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2279

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Halaman 12 / 46
Crizanlizumab Approved DB15271
biotech | CAS: 1690318-25-2

Crizanlizumab is a humanized IgG2 monoclonal antibody used to reduce the frequency of vaso-occlusive crises in patients with sickle cell disease.[L10097] Sickle cell disease is a genetically inherited condition prevalent in the Middle East, Africa, and certai…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
P-selectin
Waktu ParuhGiven a 5mg/kg dose…
Vol. DistribusiThe volume of distr…
KlirensGiven a 5mg/kg dose…
Genetik -
Crizotinib Approved DB08865
small molecule | CAS: 877399-52-5

Crizotinib is a tyrosine kinase receptor inhibitor used for the treatment of anaplastic lymphoma kinase (ALK) or ROS1-positive non-small cell lung cancer (NSCLC) tumors, as well as ALK-positive anaplastic large cell lymphoma (ALCL) and inflammatory myofibrobl…

Kategori:
AminopyridinesAnaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic Agents +32
Target Protein:
ALK tyrosine kinase receptorHepatocyte growth factor receptorProto-oncogene tyrosine-protein kinase ROS +1
Waktu ParuhFollowing single do…
Vol. DistribusiFollowing a single …
KlirensAt steady-state (25…
Genetik -
biotech

Each year it is estimated there are 45,000 snakebites in the US and 300,000 to 400,000 bites worldwide. About 8000 of these snakebites involve venomous snake species. The majority of people bitten are males and about 50% occur in the age group of 18 to 28 [F1…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Target Protein:
Group 10 secretory phospholipase A2
Waktu Paruh12 to 23 hours [FDA…
Vol. Distribusi-
KlirensThis product was sh…
Genetik -
biotech

Crotalus scutulatus antivenin is derived and purified immunoglobulin fragments obtained from other domestic animals such as sheep previously immunized with Crotalus scutulatus (also known as the _Mojave rattlesnake_ [L2856]). The final purified antivenin …

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu ParuhApproximately 15 ho…
Vol. Distribusi0.3 L/kg [FDA label]
Klirens32 mL/min (approxim…
Genetik -
Crovalimab Approved DB16128
biotech | CAS: 1917321-26-6

Crovalimab is a humanized monoclonal antibody and complement C5 inhibitor.[L50908] It consists of two heavy chains (451 amino acid residues each) and two light chains (217 amino acid residues each).[L50908] First developed by Chugai Pharmaceutical, in collabo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +7
Target Protein:
Complement C5
Waktu ParuhThe mean estimated …
Vol. DistribusiThe mean central an…
KlirensIn PNH treatment-na…
Genetik -
CRS-207 DB17323
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Vesta Therapeutics is a privately held company developing cell therapeutics for liver repair and regeneration. The Company's technology is centered on the isolation, expansion, and cryopreservation of liver cells (human hepatocytes) obtained from organ donor …

Waktu Paruh-
Vol. Distribusi-
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Genetik -
CSL324 DB16359
biotech

CSL324 is a fully human anti-G-CSFR antibody shown to have the ability to control G-CSF-mediated neutrophilia in cynomolgus macaques.[A225626] It has potential applications in various inflammatory conditions such as cystic fibrosis, inflammatory bowel disease…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
CT-001 DB18284
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
CT-011 DB05916
biotech

CT-011 is a humanized monoclonal antibody directed against a B7 family-associated protein, in patients with advanced haematological malignancies. It is directed against human PD-1 (programmed cell death 1; PDCD1), with immunomodulating and antitumor activitie…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +7
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTA018 DB05024
small molecule

CTA018 is a member of a new class of vitamin D analogues with a dual mechanism of action, called Vitamin D Signal Amplifiers. This proprietary new drug is both a potent inhibitor of CYP24 (the enzyme responsible for the breakdown of vitamin D) and a potent ac…

Target Protein:
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialVitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTx-PDE6b DB17858
biotech

CTx-PDE6b is an adeno-associated virus (AAV) based gene therapy designed to deliver a full-length non-mutated copy of the functional human _PDE6b_ gene. Being commercialied by Coave Therapeutics, it is being investigated for the treatment of retinitis pigment…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Cupric oxide Approved DB11134
small molecule | CAS: 1317-38-0

Cupric oxide, or copper (II) oxide, is an inorganic compound with the chemical formula CuO. Cupric oxide is used as a precursor in many copper-containing products such as wood preservatives and ceramics. Cupric oxide may be found in over-the-counter vitamin-m…

