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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 119 / 252
Geneticin DB04263
small molecule | CAS: 49863-47-0

Geneticin (also known as G418) is an aminoglycoside antibiotic similar in structure to gentamicin B1, produced by Micromonospora rhodorangea. Geneticin blocks polypeptide synthesis by inhibiting the elongation step in both prokaryotic and eukaryotic cells and…

Kategori:
Agents that produce neuromuscular block (indirect)AmebicidesAminoglycoside Antibacterials +8
Target Protein:
Ornithine decarboxylase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Genipin DB19124
small molecule | CAS: 6902-77-8

Genipin is under investigation in clinical trial NCT05755750 (Intratendinous Genipin Injection in Horses With Tendon Injuries).

Kategori:
AdhesivesCholagogues and CholereticsCycloparaffins +6
Waktu Paruh-
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Genistein DB01645
small molecule | CAS: 446-72-0

An isoflavonoid derived from soy products. It inhibits protein-tyrosine kinase and topoisomerase-II (DNA topoisomerases, type II) activity and is used as an antineoplastic and antitumor agent. Experimentally, it has been shown to induce G2 phase arrest in hum…

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsBCRP/ABCG2 Inhibitors +31
Target Protein:
Estrogen receptor betaNuclear receptor coactivator 1Estrogen receptor +11
Waktu Paruh-
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Genetik -
Gentamicin Approved DB00798
small molecule | CAS: 1403-66-3

Gentamicin is a bactericidal aminoglycoside that was discovered and isolated from _Micromonospora purpurea_ in 1963.[A234349] It is one of the most frequently prescribed aminoglycosides due to its spectrum of activity, low cost, and availability.[A234339,A234…

Kategori:
Agents that produce neuromuscular block (indirect)alpha-Galactosidase, antagonists & inhibitorsAminoglycoside Antibacterials +21
Target Protein:
30S ribosomal protein S1216S ribosomal RNA23S ribosomal RNA +4
Waktu ParuhOne study assessing…
Vol. Distribusi-
KlirensThe renal clearance…
Genetik -
Gentamicin C2 DB17884
small molecule | CAS: 25876-11-3

Deskripsi belum tersedia.

Kategori:
Aminoglycoside AntibacterialsAnti-Bacterial AgentsCarbohydrates +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Genz-10850 DB04289
small molecule

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Gepirone Approved DB12184
small molecule | CAS: 83928-76-1

Gepirone, an azapirone, is a pharmacologic analog of [buspirone] that acts selectively on the pre- and post-synaptic 5HT<sub>1A</sub> receptors. Although earlier clinical trials showed promising results for gepirone, its formulation as an immediate-release ta…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsCentral Nervous System Agents +12
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensAfter the administr…
Genetik -
Gepotidacin DB12134
small molecule | CAS: 1075236-89-3

Gepotidacin has been used in trials studying the treatment of Gonorrhea, Infections, Bacterial, and Infections, Respiratory Tract.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Geptanolimab DB16417
biotech | CAS: 2348469-43-0

Geptanolimab is under investigation in clinical trial NCT03502629 (Clinical Trial in Chinese Patients of Relapsed and Refractory Peripheral T Cell Lymphoma (GB226)).

Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
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Geraniol Approved DB14183
small molecule | CAS: 106-24-1

Geraniol is a monoterpene that is found within many essential oils of fruits, vegetables, and herbs including rose oil, citronella, lemongrass, lavender, and other aromatic plants. It is emitted from the flowers of many species of plant and is commonly used b…

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseMonoterpenes +2
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu ParuhIn vitro measuremen…
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAnions +8
Target Protein:
Farnesyl pyrophosphate synthase2-C-methyl-D-erythritol 2,4-cyclodiphosphate synthasePrenyltransferase +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Gestodene DB06730
small molecule | CAS: 60282-87-3

Gestodene is a progestogen hormonal contraceptive. Products containing gestoden include Meliane, which contains 20 mcg of ethinylestradiol and 75 mcg of gestodene; and Gynera, which contains 30 mcg of ethinylestradiol and 75 mcg of gestodene.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +30
Target Protein:
Progesterone receptor
Waktu Paruh16 to 18 hrs.
Vol. Distribusi-
Klirens-
Genetik -
Gestonorone caproate Approved DB14677
small molecule | CAS: 1253-28-7

Deskripsi belum tersedia.

Kategori:
Fused-Ring CompoundsNorpregnanesNorpregnenes +5
Waktu Paruh-
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Genetik -
GET-73 DB12928
small molecule | CAS: 202402-01-5

Get 73 has been investigated for the treatment of Alcohol Dependence.

