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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
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6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 122 / 134
Tenofovir disoproxil Approved DB00300
small molecule | CAS: 201341-05-1

Tenofovir disoproxil fumarate (a prodrug of tenofovir), marketed by Gilead Sciences under the trade name _Viread_, belongs to a class of antiretroviral drugs known as nucleotide analogue reverse transcriptase inhibitors (nRTIs). This drug is prescribed in co…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +19
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseHProtein P
Waktu ParuhWhen a single oral …
Vol. DistribusiThe volume of distr…
KlirensThe clearance of te…
Genetik -
small molecule | CAS: 1208229-58-6

Deskripsi belum tersedia.

Target Protein:
Nuclear factor NF-kappa-B p105 subunitTranscription factor RelBNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teplizumab Approved DB06606
biotech | CAS: 876387-05-2

Teplizumab (teplizumab-mzwv) is a humanized IgG1 kappa CD3-directed monoclonal antibody used to delay the onset of type 1 diabetes (T1D).[A241480,A241045,A241475,L44091] T1D is an autoimmune condition in which T cell-mediated destruction of pancreatic ? cells…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAntibodies +11
Target Protein:
T-cell surface glycoprotein CD3 epsilon chain
Waktu ParuhIn a 60 kg subject,…
Vol. DistribusiIn a 60 kg subject,…
KlirensIn a 60 kg subject,…
Genetik -
Tepotinib Approved DB15133
small molecule | CAS: 1100598-32-0

Tepotinib is a MET tyrosine kinase inhibitor intended to treat a variety of MET-overexpressing solid tumors.[A228058] It was originally developed in partnership between EMD Serono and the University of Texas M.D. Anderson Cancer Center in 2009 and has since b…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +23
Target Protein:
Hepatocyte growth factor receptorNischarinMelatonin receptor type 1B
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe mean apparent v…
KlirensThe apparent cleara…
Genetik -
Tepoxalin DB11466
small molecule | CAS: 103475-41-8

Tepoxalin is a nonsteroidal anti-inflammatory drug approved for veterinary use in the United States and many other countries. It is primarily used to reduce inflammation and relief of pain caused by musculoskeletal disorders such as hip dysplasia and arthriti…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +10
Target Protein:
Interleukin-4Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terameprocol DB12226
small molecule | CAS: 24150-24-1

Terameprocol has been investigated for the treatment of Brain and Central Nervous System Tumors.

Kategori:
Benzene DerivativesBenzyl CompoundsCatechols +2
Target Protein:
Transcription factor Sp1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terevalefim DB16397
small molecule | CAS: 1070881-42-3

Terevalefim is under investigation in clinical trial NCT02474667 (Reduce the Severity of DGF in Recipients of a Deceased Donor Kidney).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teriflunomide Approved DB08880
small molecule | CAS: 163451-81-8

Teriflunomide is the active metabolite of leflunomide, and it acts as an immunomodulatory agent by inhibiting pyrimidine synthesis. It is marketed under the name Aubagio® and is indicated for the treatment of multiple sclerosis, specifically relapsing forms. …

Kategori:
Acids, AcyclicAminesAnalgesics +32
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial3-hydroxy-3-methylglutaryl-coenzyme A reductaseDihydroorotate dehydrogenase (quinone), mitochondrial
Waktu ParuhThe median half-lif…
Vol. DistribusiAfter a single intr…
KlirensAfter a single IV d…
Genetik -
Teriparatide Approved DB06285
biotech | CAS: 52232-67-4

Teriparatide is a recombinant parathyroid hormone (PTH) analog and a potent osteoanabolic agent.[A251395] It is made up of the first amino(N)-terminal 34 amino acids of the human PTH.[A251395] First approved in the United States in November 2002 and in Europe…

Kategori:
Amino Acids, Peptides, and ProteinsBone Anabolic AgentsBone Density Conservation Agents +10
Target Protein:
Parathyroid hormoneParathyroid hormone/parathyroid hormone-related peptide receptor
Waktu ParuhThe half-life of te…
Vol. DistribusiThe volume of distr…
KlirensSystemic clearance …
Genetik -
TERN-101 DB16045
small molecule | CAS: 1103500-20-4

TERN-101 is under investigation in clinical trial NCT04328077 (LIFT Study: A Safety, Tolerability, Efficacy, and Pharmacokinetics Study of TERN-101 in Subjects With Non-cirrhotic Non-alcoholic Steatohepatitis (NASH)).

Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teropavimab DB18916
biotech | CAS: 2417213-72-8

Teropavimab is under investigation in clinical trial NCT05729568 (A Study of GS-5423 and GS-2872 in Combination With Capsid Inhibitor Lenacapavir in Virologically Suppressed Adults With HIV-1 Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Terpin hydrate Approved DB13163
small molecule | CAS: 2451-01-6

Terpin hydrate is an expectorant, commonly used to loosen mucus and ease congestion in patients presenting with acute or chronic bronchitis, and related pulmonary conditions. It is derived from sources such as turpentine, oregano, thyme and eucalyptus. It was…

Kategori:
AlcoholsCyclohexane MonoterpenesCyclohexanes +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TERT-572 DB17286
biotech | CAS: 255706-49-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCarrier ProteinsDNA Nucleotidyltransferases +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tertomotide DB12747
biotech | CAS: 915019-08-8

Tertomotide is under investigation in clinical trial NCT01223209 (A Study, Combination, Immunologic Study of LTX-315 as adjunct to tertomotide in Patients Following Curative Surgery for Carcinoma). It is a peptide vaccine that activates the immune system so t…

Target Protein:
Telomerase reverse transcriptase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tesamorelin Approved DB08869
biotech | CAS: 218949-48-5

Tesamorelin is a stabilized synthetic peptide analogue of the hypothalamic peptide, Growth Hormone Releasing Hormone (GHRH) indicated for the reduction of excess abdominal fat in HIV-infected patients with lipodystrophy. Lipodystrophy is a metabolic condition…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesGrowth Hormone Releasing Factor Analog +17
Target Protein:
Growth hormone-releasing hormone receptor
Waktu Paruh26 and 38 minutes i…
Vol. Distribusi9.4±3.1 L/kg in hea…
Klirens-
Genetik -
Tesetaxel DB12019
small molecule | CAS: 333754-36-2

Tesetaxel has been used in trials studying the treatment of Cancer, Melanoma, Prostate Cancer, Gastric Carcinoma, and Advanced Melanoma, among others.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tesmilifene DB04905
small molecule | CAS: 98774-23-3

Tesmilifene is a novel potentiator of chemotherapy which, when added to doxorubicin, achieved an unexpected and very large survival advantage over doxorubicin alone in a randomized trial in advanced breast cancer.

Kategori:
Antiplatelet agentsBenzene DerivativesCytochrome P-450 CYP2D6 Substrates +18
Target Protein:
ATP-dependent translocase ABCB1Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tesnatilimab DB16377
biotech | CAS: 2242758-08-1

Tesnatilimab is under investigation in clinical trial NCT04655807 (A Study of JNJ-64304500 as Add-on Therapy in Participants With Active Crohn's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Testolactone Approved DB00894
small molecule | CAS: 968-93-4

An antineoplastic agent that is a derivative of progesterone and used to treat advanced breast cancer.

Kategori:
AndrostadienesAndrostanesAndrostenes +7
Target Protein:
Aromatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Testosterone cypionate Approved DB13943
small molecule | CAS: 58-20-8

Testosterone cypionate is a synthetic derivative of testosterone in the form of an oil-soluble 17 (beta)-cyclopentylpropionate ester. Its benefit compared to other testosterone derivatives is the slow rate of release after injection and longer half-life. It w…

Kategori:
Anabolic AgentsAndrogensAndrostanes +33
Target Protein:
Androgen receptorEstrogen receptorMineralocorticoid receptor
Waktu ParuhThe half-life of te…
Vol. DistribusiThe volume of distr…
KlirensTestosterone cypion…
Genetik -
small molecule | CAS: 18625-33-7

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesAndrostenols +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Testosterone enanthate Approved DB13944
small molecule | CAS: 315-37-7

Testosterone enanthate is an esterified variant of testosterone that comes as an injectable compound with a slow-release rate. This slow release is achieved by the presence of the enanthate ester functional group attached to the testosterone molecule.[A31615…

Kategori:
Adrenal Cortex HormonesAndrogensAndrostanes +34
Target Protein:
Androgen receptorEstrogen receptorMineralocorticoid receptor
Waktu ParuhTestosterone enanth…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
small molecule | CAS: 521-15-3

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesAndrostenols +9
Target Protein:
Neocarzinostatin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Testosterone undecanoate Approved DB13946
small molecule | CAS: 5949-44-0

Testosterone undecanoate is the ester prodrug of [testosterone] and has a mid-chain fatty acid at the carbon 17? position.[L35970] It was developed via fatty acid esterification of testosterone in order to achieve orally administer testosterone.[A246594] Ther…

Kategori:
AndrogensAndrostanesAndrostenes +32
Target Protein:
Androgen receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThere is no informa…
KlirensWhile there is limi…
Genetik -
Tetrabenazine Approved DB04844
small molecule | CAS: 58-46-8

A drug formerly used as an antipsychotic but now used primarily in the symptomatic treatment of various hyperkinetic disorders. It is a monoamine depletor and used as symptomatic treatment of chorea associated with Huntington's disease. FDA approved on August…

Kategori:
Adrenergic AgentsCytochrome P-450 CYP2D6 SubstratesCytochrome P-450 Substrates +11
Target Protein:
Synaptic vesicular amine transporterD(2) dopamine receptor
Waktu ParuhThere is interindiv…
Vol. DistribusiSteady State, IV, i…
KlirensIV, 1.67 L/min in H…
Genetik -
Tetracaine Approved DB09085
small molecule | CAS: 94-24-6

Tetracaine is an ester local anaesthetic currently available in combination with lidocaine as a cream and patch.

