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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 120 / 236
Idalopirdine DB11957
small molecule | CAS: 467459-31-0

Idalopirdine has been used in trials studying the treatment of Cognition, Schizophrenia, and Alzheimer's Disease.

Kategori:
AminesAntidepressive AgentsBenzene Derivatives +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idanpramine DB13276
small molecule | CAS: 25466-44-8

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idarubicin Approved DB01177
small molecule | CAS: 58957-92-9

An orally administered anthracycline antineoplastic. The compound has shown activity against breast cancer, lymphomas and leukemias, together with the potential for reduced cardiac toxicity.

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +19
Target Protein:
DNA topoisomerase 2-betaDNADNA topoisomerase 2-alpha
Waktu Paruh22 hours
Vol. Distribusi-
Klirens-
Genetik -
Idasanutlin DB12325
small molecule | CAS: 1229705-06-9

Idasanutlin has been used in trials studying the treatment of Neoplasms, Non-Hodgkin's Lymphoma, Leukemia, Myeloid, Acute, Recurrent Plasma Cell Myeloma, and Neoplasms, Leukemia, Acute Myeloid Leukemia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Target Protein:
E3 ubiquitin-protein ligase Mdm2Receptor tyrosine-protein kinase erbB-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idazoxan DB12551
small molecule | CAS: 79944-58-4

Idazoxan has been used in trials studying the basic science of Molecular Imaging, Alzheimer Disease, and Major Depressive Disorder.

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDD-3 DB05427
biotech

IDD-3 is a therapeutic specific immunostimulant developed by IDM Pharma in partnership with sanofi-aventis. It consists of mature dendritic cells loaded with lysates from melanoma tumor cell lines. It includes Dendritophages that are dendritic cells, a type o…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idebenone Approved DB09081
small molecule | CAS: 58186-27-9

Idebenone is a synthetic analogue of ubiquinone (also known as Coenzyme Q10), a vital cell antioxidant and essential component of the Electron Transport Chain (ETC). It has been proposed that by interacting with the ETC, idebenone increases ATP production req…

Kategori:
AntioxidantsBenzoquinonesBiological Factors +9
Waktu Paruh-
Vol. DistribusiExperimental data h…
Klirens-
Genetik -
Idelalisib Approved DB09054
small molecule | CAS: 870281-82-6

Idelalisib is a phosphoinositide 3-kinase inhibitor indicated in the treatment of chronic lymphocytic leukemia (CLL), relapsed follicular B-cell non-Hodgkin lymphoma (FL), and relapsed small lymphocytic lymphoma (SLL). For the treatment of relapsed CLL, it is…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +47
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe terminal elimin…
Vol. Distribusi23 L
Klirens14.9 L/hr
Genetik -
IDN-7314 DB18073
small molecule | CAS: 254750-11-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Idraparinux DB06406
small molecule | CAS: 162610-17-5

Idraparinux, a synthetic pentasaccharide is an antithrombin-dependent inhibitor of activated factor X. It was developed for the treatment and prevention of thromboembolic events. However, clinical trials have revealed that idraparinux had lead to bleeding. As…

Kategori:
AnticoagulantsAntithrombinsCarbohydrates +6
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idrevloride DB18042
small molecule | CAS: 1416973-63-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idrocilamide DB13297
small molecule | CAS: 6961-46-2

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmino Alcohols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idronoxil DB04915
small molecule | CAS: 81267-65-4

Idronoxil is a substance that is being studied in the treatment of cancer. It belongs to the family of drugs called signal transduction inhibitors.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
E3 ubiquitin-protein ligase XIAPSphingosine kinase 1Ecto-NOX disulfide-thiol exchanger 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 56472-29-8

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, MonounsaturatedFatty Acids, Unsaturated +1
Target Protein:
Phosphatidylcholine:ceramide cholinephosphotransferase 1Phosphatidylcholine:ceramide cholinephosphotransferase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDRX-42 DB18087
small molecule | CAS: 2590556-80-0

Deskripsi belum tersedia.

