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6694

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4518 (67.5%)
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3751 (56.0%)
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81 (1.2%)
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Halaman 116 / 134
Solrikitug DB19301
biotech | CAS: 2768721-24-8

Solrikitug is under investigation in clinical trial NCT06496607 (A Study to Evaluate Solriktug in Adult Participants With Asthma).

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Somapacitan Approved DB15093
biotech | CAS: 1338578-34-9

Somapacitan, also known as NNC0195-0092,[A219136] is a growth hormone analog indicated to treat adults with growth hormone deficiency.[A219126,L15661] This human growth hormone analog differs by the creation of an albumin binding site, and prolonging the effe…

Kategori:
AlcoholsAmino AcidsAmino Acids, Cyclic +25
Target Protein:
Growth hormone receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe approximate vol…
KlirensThe apparent maximu…
Genetik -
Somatorelin DB12656
biotech | CAS: 83930-13-6

Somatorelin has been used in trials studying the treatment of Aging, Elderly, Sleep Disorders, Hormone Deficiency, and Mild Cognitive Impairment.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGrowth Hormone-Releasing Hormone, agonists +10
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Somatostatin Approved DB09099
small molecule | CAS: 38916-34-6

Somatostatin, also known as growth hormone-inhibiting hormone, is a naturally-occurring peptide hormone of 14 or 28 amino acid residues [T28] that regulates the endocrine system. It is secreted by the D cells of the islets to inhibit the release of insulin an…

Kategori:
Amino Acids, Peptides, and ProteinsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +17
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorSomatostatin receptor type 1 +4
Waktu ParuhThe half-life of en…
Vol. DistribusiThis pharmacokineti…
KlirensFollowing intraveno…
Genetik -
Somatotropin Approved DB00052
biotech | CAS: 12629-01-5

Human growth hormone (HGH), also known as somatotropin, is a peptide hormone that is synthesized and secreted by the somatotropic cells of the anterior pituitary gland.[A228183] Growth hormone plays an essential role in growth regulation during childhood as w…

Kategori:
Agents Causing Muscle ToxicityAmino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and Analogues +23
Target Protein:
Growth hormone receptorProlactin receptor
Waktu ParuhWhen somatotropin w…
Vol. DistribusiInformation is unav…
KlirensFollowing intraveno…
Genetik -
Somatrem Approved DB09098
biotech | CAS: 82030-87-3

Despite the ability of almost all contemporary recombinant growth hormones to cause definite and demonstrable increases in growth rate in patients who are administered the drug, the use of these agents continues to be mired in persistent bioethical debate [A3…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesGrowth Hormone +9
Target Protein:
Growth hormone receptorInsulin-like growth factor 1 receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiAnimal studies with…
KlirensThe clearance of so…
Genetik -
Somatrogon Approved DB14960
biotech | CAS: 1663481-09-1

Somatrogon is a long-acting recombinant human growth hormone. Growth hormone is a peptide hormone secreted by the pituitary gland that plays a crucial role in promoting longitudinal growth during childhood and adolescence and regulating metabolic function in …

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesGrowth Hormone +10
Target Protein:
Growth hormone receptor
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing subcutane…
KlirensFollowing subcutane…
Genetik -
biotech | CAS: 1088845-67-3

Somatropin pegol is under investigation in clinical trial NCT00715689 (Dose Study in Growth Hormone Deficient Adults Investigating Safety, Pharmacokinetics and Pharmacodynamics of NNC126-0083).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsEthylene Glycols +10
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Somavaratan DB12421
biotech | CAS: 1448335-08-7

Somavaratan has been used in trials studying the treatment of Growth Disorders and Adult Growth Hormone Deficiency.

