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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 122 / 252
GPI-0100 DB05929
small molecule

GPI-0100 is Avantogen’s lead adjuvanat-immunopotentiator, a key component of vaccines for boosting the immune response. The GPI-0100 adjuvant, which has been shown to significantly enhance the immune response with a variety of vaccines, has been shown to hav…

Kategori:
CarbohydratesGlycosides
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Gpi-1046 DB01951
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GPI-1485 DB05814
small molecule | CAS: 186268-78-0

GPI 1485 is a product candidate that belongs to a class of small molecule compounds called neuroimmunophilin ligands. In preclinical experiments, neuroimmunophilin ligands have been shown to repair and regenerate damaged nerves without affecting normal, heal…

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 InhibitorsCytochrome P-450 CYP3A4 Inhibitors (strength unknown) +2
Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GR270773 DB06427
small molecule

GR270773, was investigated in two clinical trials for its potential to treat sepsis: NCT00158769 (completed, comparing the effects of infusion between healthy adults and those with damaged livers) and NCT00089986 (completed with results, treatment of suspecte…

Waktu Paruh-
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Gramicidin D Approved DB00027
small molecule | CAS: 1405-97-6

Gramcidin D is a heterogeneous mixture of three antibiotic compounds, gramicidins A, B and C, making up 80%, 6%, and 14% respectively all of which are obtained from the soil bacterial species Bacillus brevis and called collectively gramicidin D. Gramcidins ar…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Dihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Granaticin B DB17273
small molecule | CAS: 19879-03-9

Deskripsi belum tersedia.

Kategori:
BenzopyransBenzoquinonesChromans +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Granisetron Approved DB00889
small molecule | CAS: 109889-09-0

A serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic and antinauseant for cancer chemotherapy patients.

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +23
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh4-6 hours in health…
Vol. Distribusi-
Klirens* 0.52 L/h/kg [Canc…
Genetik -
Granotapide DB12934
small molecule | CAS: 594842-13-4

Granotapide has been used in trials studying the treatment of Type II Diabetes Mellitus.

Kategori:
Acids, AcyclicAcids, CarbocyclicAmides +3
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Grape Approved DB10533
biotech

Grape allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Grape seed oil DB14323
biotech | CAS: 8016-21-5

Grape seed oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Grapefruit Approved DB10534
biotech

Grapefruit allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Grapefruit oil DB15663
biotech | CAS: 8016-20-4

Deskripsi belum tersedia.

Waktu Paruh-
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Graphite Approved DB18717
small molecule | CAS: 7782-42-5

Deskripsi belum tersedia.

Kategori:
CarbonElementsGraphite +1
Waktu Paruh-
Vol. Distribusi-
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Grapiprant DB12836
small molecule | CAS: 415903-37-6

Grapiprant, also known as AT-001 and CJ-023, is a drug from the piprant class. These molecules were derived from acylsulfonamide and are characterized to be a novel series of para-N-acylaminomethylbenzoic acid known to be prostaglandin receptor antagonists.[A…

Kategori:
AmidesBenzene DerivativesP-glycoprotein substrates +3
Target Protein:
Prostaglandin E2 receptor EP4 subtype
Waktu ParuhThe reported elimin…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik -
Grazoprevir Approved DB11575
small molecule | CAS: 1350514-68-9

Grazoprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nin…

Kategori:
Acids, AcyclicAmidesAnti-Infective Agents +24
Target Protein:
Genome polyprotein
Waktu ParuhThe geometric mean …
Vol. DistribusiGrazoprevir has an …
KlirensThe clearance of Gr…
Genetik -
Green bell pepper Approved DB10556
biotech

Green bell pepper allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Gremubamab DB15014
biotech | CAS: 1800381-36-5

Gremubamab is under investigation in clinical trial NCT02255760 (Phase 1 Randomized Double-blind Placebo Controlled Study to Evaluate Safety and PK of MEDI3902 in Healthy Adults).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Grepafloxacin Approved DB00365
small molecule | CAS: 119914-60-2

