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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 118 / 236
Huperzine A Approved DB04864
small molecule | CAS: 102518-79-6

Huperzine A, is a naturally occurring sesquiterpene alkaloid found in the extracts of the firmoss _Huperzia serrata_. The botanical has been used in China for centuries for the treatment of swelling, fever and blood disorders. Recently in clinical trials in C…

Kategori:
Central Nervous System AgentsCholinergic AgentsCholinesterase Inhibitors +6
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
HX-1171 DB12162
small molecule | CAS: 148081-72-5

Hx 1171 is under investigation in clinical trial NCT01548391 (A Phase I Clinical Study Study of the Safety, Tolerability, and Pharmacokinetics of HX-1171 in Healthy Male Subjects).

Kategori:
Benzene DerivativesPhenols
Waktu Paruh-
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HY-111996 DB16964
small molecule | CAS: 1380696-64-9

Deskripsi belum tersedia.

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HY10275 DB05079
small molecule

HY10275 is a novel compound specifically designed to modulate two key neurobiological mechanisms that interfere with the sleeping process. HY10275 is highly selective for histamine H1 and serotonin 5HT2a, two chemical receptors that are known to impact the ab…

Target Protein:
Histamine H1 receptor5-hydroxytryptamine receptor 2A
Waktu Paruh-
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Genetik -
small molecule | CAS: 9004-61-9

Hyaluronic acid (non-animal stabilized) is under investigation in clinical trial NCT03460158 (Prospective Evaluation of Facial Cosmetic Procedures).

Kategori:
CarbohydratesGlycosaminoglycansPolysaccharides
Waktu Paruh-
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Hyaluronidase Approved DB14740
biotech | CAS: 9001-54-1

Hyaluronidase is an enzyme used to improve the absorption and dispersion of parenterally administered fluids, drugs, and contrast agents.[L13338] The action of hyaluronidase was first described in 1936, and named in 1939.[A199026] Early research into hyaluron…

Kategori:
Blood and Blood Forming OrgansCarbon-Oxygen LyasesEnzymes +6
Target Protein:
Hyaluronic acidTransforming growth factor beta-1 proprotein
Waktu ParuhHyaluronidase has a…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
biotech | CAS: 757971-58-7

A purified preparation of the enzyme recombinant human hyaluronidase. Hyaluronidase (human recombinant) (INN Vorhyaluronidase alfa) is produced by genetically engineered Chinese Hamster Ovary (CHO) cells containing a DNA plasmid encoding for a soluble fragmen…

Kategori:
Blood and Blood Forming OrgansCarbon-Oxygen LyasesEnzymes +6
Target Protein:
Hyaluronic acidTransforming growth factor beta-1 proprotein
Waktu ParuhHyaluronidase has a…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Hyaluronidase (ovine) Approved DB00070
biotech | CAS: 488712-31-8

Highly purified sheep hyaluronidase for administration by injection into the vitreous of the eye.

Kategori:
EnzymesEnzymes and CoenzymesGlycoside Hydrolases
Target Protein:
Transforming growth factor beta-1 proprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hycanthone DB14061
small molecule | CAS: 3105-97-3

Potentially toxic, but effective antischistosomal agent, it is a metabolite of LUCANTHONE. Hycanthone was approved by the FDA in 1975 but is no longer used.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +7
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenylosuccinate synthetaseAdenylosuccinate synthetase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hydracarbazine DB09243
small molecule | CAS: 3614-47-9

Hydracarbazine is a pyridazine that has found use as an antihypertensive agent [A19790] It was once marketed in France under the tradename Normatensyl.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +3
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Hydralazine Approved DB01275
small molecule | CAS: 86-54-4

Originally developed in the 1950s as a malaria treatment, hydralazine showed antihypertensive ability and was soon repurposed.[A186841] Hydralazine is a hydrazine derivative vasodilator used alone or as adjunct therapy in the treatment of hypertension and onl…

Kategori:
Antihypertensive AgentsAntihypertensive Agents Indicated for HypertensionArteriolar Smooth Muscle, Agents Acting On +15
Target Protein:
Amine oxidase [copper-containing] 3Hypoxia-inducible factor 1-alphaProlyl 4-hydroxylase subunit alpha-1
Waktu ParuhHydralazine has a h…
Vol. DistribusiThe volume of distr…
KlirensThe majority of hyd…
Genetik -
Hydrastine DB19354
small molecule | CAS: 118-08-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingHydrastis +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Hydrastinine DB19359
small molecule | CAS: 6592-85-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIsoquinolines
Waktu Paruh-
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Genetik -
small molecule | CAS: 7647-01-0

Deskripsi belum tersedia.

