453-46-1

Figitumumab has been used in trials studying the treatment of Sarcoma, Solid Tumor, Breast Cancer, Lung Neoplasms, and Advanced Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Filaminast DB02660
small molecule | CAS: 141184-34-1

Filaminast is a phosphodiesterase 4 inhibitor (PDE4 inhibitor). As such, has potential in the treatment of asthma and chronic obstructive pulmonary disease (COPD).

Kategori:
AminesHydroxylamines
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Filanesib DB06040
small molecule | CAS: 885060-09-3

Filanesib is a potent Kinesin Spindle Protein (KSP) inhibitor that caused marked tumor regression in preclinical models of human solid tumors and human leukemias, often leading to durable responses.

Kategori:
Antimitotic AgentsAntineoplastic AgentsMitosis Modulators +2
Target Protein:
Kinesin-like protein KIF11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Filgotinib Approved DB14845
small molecule | CAS: 1206161-97-8

Rheumatoid arthritis (RA) is a chronic, autoimmune, systemic, and inflammatory disease that causes synovial joint symptoms and can limit range of motion in severe cases.[A221451,A221456] The disease is associated with extra-articular manifestations, progressi…

Kategori:
Antineoplastic and Immunomodulating AgentsArthritis, Rheumatoid, drug therapyImmunosuppressive Agents +5
Target Protein:
Tyrosine-protein kinase JAK1
Waktu ParuhThe half-life of fi…
Vol. Distribusi-
Klirens-
Genetik -
Filgrastim Approved DB00099
biotech | CAS: 121181-53-1

Filgrastim is a short-acting recombinant, non-pegylated human granulocyte colony-stimulating factor (G-CSF) analog produced by recombinant DNA technology. It has an amino acid sequence identical to endogenous G-CSF, but it is non-glycosylated unlike the endog…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBiological Factors +10
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhAfter intravenous a…
Vol. DistribusiAfter intravenous a…
KlirensClearance rates of …
Genetik -
Filibuvir DB11878
small molecule | CAS: 877130-28-4

Filibuvir has been used in trials studying the treatment of Hepatitis, Hepatitis C, and Chronic Hepatitis C.

Kategori:
PyransRNA Replicase, antagonists & inhibitorsRNA-Dependent RNA Polymerase, antagonists & inhibitors
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
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Filociclovir DB12438
small molecule | CAS: 632325-71-4

Filociclovir is under investigation in clinical trial NCT01433835 (Safety and Pharmacokinetics of Single Oral Doses of Filociclovir in Healthy Volunteers).

Waktu Paruh-
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Filorexant DB12158
small molecule | CAS: 1088991-73-4

Filorexant has been used in trials studying the prevention and treatment of Migraine, Headache, Polysomnography, Diabetic Neuropathy, Painful, and Major Depressive Disorder, Recurrent.

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Fimaporfin DB17253
small molecule | CAS: 1443547-43-0

Deskripsi belum tersedia.

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Fimasartan DB09279
small molecule | CAS: 247257-48-3

Fimasartan is an angiotensin II receptor antagonist (ARB) drug employed in the treatment of both hypertension and heart failure. It has been found to be safe when administered with hydrochlorothiazide (a diuretic) in clinical trials. Fimasartan was initially …

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin II receptor blockers (ARBs) and calcium channel blockers +8
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhThe half life of el…
Vol. Distribusi-
Klirens-
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Fimepinostat DB11891
small molecule | CAS: 1339928-25-4

Fimepinostat (CUDC-907) has been used in trials studying the treatment of lymphoma, solid tumors, breast cancer, multiple myeloma, and NUT midline carcinoma, among others.

Kategori:
Antineoplastic AgentsHistone Deacetylase InhibitorsOxazines +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Finafloxacin Approved DB09047
small molecule | CAS: 209342-40-5

Finafloxacin is a fluoroquinolone antibiotic indicated in the treatment of acute otitis externa (swimmer's ear) caused by the bacteria Pseudomonas aeruginosa and Staphylococcus aureus. Finafloxacin is marketed by Novartis under the brand Xtoro™, and was appro…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Finasteride Approved DB01216
small molecule | CAS: 98319-26-7

Finasteride is a synthetic 4-azasteroid compound [L10565] and specific inhibitor of steroid Type II 5?-reductase, which is an intracellular enzyme that converts the androgen testosterone into 5?-dihydrotestosterone (DHT). It works in a similar fashion as [dut…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +22
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 2Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 1 +1
Waktu ParuhIn healthy young su…
Vol. DistribusiThe volume of distr…
KlirensIn healthy young su…
Genetik -
Finerenone Approved DB16165
small molecule | CAS: 1050477-31-0

