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14063

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8038 (57.2%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 116 / 282
Efavirenz Approved DB00625
small molecule | CAS: 154598-52-4

Efavirenz (brand names Sustiva® and Stocrin®) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) and is used as part of highly active antiretroviral therapy (HAART) for the treatment of a human immunodeficiency virus (HIV) type 1. For HIV infectio…

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiinfectives for Systemic Use +52
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Gen Terkait:
CYP2B6
Waktu Paruh40-55 hours
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Efbemalenograstim alfa Approved DB18704
biotech | CAS: 2200269-79-8

Efbemalenograstim alfa is a long-acting recombinant fusion protein of granulocyte-colony stimulating factor (G-CSF) due to the addition of the Fc portion of human IgG2, allowing for once-per-cycle administration.[L48852,A262167] As endogenous G-CSF mediates t…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsColony-Stimulating Factors +2
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Efepoetin alfa DB19197
biotech | CAS: 1905452-78-9

Efepoetin alfa is under investigation in clinical trial NCT04155125 (A Study of Efepoetin Alfa in Treating Anaemia Associated With Chronic Kidney Diseases Patient).

Waktu Paruh-
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Efgartigimod alfa Approved DB15270
biotech | CAS: 1821402-21-4

Myasthenia gravis (MG) is an autoimmune disorder characterized by significant muscle weakness - particularly in the eye, throat, and extremities - caused by autoantibodies attacking the neuromuscular junction.[A243759] The production of IgG autoantibodies aga…

Kategori:
AntibodiesAntineoplastic and Immunomodulating AgentsGlobulins +6
Target Protein:
IgG receptor FcRn large subunit p51
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Efinaconazole Approved DB09040
small molecule | CAS: 164650-44-6

Efinaconazole is a 14 alpha-demethylase inhibitor indicated in the treatment of fungal infection of the nail, known as onychomycosis. It was approved for use in Canada and the USA in 2014 and is marketed by Valeant Pharmaceuticals North America LLC under the …

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +4
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylase
Waktu Paruh29.9 hours in healt…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2026634-47-7

Efineptakin alfa (also known as NT-I7) is a long-acting human interleukin-7 (IL-7) fusion protein that promotes T-cell development, contributing to the immune response. Compared to endogenous IL-7, NT-I7 is more stable and potent, has a longer half-life, and …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efinopegdutide DB15077
biotech | CAS: 2055640-93-0

Efinopegdutide is under investigation in clinical trial NCT03606057 (A Study to Investigate the Effect of JNJ-64565111 on Cardiac Repolarization (Corrected QT Interval) Compared With Placebo in Healthy Adults: a Thorough ECG Study Employing Placebo, JNJ-64565…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 1635395-27-5

Efizonerimod alfa is under investigation in clinical trial NCT02221960 (A Phase 1 Study to Evaluate MEDI6383 Alone and in Combination With MEDI4736 in Adult Subjects With Select Advanced Solid Tumors).

Waktu Paruh-
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Eflapegrastim Approved DB15001
biotech | CAS: 1384099-30-2

Febrile neutropenia (FN), defined as the co-occurrence of fever (temperature > 38 ?C) and severe neutropenia (ANC < 500 cells/mm<sup>3</sup>), is a potential side effect of myelosuppressive chemotherapy in which the patient develops an infection during a peri…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +20
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhIn patients with br…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ef…
Genetik -
biotech

Eflepedocokin alfa is a recombinant IL-22-Fc fusion protein manufactured in Chinese hamster ovary cells that is composed of 2 human interleukin 22 (IL-22) molecules linked to an immunoglobulin constant region (IgG2-Fc).[A225706, L27661] It is being developed …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eflornithine Approved DB06243
small molecule | CAS: 70052-12-9

Eflornithine is an irreversible ornithine decarboxylase inhibitor originally developed as a treatment for human African trypanosomiasis.[A262829] Further research has also implicated ornithine decarboxylase in other conditions like facial hirsutism and cancer…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAmino AcidsAmino Acids, Basic +15
Target Protein:
Ornithine decarboxylase
Waktu ParuhThe terminal plasma…
Vol. DistribusiEflornithine volume…
KlirensThe clearance (CL/F…
Genetik -
biotech | CAS: 1953227-87-6

Efmarodocokin alfa is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 1644543-31-6

Efmitermant alfa, a locally-acting GDF/activin ligand trap, is under investigation in clinical trial NCT03124459 (Study of ACE-083 in Patients With Charcot-marie-tooth Disease).

