Hasil Filter

6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (6694)

Halaman 120 / 134
biotech | CAS: 1580555-26-5

Talditercept alfa is under investigation in clinical trial NCT03039686 (Clinical Trial to Evaluate the Efficacy, Safety, and Tolerability of RO7239361 in Ambulatory Boys With Duchenne Muscular Dystrophy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talimogene laherparepvec Approved DB13896
biotech | CAS: 1187560-31-1

Talimogene laherparepvec is an oncolytic treatment used in local treatment of unresectable cutaneous, subcutaneous, and nodal lesions in patients with recurrent melanoma. It is a genetically administered herpes simplex virus 1 (HSV-1) that expresses human cyt…

Kategori:
AlphaherpesvirinaeAntineoplastic AgentsAntineoplastic Agents, Immunological +9
Target Protein:
Granulocyte-macrophage colony-stimulating factor
Waktu ParuhReadily accessible …
Vol. DistribusiTalimogene laherpar…
KlirensAlthough readily ac…
Genetik -
Talinolol DB11770
small molecule | CAS: 57460-41-0

Talinolol has been investigated for the basic science of Gastrointestinal Motility Disorder.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tallimustine DB15466
small molecule | CAS: 115308-98-0

Tallimustine, a benzoyl mustard derivative of distamycin A, is an alkylating agent that binds to the minor groove of DNA.[A182036,A182039] It's association with severe myelotoxicity lead to the end of its development in favour of ?-halogenoacrylamide derivati…

Kategori:
Alkylating DrugsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +6
Target Protein:
C-X-C chemokine receptor type 2DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talmapimod DB05412
small molecule | CAS: 309913-83-5

Talmapimod is the first-generation oral p38 MAP kinase inhibitor developed by Scios. It has shown to be effective to cure inflammatory diseases such as Rheumatoid Arthritis.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Mitogen-activated protein kinase 14Tumor necrosis factorInterleukin-1 beta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talniflumate DB09295
small molecule | CAS: 66898-62-2

Talniflumate, is an anti-inflammatory molecule studied and used as a mucin regulator in the treatment of cystic fibrosis, chronic obstructive pulmonary disease (COPD) and asthma [L1400]. In addition, it is used in inflammatory conditions such as rheumatoid ar…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +5
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Chloride channel protein ClC-Ka
Waktu ParuhApproximately 2h in…
Vol. DistribusiIn 12 subjects afte…
KlirensThis drug undergoes…
Genetik -
Talopram DB09190
small molecule | CAS: 7182-51-6

Talopram is a selective norepinephrine reuptake inhibitor (SNRI) that is structurally similar to citalopram and melitracen. It was researched in the 1960s and 1970s but never marketed.

Kategori:
Adrenergic Uptake InhibitorsAminesAntidepressive Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Talquetamab Approved DB16678
biotech | CAS: 2226212-40-2

Talquetamab is a IgG4-PAA bispecific G protein-coupled receptor class C group 5 member D (GPRC5D)-directed CD3 T-cell engager. It consists of two arms - anti-GPRC5D and anti-CD3 arms - linked by two interchain disulfide bonds, each arm comprising a heavy and …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic Agents +7
Target Protein:
T-cell surface glycoprotein CD3G-protein coupled receptor family C group 5 member D
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensTalquetamab clearan…
Genetik -
Talsupram DB09191
small molecule | CAS: 21489-20-3

Talsupram is a selective norepinephrine reuptake inhibitor (NRI). It was under research for the treatment of depression in 1960 and 1970 but it was never marketed. Talsupram presents a similar structure to [citalopram].

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamibarotene DB04942
small molecule | CAS: 94497-51-5

Tamibarotene is a novel synthetic retinoid for acute promyelocytic leukaemia (APL). Tamibarotene is currently approved in Japan for treatment of recurrent APL, and is undergoing clinical trials in the United States.

