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6694

Total database: 17430
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4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
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6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 121 / 134
small molecule | CAS: 374107-43-4

99mTc-Ciprofloxacin is a new formulation of ciprofloxacin (INFECTON), being investigated as a radioimaging agent for the potential diagnosis of infection, including fever of unknown origin, osteomyelitis, wound infection, abdominal abscess, pneumonia, appendi…

Kategori:
4-QuinolonesAnti-Bacterial AgentsCytochrome P-450 CYP1A2 Inhibitors +9
Target Protein:
DNA gyrase subunit BDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Technetium Tc-99m disofenin Approved DB09164
small molecule

Technetium Tc-99m disofenin is a radiopharmaceutical agent used in hepatobiliary imaging for diagnostic purposes. It is well suited for both planar and single photon tomographic scintigraphy to quantitatively measure the function of liver, gallbladder and bil…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +15
Waktu ParuhTechnetium Tc99m de…
Vol. DistribusiTechnetium Tc99M di…
KlirensTechnetium Tc 99M D…
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsLigandsOrganometallic Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Technetium Tc-99m mebrofenin Approved DB09137
small molecule | CAS: 1415247-71-0

Technetium Tc 99m Mebrofenin is a diagnostic radiopharmaceutical composed of diisopropyl-iminodiacetic acid (DISIDA) attached to a technetium-99m ion. Following intravenous injection, single photon emission computer tomography (SPECT) imaging of the liver o…

Kategori:
AminesAmino AcidsAmino Acids, Peptides, and Proteins +14
Waktu ParuhTechnetium Tc 99m d…
Vol. Distribusi-
KlirensFollowing intraveno…
Genetik -
Technetium Tc-99m medronate Approved DB09138
small molecule | CAS: 121524-79-6

Technetium (99mTc) medronic acid is a pharmaceutical product used in nuclear medicine imaging. It is composed of a technetium ion complexed with medronic acid, a type of bisphosphonate. Like other bisphosphonates used in the treatment of osteoporosis, medroni…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +11
Waktu ParuhTechnetium Tc-99m d…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 165942-79-0

Technetium Tc-99m nofetumomab merpentan (Tc-99m nm) consists of a Fab fragment of an IgG2b of the pancarcinoma murine antibody NR-LU-10.[A32115] The NR-LU-10 antibody is directed against a 40 kDa glycoprotein antigen expressed in a variety of cancers and some…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Epithelial cell adhesion moleculeB-lymphocyte antigen CD20
Waktu ParuhThe radioactive hal…
Vol. Distribusi-
Klirens-
Genetik -
Technetium Tc-99m oxidronate Approved DB09139
small molecule | CAS: 72945-61-0

Technetium Tc-99m oxidronate, also known as 99mTc-methylene diphosphonate, is a radiopharmaceutical agent. A radiopharmaceutical is defined as a medicinal formulation containing radioisotopes that are used in major clinical areas for diagnosis and/or therapy.…

Kategori:
Diagnostic RadiopharmaceuticalsDrugs that are Mainly Renally ExcretedOrganometallic Compounds +6
Waktu ParuhThe elimination of …
Vol. DistribusiThe distribution of…
KlirensDuring the first 24…
Genetik -
small molecule | CAS: 23288-61-1

Technetium Tc-99m pertechnetate is a radiopharmaceutical diagnostic agent composed of an oxoanion with the chemical formula TcO4-. Pertechnetate has a wide variety of uses within nuclear medicine as it distributes within the body to a similar extent as iodine…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 52997-54-3

A radionuclide imaging agent used primarily in scintigraphy or tomography of the heart to evaluate the extent of the necrotic myocardial process. It has also been used in noninvasive tests for the distribution of organ involvement in different types of amyloi…

Kategori:
AcidsAcids, NoncarboxylicCompounds used in a research, industrial, or household setting +17
Target Protein:
HydroxyapatiteAmorphous calcium phosphate
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Technetium Tc-99m red blood cells is a radiopharmaceutical diagnostic agent that is intravenously administered to be used in blood pool imaging, including cardiac first pass and gated equilibrium imaging and for detection of sites of gastrointestinal bleeding…

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu ParuhTechnetium Tc 99m d…
Vol. DistribusiFollowing intraveno…
Klirens-
Genetik -
Technetium Tc-99m sestamibi Approved DB09161
small molecule | CAS: 109581-73-9