Kategori:
Diet, Food, and NutritionElementsFood +6
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiFollowing exposure …
KlirensNo pharmacokinetic …
Genetik -
Cupric sulfate Approved DB06778
small molecule | CAS: 7758-98-7

Cupric sulfate is a salt created by treating cupric oxide with sulfuric acid. This forms as large, bright blue crystals containing five molecules of water (CuSO4?5H2O) and is also known as _blue vitriol_. The anhydrous salt is created by heating the hydrate t…

Kategori:
AntidotesAutonomic AgentsCentral Nervous System Agents +10
Waktu ParuhThe biological half…
Vol. DistribusiThe body of a 70 kg…
Klirens-
Genetik -
biotech

_Curcuma xanthorrhiza_ oil is extracted from _Curcuma xanthorrhiza_ Roxb., a member of the ginger family (_Zingiberaceae_) that is widely distributed in the region of Southeastern Asia [A33162]. _Curcuma xanthorrhiza_ is also known as Javanese Turmeric or Te…

Waktu ParuhThere are no pharma…
Vol. DistribusiThere are no pharma…
KlirensThere are no pharma…
Genetik -
Cusatuzumab DB15100
biotech | CAS: 1864871-20-4

CD70 is a ligand expressed on the surface of activated lymphocytes and mature dendritic cells that, in its binding to CD27 receptors, plays an important role in cell proliferation and survival. An overexpression of CD70 can result in the proliferation of mali…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Target Protein:
CD70 antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CVac Approved DB17351
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CVnCoV DB15844
biotech

The CVnCov Vaccine (or CV07050101) is in development by CureVac AG. The vaccine uses mRNA technology to create a protein associated with SARS-CoV2, and upon administration and replication, to initiate subsequent immune responses in the body. As of June 2020, …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CVnCoV Vaccine DB15843
biotech

The CVnCov Vaccine (or CV07050101) is in development by CureVac AG. The vaccine uses mRNA technology to create a protein associated with SARS-CoV2, and upon administration and replication, to initiate subsequent immune responses in the body. As of June 2020, …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyanamide DB02679
small molecule | CAS: 420-04-2

A cyanide compound which has been used as a fertilizer, defoliant and in many manufacturing processes. It often occurs as the calcium salt, sometimes also referred to as cyanamide. The citrated calcium salt is used in the treatment of alcoholism. [PubChem]

Kategori:
CarbodiimidesCyanidesImines +1
Target Protein:
Cathepsin KCarbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyanocobalamin Approved DB00115
small molecule | CAS: 68-19-9

Cyanocobalamin (commonly known as Vitamin B12) is a highly complex, essential vitamin, owing its name to the fact that it contains the mineral, cobalt. This vitamin is produced naturally by bacteria [A175276], and is necessary for DNA synthesis and cellular e…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCorrinoids +10
Target Protein:
Methionine synthaseMethylmalonyl-CoA mutase, mitochondrialMethionine synthase reductase +3
Waktu ParuhApproximately 6 day…
Vol. DistribusiCobalamin is distri…
KlirensDuring vitamin load…
Genetik -
Cyclandelate Approved DB04838
small molecule | CAS: 456-59-7

A direct-acting smooth muscle relaxant used to dilate blood vessels. It may cause gastrointestinal distress and tachycardia. Cyclandelate is not approved for use in the U.S. or Canada, but is approved in various European countries.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAntiarrhythmic agents +10
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1Liver carboxylesterase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 60-92-4

Cyclic adenosine monophosphate (cAMP, cyclic AMP or 3'-5'-cyclic adenosine monophosphate) is a molecule that is important in many biological processes; it is derived from adenosine triphosphate (ATP).

Kategori:
Adenine NucleotidesCyclic AMPHeterocyclic Compounds, Fused-Ring +8
Target Protein:
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2cAMP-dependent protein kinase type I-alpha regulatory subunitcAMP-dependent protein kinase type II-beta regulatory subunit +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cyclobenzaprine Approved DB00924
small molecule | CAS: 303-53-7

Cyclobenzaprine, a centrally-acting muscle relaxant, was first synthesized in 1961[A185039] and has been available for human use since 1977.[A184982] It was initially studied for use as antidepressant given its structural similarity to tricyclic antidepressan…

Kategori:
Agents that reduce seizure thresholdAntidepressive AgentsBenzocycloheptenes +23
Target Protein:
Alpha-2C adrenergic receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2B +7
Waktu ParuhThe effective half-…
Vol. DistribusiThe volume of distr…
KlirensThe approximate pla…
Genetik -
Cyclosporine Approved DB00091
small molecule | CAS: 59865-13-3