Waktu Paruh-
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Idursulfase Approved DB01271
biotech | CAS: 50936-59-9

Idursulfase is a purified form of human iduronate-2-sulfatase, a lysosomal enzyme. Idursulfase is produced by recombinant DNA technology in a human cell line. Idursulfase is an enzyme that hydrolyzes the 2-sulfate esters of terminal iduronate sulfate residues…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +4
Target Protein:
Dermatan sulfateHeparan sulfatePerilipin-3
Waktu Paruh44 ± 19 minu…
Vol. Distribusi-
Klirens* 3 mL/min/kg [Pati…
Genetik -
biotech | CAS: 1271734-34-9

Idursulfase beta is under investigation in clinical trial NCT01645189 (Safety and Efficacy of Hunterase).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ieramilimab DB16419
biotech | CAS: 2137049-37-5

Ieramilimab is under investigation in clinical trial NCT02460224 (Safety and Efficacy of LAG525 Single Agent and in Combination With PDR001 in Patients With Advanced Malignancies.).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ifebemtinib DB17570
small molecule | CAS: 1227948-82-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Iferanserin DB11686
small molecule | CAS: 58754-46-4

Iferanserin has been investigated for the treatment of Hemorrhoids.

Kategori:
Acids, CarbocyclicAntidepressive AgentsCentral Nervous System Depressants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ifetroban DB12321
small molecule | CAS: 143443-90-7

Ifetroban has been used in trials studying the treatment of Skin Diseases, Autoimmune Diseases, Pathologic Processes, Scleroderma, Limited, and Scleroderma, Diffuse, among others.

Kategori:
Antiplatelet agentsHematologic Agents
Target Protein:
Thromboxane A2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2407582-19-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ifidancitinib DB16191
small molecule | CAS: 1236667-40-5

Ifidancitinib is under investigation in clinical trial NCT03585296 (A Study of ATI-502 Topical Solution for the Treatment of Atopic Dermatitis).

Kategori:
Adrenal Cortex HormonesFused-Ring CompoundsNorpregnanes +4
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2484870-92-8

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Ifosfamide Approved DB01181
small molecule | CAS: 3778-73-2

Ifosfamide is a chemotherapeutic agent chemically related to the nitrogen mustards and a synthetic analog of cyclophosphamide. It is active as an alkylating agent and an immunosuppressive agent.

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +46
Target Protein:
DNANuclear receptor subfamily 1 group I member 2
Waktu Paruh7-15 hours. The eli…
Vol. DistribusiIfosfamide volume o…
Klirens* 2.4±0.33 L/h/m^2 …
Genetik -
IGN101 DB06500
biotech

IGN101 is an antibody-based cancer vaccine directed against epithelial cancers. It consists of 500 ug 17-1A antibody adsorbed on aluminum hydroxide.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IGN301 DB05117
biotech

IGN301 is a cancer vaccine based on an anti-idiotypic antibody which provokes an immune response to Lewis Y. Lewis Y is a carbohydrate molecule expressed on the surface of tumor cells of epithelial origin (e.g. lung, intestinal, breast, prostate or ovarian ca…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IKT-001Pro DB17307
small molecule

Deskripsi belum tersedia.

Kategori:
Kinase Inhibitor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IL15-NK Cell DB15725
biotech

Natural killer (NK) cells can be incubated with ‘feeder cells’ expressing certain cytokines prior to maturation to enhance their activity. In particular, incubation with IL-15 allows NK cells to lyse a broad range of fresh and cultured tumor targets that the …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ilacirnon DB16066
small molecule | CAS: 1100318-47-5

Ilacirnon (CCX-140) is under investigation in clinical trial NCT01440257 (A Study to Evaluate the Effect of CCX140-B on Urinary Albumin Excretion in Subjects With Type 2 Diabetes and Albuminuria).

Target Protein:
C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ilaprazole DB11964
small molecule | CAS: 172152-36-2

Ilaprazole has been investigated in Helicobacter Infections.

Kategori:
Anti-Ulcer AgentsBenzimidazolesGastric Acid Lowering Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ilepatril DB06604
small molecule | CAS: 473289-62-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingProdrugs
Target Protein:
NeprilysinAngiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ilepcimide DB16942
small molecule | CAS: 82857-82-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ilginatinib DB12784
small molecule | CAS: 1239358-86-1

NS-018 has been used in trials studying the treatment of Primary Myelofibrosis, Post-Polycythemia Vera Myelofibrosis, and Post-Essential Thrombocythemia Myelofibrosis.