Finerenone, or BAY 94-8862, is a mineralocorticoid receptor antagonist indicated to reduce the risk of sustained decline in glomerular filtration rate, end stage kidney disease, cardiovascular death, heart attacks, and hospitalization due to heart failure in …

Kategori:
Agents causing hyperkalemiaCytochrome P-450 CYP2C8 SubstratesCytochrome P-450 CYP3A Substrates +6
Target Protein:
Mineralocorticoid receptor
Waktu ParuhThe half life of a …
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Fingolimod Approved DB08868
small molecule | CAS: 162359-55-9

Multiple sclerosis, or MS, is a devastating inflammatory disease that often progresses and causes severe neurological, physical, and cognitive effects.[A176474] Fingolimod is a sphingosine 1-phosphate receptor modulator for the treatment of relapsing-remittin…

Kategori:
AlcoholsAminesAmino Alcohols +16
Target Protein:
D(3) dopamine receptorSphingosine kinase 1Sphingosine 1-phosphate receptor 5 +4
Waktu ParuhThe half-life of fi…
Vol. DistribusiThe volume of distr…
KlirensFingolimod blood cl…
Genetik -
FINLAY-FR-1 DB16524
biotech

FINLAY-FR-1, also known as Soberana 01, is a vaccine candidate for COVID-19 that is being led developmentally by the Finlay Vaccine Institute[L31373]. It is currently being tested in the clinical trial RPCEC00000332 (Phase I / II, randomized, controlled, adap…

Waktu Paruh-
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Finotonlimab DB18859
biotech | CAS: 2350298-85-8

Finotonlimab is under investigation in clinical trial NCT04560894 (SCT-I10A Plus SCT510 Versus Sorafenib as First-line Therapy for Advanced Hepatocellular Carcinoma).

Waktu Paruh-
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Fipaxalparant DB18124
small molecule | CAS: 1195941-38-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysophosphatidic acid receptor 1Lysophosphatidic acid receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fipexide DB13790
small molecule | CAS: 34161-24-5

Deskripsi belum tersedia.

Kategori:
Nervous SystemPsychoanalepticsPsychostimulants, Agents Used for ADHD and Nootropics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Firategrast DB12732
small molecule | CAS: 402567-16-2

Firategrast has been used in trials studying the treatment of Multiple Sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Firazorexton DB19440
small molecule | CAS: 2274802-95-6

Firazorexton is under investigation in clinical trial NCT04096560 (A Study of TAK-994 in Adults With Type 1 and Type 2 Narcolepsy).

Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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Firsocostat DB16166
small molecule | CAS: 1434635-54-7

Firsocostat is under investigation in clinical trial NCT02781584 (Safety, Tolerability, and Efficacy of Selonsertib, Firsocostat, and Cilofexor in Adults With Nonalcoholic Steatohepatitis (NASH)).

Kategori:
Acids, AcyclicButyratesEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Firtecan pegol DB14953
small molecule | CAS: 946062-05-1

Firtecan pegol is under investigation in clinical trial NCT01036113 (A Phase 2 Study of EZN-2208 in Patients With Metastatic Breast Cancer).

Kategori:
AlcoholsAlkaloidsEthylene Glycols +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fisetin DB07795
small molecule | CAS: 528-48-3

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
Cyclin-dependent kinase 6Fatty acid synthaseCyclin homolog
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fish oil Approved DB13961
biotech

Fish oil is a component of SMOFLIPID, which was FDA approved in July 2016. It is indicated in adults as a source of calories and essential fatty acids for parenteral nutrition when oral or enteral nutrition is not possible, insufficient, or contraindicated. …

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +8
Target Protein:
Diacylglycerol O-acyltransferase 2Prostaglandin G/H synthase 2Free fatty acid receptor 4 +8
Waktu ParuhThe half-life of EP…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of EP…
Genetik -
Fispemifene DB06640
small molecule | CAS: 341524-89-8

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsStilbenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fitusiran DB15002
biotech | CAS: 1499251-18-1

Fitusiran is under investigation in clinical trial NCT02554773 (An Open-label Extension Study of an Investigational Drug, ALN-AT3SC, in Patients With Moderate or Severe Hemophilia A or B).

Kategori:
Amino SugarsAntisense Elements (Genetics)Carbohydrates +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FK-614 DB12557
small molecule | CAS: 193012-35-0

FK614 has been used in trials studying the treatment of Diabetes Mellitus.

Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FK-960 DB06465
small molecule | CAS: 133920-70-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FK352B DB06484
small molecule | CAS: 143881-08-7

FK352B is a adenosine A1 antagonist that is developed for the treatment of dialysis-induced hypotension.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flavin adenine dinucleotide Approved DB03147
small molecule | CAS: 146-14-5

A condensation product of riboflavin and adenosine diphosphate. The coenzyme of various aerobic dehydrogenases, e.g., D-amino acid oxidase and L-amino acid oxidase. (Lehninger, Principles of Biochemistry, 1982, p972) Flavin adenine dinucleotide is approved f…

Kategori:
Adenine NucleotidesBiological FactorsCoenzymes +13
Target Protein:
Ribosyldihydronicotinamide dehydrogenase [quinone]Nitric oxide synthase 1Dihydropyrimidine dehydrogenase [NADP(+)] +83
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flavin mononucleotide Approved DB03247
small molecule | CAS: 146-17-8

A coenzyme for a number of oxidative enzymes including NADH DEHYDROGENASE. It is the principal form in which RIBOFLAVIN is found in cells and tissues.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +11
Target Protein:
Flavin reductase (NADPH)2-Hydroxyacid oxidase 1Pyridoxine-5'-phosphate oxidase +51
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
D-amino-acid oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cholesterol oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flavone Approved DB07776
small molecule | CAS: 525-82-6

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
AromataseGamma-aminobutyric acid receptor subunit alpha-1Androgen receptor +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flavoxate Approved DB01148
small molecule | CAS: 15301-69-6

A drug that has been used in various urinary syndromes and as an antispasmodic. Its therapeutic usefulness and its mechanism of action are not clear. It may have local anesthetic activity and direct relaxing effects on smooth muscle as well as some activity a…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAutonomic Agents +15
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flecainide Approved DB01195
small molecule | CAS: 54143-55-4

Flecainide is a Class I anti-arrhythmic agent like [encainide] and [propafenone].[A186880] Flecainide’s development began in 1966 and was first synthesized in 1972 as an attempt to generate new anesthetics.[A186931] It is used to prevent supraventricular and …

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ic +27
Target Protein:
Sodium channel protein type 4 subunit alphaSodium channel protein type 5 subunit alphaVoltage-gated inwardly rectifying potassium channel KCNH2 +1
Waktu ParuhIn healthy subjects…
Vol. DistribusiThe average volume …
KlirensThe average clearan…
Genetik -
Fleroxacin DB04576
small molecule | CAS: 79660-72-3

Fleroxacin is a broad-spectrum antimicrobial fluoroquinolone. It strongly inhibits the DNA-supercoiling activity of DNA gyrase. Fleroxacin is not an inhibitor of CYP1A2.[A39048]

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
DNA topoisomerase 2-betaDNA gyrase subunit ADNA topoisomerase 4 subunit A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fletikumab DB12356
biotech | CAS: 1357158-22-5

Fletikumab is under investigation in clinical trial NCT01038674 (Safety and Tolerability of Anti-IL-20 in Subjects With Rheumatoid Arthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flibanserin Approved DB04908
small molecule | CAS: 167933-07-5

Flibanserin is the first drug to be approved for hypoactive sexual desire disorder (HSDD) in premenopausal women by the FDA in August 2015. It was originally developed as an antidepressant medication by Boehringer Ingelheim, but showed lack of efficacy in tri…

Kategori:
Agents that produce hypertensionAntidepressive AgentsCentral Nervous System Depressants +15
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2AD(4) dopamine receptor
Waktu Paruh?11 hours
Vol. Distribusi-
Klirens-
Genetik -
Flindokalner DB16908
small molecule | CAS: 187523-35-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Genetik -
Floctafenine Approved DB08976
small molecule | CAS: 23779-99-9

Floctafenine is an anti-inflammatory analgesic similar in action to aspirin. Floctafenine inhibits prostaglandin synthesis.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +14
Waktu Paruh-
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Genetik -
Flomoxef DB11935
small molecule | CAS: 99665-00-6

Flomoxef has been used in trials studying the treatment of Urinary Tract Infection.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +9
Waktu Paruh-
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Genetik -
Florasulam DB15316
small molecule | CAS: 145701-23-1

Florasulam is under investigation in clinical trial NCT01193465 (Temperature and Humidity Among Different Anesthesia Work-station).

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
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small molecule | CAS: 956903-29-0

Florbenazine F-18 is under investigation in clinical trial NCT01515384 (A Trial of 18F-AV-133 Positron Emission Tomography (PET)).

Waktu Paruh-
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Genetik -
Menampilkan 6101–6150 dari 13591
Sebelumnya Halaman 123 / 272 Berikutnya