Cyclosporine is a calcineurin inhibitor known for its immunomodulatory properties that prevent organ transplant rejection and treat various inflammatory and autoimmune conditions. It is isolated from the fungus _Beauveria nivea_.[A174049] Initially manufactur…

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAgents that produce hypertension +45
Target Protein:
Guided entry of tail-anchored proteins factor CAMLGProtein phosphatase 3 catalytic subunit alphaCalcineurin subunit B type 2 +2
Waktu ParuhThe half-life of cy…
Vol. DistribusiThe distribution of…
KlirensCyclosporin shows a…
Genetik -
Cyclothiazide Approved DB00606
small molecule | CAS: 2259-96-3

As a diuretic, cyclothiazide inhibits active chloride reabsorption at the early distal tubule via the Na-Cl cotransporter, resulting in an increase in the excretion of sodium, chloride, and water. Thiazides like cyclothiazide also inhibit sodium ion transport…

Kategori:
Antihypertensive AgentsCardiovascular AgentsDiuretics +11
Target Protein:
Sodium/potassium-transporting ATPase subunit gammaCarbonic anhydraseCarbonic anhydrase 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cycrimine Approved DB00942
small molecule | CAS: 77-39-4

Cycrimine is a drug used to reduce levels of acetylcholine to return a balance with dopamine in the treatment and management of Parkinson's disease.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsMuscarinic Antagonists
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CYNK-001 DB15722
biotech

CYNK-001 is a novel allogenic off-the-shelf natural killer (NK) cell therapy originating from human placental CD34+ hematopoietic stem cells and enriched with CD56+/CD3-.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
CYNK-101 DB18637
biotech

CYNK-101 is an allogeneic human placental hematopoietic stem cell-derived natural killer (NK) cell therapy product that is genetically modified to express a variant of CD16 (CD16VP).

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Vol. Distribusi-
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Genetik -
Cynodon dactylon pollen Approved DB10351
biotech

Cynodon dactylon pollen, also known as bermuda grass pollen, is a standardized grass pollen extracts used for the diagnosis and treatment of allergic disease to grass pollen. It can be cutaneously, intradermally and subcutaneously administered to initiate an …

Kategori:
Allergenic ExtractsCell-mediated ImmunityGrass Pollen Allergen Extracts +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CypCaps DB17435
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cysteamine Approved DB00847
small molecule | CAS: 60-23-1

Cystinosis is a rare disease caused by mutations in the CTNS gene that encodes for cystinosin, a protein responsible for transporting cystine out of the cell lysosome. A defect in cystinosin function is followed by cystine accumulation throughout the body, es…

Kategori:
Alimentary Tract and MetabolismAminesAmino Acids and Derivatives +11
Target Protein:
SomatostatinCystineNeuropeptide Y receptor type 2
Waktu ParuhThe half-life of cy…
Vol. DistribusiCysteamine has a vo…
KlirensThe plasma clearanc…
Genetik -
CYT-6091 DB05991
small molecule

CYT-6091 (Aurimune) is an investigational small molecule made up of recombinant human tumor necrosis factor alpha (rhTNF) and thiolyated polyethylene glycol bound to the surface of 27 nm colloidal gold particles. It was under investagtion in clinical trials N…

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingElements +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
D-3082-L DB17440
biotech | CAS: 2170657-73-3

D-3082-L is one of the components of the human papilloma virus (HPV) type 16 E6/E7 synthetic long peptide (SLP) vaccine ISA101b.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
D-alpha-Tocopherol acetate Approved DB14002
small molecule | CAS: 58-95-7

Alpha-tocopherol is the primary form of vitamin E that is preferentially used by the human body to meet appropriate dietary requirements. In particular, the RRR-alpha-tocopherol (or sometimes called the d-alpha-tocopherol stereoisomer) stereoisomer is conside…

Kategori:
AntioxidantsBenzopyransBiological Factors +12
Target Protein:
SEC14-like protein 3SEC14-like protein 2Nuclear receptor subfamily 1 group I member 2 +3
Waktu Paruh_In addition to any…
Vol. Distribusi_In addition to any…
Klirens_In addition to any…
Genetik -
small molecule | CAS: 870452-26-9

