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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 121 / 236
Imetelstat Approved DB14909
small molecule | CAS: 868169-64-6

Imetelstat is a first-in-class 18-amino acid oligonucleotide that directly and competitively inhibits human telomerase.[A263973] It is used to treat anemia in patients with myelodysplastic syndromes (MDS), a group of hematologic disorders characterized by ine…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +6
Target Protein:
Telomerase reverse transcriptaseHuman telomerase RNA component
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
Klirens-
Genetik -
IMG-7289 DB15126
small molecule | CAS: 1990504-34-1

IMG-7289 is under investigation in clinical trial NCT03136185 (IMG-7289 in Patients With Myelofibrosis).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysine-specific histone demethylase 1A
Waktu Paruh-
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IMGN632 DB17337
biotech

Deskripsi belum tersedia.

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IMGN779 DB17336
biotech

Deskripsi belum tersedia.

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Imidacloprid DB11421
small molecule | CAS: 105827-78-9

Imidacloprid is a neonicotinoid, which is a class of neuro-active insecticides modeled after nicotine. Imidacloprid is a patented chemical, Imidacloprid is manufactured by Bayer Cropscience (part of Bayer AG) and sold under trade names Kohinor, Admire, Advant…

Kategori:
AgrochemicalsCholinergic AgentsCompounds used in a research, industrial, or household setting +4
Target Protein:
CHRNA7-FAM7A fusion protein
Waktu Paruh-
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Imidafenacin DB09262
small molecule | CAS: 170105-16-5

Imidafenacin is an antispasmodic agent with anticholinergic effects. It antagonizes muscarinic receptors in the bladder to reduce the frequency of urination in the treatment of overactive bladder. It is marketed in Japan under the tradenames Staybla by Ono Ph…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCytochrome P-450 CYP3A Substrates +8
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu ParuhThe half life of el…
Vol. DistribusiThe estimated volum…
KlirensThe estimated clear…
Genetik -
Imidapril DB11783
small molecule | CAS: 89371-37-9

Imidapril has been investigated for the treatment of Kidney, Polycystic, Autosomal Dominant.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +7
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh-
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small molecule | CAS: 1072-84-0

Imidazole-4-carboxylic acid is under investigation in clinical trial NCT00583895 (Safety and Efficacy Study of Imcooh Cream in Patients Suffering From Moderate Atopic Dermatitis).

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small molecule

Deskripsi belum tersedia.

Target Protein:
Endoglucanase 5A
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase pim-1
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Methionine aminopeptidase
Waktu Paruh-
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Imidocarb DB11521
small molecule | CAS: 27885-92-3

Imidocarb is a urea derivative used in veterinary medicine as an antiprotozoal agent for the treatment of infection with Babesia and other parasites.

Kategori:
AmidesAminesAnilides +7
Target Protein:
Acetylcholinesterase
Waktu Paruh-
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Imidurea Approved DB14075
small molecule | CAS: 39236-46-9

Imidurea is an antimicrobial preservative used in cosmetics. It acts as a formaldehyde releaser.

Kategori:
AmidesCell-mediated ImmunityIncreased Histamine Release +2
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Imifoplatin DB17120
small molecule | CAS: 1339960-28-9

Deskripsi belum tersedia.

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Imiglucerase Approved DB00053
biotech | CAS: 154248-97-2

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 0.09 to 0.15 L/kg
Klirens* 14.5 +/- 4.0 mL/m…
Genetik -
Imipenem Approved DB01598
small molecule | CAS: 64221-86-9

Imipenem is a semisynthetic thienamycin that has a wide spectrum of antibacterial activity against gram-negative and gram-positive aerobic and anaerobic bacteria, including many multiresistant strains.[label] It is stable to many beta-lactamases. Similar comp…

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +12
Target Protein:
Penicillin-binding protein 2Penicillin-binding protein 1BPenicillin-binding protein 1A +3
Waktu ParuhWhen given via IV i…
Vol. DistribusiThe reported volume…
KlirensThe total clearance…
Genetik -
Imipramine Approved DB00458
small molecule | CAS: 50-49-7

Imipramine, the prototypical tricyclic antidepressant (TCA), is a dibenzazepine-derivative TCA. TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +70
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +21
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhImipramine has a me…
Vol. DistribusiImipramine has a hi…
KlirensImipramine has a me…
Genetik 9 Varian
small molecule | CAS: 6829-98-7

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +10
Waktu Paruh-
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Imiquimod Approved DB00724
small molecule | CAS: 99011-02-6

Imiquimod is an immune response modifier that acts as a toll-like receptor 7 agonist. Imiquimod is commonly used topically to treat warts on the skin of the genital and anal areas. Imiquimod does not cure warts, and new warts may appear during treatment. Imiq…