Kategori:
Acid PreparationsAcidsAcids, Noncarboxylic +7
Waktu Paruh-
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Hydrochlorothiazide Approved DB00999
small molecule | CAS: 58-93-5

Hydrochlorothiazide is the most commonly prescribed thiazide diuretic.[A185138] It is indicated to treat edema and hypertension.[A185138,L8447,L8450] Hydrochlorothiazide use is common but declining in favour of angiotensin converting enzyme inhibitors.[A18513…

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +25
Target Protein:
Solute carrier family 12 member 3Angiotensin-converting enzymeCalcium-activated potassium channel subunit alpha-1
Waktu ParuhThe plasma half lif…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik -
Hydrocodone Approved DB00956
small molecule | CAS: 125-29-1

Hydrocodone is a synthetic opioid derivative of codeine.[T116] It is commonly used in combination with [acetaminophen] to control moderate to severe pain. Historically, hydrocodone has been used as a cough suppressant although this has largely been replaced b…

Kategori:
AlkaloidsAnalgesicsAntitussive Agents +23
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorSigma non-opioid intracellular receptor 1
Waktu ParuhThe half-life of el…
Vol. DistribusiThe apparent volume…
KlirensOfficial FDA labeli…
Genetik -
Hydrocortamate Approved DB00769
small molecule | CAS: 76-47-1

Hydrocortamate is a synthetic glucocorticoid used for its anti-inflammatory or immunosuppressive properties to treat inflammation due to corticosteroid-responsive dermatoses. Glucocorticoids are a class of steroid hormones characterised by an ability to bind …

Kategori:
Cytochrome P-450 CYP3A InducersCytochrome P-450 CYP3A4 InducersCytochrome P-450 CYP3A4 Inducers (strength unknown) +1
Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hydrocortisone Approved DB00741
small molecule | CAS: 50-23-7

Hydrocortisone, or cortisol, is a glucocorticoid secreted by the adrenal cortex.[A188387] Hydrocortisone is used to treat immune, inflammatory, and neoplastic conditions.[L10529,L10532,L10535,L10538,L7772,L7321] It was discovered in the 1930s by Edward Kendal…

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +55
Target Protein:
Glucocorticoid receptorAnnexin A1
Waktu ParuhTotal hydrocortison…
Vol. DistribusiTotal hydrocortison…
KlirensTotal hydrocortison…
Genetik -
small molecule | CAS: 74050-20-7

Deskripsi belum tersedia.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +25
Target Protein:
Annexin A1Glucocorticoid receptor11-beta-hydroxysteroid dehydrogenase type 2 +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Hydrocortisone butyrate Approved DB14540
small molecule | CAS: 13609-67-1

Deskripsi belum tersedia.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdministration, Topical +26
Target Protein:
Annexin A1Glucocorticoid receptor11-beta-hydroxysteroid dehydrogenase type 2 +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Hydrocortisone probutate Approved DB14543
small molecule | CAS: 72590-77-3

Deskripsi belum tersedia.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +26
Target Protein:
Annexin A1Glucocorticoid receptor11-beta-hydroxysteroid dehydrogenase type 2 +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Hydrocortisone succinate Approved DB14545
small molecule | CAS: 2203-97-6

Deskripsi belum tersedia.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +22
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hydrocortisone valerate Approved DB14544
small molecule | CAS: 57524-89-7

Deskripsi belum tersedia.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +23
Target Protein:
Annexin A1Glucocorticoid receptor11-beta-hydroxysteroid dehydrogenase type 2 +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Hydroflumethiazide Approved DB00774
small molecule | CAS: 135-09-1

A thiazide diuretic with actions and uses similar to those of hydrochlorothiazide. (From Martindale, The Extra Pharmacopoeia, 30th ed, p822)

Kategori:
AmidesAntihypertensive AgentsBenzothiadiazines +19
Target Protein:
Solute carrier family 12 member 1Carbonic anhydrase 7Carbonic anhydrase 9 +6
Waktu ParuhIt appears to have …
Vol. Distribusi-
Klirens-
Genetik -
Hydrogen DB15127
small molecule | CAS: 1333-74-0

Hydrogen is under investigation in clinical trial NCT02830854 (Molecular Hydrogen for Cognitive Function and Performance in Elderly).

Kategori:
ElementsGases
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Hydrogen fluoride Approved DB11072
small molecule | CAS: 7664-39-3

Hydrogen fluoride (Hydrofluoric acid) is a weak acid that is a precursor to almost all fluorine compounds, including pharmaceuticals such as [DB00472] (Prozac). It is used as a chemical reagent in several industrial processes such as oil refinery. It is also …

Kategori:
AcidsAcids, NoncarboxylicDental Agents +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Hydrogen iodide DB15778
small molecule | CAS: 10034-85-2

Deskripsi belum tersedia.