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Sonelokimab DB18843
biotech | CAS: 1414386-05-2

Sonelokimab is under investigation in clinical trial NCT06411379 (Study to Evaluate the Efficacy and Safety of Subcutaneous Sonelokimab Compared With Placebo in Adult Participants With Moderate to Severe Hidradenitis Suppurativa).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +9
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Sonepcizumab DB06305
biotech | CAS: 1031360-18-5

A humanized monoclonal antibody directed against sphingosine 1-phosphate (S1P) with potential antiangiogenic and antineoplastic activities. Upon administration, sonepcizumab binds S1P, which may result in the inhibition of tumor angiogenesis. S1P is the extra…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Sonidegib Approved DB09143
small molecule | CAS: 956697-53-3

Sonidegib is a Hedgehog signaling pathway inhibitor (via smoothened antagonism) developed as an anticancer agent by Novartis. It was FDA approved in 2015 for the treatment of basal cell carcinoma.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBenzene Derivatives +8
Target Protein:
Protein smoothened
Waktu ParuhHalf-life ~ 28 days…
Vol. DistribusiEstimated volume of…
Klirens-
Genetik -
biotech

Sonpiretigene isteparvovec is an ambient-light activatable Multi-Characteristic Opsin (MCO) optogenetic therapy. Developed by Nanoscope Therapeutics, it is being investigated for vision restoration in advanced retinitis pigmentosa (RP).[L46676] Sonpiretigene …

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Sorafenib Approved DB00398
small molecule | CAS: 284461-73-0

Sorafenib is a bi-aryl urea and an oral multikinase inhibitor. It targets cell surface tyrosine kinase receptors and downstream intracellular kinases that are implicated in tumour cell proliferation and tumour angiogenesis.[A255852] First approved by the FDA …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +51
Target Protein:
Serine/threonine-protein kinase B-rafEpidermal growth factor receptorRAF proto-oncogene serine/threonine-protein kinase +8
Waktu ParuhThe mean eliminatio…
Vol. DistribusiSorafenib is widely…
Klirens-
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Sorbitol Approved DB01638
small molecule | CAS: 50-70-4

A polyhydric alcohol with about half the sweetness of sucrose. Sorbitol occurs naturally and is also produced synthetically from glucose. It was formerly used as a diuretic and may still be used as a laxative and in irrigating solutions for some surgical proc…

Kategori:
AlcoholsAlimentary Tract and MetabolismBlood and Blood Forming Organs +22
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Sotagliflozin Approved DB12713
small molecule | CAS: 1018899-04-1

Sotagliflozin is a dual inhibitor of SGLT1 and SGLT2, the first of its kind,[A244499] which is approved for use in the EU, in combination with insulin, to improve glycemic control in patients with type 1 diabetes mellitus (T1DM) and a BMI ?27 kg/m<sup>2</sup>…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 InhibitorsBlood Glucose Lowering Agents +24
Target Protein:
Sodium/glucose cotransporter 2Sodium/glucose cotransporter 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiSotagliflozin has a…
KlirensIn healthy voluntee…
Genetik -
Sotigalimab DB16413
biotech | CAS: 2305607-45-6

Sotigalimab is under investigation in clinical trial NCT03123783 (CD40 Agonistic Antibody APX005M in Combination With Nivolumab).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Sotrastaurin DB12369
small molecule | CAS: 425637-18-9

Sotrastaurin has been used in trials studying the basic science and treatment of Uveal Melanoma, Richter Syndrome, Prolymphocytic Leukemia, Recurrent Mantle Cell Lymphoma, and Recurrent Small Lymphocytic Lymphoma, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein kinase C theta typeProtein kinase C beta typeProtein kinase C alpha type
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Sovesudil DB18812
small molecule | CAS: 1333400-14-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene Derivatives
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Sovleplenib DB17557
small molecule | CAS: 1415792-84-5

Sovleplenib is a novel, investigational, selective small molecule inhibitor for oral administration targeting spleen tyrosine kinase (Syk). It is under investigation in clinical trial NCT03483948 (Phase I Study of Hmpl-523+azacitidine in Elderly Patients With…

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Soy sterol DB11325
biotech | CAS: 129311-52-0

Deskripsi belum tersedia.