Kategori:
Acids, CarbocyclicBenzene DerivativesNaphthalenes
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tamoxifen Approved DB00675
small molecule | CAS: 10540-29-1

Tamoxifen is a non-steroidal antiestrogen used to treat estrogen receptor positive breast cancers as well as prevent the incidence of breast cancer in high risk populations.[A1025,L7799,L7802] Tamoxifen is used alone or as an adjuvant in these treatments.[L77…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +64
Target Protein:
Estrogen receptorEstrogen receptor betaProtein kinase C +7
Gen Terkait:
CYP2D6 F5
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ta…
Genetik 2 Varian
biotech

Tanacetum cinerariifolium flower allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tandamine DB09192
small molecule | CAS: 42408-80-0

Tandamine was researched in 1970s as an antidepressant but was never commercialized. Tandamine is an analog of pirandamine and it acts as a selective serotonin reuptake inhibitor (SSRI).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tanespimycin DB05134
small molecule | CAS: 75747-14-7

Tanespimycin, manufactured by Conforma Therapeutics is under development as a small molecule inhibitor of heat shock protein 90 (HSP90). It is developed for the treatment of several types of cancer, solid tumors or chronic myelogenous leukemia.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tangerine peel DB14316
biotech

Tangerine peel is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tannic acid Approved DB09372
small molecule | CAS: 1401-55-4

Tannic acid is a polyphenolic compound. It is a type of the commercially available tannins. It acts as a weak acid. Tannic acid is found in the nutgalls formed by insects on twigs of certain oak trees (Quercus infectoria and other Quercus species). It is remo…

Kategori:
Benzene DerivativesBiopolymersCompounds used in a research, industrial, or household setting +4
Target Protein:
Anoctamin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tapinarof Approved DB06083
small molecule | CAS: 79338-84-4

Tapinarof is a novel, first-in-class, small-molecule AhR agonist that is indicated for the treatment of adult psoriasis. It is available as a topical cream to be applied to the affected area once daily.[L41845, A248790] Tapiranof was first discovered as a met…

Kategori:
AntipsoriaticsAntipsoriatics for Topical UseAryl Hydrocarbon Receptor Agonist +11
Target Protein:
Aryl hydrocarbon receptor
Waktu ParuhDue to the insuffic…
Vol. DistribusiThe Vss of tapinaro…
Klirens-
Genetik -
Tarafenacin DB18810
small molecule | CAS: 385367-47-5

Deskripsi belum tersedia.

Target Protein:
Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Taraxacum officinale leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taraxacum officinale pollen Approved DB10755
biotech

Taraxacum officinale pollen is the pollen of the Taraxacum officinale plant. Taraxacum officinale pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2411896-53-0

Tarcocimab tedromer is under investigation in clinical trial NCT06270836 (A Study to Evaluate the Efficacy and Safety of Tarcocimab Tedromer Compared With Sham Treatment in Participants With Moderately Severe to Severe Non-proliferative Diabetic Retinopathy (…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarenflurbil DB05289
small molecule | CAS: 51543-40-9

Tarenflurbil is an investigational drug that was studied in patients with mild Alzheimer's disease. It is a selective amyloid lowering agent (SALA) that reduces levels of the toxic peptide amyloid beta 42 (A?42) in cultured human cells and in animal models. A…

Kategori:
Acids, AcyclicAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tarlatamab Approved DB17256
biotech | CAS: 2307488-83-9

Tarlatamab is a first-in-class T-cell engager used to treat extensive-stage small cell lung cancer.[L50748] It is a bispecific monoclonal antibody that targets CD3 expressed on the surface of T-cells and delta-like ligand 3 (DLL3), an inhibitory ligand that s…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalBispecific Monoclonal Antibodies +5
Target Protein:
Delta-like protein 3T-cell surface glycoprotein CD3
Waktu ParuhThe median terminal…
Vol. DistribusiAt steady-state, th…
KlirensThe systemic cleara…
Genetik -
TAS-102 DB08937
small molecule | CAS: 733030-01-8

TAS-102 (Taiho Pharma USA, Inc.) is an anti-cancer drug under development and in stage 3 clinical trials for the treatment of colorectal cancer. It is composed of the thymidine phosphorylase inhibitor (TPI) tipiracil and the cytotoxin trifluridine. Trifluridi…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TAS-106 DB06656
small molecule | CAS: 180300-43-0

TAS-106 is a new nucleoside antimetabolite. TAS-106 has demonstrated strong antitumor activity without serious toxicity in nude rat models bearing human tumours [A31693].

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taselisib DB12108
small molecule | CAS: 1282512-48-4

Taselisib has been used in trials studying the treatment and basic science of LYMPHOMA, Breast Cancer, Ovarian Cancer, Solid Neoplasm, and HER2/Neu Negative, among others.