Kategori:
Adjuvants, ImmunologicAminoquinolinesAntineoplastic Agents +17
Target Protein:
Toll-like receptor 7Toll-like receptor 8
Waktu Paruh20 hours (topical d…
Vol. Distribusi-
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Imlifidase Approved DB15258
biotech | CAS: 1947415-68-0

Chronic kidney disease (CKD) is a progressive and irreversible disease that represents a significant burden for both the individual and healthcare system at large.[A225916] Currently available treatments for end-stage renal disease are limited to dialysis and…

Kategori:
Antineoplastic and Immunomodulating AgentsEndopeptidasesImmunosuppressive Agents +2
Target Protein:
IgG heavy chain
Waktu ParuhThe mean distributi…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
IMM-0306 DB19309
biotech

IMM-0306 (bispecific antibody-trap selectively targeting cd47 and cd20) is under investigation in clinical trial NCT05805943 (Study of IMM0306 in Patients With Relapsed or Refractory Cd20-positive B-cell Non-hodgkin's Lymphoma).

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IMM101 DB15851
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma [PMID: 21930686; PMID: 30107850; PMID: …

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Immucin DB17403
biotech

Deskripsi belum tersedia.

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Genetik -
biotech | CAS: 1807503-77-0

Deskripsi belum tersedia.

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Implitapide DB04852
small molecule | CAS: 177469-96-4

Implitapide is a microsomal triglyceride transfer protein (MTP)-inhibitor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
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IMT-288 DB19068
small molecule | CAS: 637771-94-9

IMT-288 is under investigation in clinical trial NCT01730638 (Immunotep for Patients With Medullary Thyroid Carcinoma.).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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IMT504 DB17792
biotech

IMT504, a non-CpG 24-mer oligodeoxynucleotide, is an immunomodulatory oligonucleotide currently being investigated as a rabies vaccine.[A259467]

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
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Imvotamab DB17331
biotech

Deskripsi belum tersedia.

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IN01 DB16434
biotech

The IN01 Vaccine, sponsored by the Instituto Oncologico Dr Rosell, IN3BIO, and PANGAEA, is a compound containing recombinant bacteria[L30543]. These cultures contain EGF-4-EGF with the cholera toxin B-subunit domain G33D sequence[L30543]. Administration of th…

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biotech

Developed by Sinopharm's Wuhan Institute of Biological Products co., this vaccine consists of the WIV04 strain of SARS-CoV-2. This strain was isolated from a patient in Wuhan, cultivated in a Vero cell line, and then subsequently inactivated using B-propiolac…

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biotech

The SARS-CoV-2 Inactivated Vaccine is a purified vaccine that contains multiple antigens from the virus and is inactivated in Vero Cells[A219758]. This vaccine specifically was developed in collaboration with the Chinese Academy of Medical Sciences, West Chin…

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Inalimarev DB17332
biotech | CAS: 685563-13-7

Deskripsi belum tersedia.

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Inarigivir DB15062
small molecule | CAS: 475650-36-3

Inarigivir is under investigation in clinical trial NCT03434353 (Study to Evaluate the Antiviral Activity of Inarigivir (GS-9992) Plus Tenofovir Alafenamide (TAF) for 12 Weeks in Adults With Chronic Hepatitis B (CHB)).

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Inavolisib Approved DB15275
small molecule | CAS: 2060571-02-8

_PIK3CA_ is one of the most frequently mutated oncogenes, with the resulting mutated p110? protein it encodes playing a central role in tumor cell proliferation.[A264563] Chemotherapeutic agents targeting the PI3K p110? catalytic subunit have shown antitumor …

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +4
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe total clearance…
Genetik -
Inbakicept DB16479
biotech | CAS: 2135939-52-3

Inbakicept is a dimeric human IL-15 receptor ? (IL-15R?) sushi domain/human IgG1 Fc fusion protein. It is one of the active ingredients in Anktiva, a combination product also containing [nogapendekin alfa], where a single inbakicept is complexed with two noga…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsExperimental Unapproved Treatments for COVID-19 +4
Target Protein:
Interleukin-2 receptor subunit betaCytokine receptor common subunit gamma
Waktu Paruh-
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Incadronic acid DB06255
small molecule | CAS: 124351-85-5

Incadronate, or YM-175,[A202769] is a nitrogen containing bisphosphonate. Along with being investigated to treat hypercalcemia of malignancy,[A202862] it has also been investigated in the treatment of myeloma, leukemia, and other cancers.[A14426,A14431,A14427…

Kategori:
Antineoplastic AgentsBisphosphonatesBone Density Conservation Agents +2
Target Protein:
Farnesyl pyrophosphate synthaseCaspase-3Caspase-4 +1
Waktu ParuhIncadronate has a b…
Vol. Distribusi-
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INCB-054329 DB16894
small molecule | CAS: 1628607-64-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic Agents
Waktu Paruh-
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INCB-057643 DB16054
small molecule | CAS: 1820889-23-3

INCB-057643 is under investigation in clinical trial NCT02959437 (Azacitidine Combined With Pembrolizumab and Epacadostat in Subjects With Advanced Solid Tumors (ECHO-206)).