Technetium Tc-99m sestamibi (commonly sestamibi) is a pharmaceutical agent used in nuclear medicine imaging. The drug is a coordination complex consisting of the radioisotope technetium-99m bound to six methoxyisobutylisonitrile (MIBI) ligands, hence the name…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +10
Waktu ParuhTechnetium Tc 99m d…
Vol. Distribusi-
KlirensThe effective half-…
Genetik -
Technetium Tc-99m succimer Approved DB09436
small molecule | CAS: 65438-08-6

Technetium Tc-99m (<sup>99m</sup>Tc) succimer, also known as technetium Tc-99m dimercaptosuccinic acid (DMSA),[A245643] is a radioactive diagnostic agent used to evaluate functional renal tissue and tubular function in patients with renal parenchymal disorder…

Kategori:
Acids, AcyclicCompounds used in a research, industrial, or household settingDiagnostic Radiopharmaceuticals +14
Waktu ParuhTechnetium Tc-99m d…
Vol. DistribusiThere is no informa…
KlirensThere is no informa…
Genetik -
small molecule | CAS: 1262984-82-6

Technetium Tc-99m tilmanocept is a radiopharmaceutical diagnostic imaging agent approved by the U.S. Food and Drug Administration (FDA) for the imaging of lymph nodes with or without scintigraphic imaging. It is a macromolecule consisting of multiple units of…

Kategori:
Diagnostic RadiopharmaceuticalsRadioactive Diagnostic AgentRadiopharmaceutical Activity +2
Target Protein:
Macrophage mannose receptor 1
Waktu ParuhTechnetium Tc99m ti…
Vol. Distribusi-
KlirensIn dose-ranging cli…
Genetik -
Teclistamab Approved DB16655
biotech | CAS: 2119595-80-9

Teclistamab is an IgG4-PAA bispecific antibody that targets the CD3 receptor expressed on the surface of T cells and B cell maturation antigen (BCMA) expressed on malignant multiple myeloma cells.[A253587] Teclistamab consists of an anti-BCMA arm and an anti-…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +8
Target Protein:
T-cell surface glycoprotein CD3Tumor necrosis factor receptor superfamily member 17
Waktu ParuhBased on non-compar…
Vol. DistribusiThe mean (CV%) volu…
KlirensTeclistamab exhibit…
Genetik -
Tecovirimat Approved DB12020
small molecule | CAS: 869572-92-9

The World Health Organization declared smallpox, a contagious and sometimes fatal infectious disease, eradicated in 1980. However, there have been longstanding concerns that smallpox may be used as a bioweapon.[A35133,L3614] Tecovirimat is an antiviral drug t…

Kategori:
Acids, CarbocyclicAmidesAnti-Infective Agents +27
Target Protein:
Envelope protein F13
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Tedizolid Approved DB14569
small molecule | CAS: 856866-72-3

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +5
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Tedizolid phosphate Approved DB09042
small molecule | CAS: 856867-55-5

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntidepressive Agents +10
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Teduglutide Approved DB08900
biotech | CAS: 197922-42-2

Teduglutide is a glucagon-like peptide-2 (GLP-2) analogue. It is made up of 33 amino acids and is manufactured using a strain of Escherichia coli modified by recombinant DNA technology. Teduglutide differs from GLP-2 by one amino acid (alanine is substituted …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnalogs/Derivatives +15
Target Protein:
Glucagon-like peptide 2 receptor
Waktu ParuhTerminal half-life,…
Vol. DistribusiVd, healthy subject…
KlirensPlasma clearance, h…
Genetik -
biotech | CAS: 2143580-10-1

Tefidsogene civaparvovec, formerly known as SB-913, is an investigational therapy for genome editing. It consists of an adeno-associated virus (AAV) type 2/6 vector and a zinc finger nuclease (ZFN) system that inserts a correct copy of the Iduronate 2-Sulfata…

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tefinostat DB15321
small molecule | CAS: 914382-60-8

Tefinostat is under investigation in clinical trial NCT02759601 (Dose Escalation Trial of Tefinostat for Cancer Associated Inflamation in Hepatocellular Carcinoma (HCC)).

