Hasil Filter

16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

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Hasil Pencarian (16004)

Halaman 123 / 321
Dextranomer DB13560
small molecule | CAS: 56087-11-7

Deskripsi belum tersedia.

Kategori:
BiopolymersCarbohydratesCicatrizants +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 142985-55-5

Deskripsi belum tersedia.

Kategori:
BiopolymersCarbohydratesDietary Carbohydrates +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextroamphetamine Approved DB01576
small molecule | CAS: 51-64-9

Dextroamphetamine is the dextrorotatory enantiomer of amphetamine[A2505]. Dextroamphetamine was approved by the FDA in 2001 for the treatment of attention deficit hyperactivity disorder[L6010,Label].

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +19
Target Protein:
Synaptic vesicular amine transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +3
Waktu Paruh11.75 hours.[Label]…
Vol. Distribusi195L.[A177247]
Klirens17L/h.[A177247]
Genetik -
Dextromethadone DB15198
small molecule | CAS: 5653-80-5

Dextromethadone is under investigation in clinical trial NCT00588640 (Study of D-Methadone in Patients With Chronic Pain).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextromethorphan Approved DB00514
small molecule | CAS: 125-71-3

Dextromethorphan is a levorphanol derivative and codeine analog commonly used as a cough suppressant and also a drug of abuse.[A215412] Although similar in structure to other opioids, it has minimal interaction with opioid receptors.[A215412] Dextromethorp…

Kategori:
AlkaloidsAnticholinergic AgentsAntidepressive Agents +37
Target Protein:
Sigma non-opioid intracellular receptor 1AromataseGlutamate receptor ionotropic, NMDA 3A +13
Gen Terkait:
CYP2D6 CYP2D6
Waktu ParuhDextromethorphan ha…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik 2 Varian
Dextromoramide DB01529
small molecule | CAS: 357-56-2

An opioid analgesic structurally related to methadone and used in the treatment of severe pain. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1070)

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextropropoxyphene Approved DB00647
small molecule | CAS: 469-62-5

Dextropropoxyphene is an opioid analgesic manufactured by Eli Lilly and Company. It is used in the symptomatic treatment of mild pain. It displays antitussive and local anaesthetic actions. Due to the risk of cardiac arrhythmias and overdose, possibly leading…

Kategori:
Acids, AcyclicAgents that reduce seizure thresholdAnalgesics +22
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +2
Waktu Paruh6-12 hours
Vol. Distribusi* 16 L/kg
Klirens* 2.6 L/min
Genetik -
Dextrorphan DB14682
small molecule | CAS: 125-73-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsCentral Nervous System AgentsCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextrose, unspecified form Approved DB09341
small molecule

Glucose is a simple sugar (monosaccharide) generated during phosynthesis involving water, carbon and sunlight in plants. It is produced in humans via hepatic gluconeogenesis and breakdown of polymeric glucose forms (glycogenolysis). It circulates in human cir…

Kategori:
Caloric AgentsCardiac FunctionCompounds used in a research, industrial, or household setting +4
Waktu ParuhThe approximate hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean metabolic …
Genetik -
Dextrothyroxine Approved DB00509
small molecule | CAS: 51-49-0

The major hormone derived from the thyroid gland. Thyroxine is synthesized via the iodination of tyrosines (monoiodotyrosine) and the coupling of iodotyrosines (diiodotyrosine) in the thyroglobulin. Thyroxine is released from thyroglobulin by proteolysis and …

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +5
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor betaThyroid peroxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexverapamil DB14063
small molecule | CAS: 38321-02-7

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAminesAntiarrhythmic agents +14
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dezamizumab DB15153
biotech | CAS: 1662664-56-3

Dezamizumab is under investigation in clinical trial NCT03417830 (Biodistribution of 89Zirconium-labelled GSK2398852 Using PET Imaging).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dezapelisib DB16137
small molecule | CAS: 1262440-25-4

Dezapelisib is under investigation in clinical trial NCT02456675 (INCB040093 and INCB040093 Combined With Itacitinib (INCB039110) in Relapsed/refractory Hodgkin Lymphoma).

Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dezocine Approved DB01209
small molecule | CAS: 53648-55-8

Dezocine is a partial opiate drug and is used for pain management. Dezocine is a very effective alternative to fentanyl when administered during outpatient laparoscopy, although is associated with an increased incidence of postoperative nausea.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +8
Target Protein:
Mu-type opioid receptorKappa-type opioid receptor
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
DF-1001 DB18231
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DFV890 DB16461
small molecule

DFV890 is under investigation in multiple clinical trials for its efficacy, safety, and tolerability across various conditions: NCT06031844 (coronary heart disease with elevated hsCRP), NCT04886258 (symptomatic knee osteoarthritis), NCT06097663 (coronary hear…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DG041 DB05027
small molecule

DG041 is a novel, first-in-class, orally-administered small molecule developmented for the prevention of arterial thrombosis and its complications. DG041, an anti-platelet compound, has shown to be a selective and potent antagonist of the EP3 receptor for p…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DG051 DB05177
small molecule

DG051 is a novel small-molecule inhibitor of leukotriene A4 hydrolase (LTA4H), the protein made by one of the genes in the leukotriene pathway that has been shown to link to risk of heart attack. DG051 is designed to decrease risk of heart attack by decreasin…

Target Protein:
Leukotriene A-4 hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1382469-39-7

Di-2-pyridylketone 4-cyclohexyl-4-methyl-3-thiosemicarbazone is under investigation in clinical trial NCT02688101 (Dose-finding and Pharmacokinetic Study of DpC, Administered Orally to Patients With Advanced Solid Tumors).

Kategori:
SemicarbazidesSemicarbazonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DI-87 DB18027
small molecule | CAS: 2107280-55-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
ADP/ATP translocase 1Bactericidal permeability-increasing protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Prosaposin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diacerein Approved DB11994
small molecule | CAS: 13739-02-1

Diacerein is a prodrug which is metabolized to rhein. It is currently approved in France for the treatment of osteoarthritis although the use of diacerein is restricted due to the side effects including severe diarrhea [L780]. Diacerein is under investigation…

Kategori:
AnthracenesAnti-Inflammatory AgentsAntiinflammatory and Antirheumatic Products +12
Target Protein:
Interleukin-1 betaOxysterols receptor LXR-alphaOxysterols receptor LXR-beta +7
Waktu Paruh4-10h [A19300].
Vol. Distribusi15-60L [A19300].
KlirensTotal CL is 1.5L/h …
Genetik -
Diacetyl benzoyl lathyrol Approved DB11260
small molecule | CAS: 218916-52-0

Diacetyl benzoyl lathyrol is an active ingredient in whitening creams. It is also reported to be a skin conditioning agent.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Trypsin-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3148-72-9

Diaminohydroxypropanetetraacetic acid has been investigated for the treatment of Vascular Disease, Coronary Disease, Myocardial Ischemia, Coronary Restenosis, and Coronary Artery Disease, among others.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diaminopyrimidine oxide Approved DB18756
small molecule | CAS: 74638-76-9

Diaminopyrimidine oxide is a compound similar to [minoxidil] which is used to aid in hair growth.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diamorphine Approved DB01452
small molecule | CAS: 561-27-3

Diamorphine (heroin) is a narcotic analgesic that may be habit-forming. It is a controlled substance (opium derivative) listed in the U.S. Code of Federal Regulations, Title 21 Parts 329.1, 1308.11 (1987). Sale is forbidden in the United States by Federal sta…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +16
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Waktu ParuhIn humans, administ…
Vol. DistribusiData regarding the …
KlirensSome studies have d…
Genetik -
Diampromide DB01502
small molecule | CAS: 552-25-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dianexin DB15000
biotech | CAS: 1352413-49-0

Dianexin is under investigation in clinical trial NCT00615966 (Phase 2 Study of the Safety of Diannexin in Kidney Transplant Recipients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 23261-20-3

Dianhydrogalactitol has been used in trials studying the treatment of GBM, Glioma, Glioblastoma, Brain Cancer, and Glioblastoma Multiforme.

Kategori:
AlcoholsAlkylating DrugsAntineoplastic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dianicline DB12125
small molecule | CAS: 292634-27-6

Dianicline has been used in trials studying the treatment of Smoking, Smoking Cessation, and Tobacco Use Cessation.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit beta-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DiaPep 277 DB06651
small molecule | CAS: 179822-83-4

DiaPep 277 is a 24-mer laboratory-made peptide derived from Hsp60(437-460).