Grepafloxacin is an oral broad-spectrum quinoline antibacterial agent used to treat bacterial infections. Due to the QTc-prolonging potential, as indicated by the changes in the QT interval on the electrocardiogram, and the risk for cardiovascular adverse eve…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu Paruh15 ± 3 hours
Vol. Distribusi-
Klirens-
Genetik -
Gresonitamab DB18210
biotech | CAS: 2413817-97-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Grn163l DB05036
small molecule

GRN163L is a novel anti-cancer drug. It has been characterized preclinically and shown to inhibit telomerase in human tumor cells of many cancer types (including lung, breast, prostate, liver, and early stage of human breast cancer), in both cell culture syst…

Target Protein:
Telomerase-binding protein EST1AN-terminal kinase-like proteinProstaglandin E synthase 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GRObeta DB18205
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 141925-59-9

Growth hormone-releasing peptide 1 is under investigation in clinical trial NCT00381602 (A Phase II, Randomized, Cross-over, Vehicle-controlled, Double-blind, Multicenter Study of the Safety, Pharmacodynamics, and Preliminary Efficacy of GHRP-1/AG in Subjects…

Kategori:
Amino Acids, Peptides, and ProteinsGrowth Hormone-Releasing HormonePeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GS 0573 DB08843
small molecule | CAS: 113852-41-8

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsHeterocyclic Compounds, Fused-RingImmunologic Factors +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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GS-441524 DB15686
small molecule | CAS: 1191237-69-0

GS-441524 is an adenosine nucleotide analog antiviral, similar to [remdesivir].[A203057,L13239] This molecule was patented in 2009.[L13775] _In vitro_ studies of GS-441524 have determined it has a higher EC<sub>50</sub> than remdesivir against a number of vir…

Kategori:
Adenine NucleotidesAnti-Infective AgentsAntiviral Agents +10
Target Protein:
Replicase polyprotein 1abRNA-directed RNA polymerase L
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GS-5745 DB12296
biotech | CAS: 1518996-49-0

GS-5745 has been used in trials studying the treatment of Tumors, Breast Cancer, Crohn's Disease, Colorectal Cancer, and Pancreatic Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GS-6620 DB15222
small molecule | CAS: 1350735-70-4

GS-6620 is under investigation in clinical trial NCT01316237 (A Study Evaluating the Safety, Tolerability, Pharmacokinetics and Antiviral Activity of GS-6620 in Treatment Naïve Subjects With Chronic Hepatitis C Virus Infection).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GS-9191 DB15084
small molecule | CAS: 859209-84-0

GS-9191 is under investigation in clinical trial NCT00499967 (Safety and Effectiveness Study of an Experimental Topical Ointment (GS-9191) for the Treatment of Genital Warts).

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Waktu Paruh-
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Klirens-
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GS-9256 DB12876
small molecule | CAS: 1001094-46-7

GS-9256 has been used in trials studying the treatment of HCV Infection and Chronic Hepatitis C Infection.

Kategori:
AcidsAcids, NoncarboxylicAmino Acids, Peptides, and Proteins +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GS030-DP DB17847
biotech

GS030-DP is an optogenetic gene therapy being investigated for the treatment of retinitis pigmentosa. It targets retinal ganglion cells that encodes a light-sensitive channelrhodopsin, ChrimsonR-tdTomato (ChR-tdT), delivered by an AAV2.7m8 vector. It is a com…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSBR-1290 DB18551
small molecule

GSBR-1290 is a small molecule agonist of the GLP-1 receptor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-1004723 DB12806
small molecule | CAS: 955359-72-5

Gsk1004723 has been investigated for the treatment of Allergic Rhinitis and Rhinitis, Allergic, Seasonal.

Kategori:
Histamine AntagonistsHistamine H1 AntagonistsPyridazines
Target Protein:
Histamine H3 receptorHistamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-1059615 DB11962
small molecule | CAS: 958852-01-2

GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, Solid Tumor Cancer, and Metastatic Breast Cancer.

Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 3-kinase catalytic subunit type 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-1292263 DB12627
small molecule | CAS: 1032823-75-8

GSK1292263 has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.

Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-1521498 DB12886
small molecule | CAS: 1007573-18-3

GSK1521498 has been used in trials studying the treatment of Obesity and Alcoholism.