D-fluoromethyltyrosine F-18 is under investigation in clinical trial NCT01089998 (PET/CT Imaging for Radiation Dosimetry, Plasma Pharmacokinetics, Safety and Tolerability in Healthy Volunteers and Safety, Tolerability and Diagnostic Performance of BAY86-9596 …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
D-glucose Approved DB01914
small molecule | CAS: 50-99-7

Glucose is a simple sugar (monosaccharide) generated during phosynthesis involving water, carbon and sunlight in plants. It is produced in humans via hepatic gluconeogenesis and breakdown of polymeric glucose forms (glycogenolysis). It circulates in human cir…

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +11
Waktu ParuhThe approximate hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean metabolic …
Genetik -
D-Glutamine DB02174
small molecule | CAS: 5959-95-5

A non-essential amino acid present abundantly throughout the body and is involved in many metabolic processes. It is synthesized from glutamic acid and ammonia. It is the principal carrier of nitrogen in the body and is an important energy source for many cel…

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Glutamate racemase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Phosphoheptose isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
D-Lactic acid DB03066
small molecule | CAS: 10326-41-7

A normal intermediate in the fermentation (oxidation, metabolism) of sugar. The concentrated form is used internally to prevent gastrointestinal fermentation. (From Stedman, 26th ed)

Kategori:
Hydroxy AcidsLactates
Target Protein:
(S)-2-haloacid dehalogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 27251-84-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesHexosephosphatesSugar Phosphates
Target Protein:
Phosphomannomutase/phosphoglucomutase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1986-14-7

Deskripsi belum tersedia.

Target Protein:
AlgQ1AlgQ2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
D-Proline DB02853
small molecule | CAS: 344-25-2

D-proline is an isomer of the naturally occurring amino acid, L-Proline. D-amino acids have been found in relatively high abundance in human plasma and saliva [A19262]. These amino acids may be of bacterial origin, but there is also evidence that they are end…

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Vol. Distribusi-
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Genetik -
small molecule | CAS: 10162-32-0

A pteridine derivative present in body fluids; elevated levels result from immune system activation, malignant disease, allograft rejection, and viral infections. (From Stedman, 26th ed) Neopterin also serves as a precursor in the biosynthesis of biopterin.

Kategori:
CoenzymesEnzymes and CoenzymesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
D-Tryptophan DB03225
small molecule | CAS: 153-94-6

Tryptophan is one of the 20 standard amino acids, as well as an essential amino acid in the human diet. It is encoded in the standard genetic code as the codon UGG. The D-stereoisomer is occasionally found in naturally produced peptides (for example, the mari…

Target Protein:
Hydroxycarboxylic acid receptor 3D-amino-acid oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2365353-63-3

Dabocemagene autoficel is an _ex vivo_, autologous cell-based gene therapy. It comprises autologous dermal fibroblasts genetically modified to express functional type VII collagen. Developed by Castle Creek Biosciences Inc., dabocemagene autoficel is being in…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Dacetuzumab DB12589
biotech | CAS: 880486-59-9

Dacetuzumab has been used in trials studying the treatment of Multiple Myeloma, Non-Hodgkin Lymphoma, Leukemia, Lymphocytic, Chronic, and Lymphoma, Large B-Cell, Diffuse. It is a humanized anti-CD40 antibody and induces cytotoxicity in human multiple myeloma …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Tumor necrosis factor receptor superfamily member 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Daclizumab DB00111
biotech | CAS: 152923-56-3

Humanized IgG1 Mab that binds to the human interleukin-2 receptor (anti-Tac or anti-CD25). Daclizumab is a composite of human (90%) and murine (10%) antibody sequences. The human sequences were derived from the constant domains of human IgG1 and the variable …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Interleukin-2 receptor subunit alphaInterleukin-2 receptor subunit betaLow affinity immunoglobulin gamma Fc region receptor III-B +9
Waktu Paruh11-38 days
Vol. Distribusi-
Klirens-
Genetik -
biotech

Dalcinonacog alfa is a recombinant human factor IX (FIX) variant. It is being investigated for the treatment of hemophilia B.[A259058]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Danaparoid Approved DB06754
small molecule | CAS: 308068-55-5

Danaparoid is a low-molecular-weight heparinoid with an average molecular weight of 5500 Daltons consisting of a mixture of glycosaminoglycans [A32565]. The active constituents are heparan, dermatan and [DB09301] [T28], and they are isolated from the porcine …

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +9
Target Protein:
Antithrombin-III
Waktu ParuhPharmacokinetic stu…
Vol. DistribusiPharmacokinetic stu…
KlirensPharmacokinetic stu…
Genetik -
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