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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 122 / 282
ET-101 DB18255
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ET140203 DB17196
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Etacrynic acid Approved DB00903
small molecule | CAS: 58-54-8

A compound that inhibits symport of sodium, potassium, and chloride primarily in the ascending limb of Henle, but also in the proximal and distal tubules. This pharmacological action results in excretion of these ions, increased urinary output, and reduction …

Kategori:
AcetatesAcids, AcyclicAgents that produce neuromuscular block (indirect) +16
Target Protein:
Solute carrier family 12 member 1Sodium/potassium-transporting ATPase subunit alpha-1Lymphoid enhancer-binding factor 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etafedrine Approved DB11587
small molecule | CAS: 48141-64-6

Etafedrine (INN) or ethylephedrine is a long-acting bronchodilator and has been an ingredient combined with other drugs in the brand names Nethaprin [A32757] and Dalmacol [L2568]. It was previously available as both the free base and as the hydrochloride salt…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +10
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIt has a plasma hal…
Vol. DistribusiSimilar to ephedrin…
Klirens-
Genetik -
Etalocib DB12850
small molecule | CAS: 161172-51-6

Etalocib has been used in trials studying the treatment of Pancreatic Cancer, Carcinoma, Non-Small-Cell Lung, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Acids, CarbocyclicBenzene Derivatives
Target Protein:
Leukotriene B4 receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etamicastat DB15288
small molecule | CAS: 760173-05-5

Etamicastat is under investigation in clinical trial NCT02840565 (Tolerability, Pharmacokinetics and Pharmacodynamics of Six Multiple Rising Dose Regimens of BIA 5-453).

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Dopamine beta-hydroxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etamiphylline DB13592
small molecule | CAS: 314-35-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnti-Asthmatic AgentsAutonomic Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etamsylate DB13483
small molecule | CAS: 2624-44-4

Deskripsi belum tersedia.

Kategori:
ArylsulfonatesArylsulfonic AcidsBenzene Derivatives +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etanercept Approved DB00005
biotech | CAS: 185243-69-0

Dimeric fusion protein consisting of the extracellular ligand-binding portion of the human 75 kilodalton (p75) tumor necrosis factor receptor (TNFR) linked to the Fc portion of human IgG1.[L14862,A216522] The Fc component of etanercept contains the CH2 domain…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +18
Target Protein:
Tumor necrosis factorLymphotoxin-alphaHigh affinity immunoglobulin gamma Fc receptor I +6
Waktu ParuhEtanercept has a me…
Vol. DistribusiPopulation pharmaco…
KlirensEtanercept has a me…
Genetik -
Etanidazole DB12736
small molecule | CAS: 22668-01-5

Etanidazole has been used in trials studying the diagnostic of Adult Ependymoma, Malignant Ascites, Adult Gliosarcoma, Adult Mixed Glioma, and Adult Glioblastoma, among others.

Kategori:
Antineoplastic AgentsImidazolesNitro Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etaracizumab DB12213
biotech | CAS: 892553-42-3

Etaracizumab has been investigated for the treatment of Psoriasis, Renal Cell Carcinoma, Stage IV Renal Cell Cancer, Recurrent Renal Cell Cancer, and Stage III Renal Cell Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etarfolatide DB11810
small molecule | CAS: 479578-27-3

Etarfolatide has been used in trials studying the treatment and diagnostic of Breast Neoplasms, Non Small Cell Lung Cancer, and Adenocarcinoma of the Lung.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etavopivat DB18176
small molecule | CAS: 2245053-57-8

Etavopivat is a small molecule activator of erythrocyte pyruvate kinase (PKR) under investigation for the treatment of sickle cell disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etazolate DB05881
small molecule

EHT 0202 is developed to treat neurodegenerative disorders by ExonHit Therapeutics.