Kategori:
Acid Anhydride HydrolasesAdenosine TriphosphatasesAmino Acids, Peptides, and Proteins +10
Target Protein:
60 kDa heat shock protein, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diatrizoate Approved DB00271
small molecule | CAS: 117-96-4

A commonly used x-ray contrast medium. As diatrizoate meglumine and as Diatrizoate sodium, it is used for gastrointestinal studies, angiography, and urography.

Kategori:
Acids, CarbocyclicAlcoholsAmino Sugars +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diazepam Approved DB00829
small molecule | CAS: 439-14-5

A benzodiazepine with anticonvulsant, anxiolytic, sedative, muscle relaxant, and amnesic properties and a long duration of action. Its actions are mediated by enhancement of gamma-aminobutyric acid activity. It is used in the treatment of severe anxiety disor…

Kategori:
Adjuvants, AnesthesiaAnestheticsAnesthetics, General +40
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhDiazepam has a biph…
Vol. DistribusiIn young healthy ma…
KlirensThe clearance of di…
Genetik -
Diazepinomicin DB12420
small molecule | CAS: 733035-26-2

Diazepinomicin has been used in trials studying the treatment of Glioblastoma Multiforme. It is a proprietary first-in-class small molecule with the potential to treat multiple solid tumours like the well known chemotherapeutics, doxorubicin and mitomycin C. …

Kategori:
Heterocyclic Compounds, Fused-RingTerpenes
Target Protein:
Translocator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diaziquone DB17174
small molecule | CAS: 57998-68-2

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAzirinesCompounds used in a research, industrial, or household setting +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diazolidinylurea Approved DB14173
small molecule | CAS: 78491-02-8

Deskripsi belum tersedia.

Kategori:
AmidesCell-mediated ImmunityIncreased Histamine Release +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diazoxide Approved DB01119
small molecule | CAS: 364-98-7

Diazoxide is a non-diuretic benzothiadiazine derivative that activates ATP-sensitive potassium channels.[A255647,L44612] It is chemically related to thiazide diuretics but does not inhibit carbonic anhydrase and does not have chloriuretic or natriuretic activ…

Kategori:
Antihypertensive AgentsArteriolar Smooth Muscle, Agents Acting OnBenzothiadiazines +12
Target Protein:
ATP-sensitive inward rectifier potassium channel 11Mitochondrial ATP synthase F1 domain
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe apparent volume…
KlirensIn subjects with no…
Genetik -
Dibekacin Approved DB13270
small molecule | CAS: 34493-98-6

Dibekacin is an aminoglycoside antibiotic marketed in Japan [L5623].

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dibenzepin Approved DB13225
small molecule | CAS: 4498-32-2

Dibenzepin is approved for use in Europe.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dibotermin alfa Approved DB11639
biotech | CAS: 246539-15-1

Dibotermin alfa is a recombinant human bone morphogenetic protein-2 (rhBMP-2) derived from a recombinant Chinese Hamster Ovary (CHO) cell line [FDA Label]. It is implanted in patients undergoing bone surgeries or those with fractures. BMPs are subfamily of th…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBone Morphogenetic Proteins +7
Target Protein:
Bone morphogenetic protein receptor type-2Bone morphogenetic protein receptor type-1A
Waktu ParuhWhen injected intra…
Vol. Distribusi-
KlirensAt the site of impl…
Genetik -
small molecule | CAS: 29096-93-3

At low concentrations, this compound inhibits reduction of conventional hydrophilic electron acceptors, probably acting as a plastoquinone antagonist. At higher concentrations, it acts as an electron acceptor, intercepting electrons either before or at the si…

Kategori:
BenzoquinonesQuinones
Target Protein:
Cytochrome fCytochrome b6-f complex subunit 5Cytochrome b6-f complex subunit 6 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dibromotyrosine DB07637
small molecule | CAS: 300-38-9

Deskripsi belum tersedia.

Kategori:
Antithyroid agentsSystemic Hormonal Preparations, Excl. Sex Hormones and InsulinsThyroid Products
Target Protein:
Erythropoietin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 496-00-4

Deskripsi belum tersedia.

Kategori:
AmidinesAnti-Infective AgentsAnti-Infective Agents, Local +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dibunate DB13796
small molecule | CAS: 14992-58-6

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 84-74-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAntiparasitic Products, Insecticides and RepellentsCompounds used in a research, industrial, or household setting +4
Target Protein:
Transient receptor potential cation channel subfamily A member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6101–6150 dari 16004
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