Kategori:
Antineoplastic AgentsAzepinesPhosphatidylinositol 3-Kinases, antagonists & inhibitors
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tasimelteon Approved DB09071
small molecule | CAS: 609799-22-6

Tasimelteon is a selective dual melatonin receptor agonist indicated for the treatment of Non-24-Hour Sleep-Wake Disorder (N24HSWD). Occurring commonly in blind individuals without light perception, this condition is often characterized by periods of night-ti…

Kategori:
Central Nervous System DepressantsCycloparaffinsCytochrome P-450 CYP1A2 Substrates +11
Target Protein:
Melatonin receptor type 1AMelatonin receptor type 1B
Waktu ParuhThe observed mean e…
Vol. DistribusiThe apparent oral v…
Klirens-
Genetik -
Tasisulam DB11941
small molecule | CAS: 519055-62-0

Tasisulam has been used in trials studying the treatment and basic science of Melanoma, Lymphoma, Solid Tumors, Breast Cancer, and Ovarian Cancer, among others.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TASO-001 DB17463
biotech

TASO-001 is a transforming growth factor (TGF)-beta 2 specific antisense oligodeoxynucleotide.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tasonermin Approved DB11626
biotech | CAS: 94948-59-1

Tasonermin is recombinant soluble form tumor necrosis factor α produced via _Escherichia coli_ cell culture. It was approved for use by the European Medicines Agency in April of 1999 for use as an adjunt to surgery for the subsequent removal of the tum…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating Agents
Target Protein:
Tumor necrosis factor receptor superfamily member 1ATumor necrosis factor receptor superfamily member 1B
Waktu ParuhTasonermin has a te…
Vol. DistribusiThe estimated volum…
KlirensClearance was estim…
Genetik -
Taspoglutide DB14027
small molecule | CAS: 275371-94-3

Taspoglutide is a pharmaceutical drug, a glucagon-like peptide-1 agonist (GLP-1 agonist), under investigation for treatment of type 2 diabetes being codeveloped by Ipsen and Roche. In September 2010 Roche halted Phase III clinical trials due to incidences of …

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsGastrointestinal Hormones +5
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taurine Approved DB01956
small molecule | CAS: 107-35-7

Taurine, whose chemical name is 2-aminoethanesulfonic acid, is one of the most abundant amino acids in several organs. It plays important role in essential biological processes.[A31396] This conditional amino acid can be either be manufactured by the body or …

Kategori:
AlkanesAlkanesulfonic AcidsAmino Acids +5
Target Protein:
Glutamate receptor ionotropic, NMDA 2BGlycine receptor subunit betaGlycine receptor subunit alpha-2 +6
Waktu ParuhOral administration…
Vol. DistribusiThe distribution of…
KlirensThe clearance rate …
Genetik -
small molecule | CAS: 516-35-8

Taurochenodeoxycholic acid is an experimental drug that is normally produced in the liver. Its physiologic function is to emulsify lipids such as cholesterol in the bile. As a medication, taurochenodeoxycholic acid reduces cholesterol formation in the liver, …

Kategori:
AlkanesAlkanesulfonic AcidsBile Acids and Salts +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taurocholic acid Approved DB04348
small molecule | CAS: 81-24-3

The product of conjugation of cholic acid with taurine. Its sodium salt is the chief ingredient of the bile of carnivorous animals. It acts as a detergent to solubilize fats for absorption and is itself absorbed. It is used as a cholagogue and cholerectic.

Kategori:
AcidsAcids, NoncarboxylicAlkanes +30
Target Protein:
Ileal sodium/bile acid cotransporterG-protein coupled bile acid receptor 1Bile salt-activated lipase +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Taurolidine Approved DB12473
small molecule | CAS: 19388-87-5

Taurolidine is an antimicrobial used for the prevention of catheter-related infections. It is a derivative of the amino acid [taurine]. It was first synthesized in the 1970s and was originally used as a prophylactic against intraperitoneal bacterial infect…

Kategori:
AlkanesAlkanesulfonic AcidsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75018-71-2

Deskripsi belum tersedia.

Kategori:
Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tauroursodeoxycholic acid Approved DB08834
small molecule | CAS: 14605-22-2

Tauroursodeoxycholic acid, also known as ursodoxicoltaurine, is a highly hydrophilic tertiary bile acid [A249070] that is produced in humans at a low concentration.[A249070] It is a taurine conjugate of [ursodeoxycholic acid] [A249065] with comparable therape…

Kategori:
Alimentary Tract and MetabolismBile acids and derivativesBile Acids and Salts +10
Target Protein:
Integrin alpha-5
Waktu Paruh-
Vol. DistribusiThere is evidence t…
Klirens-
Genetik -
Tavaborole Approved DB09041
small molecule | CAS: 174671-46-6

