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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 118 / 252
Ganstigmine DB06525
small molecule | CAS: 457075-21-7

Ganstigmine is an orally active, geneserine derived, carbamate-based acetylcholinesterase inhibitor developed for the treatment of Alzheimer's disease.

Kategori:
Acids, AcyclicCarbamates
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gantacurium DB05710
small molecule | CAS: 758669-50-0

Gantacurium chloride is a new, investigational, non-depolarizing ultra-short acting neuromuscular blocker. It is being developed by Avera Pharmaceuticals.

Kategori:
Anticholinergic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Neuronal acetylcholine receptor subunit alpha-3
Waktu Paruh3.09±0.21 minutes
Vol. Distribusi-
Klirens-
Genetik -
Gantenerumab DB12034
biotech | CAS: 1043556-46-2

Alzheimer's disease (AD) is the most common cause of dementia in elderly patients, with classical histopathological hallmarks including extracellular amyloid-beta (A?) plaques and intraneuronal neurofibrillary tangles (NFTs). As the classical view of AD patho…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhGantenerumab admini…
Vol. Distribusi-
Klirens-
Genetik -
Garadacimab DB15629
biotech | CAS: 2162134-62-3

Garadacimab is under investigation in clinical trial NCT04281524 (A Clinical Study to Test the Efficacy and Safety of CSL312 on Catheter-associated Blood Clot Formation in Subjects With Cancer Who Receive Chemotherapy Through a PICC Line).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Garcinia gummi-gutta fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Garenoxacin DB06160
small molecule | CAS: 194804-75-6

Garenoxacin, a quinolone antibiotic, is being investigated for the treatment of gram-positive and gram-negative bacterial infections.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garetosmab DB16379
biotech | CAS: 2097125-54-5

Fibrodysplasia ossificans progressiva (FOP) is a rare autosomal dominant disorder of episodic, progressive heterotropic ossification. FOP is characterized by episodic inflammatory episodes, which may be precipitated by trauma, including immunizations and mino…

Target Protein:
Inhibin beta A chain
Waktu Paruh-
Vol. DistribusiGaretosmab had a st…
KlirensWhen administered a…
Genetik -
Garivulimab DB16670
biotech | CAS: 2342597-81-1

Garivulimab is under investigation in clinical trial NCT03379259 (Study of BGB-A333 Alone and in Combination With Tislelizumab in Advanced Solid Tumors).

Waktu Paruh-
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Garlic Approved DB10532
biotech | CAS: 8008-99-9

Garlic allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityHerbs and Natural ProductsIncreased Histamine Release +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garlic oil DB15989
biotech | CAS: 8000-78-0

Deskripsi belum tersedia.

Kategori:
AlkenesAnionsAnticarcinogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gartisertib DB18770
small molecule | CAS: 1613191-99-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 100040-31-1

Gastric inhibitory polypeptide is under investigation in clinical trial NCT03081676 (The Effect of GIP and GLP-1 on Insulin and Glucagon Secretion in Patients With HNF1A-diabetes Treated With or Without Sulphonylurea).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsGastrointestinal Agents +9
Waktu Paruh-
Vol. Distribusi-
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Gatifloxacin Approved DB01044
small molecule | CAS: 112811-59-3

Gatifloxacin is an antibiotic agent and a member of the fourth-generation fluoroquinolone family. It works by inhibiting the bacterial enzymes DNA gyrase and topoisomerase IV. It was first introduced by Bristol-Myers Squibb in 1999 under the brand name Tequin…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh7-14 hours
Vol. Distribusi-
Klirens-
Genetik -
Gatipotuzumab DB18861
biotech | CAS: 1264737-26-9

Gatipotuzumab is under investigation in clinical trial NCT01899599 (Pankomab-gex™ Versus Placebo as Maintenance Therapy in Advanced Ovarian Cancer).

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Gatralimab DB16528
biotech | CAS: 1826020-80-7

Gatralimab is under investigation in clinical trial NCT02389452 (Study of Safety and Efficacy of 6 Ml Synvisc-one (Hylan G-F 20) in Indian Patients With Symptomatic Osteoarthritis of Knee(s) After Initial and Repeat Treatment).

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Gavestinel DB06741
small molecule | CAS: 153436-22-7

Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Gavestinel displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites and is o…

Kategori:
Excitatory Amino Acid AgentsExcitatory Amino Acid AntagonistsGlycine Agents +5
Target Protein:
Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2Glycine receptor subunit alpha-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gavilimomab DB06545
biotech | CAS: 244096-20-6

Deskripsi belum tersedia.

Waktu Paruh-
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Gavorestat DB16707
small molecule | CAS: 2170729-29-8

Gavorestat is under investigation in clinical trial NCT04902781 (Clinical Benefit, Safety, PK and PD Study of AT-007 in Pediatric Subjects With Classic Galactosemia).

Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GB-115 DB19204
small molecule | CAS: 678996-63-9

GB-115 is under investigation in clinical trial NCT05586789 (A Study of the Efficacy and Safety of Ranquilon Tablets in Patients With Anxiety in Neurasthenia and Adjustment Disorders).

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
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GB1211 DB17499
small molecule | CAS: 1978336-95-6

GB1211 is an orally active galectin-3 (Gal-3) inhibitor.

Waktu Paruh-
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GBR-12783 DB17027
small molecule | CAS: 145428-33-7

A selective inhibitor of dopamine uptake.[A252997]

Kategori:
Dopamine AgentsDopamine AgonistsDopamine Uptake Inhibitors +3
Waktu Paruh-
Vol. Distribusi-
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GC-373 DB15797
small molecule

GC-373 is a peptide aldehyde which is metabolized from the bisulfide adduct, [GC-376 free acid][A219031,A219036]. It is an inhibitor of M<sup>pro</sup> (otherwise known as 3CL<sup>pro</sup>), a viral encoded protease that cleaves and activates functional prot…

Kategori:
AmidesAmino AcidsAmino Acids, Branched-Chain +3
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1417031-79-8

GC-376 is a 3C-like protease (3CL<sup>pro</sup> or M<sup>pro</sup>) inhibitor that stops the cleavage and activation of functional viral proteins required for replication and transcription in host cells[A219036]. The compound is known as a direct acting antiv…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +15
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GC5107 DB17604
biotech

GC5107 is an investigational intravenous immunoglobulin. It is marketed as IVIG-SN.

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GCS-100 DB17566
biotech

Deskripsi belum tersedia.

Kategori:
Carbohydrates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0134 DB17079
small molecule | CAS: 1637394-01-4

Deskripsi belum tersedia.

Waktu Paruh-
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GDC-0152 DB12380
small molecule | CAS: 873652-48-3

GDC-0152 has been used in trials studying the treatment of Solid Cancers.

Kategori:
Cycloparaffins
Target Protein:
E3 ubiquitin-protein ligase XIAP
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0425 DB14791
small molecule | CAS: 1627539-18-7

GDC-0425 is under investigation in clinical trial NCT01359696 (A Study Evaluating the Safety, Tolerability, and Pharmacokinetics of GDC-0425 Administered With and Without Gemcitabine in Patients With Refractory Solid Tumors or Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
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GDC-0810 DB12253
small molecule | CAS: 1365888-06-7

ARN-810 has been used in trials studying the basic science and treatment of Breast Cancer.

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0927 DB14934
small molecule | CAS: 2100830-77-9

GDC-0927 is under investigation in clinical trial NCT02316509 (A Study of GDC-0927 in Postmenopausal Women With Locally Advanced or Metastatic Estrogen Receptor Positive Breast Cancer).

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GDC-1971 DB17487
small molecule | CAS: 2377352-49-1

Deskripsi belum tersedia.

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Vol. Distribusi-
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GDP-L-fucose DB18689
small molecule | CAS: 15839-70-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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GE-2270A DB02975
small molecule | CAS: 134861-34-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +2
Target Protein:
Elongation factor Tu
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 921195-93-9

GED-0507-34-Levo is under investigation in clinical trial NCT02808390 (Efficacy and Safety Study of Ged-0507-34-levo for Treatment of UC).

Kategori:
Acids, CarbocyclicAmines
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gedivumab DB15277
biotech | CAS: 1807954-17-1

Gedivumab is under investigation in clinical trial NCT01877785 (A Study of MHAA4549A to Assess Safety And Pharmacokinetics in Healthy Volunteers).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Gedocarnil DB13534
small molecule | CAS: 109623-97-4

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsHypnotics (Nonbenzodiazepine) +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gefapixant Approved DB15097
small molecule | CAS: 1015787-98-0

It has been estimated that 5-10% of adults globally suffer from chronic cough, which is defined as a cough lasting longer than eight weeks.[L48601] A subset of these patients remain symptomatic despite thorough investigation and treatment, termed refractory c…

Kategori:
AmidesBCRP/ABCG2 SubstratesBenzene Derivatives +8
Target Protein:
P2X purinoceptor 3P2X purinoceptor 2
Waktu ParuhThe terminal half-l…
Vol. DistribusiBased on population…
KlirensPopulation pharmaco…
Genetik -
Gefarnate DB12079
small molecule | CAS: 51-77-4

Gefarnate has been investigated for the treatment and prevention of Stomach Ulcer, Duodenal Ulcer, and Cardio-cerebrovascular Disease.