Kategori:
Acids, CarbocyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAminobenzoates +23
Target Protein:
Ryanodine receptor 1Sodium channel protein type 10 subunit alphaRyanodine receptor 2 +1
Waktu ParuhTetracaine is hydro…
Vol. DistribusiTetracaine is rapid…
KlirensTetracaine is hydro…
Genetik -
Tetrachlorodecaoxide Approved DB05389
small molecule | CAS: 92047-76-2

WF10 is a chlorite-based, immunomodulating drug is developed by Nuvo Research Inc. Certain preclinical evidence and clinical pilot data suggest that WF10 may be effective in treating certain cancers. The Corporation believes the research to-date demonstrates …

Kategori:
AnionsCompounds used in a research, industrial, or household settingElectrolytes +7
Target Protein:
E3 ubiquitin-protein transferase MAEAScavenger receptor cysteine-rich type 1 protein M130
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tetracosactide Approved DB01284
small molecule | CAS: 16960-16-0

Tetracosactide (also known as Cosyntropin) is a synthetic peptide that is identical to the 24-amino acid segment (sequence: SYSMEHFRWGKPVGKKRRPVKVYP) at the N-terminal of adrenocorticotropic hormone. ACTH (1-24), a segment similar in all species, contains the…

Kategori:
AdrenalsAdrenocortical InsufficiencyAdrenocorticotropic Hormone +16
Target Protein:
Adrenocorticotropic hormone receptor
Waktu ParuhAbout 15 minutes fo…
Vol. Distribusi-
Klirens-
Genetik -
Tetracycline Approved DB00759
small molecule | CAS: 60-54-8

Tetracycline is a broad spectrum polyketide antibiotic produced by the Streptomyces genus of Actinobacteria. It exerts a bacteriostatic effect on bacteria by binding reversible to the bacterial 30S ribosomal subunit and blocking incoming aminoacyl tRNA from b…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAnti-Bacterial Agents +32
Target Protein:
30S ribosomal protein S730S ribosomal protein S1430S ribosomal protein S3 +6
Waktu Paruh6-12 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 300-52-7

Sodium tetradecyl sulfate is an anionic surface-active agent which is used for its wetting properties in the industry and is also used in medicine as a blood vessel irritant and sclerosing agent for hemorrhoids and varicose veins [L2031]. Sodium tetradecyl…

Kategori:
Drugs that are Mainly Renally Excreted
Target Protein:
Endothelial protein C receptor
Waktu Paruh-
Vol. DistribusiIn humans, a large …
Klirens-
Genetik -
small molecule | CAS: 2921-20-2

Deskripsi belum tersedia.

Kategori:
AnionsAntioxidantsBiological Factors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 66-40-0

Tetraethylammonium is an experimental drug with no approved indication or marketed formulation. The only marketed drug containing tetraethylammonium was a combination drug called Fosglutamina B6, but this drug has now been discontinued. As an experimental age…

Kategori:
AminesCardiovascular AgentsGanglion Blockers +9
Target Protein:
Potassium voltage-gated channel subfamily KQT member 3Potassium channel subfamily T member 2Potassium channel subfamily T member 1 +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Tetraferric tricitrate decahydrate is an iron containing phosphate binder used to treat hyperphosphatemia and iron deficiency anemia in adults with chronic kidney disease.[A25965] Tetraferric tricitrate decahydrate was granted FDA approval on 5 September 2…

Kategori:
Anemia, Iron-DeficiencyDrugs for Treatment of Hyperkalemia and HyperphosphatemiaIron Compounds +2
Target Protein:
Transferrin receptor protein 1Iron(3+)-hydroxamate-binding protein FhuD
Waktu Paruh-
Vol. Distribusi-
KlirensData regarding the …
Genetik -
small molecule | CAS: 53008-15-4

Deskripsi belum tersedia.