Tavaborale is a novel, boron-based topical antifungal medication for the treatment of onychomycosis, a fungal infection of the nail and nail bed due to *Trichophyton rubrum* or *Trichophyton mentagrophytes* infection. Tavaborole functions by inhibiting Leucyl…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +4
Target Protein:
leucine--tRNA ligase
Waktu Paruh28.5 hr
Vol. Distribusi-
Klirens-
Genetik -
Tazobactam Approved DB01606
small molecule | CAS: 89786-04-9

Tazobactam is an antibiotic of the beta-lactamase inhibitor class that prevents the breakdown of other antibiotics by beta-lactamase enzyme producing organisms. It is combined with [Piperacillin] and [Ceftolozane] for the treatment of a variety of bacterial i…

Kategori:
AmidesAnti-Infective AgentsAntibacterials for Systemic Use +15
Target Protein:
Beta-lactamaseBeta-lactamase TEMBeta-lactamase Ohio-1 +1
Waktu ParuhPiperacillin-tazoba…
Vol. Distribusi18.2 L when given w…
KlirensBecause tazobactam …
Genetik -
TB-402 DB06050
biotech

TB-402 is a human antibody binding to Factor VIII, which plays a crucial role in the coagulation of the blood. It is expected to be developed as a potential treatment to prevent blood clot formation in connection with certain types of heart arrhythmia, such a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Coagulation factor VIII
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TBA-7371 DB16243
small molecule | CAS: 1494675-86-3

TBA-7371 is under investigation in clinical trial NCT04176250 (Early Bactericidal Activity of TBA-7371 in Pulmonary Tuberculosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TBI-223 DB18911
small molecule | CAS: 2071265-08-0

TBI-223 is under investigation in clinical trial NCT06192160 (Trial of Novel Regimens for the Treatment of Pulmonary Tuberculosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TC-5231 DB05333
small molecule

TC-5231 is a small molecule that has been under investigation as an oral treatment for ADHD (Attention Deficit/Hyperactivity Disorder). TC-5231 is mecamylamine hydrochloride, the active ingredient in FDA-approved product, Inversine, but in a lower dose than I…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TD-0903 DB16463
small molecule | CAS: 2412496-23-0

TD-0903 was investigated in clinical trials for its potential to treat acute lung injury (ALI) associated with COVID-19, including NCT04350736, NCT05091723 (a pharmacokinetics study in healthy participants with supplemental oxygenation), and NCT04402866 (focu…

Kategori:
AzetinesExperimental Unapproved Treatments for COVID-19Heterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TD-2749 DB05905
small molecule | CAS: 863248-59-3

TD-2749 is selective 5-HT4 agonists discovered by Theravance through the application of multivalent drug design in a drug discovery program dedicated to finding new medicines for GI motility disorders such as chronic constipation, constipation-predominant irr…

Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tebapivat DB19338
small molecule

Tebapivat is under investigation in clinical trial NCT05490446 (A Study of Tebapivat (AG-946) in Participants With Anemia Due to Lower-risk Myelodysplastic Syndromes (LR-MDS)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tebentafusp Approved DB15283
biotech | CAS: 1874157-95-5

Tebentafusp is a gp100 peptide-HLA-directed CD3 T cell engager.[L39995] It is a bispecific, fusion protein and first-in-class drug of immune-mobilizing monoclonal T cell receptors against cancer (ImmTACs), a recently developed cancer immunotherapy with a nove…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +6
Target Protein:
Melanocyte protein PMEL
Waktu ParuhThe median terminal…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Teceleukin DB15389
biotech | CAS: 136279-32-8

Teceleukin is under investigation in clinical trial NCT03610490 (Autologous Tumor Infiltrating Lymphocytes MDA-TIL in Treating Patients With Recurrent or Refractory Ovarian Cancer, Osteosarcoma, or Pancreatic Ductal Adenocarcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tecemotide DB12568
biotech | CAS: 221214-84-2

Tecemotide has been used in trials studying the treatment of Prostate Cancer and Carcinoma, Non-Small-Cell Lung.

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsCarbohydrates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 154361-49-6

Reduced Fab fragment of the murine IgG1 monoclonal antibody IMMU-4 (also called NP-4) with specificity for carcinoembryonic antigen (CEA) covalently labeled with Technitium 99. The molecule has a molecular weight of ~54,000 Daltons.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +9
Target Protein:
Cell adhesion molecule CEACAM1
Waktu ParuhApproximately 1 hour
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5951–6000 dari 6694
Sebelumnya Halaman 120 / 134 Berikutnya