Target Protein:
Tyrosine-protein kinase JAK2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ilodecakin DB06449
small molecule | CAS: 149824-15-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iloperidone Approved DB04946
small molecule | CAS: 133454-47-4

Iloperidone is a benzisoxazole [A263557] and an atypical antipsychotic agent that was first approved by the FDA on May 6, 2009.[A3024] It is considered to be a second-generation antipsychotic drug [A263552] with multiple receptor binding profile, although it …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +31
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +14
Waktu ParuhThe observed mean e…
Vol. DistribusiThe apparent volume…
KlirensIloperidone has an …
Genetik -
Iloprost Approved DB01088
small molecule | CAS: 78919-13-8

Iloprost is an analog of prostacyclin (PGI2; epoprostenol), an endogenous prostanoid mainly produced in the vascular endothelium. It is more stable than prostacyclin, which is short-lived.[A263326] Iloprost consists of a mixture of the 4R and 4S diastereoisom…

Kategori:
Agents Causing Muscle ToxicityAntiplatelet agentsAutacoids +16
Target Protein:
Prostacyclin receptorProstaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype +6
Waktu ParuhThe half-life of il…
Vol. DistribusiFollowing intraveno…
KlirensClearance in normal…
Genetik -
Ilorasertib DB11694
small molecule | CAS: 1227939-82-3

Ilorasertib has been used in trials studying the treatment of Myelodysplasia, Solid Neoplasm, Advanced Cancers, Advanced Solid Tumors, and Acute Myelogenous Leukemia, among others.

Kategori:
AmidesAminesAntineoplastic Agents +4
Target Protein:
Aurora kinase AAurora kinase BAurora kinase C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ILS-920 DB15422
small molecule | CAS: 892494-07-4

ILS-920 is under investigation in clinical trial NCT00827190 (Study Evaluating Single Ascending Doses Of ILS-920).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iluzanebart DB18275
biotech | CAS: 2733621-19-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1422365-93-2

Deskripsi belum tersedia.

Kategori:
Amidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IMAB027 DB17282
biotech

IMAB027 is a chimeric monoclonal antibody against Claudin 6.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imagabalin DB12105
small molecule | CAS: 610300-07-7

Imagabalin has been investigated in Generalized Anxiety Disorder.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Anxiety AgentsCentral Nervous System Depressants
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imalumab DB15558
biotech | CAS: 1430205-07-4

Imalumab is under investigation in clinical trial NCT02540356 (Phase 1/2a Two-arm Dose-escalation Study of BAX69 in Subjects With Malignant Ascites of Ovarian Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imaradenant DB16192
small molecule | CAS: 1321514-06-0

Imaradenant is under investigation in clinical trial NCT03381274 (Oleclumab (MEDI9447) Egfrm NSCLC Novel Combination Study).

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imatinib Approved DB00619
small molecule | CAS: 152459-95-5

Imatinib is a small molecule kinase inhibitor that revolutionized the treatment of cancer, particularly chronic myeloid leukemia, in 2001.[A249305] It was deemed a "miracle drug" due to its clinical success, as oncologist Dr. Brian noted that "complete hemato…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +51
Target Protein:
Breakpoint cluster region proteinInduced myeloid leukemia cell differentiation protein Mcl-1Mast/stem cell growth factor receptor Kit +8
Waktu ParuhFollowing oral admi…
Vol. DistribusiPopulation pharmaco…
KlirensTypically, clearanc…
Genetik -
IMCY-0141 DB17019
biotech

IMCY-0141 is a synthetic peptide based on MOG (Myelin Oligodendrocyte Glycoprotein), a dominant autoantigen, designed to stop the progression of multiple sclerosis (MS) and the destruction of the myelin sheath protecting the nerves.[L43287]

Waktu Paruh-
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Imdusiran DB19014
biotech | CAS: 2839476-19-4

Imdusiran is under investigation in clinical trial NCT06245291 (Study of Imdusiran (AB-729) in Combination With Intermittent Dosing of Durvalumab in Subjects With Chronic HBV Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imeglimin DB12509
small molecule | CAS: 775351-65-0

Imeglimin has been used in trials studying the treatment of Type 2 Diabetes Mellitus.

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsDrugs Used in Diabetes
Target Protein:
5'-AMP-activated protein kinase catalytic subunit alpha-15'-AMP-activated protein kinase subunit beta-15'-AMP-activated protein kinase subunit gamma-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imelasomeran Approved DB17090
biotech | CAS: 2763208-92-8

Imelasomeran was first approved in Canada on September 1, 2022, as one-half of Moderna's Spikevax Bivalent COVID-19 mRNA vaccine.[L45320] It encodes for the viral spike protein of the Omicron BA.1 variant of SARS-CoV-2, a particularly infectious variant of co…

Kategori:
COVID-19 VaccinesmRNA VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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