Waktu Paruh-
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Gevokizumab DB12119
biotech | CAS: 1129435-60-4

Gevokizumab has been used in trials studying the treatment of Acne Vulgaris, Osteoarthritis, Behcet's Uveitis, Pyoderma Gangrenosum, and Behcet's Disease Uveitis, among others. Gevokizumab acts as a modulator of cytokine imbalance in IL-1 mediated disease sta…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Interleukin-1 beta
Waktu Paruh-
Vol. Distribusi-
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GFH-925 DB17481
small molecule

GFH-925 is an irreversibly covalent inhibitor of KRAS G12C.

Waktu Paruh-
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GFT14 DB05061
small molecule

GFT14 is a new class of medicaction for treatment of cardiometabolic disease. GFT14 aims to target mixed dyslipidemia of type IIb (high levels of triglycerides and LDL-C) as one of the major indications of cardiometabolic disease. GFT14 is destined to improv…

Waktu Paruh-
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GI heptapeptide DB15070
biotech

GI heptapeptide is under investigation in clinical trial NCT01391208 (Esophageal Protocol for Detection of Neoplasia in the Digestive Tract).

Waktu Paruh-
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GI-181771X DB12309
small molecule | CAS: 305366-98-7

Gski181771 X is under investigation in clinical trial NCT00600743 (Effect of a CCK-1R Agonist on Food Intake in Humans).

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-RingReceptor, Cholecystokinin A, agonists
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-4000 DB05698
biotech

A vaccine containing a heat-killed recombinant <em>Saccharomyces cerevisiae</em> yeast transfected with mutated forms of Ras, an oncogene frequently found in solid tumors, with potential immunostimulant and antitumor activity. [L112]

Waktu Paruh-
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GI-5005 DB05942
biotech | CAS: 1001913-27-4

GI-5005 is GlobeImmune's lead infectious disease product from its proprietary Tarmogen active immunotherapy platform for the treatment of chronic hepatitis C infection. GI-5005 is whole, heat-killed recombinant yeast genetically modified to express HCV-specif…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +5
Waktu Paruh-
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Genetik -
GI-6207 DB17532
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-6301 DB17533
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Gibberella fujikuroi Approved DB15511
biotech

Gibberella fujikuroi allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Genetik -
small molecule | CAS: 77-06-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +5
Target Protein:
Arylacetamide deacetylase-like 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gibberellin A4 DB07815
small molecule | CAS: 468-44-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +2
Target Protein:
Arylacetamide deacetylase-like 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Giloralimab DB18862
biotech | CAS: 2226292-20-0

Giloralimab is under investigation in clinical trial NCT04807972 (Study to Evaluate Adverse Events and Change in Disease Activity When Intravenous (IV) Infusion of ABBV-927 Is Administered in Combination With IV Modified FOLFIRINOX (Mffx) With or Without IV B…

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Gilteritinib Approved DB12141
small molecule | CAS: 1254053-43-4

Gilteritinib, also known as ASP2215, is a small molecule part of the FLT3 tyrosine kinase inhibitors that presented a greater selectivity and potency when compared with other agents from this group.[A40036] It is a pyrazinecarboxamide derivative that showed h…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +16
Target Protein:
Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase receptor UFOALK tyrosine kinase receptor +1
Waktu ParuhThe reported median…
Vol. DistribusiThe estimated appar…
KlirensThe estimated clear…
Genetik -
Gimeracil Approved DB09257
small molecule | CAS: 103766-25-2

Gimeracil is an adjunct to antineoplastic therapy, used to increase the concentration and effect of the main active componets within chemotherapy regimens. Approved by the European Medicines Agency (EMA) in March 2011, Gimeracil is available in combination wi…

Kategori:
Drugs that are Mainly Renally Excreted
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
Klirens-
Genetik -
Gimsilumab DB15280
biotech | CAS: 1648796-29-5

Gimsilumab is under investigation in clinical trial NCT01357759 (Safety and Tolerability of MORAb-022 in Healthy and Rheumatoid Arthritis Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gingerol DB19255
small molecule | CAS: 23513-14-6

Gingerol is under investigation in clinical trial NCT05882864 (Efficacy of Ginger Muco-bioadhesive Gel in Management of Oral Lichen Planus With Immunohistochemical Analysis).

Kategori:
AlcoholsBenzene DerivativesLipids +2
Target Protein:
Transient receptor potential cation channel subfamily A member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginkgo biloba Approved DB01381
biotech | CAS: 90045-36-6

_Ginkgo biloba_ extract contains a group of terpene lactones (notably, ginkgolides and diterpenes) and ginkgo flavone glycosides (notably, ginkgetin, bilobetin, and sciadopitysin) that have antioxidant and vasoactive properties.[A232389] Most of the studies t…

Kategori:
Anti-Dementia DrugsBiological ProductsBlood Circulation +27
Target Protein:
Sodium-dependent noradrenaline transporterPhospholipase A2, membrane associatedGlycine receptor subunit alpha-1 +5
Waktu ParuhUnpublished human d…
Vol. DistribusiNo data available.
KlirensNo data available.
Genetik -
biotech

Ginkgo biloba leaf oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Ginkgolide A DB06743
small molecule | CAS: 15291-75-5

Ginkgolide A is a highly active PAF antagonist cage molecule that is isolated from the leaves of the Ginkgo biloba tree. Shows potential in a wide variety of inflammatory and immunological disorders.