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ETBX-021 DB17528
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
ETBX-041 DB17182
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ETBX-051 DB17529
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etelcalcetide Approved DB12865
small molecule | CAS: 1262780-97-1

Etelcalcetide is a calcimimetic drug for the treatment of secondary hyperparathyroidism in patients undergoing hemodialysis. Etelcalcetide was approved (trade name Parsabiv) for the treatment of secondary hyperparathyroidism (HPT) in adult patients with chron…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Parathyroid AgentsCalcium Homeostasis +3
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh3 to 4 days
Vol. Distribusi796 L
Klirens7.66 L/hr
Genetik -
Eteplirsen Approved DB06014
biotech | CAS: 1173755-55-9

Eteplirsen is a synthetic antisense oligonucleotide and a phosphorodiamidate morpholino oligomer. It consists of a six-membered morpholino ring replacing the five-membered ribofuranosyl rings found in natural DNA and RNA.[L40015] Duchenne muscular dystrop…

Kategori:
Antisense OligonucleotidesMorpholinesMusculo-Skeletal System +5
Target Protein:
DMD-001 gene (exon 51 target site)
Waktu ParuhThe elimination hal…
Vol. DistribusiFollowing weekly in…
KlirensThe total clearance…
Genetik -
Etesevimab DB15897
biotech | CAS: 2423948-94-9

Etesevimab (LY-CoV016, also known as JS016) is a fully human and recombinant monoclonal antibody that targets the SARS-CoV-2 surface spike protein receptor binding domain.[L16651,L16661] Under the EUA granted in February 2021, etesevimab is used in combinatio…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etevritamab DB17211
biotech | CAS: 2329692-74-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethacridine DB13190
small molecule | CAS: 442-16-0

Deskripsi belum tersedia.

Kategori:
Acridine DerivativesAcridinesAminoacridines +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethadione DB13799
small molecule | CAS: 520-77-4

Deskripsi belum tersedia.

Kategori:
AnticonvulsantsCentral Nervous System DepressantsNervous System +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethambutol Approved DB00330
small molecule | CAS: 74-55-5

Ethambutol is a bacteriostatic agent indicated alongside medications such as [isoniazid], [rifampin], and [pyrazinamide] in the treatment of pulmonary tuberculosis.[L31743] Ethambutol was first described in the literature in 1961.[A229048] It was developed ou…

Kategori:
AminesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
Probable arabinosyltransferase CProbable arabinosyltransferase BProbable arabinosyltransferase A
Waktu ParuhEthambutol has a ha…
Vol. DistribusiPatients coinfected…
KlirensPatients coinfected…
Genetik -
small molecule | CAS: 594-45-6

Deskripsi belum tersedia.

Kategori:
AlkanesAlkanesulfonic AcidsHydrocarbons, Acyclic +3
Target Protein:
Platelet basic proteinPhosphonoacetaldehyde hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethanolamine DB03994
small molecule | CAS: 141-43-5

A viscous, hygroscopic amino alcohol with an ammoniacal odor. It is widely distributed in biological tissue and is a component of lecithin. It is used as a surfactant, fluorimetric reagent, and to remove CO2 and H2S from natural gas and other gases.

Kategori:
AlcoholsAminesAmino Alcohols +4
Target Protein:
Surface protein AAnnexin A3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethanolamine oleate Approved DB06689
small molecule | CAS: 2272-11-9

Ethanolamine oleate is a mild sclerosing agent. It is composed of ethanolamine, a basic substance, which when combined with oleic acid forms a clear, straw to pale yellow colored, deliquescent oleate.

Kategori:
Antivaricose TherapyCardiovascular AgentsCompounds used in a research, industrial, or household setting +10
Target Protein:
Calcium ionsCoagulation factor XII
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethaselen DB15051
small molecule | CAS: 217798-39-5

Ethaselen is under investigation in clinical trial NCT02166242 (Ethaselen for the Treatment of Thioredoxin Reductase High Expression Advanced Non-small Cell Lung Cancers).

Kategori:
Selenium Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethchlorvynol Approved DB00189
small molecule | CAS: 113-18-8

Ethchlorvynol is a sedative and hypnotic drug. It has been used to treat insomnia, but has been largely superseded and is only offered where an intolerance or allergy to other drugs exists.

Kategori:
AlcoholsCentral Nervous System AgentsCentral Nervous System Depressants +4
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit alpha-1GABA(A) Receptor
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Etheno-NAD DB02483
small molecule

Deskripsi belum tersedia.

Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2L-lactate dehydrogenase A chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etheno-Nadp DB03732
small molecule

Deskripsi belum tersedia.

Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethinamate Approved DB01031
small molecule | CAS: 126-52-3

Ethinamate is a short-acting sedative-hypnotic medication used to treat insomnia. Like many such similar medications, the regular use of ethinamate can result in the development of drug tolerance in a patient. Nevertheless, the medication itself is generally …

Kategori:
Acids, Acyclic
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 1
Waktu Paruh2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Ethinylestradiol Approved DB00977
small molecule | CAS: 57-63-6

Ethinylestradiol was first synthesized in 1938 by Hans Herloff Inhoffen and Walter Hohlweg at Schering.[A191107] It was developed in an effort to create an estrogen with greater oral bioavailability.[A191107] These properties were achieved by the substitution…

Kategori:
Adrenal Cortex HormonesAntineoplastic and Immunomodulating AgentsBSEP/ABCB11 inducers +48
Target Protein:
Estrogen receptorNuclear receptor subfamily 1 group I member 2
Waktu ParuhA 30µg oral dose ha…
Vol. DistribusiA 30µg oral dose ha…
KlirensEthinylestradiol ha…
Genetik -
Ethionamide Approved DB00609
small molecule | CAS: 536-33-4

A second-line antitubercular agent that inhibits mycolic acid synthesis. It also may be used for treatment of leprosy. (From Smith and Reynard, Textbook of Pharmacology, 1992, p868)

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiinfectives for Systemic Use +9
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]Nuclear factor erythroid 2-related factor 2Catalase-peroxidase
Waktu Paruh2 to 3 hours
Vol. Distribusi* 93.5 L [healthy v…
Klirens-
Genetik -
Ethosuximide Approved DB00593
small molecule | CAS: 77-67-8

An anticonvulsant especially useful in the treatment of absence seizures unaccompanied by other types of seizures.

Kategori:
Agents causing hyperkalemiaAnti-epileptic AgentAntiarrhythmic agents +18
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1G
Waktu Paruh53 hours
Vol. Distribusi-
Klirens-
Genetik -
Ethotoin Approved DB00754
small molecule | CAS: 86-35-1

Ethotoin is a hydantoin derivative and anticonvulsant. Ethotoin exerts an antiepileptic effect without causing general central nervous system depression. The mechanism of action is probably very similar to that of phenytoin. The latter drug appears to stabili…

Kategori:
Anti-epileptic AgentAnticonvulsantsCardiovascular Agents +14
Target Protein:
Sodium channel protein type 5 subunit alphaNuclear receptor subfamily 1 group I member 2
Waktu Paruh3 to 9 hours
Vol. Distribusi-
Klirens-
Genetik -
Ethoxyquin DB16866
small molecule | CAS: 91-53-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethoxzolamide DB00311
small molecule | CAS: 452-35-7

Ethoxzolamide is a sulfonamide used as diuretic and in glaucoma. It inhibits carbonic anhydrase activity in proximal renal tubules to decrease reabsorption of water, sodium, potassium, bicarbonate. Its pharmacological activity thus confers the risk for hypoka…

Kategori:
AmidesBenzothiazolesCarbonic Anhydrase Inhibitors +9
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 4Carbonic anhydrase 7 +2
Waktu Paruh2.5-5.5 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Lactase/phlorizin hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15400-53-0

Deskripsi belum tersedia.

Target Protein:
Dihydroneopterin aldolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Dual specificity protein kinase CLK1Dual specificity tyrosine-phosphorylation-regulated kinase 1ADual specificity protein kinase CLK3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase, inducibleNitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 686723-15-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 548-00-5

Ethyl biscoumacetate is a courmarin that is used as an anticoagulant. It has actions similar to those of Warfarin. (From Martindale, The Extra Pharmacopoeia, 30th ed, p226)

Kategori:
4-HydroxycoumarinsAnticoagulantsBenzopyrans +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethyl butyrate DB15454
small molecule | CAS: 105-54-4

Ethyl butyrate is under investigation in clinical trial NCT03202342 (fMRI of Hypothalamic Responses to Taste, Temperature and Glucose).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethyl chloride Approved DB13259
small molecule | CAS: 75-00-3

Ethyl chloride, or chloroethane, has a chemical formula C2H5Cl. It was commonly used in the production of tetraethyllead (TEL), which is an additive for gasoline. It was also used in other commerical applications as a chemical reagent. It is still used in the…

Kategori:
AnestheticsAnesthetics, LocalCentral Nervous System Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1623-14-9

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAnions +7
Target Protein:
CholinesteraseParathion hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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