Waktu Paruh-
Vol. Distribusi-
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Efmoroctocog alfa Approved DB11607
biotech | CAS: 1270012-79-7

Efmoroctocog alfa is a fully recombinant factor VIII-Fc fusion protein (rFVIIIFc) with an extended half-life compared with conventional factor VIII (FVIII) preparations, including recombinant FVIII (rFVIII) products such as [DB13999][A31551]. It is an antihem…

Kategori:
HemostaticsHuman Antihemophilic Factors
Target Protein:
von Willebrand factor
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Efocipegtrutide DB18194
biotech | CAS: 2513399-19-2

Efocipegtrutide is a long-acting, monomeric peptide triple agonist.

Waktu Paruh-
Vol. Distribusi-
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Efonidipine DB09235
small molecule | CAS: 111011-63-3

Efonidipine is a calcium channel blocker of the _dihydropyridine class_, commercialized by Shionogi & Co. (Japan). Initially, it was marketed in 1995 under the trade name, _Landel_. The drug has been shown to block T-type in addition to L-type calcium channel…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +22
Target Protein:
Voltage gated L-type calcium channelVoltage-dependent calcium channelVoltage-dependent T-type calcium channel +4
Waktu ParuhThe peak plasma con…
Vol. Distribusi-
Klirens-
Genetik -
Efpeglenatide DB15650
biotech | CAS: 1296200-77-5

Efpeglenatide is under investigation in clinical trial NCT03713684 (Efficacy and Safety of Efpeglenatide Versus Placebo in Patients With Type 2 Diabetes Mellitus Inadequately Controlled With Basal Insulin Alone or in Combination With Oral Antidiabetic Drug(s)…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +2
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efprezimod alfa DB16448
biotech

CD24Fc is a biological immunomodulator originally developed to address graft-versus-host disease in stem cell transplantation in leukemia patients.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
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Efruxifermin DB19012
biotech | CAS: 2375240-92-7

Efruxifermin is under investigation in clinical trial NCT06215716 (A Study Evaluating Efruxifermin in Subjects With Non-cirrhotic Nonalcoholic Steatohepatitis (Nash)/metabolic Dysfunction-associated Steatohepatitis (MASH) and Fibrosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1905448-17-0

Eftansomatropin alfa (GX-H9) comprises a recombinant human growth hormone fused to hyFc, a synthetic hybrid Fc fragment.[L48275] It is under investigation for the treatment of growth hormone deficiency.

Kategori:
Amino Acids, Peptides, and ProteinsGrowth HormoneHormones +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1800476-36-1

Eftilagimod alfa is under investigation in clinical trial NCT02614833 (IMP321 (Eftilagimod Alpha) as Adjunctive to a Standard Chemotherapy Paclitaxel Metastatic Breast Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Differentiation +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eftrenonacog alfa Approved DB11608
biotech | CAS: 1270012-74-2

Eftrenonacog alfa is a long-acting recombinant fusion protein used in the treatment of hemophilia B. It is comprised of a single molecule of human factor IX (FIX) covalently linked to the constant region (Fc) domain of human IgG1 via recombinant DNA technolog…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +15
Target Protein:
IgG receptor FcRn large subunit p51
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Efungumab DB16151
biotech | CAS: 762260-74-2

Efungumab is under investigation in clinical trial NCT00217815 (Preliminary Study of Mycograb and Docetaxel in Advanced Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efzofitimod DB16453
biotech

Efzofitimod (ATYR1923) is a fusion protein comprised of the immuno-modulatory domain of histidyl tRNA synthetase fused to the FC region of a human antibody. It is a selective modulator of neuropilin-2 that downregulates the innate and adaptive immune response…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Neuropilin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Egaptivon pegol DB05202
biotech | CAS: 934868-74-3