Kategori:
IndenesReceptors, Opioid, mu
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-239512 DB15120
small molecule | CAS: 720691-69-0

GSK-239512 is under investigation in clinical trial NCT00474513 (An Imaging Study to Investigate the Distribution of GSK239512 in the Brain.).

Kategori:
Heterocyclic Compounds, Fused-RingHistamine Antagonists
Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-256066 DB12137
small molecule | CAS: 801312-28-7

Gsk256066 has been used in trials studying the treatment and diagnostic of SAR, Asthma, Mild Asthma, Allergic Rhinitis, and Seasonal Allergic Rhinitis, among others.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPhosphodiesterase 4 Inhibitors +3
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
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GSK-2636771 DB11795
small molecule | CAS: 1372540-25-4

GSK2636771 has been used in trials studying the treatment of CANCER, LYMPHOMA, Solid Neoplasm, Recurrent Solid Neoplasm, and Advanced Malignant Neoplasm, among others.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsOxazines +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
Waktu Paruh-
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Genetik -
GSK-269962A DB17030
small molecule | CAS: 850664-21-0

GSK-269962A is a Rho kinase (ROCK) inhibitor with both ROCK1 and ROCK2 affinity.[A253012]

Kategori:
Oxazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-2879552 DB16895
small molecule | CAS: 1401966-69-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesCycloparaffins
Target Protein:
Lysine-specific histone demethylase 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-2881078 DB16888
small molecule | CAS: 1539314-06-1

Deskripsi belum tersedia.

Kategori:
Anabolic AgentsHeterocyclic Compounds, Fused-RingHormones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-2982772 DB16875
small molecule | CAS: 1622848-92-3

Deskripsi belum tersedia.

Target Protein:
Receptor-interacting serine/threonine-protein kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-3117391 DB15440
small molecule | CAS: 1018673-42-1

GSK-3117391 is under investigation in clinical trial NCT02965599 (Efficacy, Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of GSK3117391 in Subjects With Rheumatoid Arthritis).

Waktu Paruh-
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GSK-356278 DB12542
small molecule | CAS: 720704-34-7

Gsk356278 has been used in trials studying the treatment and basic science of Anxiety Disorders, Huntington Disease, Depressive Disorder, Huntingtons Disease, and Depressive Disorder, Major, among others.

Kategori:
OxazolesSulfur Compounds
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-364735 DB13119
small molecule | CAS: 863434-13-3

GSK-364735 (Naphthyridinone) has been used in trials studying the treatment of HIV-1 Infection and Infection, Human Immunodeficiency Virus.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-376501 DB12654
small molecule | CAS: 1010412-80-2

GSK376501 has been used in trials studying the treatment and diagnostic of Type 2 Diabetes Mellitus.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-690693 DB12745
small molecule | CAS: 937174-76-0

GSK690693 has been used in trials studying the treatment of Tumor, CANCER, and Lymphoma.

Kategori:
Oxazoles
Target Protein:
RAC-gamma serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-923295 DB06097
small molecule

GSK-923295 is a small-molecule inhibitor of the mitotic kinesin centromere-associated protein E (CENP-E), and the third novel drug candidate to arise from Cytokinetics' broad strategic alliance with GlaxoSmithKline (GSK). GSK-923295 demonstrated a broad spect…

Target Protein:
Centromere-associated protein E
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-945237 DB15345
small molecule | CAS: 944406-54-6

GSK-945237 is under investigation in clinical trial NCT01039610 (A Single Center Four Part Study in Healthy Adult Subjects to Evaluate: the Safety, Tolerability and Pharmacokinetics of a Single Oral Dose and Repeat Escalating Oral Doses of GSK945237; the Effe…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Klirens-
Genetik -
GSK159797 DB05043
small molecule

GSK159797 ('797) is an inhaled, longer-acting Beta2 agonist developed for the treatment of respiratory disease such as asthma and COPD.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
GSK2245035 DB16076
small molecule | CAS: 1207629-49-9

GSK2245035 is under investigation in clinical trial NCT02833974 (Effect of the GSK2245035 on the Allergen-induced Asthmatic Response).

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6051–6100 dari 12560
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