Kategori:
Biological FactorsCholestanesFused-Ring Compounds +5
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Soybean oil Approved DB09422
biotech | CAS: 8001-22-7

Derived from soybeans, soybean oil is a common vegetable oil and a source of polyunsaturated and saturated fatty acids. It is a complex mixture of triglycerides where per 100 g, soybean oil has 16 g of saturated fat, 23 g of monounsaturated fat, and 58 g of p…

Kategori:
Biological ProductsCaloric AgentsComplex Mixtures +12
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. DistribusiAfter triglycerides…
KlirensThe elimination rat…
Genetik -
SP1049C DB04978
small molecule

SP1049C is a novel anthracycline chemotherapeutic agent containing [doxorubicin] and two nonionic pluronic block copolymers.[A260416] It is designed to overcome drug resistance in a number of cancers. It has successfully completed Phase 1 trials. Phase 2 resu…

Kategori:
AlcoholsAnthracyclinesCarbohydrates +8
Target Protein:
DNA topoisomerase 2-alpha
Waktu Paruh-
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Spaglumic acid DB08835
small molecule | CAS: 4910-46-7

Spaglumic acid is the ?-aspartyl isoform of N-Acetyl-l-aspartylglutamate (isospaglumic Acid is N-(N-Acetyl-l-?-aspartyl)-l-glutamic acid). In eye drops, spaglumic acid is either a magnesium or sodium salt of N-Acetyl-l-aspartylglutamate. Spaglumic acid is a m…

Kategori:
Antiallergic Agents, Excl. CorticosteroidsDecongestants and AntiallergicsMast Cell Stabilizers +3
Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi-
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Sparfloxacin Approved DB01208
small molecule | CAS: 110871-86-8

Sparfloxacin is a fluoroquinolone antibiotic indicated for bacterial infections. Sparfloxacin exerts its antibacterial activity by inhibiting DNA gyrase, a bacterial topoisomerase. DNA gyrase is an essential enzyme which controls DNA topology and assists in D…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu ParuhMean terminal elimi…
Vol. Distribusi-
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Sparfosic acid DB03459
small molecule | CAS: 51321-79-0

Sparfosic acid is a solid. This compound belongs to the n-acyl-alpha amino acids. These are compounds containing an alpha amino acid which bears an acyl group at the terminal nitrogen atom. This substance is known to target aspartate carbamoyltransferase cata…

Kategori:
AcetatesAcids, AcyclicAmino Acids +12
Target Protein:
Aspartate carbamoyltransferase catalytic chainMultifunctional protein CAD
Waktu Paruh-
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Sparsentan Approved DB12548
small molecule | CAS: 254740-64-2

Sparsentan is a dual antagonist of the endothelin type A receptor (ET<sub>A</sub>R) and the angiotensin II (Ang II) type 1 receptor (AT<sub>1</sub>R) with a similar affinity for both (9.3 nM for ET<sub>A</sub>R and 0.8 nM for AT<sub>1</sub>R).[A257330,L45300]…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAmidesAngiotensin 2 Receptor Blocker +30
Target Protein:
Endothelin-1 receptorType-1 angiotensin II receptorType-2 angiotensin II receptor
Waktu ParuhSparsentan has an e…
Vol. DistribusiAt the approved rec…
KlirensSparsentan has a ti…
Genetik -
Sparsomycin DB04222
small molecule | CAS: 1404-64-4

An antitumor antibiotic produced by Streptomyces sparsogenes. It inhibits protein synthesis in 70S and 80S ribosomal systems. [PubChem]

Kategori:
Antibiotics, AntineoplasticAntineoplastic AgentsEnzyme Inhibitors +3
Waktu Paruh-
Vol. Distribusi-
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Spartalizumab DB14892
biotech | CAS: 1935694-88-4

Spartalizumab is under investigation in clinical trial NCT02605967 (Safety and Efficacy Study of PDR001 in Patients With Recurrent or Metastatic Nasopharyngeal Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
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Sparteine DB06727
small molecule | CAS: 90-39-1