Kategori:
AmidesAminesAniline Compounds +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tegafur Approved DB09256
small molecule | CAS: 17902-23-7

Tegafur (INN, BAN, USAN) is a prodrug of [DB00544] (5-FU), an antineoplastic agent used as the treatment of various cancers such as advanced gastric and colorectal cancers. It is a pyrimidine analogue used in combination therapies as an active chemotherapeuti…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +22
Target Protein:
Thymidylate synthase
Gen Terkait:
DPYD DPYD DPYD +4
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensNo pharmacokinetic …
Genetik 7 Varian
Tegafur-uracil Approved DB09327
small molecule | CAS: 74578-38-4

Tegafur-uracil is an anti-tumor compound containing tegafur (1-(2-tetrahydrofuryl)-5-fluorouracil) and uracil in a molar ratio of 1:4. It was developed as an anti-cancer therapy by Taiho Pharmaceutical Co Ltd.[A32073] It is approved in different countries but…

Kategori:
Cytochrome P-450 CYP2A6 SubstratesCytochrome P-450 Substrates
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Thymidylate synthaseRNA +1
Waktu ParuhThe presence of ura…
Vol. DistribusiThe volume of distr…
KlirensThe reported cleara…
Genetik -
Tegaserod Approved DB01079
small molecule | CAS: 145158-71-0

Novartis' brand name Zelnorm (tegaserod) had originally received approval from the US FDA in 2002 for the treatment of irritable bowel syndrome with constipation (IBS-C).[L5918,F4229] It was, however, voluntarily withdrawn from widespread use in the US market…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsBCRP/ABCG2 Substrates +25
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A +1
Waktu ParuhThe mean terminal e…
Vol. DistribusiAlthough tegaserod …
KlirensAlthough tegaserod …
Genetik -
Tegoprazan DB16690
small molecule | CAS: 942195-55-3

Tegoprazan (also known as CJ-12420) is a novel therapeutic developed by CJ Healthcare Corp for treating acid-related gastrointestinal diseases.[A234215, A234220] This drug is a potent and high-selective potassium-competitive acid blocker (P-CAB) with a fast o…

Kategori:
Alimentary Tract and MetabolismDrugs for Acid Related DisordersDrugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord) +2
Target Protein:
Sodium/Potassium Transporting ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Teicoplanin Approved DB06149
small molecule | CAS: 61036-62-2

Teicoplanin is a glycopeptide antibiotic consisting of a mixture of several compounds, five major (named teicoplanin A2-1 through A2-5) and four minor (named teicoplanin RS-1 through RS-4). All teicoplanins share a same glycopeptide core, teicoplanin A3-1, bu…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
D-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycan
Waktu Paruh70-100 hours
Vol. Distribusi-
Klirens-
Genetik -
TEL540-548 DB17461
biotech

TEL540-548 is a recombinant peptide consisting of the amino acid residues 540 to 548 of the human telomerase reverse transcriptase (hTERT).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telaprevir Approved DB05521
small molecule | CAS: 402957-28-2

Telaprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine…

Kategori:
Amino Acids, Peptides, and ProteinsAntiinfectives for Systemic UseAntiviral Agents +21
Target Protein:
Genome polyproteinGenome polyproteinSolute carrier organic anion transporter family member 1B1 +1
Waktu ParuhTelaprevir has a ha…
Vol. DistribusiThe estimated appar…
KlirensTelaprevir has an e…
Genetik -
small molecule | CAS: 198414-31-2

Telapristone acetate, an orally-available, selective progesterone receptor modulator, is in development to alleviate symptoms associated with both uterine fibroids and endometriosis.

Kategori:
Fused-Ring CompoundsNorpregnanesNorsteroids +1
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telatinib DB15393
small molecule | CAS: 332012-40-5

Telatinib is under investigation in clinical trial NCT03817411 (Telatinib in Combination With Capecitabine/ Oxaliplatin in 1st Line Gastric or GEJ Cancer).

Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telavancin Approved DB06402
small molecule | CAS: 372151-71-8

Telavancin is a semi-synthetic derivative of vanocymycin that has bactericidal activity against Methicillin-resistant Staphylococcus aureus (MRSA) and other gram-positive bacteria. MRSA is an important pathogen capable of causing hospital-acquired pneumonia …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Neuronal acetylcholine receptor subunit alpha-3Corticotropin-releasing factor receptor 1
Waktu ParuhTerminal eliminatio…
Vol. DistribusiVss, healthy subjec…
KlirensCl, healthy subject…
Genetik -
Telbivudine Approved DB01265
small molecule | CAS: 3424-98-4

Telbivudine is a synthetic thymidine nucleoside analog with specific activity against the hepatitis B virus. Telbivudine is orally administered, with good tolerance, lack of toxicity and no dose-limiting side effects.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +13
Target Protein:
DNAProtein P
Waktu ParuhApproximately 15 ho…
Vol. Distribusi-
Klirens* 7.6 +/- 2.9 L/h […
Genetik -
Telcagepant DB12228
small molecule | CAS: 781649-09-0

Telcagepant has been investigated for the treatment of Migraine. It is an antagonist of the receptor for calcitonin gene-related peptide (CGRP), a primary neuropeptide involved in the pathophysiology of migraine. CGRP and its receptors are found in areas of t…

Target Protein:
Calcitonin gene-related peptide type 1 receptorCalcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telitacicept DB18312
biotech | CAS: 2136630-26-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Telithromycin Approved DB00976
small molecule | CAS: 191114-48-4

Telithromycin, a semi-synthetic erythromycin derivative, belongs to a new chemical class of antibiotics called ketolides. Ketolides have been recently added to the macrolide-lincosamide-streptogramin class of antibiotics. Similar to the macrolide antibiotics,…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +23
Target Protein:
23S ribosomal RNA
Waktu ParuhMain elimination ha…
Vol. Distribusi* 2.9 L/kg
Klirens-
Genetik -
Telmisartan Approved DB00966
small molecule | CAS: 144701-48-4

Telmisartan is an angiotensin II receptor antagonist (ARB) used in the management of hypertension. Generally, angiotensin II receptor blockers (ARBs) such as telmisartan bind to the angiotensin II type 1 (AT1) receptors with high affinity, causing inhibition …

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +24
Target Protein:
Peroxisome proliferator-activated receptor gammaType-1 angiotensin II receptor
Waktu ParuhTelmisartan display…
Vol. DistribusiTelmisartan has a v…
KlirensTelmisartan has a t…
Genetik -
Telotristat ethyl Approved DB12095
small molecule | CAS: 1033805-22-9

Telotristat ethyl is a prodrug of telotristat that was approved by the FDA in March 2017 as Xermelo.[L43342] It was previously referred to as telotristat etiprate, the hippurate salt form; however, the FDA recommends the use of the name of the neutral form ra…

Kategori:
AntidiarrhealsCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +20
Target Protein:
Tryptophan 5-hydroxylase 2Tryptophan 5-hydroxylase 1
Waktu ParuhFollowing a single …
Vol. DistribusiThe estimated appar…
KlirensThe apparent total …
Genetik -
Temafloxacin DB01405
small molecule | CAS: 108319-06-8

Temafloxacin is an antibiotic agent belonging to the fluoroquinolone drug class. It was first approved for use in the U.S. market in 1992, but was withdrawn shortly due to the reports of serious adverse reactions, such as allergic reactions and hemolyric anem…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu ParuhApproximately 8 hou…
Vol. Distribusi-
Klirens-
Genetik -
Temazepam Approved DB00231
small molecule | CAS: 846-50-4

Temazepam, like many other similar and related benzodiazepines, acts as a gamma-aminobutyric acid (GABA) modulator and is capable of eliciting a variety of actions including sedation, hypnosis, skeletal muscle relaxation, anticonvulsant activity, and anxiolyt…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepine hypnotics and sedatives +18
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensStudies regarding t…
Genetik -
Temefos DB12231
small molecule | CAS: 3383-96-8

Diphos has been used in trials studying the treatment of Plasmodium Falciparum Malaria.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Temelimab DB15634
biotech | CAS: 1393641-34-3

Temelimab is under investigation in clinical trial NCT02782858 (Clinical Trial Assessing the HERV-W Env Antagonist Gnbac1 for Efficacy in MS).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Temocillin Approved DB12343
small molecule | CAS: 66148-78-5

Temocillin has been investigated in Infection, Liver Dysfunction, and Urinary Tract Infection.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Temoporfin Approved DB11630
small molecule | CAS: 122341-38-2