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsDrugs for Acid Related Disorders +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Gefitinib Approved DB00317
small molecule | CAS: 184475-35-2

Gefitinib (originally coded ZD1839) is a drug used in the treatment of certain types of cancer. Acting in a similar manner to erlotinib (marketed as Tarceva), gefitinib selectively targets the mutant proteins in malignant cells. It is marketed by AstraZeneca …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +25
Target Protein:
Epidermal growth factor receptor
Gen Terkait:
EGFR EGFR EGFR +1
Waktu Paruh48 hours [IV admini…
Vol. Distribusi* 1400 L [IV admini…
Klirens* 595 mL/min [IV ad…
Genetik 4 Varian
Gefurulimab DB18928
biotech | CAS: 2456407-94-4

Gefurulimab is under investigation in clinical trial NCT05556096 (Safety and Efficacy of ALXN1720 in Adults With Generalized Myasthenia Gravis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Geldanamycin DB02424
small molecule | CAS: 30562-34-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Infective AgentsAntibiotics, Antineoplastic +7
Target Protein:
Heat shock protein HSP 90-alphaEndoplasminHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GEM-231 DB05798
biotech | CAS: 255810-66-3

GEM231 is a second-generation antisense oligonucleotide targeting the mRNA of the R1alpha regulatory subunit of cAMP dependent protein kinase. A monoclonal antibody combined with a toxic substance that is used treat certain types of acute myeloid leukemia in …

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
cAMP-dependent protein kinase type II-alpha regulatory subunitcAMP-dependent protein kinase type I-alpha regulatory subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemcabene DB05123
small molecule | CAS: 183293-82-5

Gemcabene is a new drug that lowers low-density lipoprotein cholesterol (LDL-C), decreases triglycerides, and raises high-density lipoprotein cholesterol (HDL-C).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemcitabine Approved DB00441
small molecule | CAS: 95058-81-4

Gemcitabine is a nucleoside analog and a chemotherapeutic agent. It was originally investigated for its antiviral effects, but it is now used as an anticancer therapy for various cancers.[A233135] Gemcitabine is a cytidine analog with two fluorine atoms repla…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +23
Target Protein:
DNARibonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit +2
Gen Terkait:
RRM1
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn patients with va…
KlirensFollowing intraveno…
Genetik 1 Varian
small molecule | CAS: 210829-30-4

Gemcitabine elaidate has been used in trials studying the treatment of Solid Tumor, Lung Cancer, Non-small-cell Lung Cancer, and Metastatic Pancreatic Adenocarcinoma.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemfibrozil Approved DB01241
small molecule | CAS: 25812-30-0

Gemfibrozil is a fibric acid agent, similar to [clofibrate], used to treat Type IIb, IV, and V hyperlipidemias.[A185777,L8525] Gemfibrozil is not a first line treatment and is prescribed to patients who have not responded adequately to weight loss, diet, exer…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +53
Target Protein:
Peroxisome proliferator-activated receptor alphaLipoprotein lipaseSolute carrier organic anion transporter family member 1B1 +3
Waktu ParuhGemfibrozil has a p…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ge…
Genetik -
Gemifloxacin Approved DB01155
small molecule | CAS: 175463-14-6

Gemifloxacin is a quinolone antibacterial agent with a broad-spectrum activity that is used in the treatment of acute bacterial exacerbation of chronic bronchitis and mild-to-moderate pneumonia. It is available in oral formulations. Gemifloxacin acts by inhib…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu Paruh7 (&plusmn; 2) hours
Vol. Distribusi* 1.66 to 12.12 L/kg
Klirens* renal cl=11.6+/- …
Genetik -
biotech

Gemogenovatucel-T is a bi-shRNA furin/Granulocyte Macrophage Colony Stimulating Factor (GMCSF) Augmented autologous tumour cell vaccine. Furin is a convertase involved in the activation of TGF?-1 and TGF?-2.[A255163] Gemogenovatucel-T is being investigated in…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemtuzumab ozogamicin Approved DB00056
biotech | CAS: 220578-59-6

Gemtuzumab ozogamicin is a recombinant humanized IgG4 kappa antibody which is conjugated with calicheamicin derivative, a cytotoxic antitumor antibiotic isolated from fermentation of Micromonospora echinospora ssp. calichensis. Gemtuzumab ozogamicin has appro…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +28
Target Protein:
Myeloid cell surface antigen CD33Low affinity immunoglobulin gamma Fc region receptor III-BLow affinity immunoglobulin gamma Fc region receptor III-A +1
Waktu ParuhIn pediatric patien…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
GEN-001 DB17518
biotech

Deskripsi belum tersedia.

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Menampilkan 5851–5900 dari 12560
Sebelumnya Halaman 118 / 252 Berikutnya