Kategori:
DiterpenesTerpenes
Target Protein:
Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2Glycine receptor subunit alpha-3 +1
Waktu Paruh-
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ginkgolide-C DB06745
small molecule | CAS: 15291-76-6

Deskripsi belum tersedia.

Kategori:
DiterpenesTerpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ginkgolide-M DB06747
small molecule | CAS: 15291-78-8

Deskripsi belum tersedia.

Waktu Paruh-
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Ginseng DB01404
biotech | CAS: 50647-08-0

Ginseng is promoted as an adaptogen (a product that increases the body's resistance to stress), one which can to a certain extent be supported with reference to its anticarcinogenic and antioxidant properties. Ginseng is also known to contain phytoestrogens.

Kategori:
AngiospermsAraliaceaeBiological Products +11
Target Protein:
Aryl hydrocarbon receptorInterleukin-6Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginsenoside B2 DB14815
small molecule | CAS: 52286-59-6

Ginsenoside B2 is under investigation in clinical trial NCT00781534 (A Clinical Trial of Ginseng in Diabetes).

Kategori:
CarbohydratesGlycosidesPanax +3
Waktu Paruh-
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Ginsenoside Rb1 DB06749
small molecule | CAS: 41753-43-9

Ginsenosides are a class of steroid glycosides, and triterpene saponins, found exclusively in the plant genus Panax (ginseng). Ginsenosides have been the target of research, as they are viewed as the active compounds behind the claims of ginseng's efficacy. B…

Kategori:
CarbohydratesGlycosidesOATP1B3 inhibitors +4
Target Protein:
Solute carrier organic anion transporter family member 1B3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginsenoside Rd DB19256
small molecule | CAS: 52705-93-8

Ginsenoside Rd is under investigation in clinical trial NCT00815763 (Efficacy and Safety of Ginsenoside-rd for Acute Ischemic Stroke).

Kategori:
CarbohydratesGlycosidesPanax +3
Waktu Paruh-
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Ginsenoside Rg1 DB06750
small molecule | CAS: 22427-39-0

Ginsenosides are a class of steroid glycosides, and triterpene saponins, found exclusively in the plant genus Panax (ginseng). Ginsenosides have been the target of research, as they are viewed as the active compounds behind the claims of ginseng's efficacy. B…

Kategori:
CarbohydratesCentral Nervous System AgentsGlycosides +4
Target Protein:
Solute carrier organic anion transporter family member 1B3
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Ginsenoside Rg3 DB19257
small molecule | CAS: 14197-60-5

Ginsenoside Rg3 is under investigation in clinical trial NCT01757366 (Safety and Efficacy of Ginsenoside Rg3 in Combination With First-line Chemotherapy in Advanced Gastric Cancer).

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicCarbohydrates +5
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginsenosides DB14152
small molecule | CAS: 74749-74-9

Dammarane type triterpene saponins based mainly on the aglycones, protopanaxadiol and protopanaxatriol.

Kategori:
CarbohydratesGlycosidesSaponins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Giredestrant DB19125
small molecule | CAS: 1953133-47-5

Giredestrant is under investigation in clinical trial NCT06065748 (A Study to Evaluate Efficacy and Safety of Giredestrant Compared With Fulvestrant (Plus a CDK4/6 Inhibitor), in Participants With Er-positive, Her2-negative Advanced Breast Cancer Resistant to…

Kategori:
Heterocyclic Compounds, Fused-RingIndole AlkaloidsIndoles +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Girentuximab DB05304
biotech | CAS: 916138-87-9

Girentuximab is a monoclonal chimeric (mouse/human) antibody directed against carbonic anhydrase IX, an antigen expressed in 95% of clear cell renal cell carcinomas (RCC).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Carbonic anhydrase 9Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1011710-99-8

Girentuximab I-124 is under investigation in clinical trial NCT01762592 (REDECT 2: REnal Masses: Pivotal Trial to DEteCT Clear Cell Renal Cell Carcinoma With PET/CT).

Waktu Paruh-
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Giripladib DB15426
small molecule | CAS: 865200-20-0

Giripladib is under investigation in clinical trial NCT00396955 (A Study Comparing 4 Dose Regimens of PLA-695, Naproxen, and Placebo In Subjects With Osteoarthritis Of The Knee).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2166101-71-7

Giroctocogene fitelparvovec is under investigation in clinical trial NCT04370054 (Study to Evaluate the Efficacy and Safety of PF-07055480 in Moderately Severe to Severe Hemophilia a Adults).

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Gitoformate DB13537
small molecule | CAS: 10176-39-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesCardanolidesCardenolides +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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