Egaptivon pegol, formerly known as ARC1779, is a therapeutic aptamer antagonist of the A1 domain of von Willebrand Factor (vWF), the ligand for receptor glycoprotein 1b on platelets. Egaptivon pegol is being investigated for the treatment of thrombotic thromb…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +2
Target Protein:
von Willebrand factorPlatelet glycoprotein Ib alpha chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EGEN-001 DB05953
small molecule

EGEN-001 is a novel non-viral vector consisting of a plasmid DNA encoding the human gene for interleukin 12 (IL-12) and a biocompatible, biodegradable delivery polymer with potential antineoplastic activity.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Egg Approved DB10529
biotech

Egg allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Egg phospholipids Approved DB14233
biotech | CAS: 93685-90-6

Egg phospholipids are primarily a mixture of naturally occurring phospholipids which are isolated from the egg yolk. Egg phospholipids are available as an intravenous fat emulsion indicated as a source of calories for patients requiring parenteral nutrition.

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Genetik -
Egg white Approved DB10528
biotech | CAS: 9006-50-2

Egg white allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EGS21 DB05056
small molecule

EGS21(TM) is a beta-D-glucosylceramide (GC) compound. It is a potential therapeutic for treating immune mediated disorders. GC is a glycolipid that has been shown by Enzo scientists and collaborators to act as an anti-inflammatory agent in animal model sy…

Waktu Paruh-
Vol. Distribusi-
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EGT-201 DB17648
biotech

EGT-201 is an adeno-associated viral vector serotype 9 (AAV9) vector-based gene therapy consisting of the alpha-N-acetyglucosaminidase (NAGLU) transgene. Developed by Esteve Pharmaceuticals, it is being investigated for Sanfilippo syndrome type B.[L45939]

Waktu Paruh-
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EGT-301 DB17649
biotech

EGT-301 is a gene therapy being investigated for Hunter Syndrome. It consists of an adeno-associated viral vector serotype 9 (AAV9) containing the human Iduronate-2-sulfatase (I2S) transgene designed to restore I2S functional deficiency in patients with Hunte…

Waktu Paruh-
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Genetik -
EHP-102 DB16933
small molecule | CAS: 1807652-43-2

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Elacestrant Approved DB06374
small molecule | CAS: 722533-56-4

Elacestrant is a non-steroidal small molecule and an estrogen receptor (ER) antagonist.[A256838,L44918] In January 2023, it was approved by the FDA for the treatment of ER-positive, HER2-negative, ESR1-mutated advanced or metastatic breast cancer.[L44918,L449…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Estrogen receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiElacestrant has an …
KlirensElacestrant has an …
Genetik -
Elacridar DB04881
small molecule | CAS: 143664-11-3

Elacridar (GW120918) is an oral bioenhancer that targets multiple drug resistance in tumors. In many cases, the appearance of multidrug resistance in cancer is due to a change in expression of protein inhibitors. As of August 2007 elacridar was not listed on …

Kategori:
BCRP/ABCG2 InhibitorsBenzocycloheptenesDrug Resistance, Multiple +3
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elacytarabine DB05494
small molecule | CAS: 188181-42-2

Elacytarabine is a fatty acid derivative of [cytarabine], an approved cytotoxic cancer drug. Cytarabine has limitations such as minimal uptake in solid tumours and is only used to treat leukaemia. Elacytarabine is designed to overcome this limitation and has …

Kategori:
ArabinonucleosidesFatty AcidsLipids +4
Target Protein:
Deoxycytidine kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eladocagene exuparvovec Approved DB16780
biotech | CAS: 2098615-91-7

Eladocagene exuparvovec is a recombinant adeno-associated virus-2 (AAV2)-based gene therapy that expresses human aromatic L-amino acid decarboxylase (AADC), and it is used to treat AADC deficiency, a fatal and rare genetic disorder that causes severe disabili…

Kategori:
Adeno-associated Viral Vector TherapiesAlimentary Tract and MetabolismEnzymes +2
Waktu ParuhNot available.
Vol. DistribusiThe biodistribution…
KlirensNot available.
Genetik -
Elafibranor Approved DB05187
small molecule | CAS: 923978-27-2