Sparteine is a plant alkaloid derived from _Cytisus scoparius_ and _Lupinus mutabilis_ which may chelate calcium and magnesium. It is a sodium channel blocker, so it falls in the category of class 1a antiarrhythmic agents. Sparteine is not currently FDA-appro…

Kategori:
AlkaloidsAntiarrhythmic agentsAntiarrhythmics, Class I +13
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SPC2968 DB06351
biotech

SPC2968 is a synthetic antisense oligodeoxynucleotide targeting hypoxia-inducible factor-1alpha (HIF-1alpha). It was under investigation in clinical trial NCT02564614 (A Study of Hypoxia-inducible Factor 1a (HIF1A) Messenger Ribonucleic Acid (mRNA) Antagonist…

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Spectinomycin Approved DB00919
small molecule | CAS: 1695-77-8

An antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +5
Target Protein:
30S ribosomal protein S12
Waktu Paruh1 to 3 hours in pat…
Vol. Distribusi-
Klirens-
Genetik -
Spermidine DB03566
small molecule | CAS: 124-20-9

Spermidine is a polyamine formed from putrescine. It is found in almost all tissues in association with nucleic acids. It is found as a cation at all pH values, and is thought to help stabilize some membranes and nucleic acid structures. It is a precursor of …

Kategori:
AminesBiogenic AminesBiogenic Polyamines +2
Target Protein:
Thioredoxin reductase 1, cytoplasmicBeta-1 adrenergic receptorBeta-2 adrenergic receptor +2
Waktu Paruh-
Vol. Distribusi-
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Spermine DB00127
small molecule | CAS: 71-44-3

Spermine is a spermidine-derived biogenic polyamine found as a polycation at all pH values. Found in various tissues and organisms, it often acts as an essential growth factor in some bacterial species. Spermine is associated with nucleic acids, particularly …

Kategori:
AminesBiogenic AminesBiogenic Polyamines +4
Target Protein:
Spermine synthaseCarbonic anhydrase 4Glutamate receptor ionotropic, NMDA 1 +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Spesolimab Approved DB15626
biotech | CAS: 2097104-58-8

Spesolimab is an interleukin-36 (IL-36) receptor antagonist. It is a humanized monoclonal immunoglobulin G1 antibody that was produced in Chinese hamster ovary (CHO) cells by recombinant DNA technology. The biosimilar of the drug, spesolimab-sbzo, was first a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-1 receptor-like 2
Waktu ParuhThe terminal half-l…
Vol. DistribusiBased on the popula…
KlirensIn the linear dose …
Genetik -
SPH-3127 DB19108
small molecule | CAS: 1399849-02-5

SPH-3127 is under investigation in clinical trial NCT05359068 (Study to Evaluate the Efficacy and Safety of SPH3127 in Patients With Mild-moderate Essential Hypertension).

Kategori:
Oxazines
Waktu Paruh-
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Spinosad Approved DB08823
small molecule | CAS: 168316-95-8

Spinosad is a pediculicide mixture of spinosyn A and spinosyn D (in an approximately 5:1 ratio, respectively) used in the topical treatment of head lice in children (four years old and older) and in adults. Spinosad is an insecticide based on a compound found…

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +6
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. DistribusiNo distribution if …
Klirens-
Genetik -
Spiradoline DB12704
small molecule | CAS: 87151-85-7

Spiradoline has been investigated for the basic science of Bipolar Depression.

Kategori:
AnalgesicsAntiarrhythmic agentsCardiovascular Agents +6
Target Protein:
Kappa-type opioid receptor
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Spiramycin Approved DB06145
small molecule | CAS: 24916-50-5

Spiramycin is a primarily bacteriostatic macrolide antimicrobial agent with activity against Gram-positive cocci and rods, Gram-negative cocci and also Legionellae, mycoplasmas, chlamydiae, some types of spirochetes, Toxoplasma gondii and Cryptosporidium. Sp…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +14
Target Protein:
50S ribosomal protein L3
Waktu ParuhIntravenous: Young…
Vol. DistribusiThe tissue distribu…
Klirens80% of the administ…
Genetik -
biotech

Deskripsi belum tersedia.