Waktu Paruh-
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Hydrogen peroxide Approved DB11091
small molecule | CAS: 7722-84-1

Hydrogen peroxide is the simplest peroxide with a chemical formula H2O2. Hydrogen peroxide is an unstable compound in the presence of a base or catalyst, and is typically stored with a stabilizer in a weakly acidic solution. If heated to its boiling point, it…

Kategori:
Alimentary Tract and MetabolismAnionsAnti-Infective Agents +19
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. DistribusiTarget organs affec…
Klirens-
Genetik -
small molecule | CAS: 97281-48-6

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
biotech | CAS: 8016-70-4

Extracted from the seeds of the soybean (Glycine soja), hydrogenated soybean oil is a major food fat used in the production of margarine, shortening, and salad and cooking oils. According to the FDA, hydrogenated soybean oil is generally recognized as safe (G…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Nephrotoxic agents
Target Protein:
Beta-lactamaseBeta-lactamase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 68607-88-5

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 1236208-20-0

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
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Hydromorphone Approved DB00327
small molecule | CAS: 466-99-9

Hydromorphone is a pure opioid,[A176468] a semi-synthetic hydrogenated ketone derivative of [morphine] that has been available clinically since 1920. Structurally, hydromorphone derived from [morphine] in the modification of the hydroxyl group in the carbon 6…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +22
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhThe half-life of hy…
Vol. DistribusiThe volume of distr…
KlirensThe mean plasma cle…
Genetik -
Hydronidone DB06299
small molecule | CAS: 851518-71-3

Hydronidone has antifibrotic activity.

Kategori:
Pyridines
Waktu Paruh-
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Genetik -
Hydroquinidine DB15300
small molecule | CAS: 1435-55-8

Hydroquinidine is under investigation in clinical trial NCT00927732 (Hydroquinidine Versus Placebo in Patients With Brugada Syndrome).

Kategori:
AlkaloidsAntiarrhythmic agentsAntiarrhythmics, Class I +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hydroquinine DB13718
small molecule | CAS: 522-66-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntiarrhythmic agentsAutonomic Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Collagenase 3Stromelysin-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 821-33-0

Deskripsi belum tersedia.

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Hydroxychloroquine Approved DB01611
small molecule | CAS: 118-42-3

Hydroxychloroquine is a racemic mixture consisting of an R and S enantiomer.[A183047] Hydroxychloroquine is an aminoquinoline like [chloroquine].[L8072] It is a commonly prescribed medication in the treatment of uncomplicated malaria, rheumatoid arthritis, ch…

Kategori:
AminoquinolinesAnti-Infective AgentsAntimalarials +22
Target Protein:
Toll-like receptor 7Toll-like receptor 9DNA +1
Waktu ParuhA half-life of 123.…
Vol. DistribusiHydroxychloroquine …
KlirensThe clearance of hy…
Genetik -
Hydroxycitronellal Approved DB14187
small molecule | CAS: 107-75-5

Hydroxycitronellal is a synthetic fragrance that is widely used in many cosmetics and hygiene products such as deodorants, soaps, antiseptics, and other household items. It has the smell of lilac, lily, and lily of the valley [A34269]. Hydroxycitronellal has …

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleasePerfume +1
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu ParuhThe mean eliminatio…
Vol. DistribusiTmax was found to b…
Klirens-
Genetik -
Hydroxyethyl Starch Approved DB09106
small molecule | CAS: 9005-27-0

Hydroxyethyl starch (HES/HAES) is a nonionic starch derivative. Hydroxyethyl starches (HES) are synthetic colloids commonly used for fluid resuscitation to replace intravascular volume. HES is a general term and can be sub-classified according to average mol…

Kategori:
Blood and Blood Forming OrgansBlood and Related ProductsBlood Substitutes +14
Waktu ParuhTerminal half-life …
Vol. Distribusi5.9 L.
Klirens31.4 mL/min
Genetik -
small molecule | CAS: 7647-63-4

Deskripsi belum tersedia.

Kategori:
Antihistamines for Systemic UsePhenothiazine Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hydroxyfasudil DB04707
small molecule | CAS: 105628-72-6

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIsoquinolinesPiperazines +3
Target Protein:
Chloride channel protein 2Rho-associated protein kinase 1cAMP-dependent protein kinase catalytic subunit alpha +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 68-96-2

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +17
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Hydroxyprogesterone caproate Approved DB06789
small molecule | CAS: 630-56-8

Hydroxyprogesterone caproate is a synthetic steroid hormone that is similar to medroxyprogesterone acetate and megestrol acetate. It is an ester derivative of 17?-hydroxyprogesterone formed from caproic acid (hexanoic acid). Hydroxyprogesterone caproate was p…

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsCombination Contraceptives (with Estrogen and derivatives) +26
Target Protein:
Progesterone receptor
Waktu ParuhHalf-life = 16 days…
Vol. DistribusiHydroxyprogesterone…
KlirensClearance is highly…
Genetik -
Hydroxyproline DB08847
small molecule | CAS: 51-35-4

Hydroxyproline is a neutral heterocyclic protein amino acid. It is found in collagen and as such it is common in many gelatin products. Hydroxyproline is mostly used as a diagnostic marker of bone turnover and liver fibrosis. Therapeutically, hydroxyproline i…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 128446-35-5

Hydroxypropyl betadex is under investigation in clinical trial NCT03471143 (Study of IV VTS-270 for Infantile Liver Disease Associated With Niemann-Pick Disease, Type C).

Kategori:
beta-CyclodextrinsCarbohydratesCompounds used in a research, industrial, or household setting +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5851–5900 dari 11778
Sebelumnya Halaman 118 / 236 Berikutnya