Elafibranor is a dual peroxisome proliferator-activated receptor (PPAR) ? and ?/? agonist [A263833] that works to inhibit bile acid synthesis.[L50768] On June 10, 2024, elafibranor was granted accelerated approval by the FDA for the treatment of primary bilia…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBCRP/ABCG2 Inhibitors +21
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor gamma
Waktu ParuhFollowing a single …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent t…
Genetik -
Elagolix Approved DB11979
small molecule | CAS: 834153-87-6

Elagolix has been used in trials studying the basic science and treatment of Endometriosis, Folliculogenesis, Uterine Fibroids, Heavy Uterine Bleeding, and Heavy Menstrual Bleeding. As of 24 July 2018, however, the U.S. Food and Drug Administration (FDA) appr…

Kategori:
Anti-Gonadotropin-Releasing HormonesAntigonadotropins and Similar AgentsCytochrome P-450 CYP2C19 Inhibitors +16
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe terminal phase …
Vol. DistribusiThe apparent volume…
KlirensThe oral clearance …
Genetik -
Elaidamide DB03784
small molecule | CAS: 4303-70-2

Deskripsi belum tersedia.

Target Protein:
Phospholipase A2, membrane associated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elamipretide DB11981
small molecule | CAS: 736992-21-5

Elamipretide has been used in trials studying the treatment of Leber's Hereditary Optic Neuropathy.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elapegademase Approved DB14712
biotech | CAS: 1709806-75-6

Elapegademase is a PEGylated recombinant adenosine deaminase. It can be defined molecularly as a genetically modified bovine adenosine deaminase with a modification in cysteine 74 for serine and with about 13 methoxy polyethylene glycol chains bound via carbo…

Kategori:
Adenosine Deaminase InhibitorsAdjuvants, ImmunologicAmino Acids, Peptides, and Proteins +12
Target Protein:
Adenosine
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Elbasvir Approved DB11574
small molecule | CAS: 1370468-36-2

Elbasvir is a direct-acting antiviral medication used as part of combination therapy to treat chronic hepatitis C, an infectious liver disease caused by infection with hepatitis C virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine d…

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +18
Target Protein:
Nonstructural protein 5A
Waktu ParuhThe geometric mean …
Vol. DistribusiElbasvir has an est…
KlirensThe clearance of el…
Genetik -
Elcatonin DB13742
small molecule | CAS: 60731-46-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Parathyroid AgentsBone Density Conservation Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eldecalcitol DB05295
small molecule | CAS: 104121-92-8

Eldecalcitol (ED-71), a vitamin D analog, is a more potent inhibitor of bone resorption than alfacalcidol in an estrogen-deficient rat model of osteoporosis. Eldecalcitol, effectively and safely increased lumbar and hip bone mineral density (BMD) in osteopor…

Kategori:
Bone Density Conservation AgentsFused-Ring CompoundsSecosteroids +4
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elebsiran DB19018
biotech | CAS: 2648009-64-5

Elebsiran is under investigation in clinical trial NCT05461170 (SOLSTICE: Combination Therapy for the Treatment of Chronic Hepatitis D Infection.).

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Eleclazine DB12394
small molecule | CAS: 1443211-72-0

Eleclazine has been used in trials studying the treatment of LQT2 Syndrome, Long QT Syndrome, Ischemic Heart Disease, Ventricular Arrhythmia, and Long QT Syndrome Type 3, among others.

Kategori:
Azepines
Waktu Paruh-
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Elenbecestat DB15391
small molecule | CAS: 1388651-30-6

Elenbecestat is under investigation in clinical trial NCT02956486 (A 24-Month Study to Evaluate the Efficacy and Safety of Elenbecestat (E2609) in Subjects With Early Alzheimer's Disease).

Target Protein:
Beta-secretase 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Elenestinib DB18489
small molecule | CAS: 2505078-08-8

Elenestinib is a selective KIT inhibitor.

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Genetik -
Elesclomol DB05719
small molecule | CAS: 488832-69-5

Elesclomol is a novel, injectable, drug candidate that kills cancer cells by elevating oxidative stress levels beyond a breaking point, triggering programmed cell death. In preclinical models elesclomol showed potent killing of a broad range of cancer cell ty…

Kategori:
AmidesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
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Genetik -
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