Kategori:
Blood and Blood Forming OrgansHemostaticsLocal Hemostatics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Blasticidin-S deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 31262-37-0

Tetrahydrocannabivarin (THCV) is a propyl analogue of tetrahydrocannabinol (?9-THC), one of the primary pharmacological components of [Medical Cannabis]. ?9-THC is currently available in several synthetic forms, including [Dronabinol], while purified or isola…

Kategori:
Agents that produce hypertensionAntidepressive AgentsCentral Nervous System Depressants +3
Target Protein:
Transient receptor potential cation channel subfamily V member 3Cannabinoid receptor 1G-protein coupled receptor 55 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 135-16-0

Tetrahydrofolic acid is a folic acid derivative that is produced from dihydrofolic acid after conversion by dihydrofolate reductase. It is converted into 5,10-methylenetetrahydrofolate by serine hydroxymethyltransferase. It is a soluble coenzyme in many react…

Kategori:
CoenzymesDietary SupplementsEnzymes and Coenzymes +7
Target Protein:
C-1-tetrahydrofolate synthase, cytoplasmicBifunctional methylenetetrahydrofolate dehydrogenase/cyclohydrolase, mitochondrialAminomethyltransferase, mitochondrial +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 67-30-1

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 16330-92-0

Tetrathiomolybdate is an oral, small-molecule, anticopper agent that is highly specific for lowering the levels of free copper in serum. COPREXA has completed pivotal clinical trials for the treatment of neurologic Wilson's disease. It is also developed for f…

Kategori:
Adenosine Triphosphatases, antagonists & inhibitorsAngiogenesis Modulating AgentsAntineoplastic Agents +10
Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tetryzoline Approved DB06764
small molecule | CAS: 84-22-0

Tetryzoline, also known as tetrahydrozoline, is a derivative of imidazoline with central and peripheral alpha (?)-adrenergic properties.[A231769] Available since the 1950s, tetryzoline is a selective ?<sub>1</sub>-receptor agonist [A231774] that is used as a…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +20
Target Protein:
Alpha-1 adrenergic receptorsAlpha-2C adrenergic receptorAlpha-2 adrenergic receptors
Waktu ParuhFollowing ocular ad…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Tezacaftor Approved DB11712
small molecule | CAS: 1152311-62-0

Tezacaftor is a drug of the cystic fibrosis transmembrane conductance regulator (CFTR) potentiator class.[L1595] It was developed by Vertex Pharmaceuticals and FDA approved in combination with [ivacaftor] to manage cystic fibrosis.[L6814] This drug was approv…

Kategori:
BCRP/ABCG2 InhibitorsBCRP/ABCG2 SubstratesCytochrome P-450 CYP1A2 Inhibitors +33
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Tezacitabine DB06433
small molecule | CAS: 171176-43-5

A synthetic purine nucleoside analogue with potential antineoplastic activity.

Kategori:
Antineoplastic AgentsDeoxyribonucleosidesEnzyme Inhibitors +6
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tezepelumab Approved DB15090
biotech | CAS: 1572943-04-4

Asthma is a heterogeneous chronic obstructive respiratory disease with both "type 2" (T2) and T2-low endotypes characterized by reduced airflow, chronic inflammation, and airway remodelling.[A243764, A243769] Thymic stromal lymphopoietin (TSLP), an innate ple…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Thymic stromal lymphopoietin
Waktu ParuhTezepelumab has an …
Vol. DistribusiTezepelumab has a c…
KlirensTezepelumab has an …
Genetik -
TG-100801 DB05075
small molecule | CAS: 867331-82-6

TG100801 is a topically applied kinase inhibitor in macular degeneration patients. It is administered noninvasively as an eye drop and is designed to suppress VEGF mediated leakage and additional kinase targets associated with inflammation, edema, and angioge…

Kategori:
Benzene Derivatives
Target Protein:
Vascular endothelial growth factor CVascular endothelial growth factor DVascular endothelial growth factor A, long form +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG01 vaccine DB17123
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG4010 DB06584
biotech | CAS: 350485-85-7

A bivalent cancer vaccine comprised of a modified vaccinia virus Ankara (MVA) strain encoding human mucin 1 (MUC1) and interleukin-2 (IL-2) with potential immunostimulating and antineoplastic activities. Originally developed for the eradication of smallpox, M…

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsCarbohydrates +6
Target Protein:
Mucin-1Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TG4023 DB06108
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TGAAC09 DB06363
biotech

tgAAC09 is an investigational vaccine that utilizes an AAV vector to deliver genes that encode HIV proteins. It was under investigation in clinical trials NCT00482027 and NCT00888446 for the treatment of HIV Infection.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TGAAC94 DB06175
small molecule

tgAAC94 is a recombinant adeno-associated virus serotype 2 (AAV2) vector containing the cDNA for a human tumor necrosis factor receptor (TNFR)-immunoglobulin (IgG1) Fc fusion (TNFR:Fc) gene. It was under investigation in clinical trials to treat Inflammatory …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
tgAAG-76 DB18421
biotech

tgAAG-76 consists of a recombinant adeno-associated virus (serotype 2) (rAAV2) gene transfer agent expressing RPE65.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6051–6100 dari 6694
Sebelumnya Halaman 122 / 134 Berikutnya