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SPL23-2 DB17866
biotech

SPL23-2 is an antisense oligonucleotide (ASO) targeting the W1282X nonsense mutation associated with a severe form of cystic fibrosis.[L46767]

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Squalene Approved DB11460
small molecule | CAS: 111-02-4

Squalene is originally obtained from shark liver oil. It is a natural 30-carbon isoprenoid compound and intermediate metabolite in the synthesis of cholesterol. It is not susceptible to lipid peroxidation and provides skin protection. It is ubiquitously distr…

Kategori:
AlkenesHydrocarbons, AcyclicPolyenes +2
Waktu Paruh-
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small molecule | CAS: 2892-62-8

Squaric acid dibutyl ester is under investigation in clinical trial NCT01971385 (Safety and Efficacy of Squaric Acid Dibutyl Ester for the Treatment of Herpes Labialis).

Kategori:
Adjuvants, ImmunologicAllergensAntigens +3
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SR-9009 DB14013
small molecule | CAS: 1379686-30-2

SR-9009 is a REV-ERB agonist. SR-9011 has been demonstrated that it is specifically lethal to cancer cells and oncogene-induced senescent cells, including melanocytic naevi, and has no effect on the viability of normal cells or tissues [A32628].

Kategori:
Sulfur Compounds
Target Protein:
Nuclear receptor subfamily 1 group D member 1Nuclear receptor subfamily 1 group D member 2
Waktu Paruh-
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SR-9011 DB14014
small molecule | CAS: 1379686-29-9

SR-9011 is a REV-ERB agonist. SR-9011 has been demonstrated that it is specifically lethal to cancer cells and oncogene-induced senescent cells, including melanocytic naevi, and has no effect on the viability of normal cells or tissues [A32628].

Kategori:
Sulfur Compounds
Target Protein:
Nuclear receptor subfamily 1 group D member 2Nuclear receptor subfamily 1 group D member 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SRP 299 DB05440
small molecule

SRP 299 is a preparation of killed Mycobacterium vaccae that has been tested in uses related to inhibiting periodontal disease, in treating asthma and in treating eczema, itching and inflammation. Mycobacterium vaccae is a non-pathogenic, saprophytic bacteria…

Kategori:
Biological ProductsComplex MixturesVaccines
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SRP-6004 DB16998
biotech

A recombinant AAVrh74 gene therapy expressing the dysferlin transgene under control of a muscle-specific promoter (rAAVrh74.MHCK7.DYSF.DV).

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SRT-2104 DB12186
small molecule | CAS: 1093403-33-8

SRT2104 has been investigated for the basic science and treatment of Sepsis, PSORIASIS, Atrophy, Muscular, and Diabetes Mellitus, Type 2.

Kategori:
Enzyme ActivatorsHeterocyclic Compounds, Fused-Ring
Target Protein:
NAD-dependent protein deacetylase sirtuin-1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SS1(dsFv)-PE38 DB17579
biotech

SS1(dsFv)-PE38 is a recombinant anti-mesothelin immunotoxin. SS1(dsFv)-PE38 is under investigation in clinical trial NCT01051934 (A Phase I Trial of SS1 (Dsfv) PE38 With Paclitaxel, Carboplatin, and Bevacizumab in Subjects With Unresectable Non-small Cell Lun…

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ST-101 DB12621
biotech | CAS: 887603-94-3

ST-101 is a small peptide antagonist of C/EBP? and T-type calcium channel activator. ST101 has been used in trials studying the treatment of Essential Tremor and Alzheimer's Disease.[A260411]

Kategori:
Indenes
Waktu Paruh-
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