Kategori:
AcidsAcids, NoncarboxylicAntineoplastic Agents +1
Waktu Paruh-
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INCB-086550 DB18901
small molecule | CAS: 2230911-59-6

INCB-086550 is under investigation in clinical trial NCT04629339 (Study of INCB086550 in Select Solid Tumors).

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INCB-9471 DB12960
small molecule | CAS: 869769-98-2

INCB-9471 is a novel, orally available CCR5 antagonist that is part of a new class of drugs to treat HIV/AIDS. It is a potent, selective inhibitor of the HIV-1 virus.

Kategori:
Receptors, CCR4, antagonists & inhibitors
Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
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INCB052793 DB17567
small molecule

Deskripsi belum tersedia.

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INCB13739 DB05064
small molecule

INCB13739 is developed as a new treatment for type 2 diabetes. It is an orally available small molecule inhibitor of 11beta-HSD1 (11-beta hydroxysteroid dehydrogenase type 1). 11beta-HSD1 is an enzyme that appears to be critical to the development of type 2…

Kategori:
11-beta-Hydroxysteroid Dehydrogenase Type 1, antagonists & inhibitorsAmidesSulfones +1
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1
Waktu Paruh-
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INCB7839 DB05033
small molecule

INCB7839 is a novel, orally available ADAM metalloprotease inhibitor that is designed to block activation of the epidermal growth factor (EGFR) pathways. It represents a potentially important new class of targeted breast cancer therapy. It has shown promising…

Target Protein:
Disintegrin and metalloproteinase domain-containing protein 9
Waktu Paruh-
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Inclisiran Approved DB14901
biotech | CAS: 1639324-58-5

Inclisiran is a long-acting, synthetic small interfering RNA (siRNA) directed against proprotein convertase subtilisin-kexin type 9 (PCSK9), which is a serine protease that regulates plasma low-density lipoprotein cholesterol (LDL-C) levels. By binding to PCS…

Kategori:
Antisense Elements (Genetics)Compounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +16
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThere is limited in…
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAlcoholsCarbohydrates +7
Waktu Paruh-
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Incyclinide DB11647
small molecule | CAS: 15866-90-7

Incyclinide has been used in trials studying the treatment of HIV Infection, AIDS-related Kaposi Sarcoma, Brain and Central Nervous System Tumors, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Naphthacenes
Target Protein:
72 kDa type IV collagenase
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Indacaterol Approved DB05039
small molecule | CAS: 312753-06-3

Indacaterol is a novel, ultra-long-acting, rapid onset ?(2)-adrenoceptor agonist developed for Novartis for the once-daily management of asthma and chronic obstructive pulmonary disease. It was approved by the European Medicines Agency (EMA) on 30 November 20…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +17
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIndacaterol serum c…
Vol. DistribusiAfter intravenous i…
KlirensRenal clearance of …
Genetik -
Indalpine DB08953
small molecule | CAS: 63758-79-2

Indalpine was one of the first selective serotonin reuptake inhibitors to reach the American market. It was initially marketed by Pharmuka. However, after the emergence of widespread concern regarding adverse effects caused by SSRIs, and reported hematologica…

Kategori:
Antidepressive AgentsCentral Nervous System AgentsCentral Nervous System Depressants +16
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Indanazoline DB13827
small molecule | CAS: 40507-78-6

Deskripsi belum tersedia.

Kategori:
Nasal PreparationsSympathomimetics, Plain
Waktu Paruh-
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Indapamide Approved DB00808
small molecule | CAS: 26807-65-8

The most significant modifiable risk factor for cardiovascular disease and the most prominent contributor to all-cause mortality is hypertension.[A204155] Characterized by an office blood pressure of ?140/90, hypertension is pervasive and impacts an estimated…

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +26
Target Protein:
Solute carrier family 12 member 3Potassium voltage-gated channel subfamily KQT member 1
Waktu ParuhIndapamide is chara…
Vol. DistribusiSome sources report…
KlirensIndapamide's renal …
Genetik -
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