Temoporfin is a photosensitizing agent used in the treatment of squamous cell carcinoma of the head and neck [FDA Label]. It was first authorized for market by the European Medicines Agency in October 2001. It is currently available under the brand name Fosca…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBiological Factors +8
Waktu ParuhTerminal plasma hal…
Vol. DistribusiThe volume of distr…
KlirensTemoporfin is clear…
Genetik -
Temozolomide Approved DB00853
small molecule | CAS: 85622-93-1

Refractory anaplastic astrocytoma (WHO grade III) and Glioblastoma multiforme (WHO grade IV) are primary malignant brain tumours with poor prognosis and limited treatment options. Despite considerable genetic heterogeneity, these tumours often have impaired D…

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +13
Target Protein:
DNA
Waktu ParuhTemozolomide has a …
Vol. DistribusiTemozolomide has a …
KlirensTemozolomide has a …
Genetik -
Temsirolimus Approved DB06287
small molecule | CAS: 162635-04-3

Temsirolimus is a derivative of sirolimus used in the treatment of renal cell carcinoma (RCC). It was developed by Wyeth Pharmaceuticals under the trade name Torisel. Temsirolimus was approved by the FDA in late May 2007 as well as the European Medicines Agen…

Kategori:
Agents causing angioedemaAnti-Bacterial AgentsAntineoplastic Agents +32
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu ParuhTemsirolimus exhibi…
Vol. Distribusi172 L in whole bloo…
Klirens16.2 L/h (22%)
Genetik -
Tenamfetamine DB01509
small molecule | CAS: 4764-17-4

An amphetamine derivative that inhibits uptake of catecholamine neurotransmitters. It is a hallucinogen. It is less toxic than its methylated derivative but in sufficient doses may still destroy serotonergic neurons and has been used for that purpose experime…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +17
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tenecteplase Approved DB00031
biotech | CAS: 191588-94-0

Tenecteplase is a tissue plasminogen activator (tPA) developed from modifications of natural human tPA complementary DNA (cDNA). It is a 527 amino acid with a substitution of threonine 103 with asparagine and substitution of asparagine 117 with glutamine with…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +17
Target Protein:
Plasminogen
Waktu Paruh1.9 hours (mammalia…
Vol. Distribusi-
Klirens* 99 - 119 mL/min […
Genetik -
Tengonermin DB16689
biotech | CAS: 1960461-99-7

Tengonermin, also known as NGR-hTNF, is a vascular-targeting drug.[A233265] It is a recombinant protein and peptide-targeted agent consisting of the human Tumour Necrosis Factor-? (TNF-?) conjugated with the CNGRCG peptide.[L33050] This drug works by modifyin…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Proteins +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tenocyclidine DB01520
small molecule | CAS: 21500-98-1

Tenocyclidine (TCP, thienyl cyclohexylpiperidine) is a dissociative anesthetic drug with stimulant and hallucinogenic effects. It is more potent than phencyclidine and hence, this drug was classified under the schedule 1 in 1970.

Kategori:
Central Nervous System AgentsCompounds used in a research, industrial, or household settingIllicit Drugs +5
Target Protein:
Glutamate receptor ionotropic, NMDA 3AGlutamate receptor ionotropic, NMDA 3BGlutamate receptor ionotropic, NMDA 2A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tenofovir DB14126
small molecule | CAS: 147127-20-6

Tenofovir is an acyclic nucleotide diester analog of adenosine monophosphate.[A37693] In the most strict sense and due to the fact that it presents a phosphate group bound to the nitrogenous base, it is determined as an actual nucleotide analog.[A37693] The a…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +16
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyproteinReverse transcriptase +1
Waktu ParuhThe reported half-l…
Vol. DistribusiAccumulation of ten…
KlirensThe clearance of te…
Genetik -
Tenofovir alafenamide Approved DB09299
small molecule | CAS: 379270-37-8

Tenofovir alafenamide is a novel [tenofovir] prodrug developed in order to improve renal safety when compared to the counterpart [tenofovir disoproxil].[A178060] Both of these prodrugs were first created to cover the polar phosphonic acid group on tenofovir b…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntiinfectives for Systemic Use +25
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyproteinReverse transcriptase +1
Waktu ParuhThe reported half-l…
Vol. DistribusiIn clinical trials,…
KlirensThe reported cleara…
Genetik -
Menampilkan 6001–6050 dari 6694
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