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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 115 / 272
Epitestosterone DB07768
small molecule | CAS: 481-30-1

Epitestosterone is the 17-alpha isomer of testosterone, derived from pregnenolone via the delta5-steroid pathway, and via 5-androstene-3-beta,17-alpha-diol. Epitestosterone acts as an antiandrogen in various target tissues. The ratio between testosterone/epit…

Kategori:
AndrostanesAndrostenesAndrostenols +7
Target Protein:
Aldo-keto reductase family 1 member C1Aldo-keto reductase family 1 member C2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epitizide DB13989
small molecule | CAS: 1764-85-8

Epitizide is an agent, commonly found in combination [triamterene], used to produce diuresis.

Kategori:
DiureticsLow-Ceiling Diuretics and Potassium-Sparing AgentsSodium Chloride Symporter Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EpiVacCorona DB16439
biotech

EpiVacCorona Vaccine, developed by the Vektor State Research Center of Virology and Biotechnology in Russia, is based on peptide-antigens that facilitate immunity to the SARS-CoV-2 virus[L30608]. It is currently being tested in Phase I/II clinical trials for …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eplivanserin DB12177
small molecule | CAS: 130579-75-8

Eplivanserin has been used in trials studying the treatment of Sleep, Insomnia, Chronic Pain, Fibromyalgia, and Primary Insomnia, among others.

Kategori:
Antidepressive AgentsBenzene DerivativesCardiovascular Agents +8
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eplontersen Approved DB16199
biotech | CAS: 1637600-16-8

Eplontersen is a transthyretin-directed antisense oligonucleotide with 3 covalently linked e N-acetyl galactosamine residues for hepatic delivery. It was previously investigated as a potential treatment for hereditary transthyretin-mediated amyloidosis.[A2629…

Kategori:
Antisense OligonucleotidesNervous SystemNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Transthyretin mRNA
Waktu ParuhThe terminal elimin…
Vol. DistribusiEplontersen is expe…
KlirensThe clearance was e…
Genetik -
Epoetin beta DB19434
biotech | CAS: 122312-54-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epoetin delta Approved DB11624
biotech | CAS: 261356-80-3

Epoetin Delta is an ingredient in the EMA-withdrawn product Dynepo.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epofolate DB12266
small molecule | CAS: 958646-17-8

Epofolate has been used in trials studying the treatment of Advanced Solid Tumors. Epofolate (BMS-753493) is a folate conjugate of the epothilone analog BMS-748285 that was designed to selectively target folate receptor expressing cancer cells. In Phase I/IIa…

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsCytochrome P-450 CYP3A Inhibitors +9
Target Protein:
Folate receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epomediol DB13802
small molecule | CAS: 1310101-21-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyCholagogues and Choleretics +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epoprostenol Approved DB01240
small molecule | CAS: 35121-78-9

A prostaglandin that is a powerful vasodilator and inhibits platelet aggregation. It is biosynthesized enzymatically from prostaglandin endoperoxides in human vascular tissue. The sodium salt has been also used to treat primary pulmonary hypertension.

Kategori:
AnticoagulantsAntihypertensive AgentsAntiplatelet agents +19
Target Protein:
Prostacyclin synthaseP2Y purinoceptor 12Prostacyclin receptor
Waktu ParuhThe in vitro half-l…
Vol. Distribusi* 357 mL/kg
Klirens-
Genetik -
Epothilone D DB01873
small molecule | CAS: 189453-10-9

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntimitotic AgentsAntineoplastic Agents +9
Target Protein:
Tubulin beta chainTubulin beta-1 chainTubulin beta-4B chain +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epratuzumab DB04958
biotech | CAS: 205923-57-5

Epratuzumab is a humanized monoclonal antibody derived from the murine IG2a monoclonal antibody, LL2 (EPB-2). This agent may subsequently be well matched for use in oncology and the treatment of inflammatory autoimmune disorders, such as lupus.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
B-cell receptor CD22
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprenetapopt DB11684
small molecule | CAS: 5291-32-7

Eprenetapopt has been used in trials studying the treatment of Prostatic Neoplasms, Hematologic Neoplasms, and Platinum Sensitive Recurrent High-grade Serous Ovarian Cancer With Mutated p53.

Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprinomectin DB11405
small molecule | CAS: 123997-26-2

Deskripsi belum tersedia.

Kategori:
AgrochemicalsAnthelminticsAnti-Bacterial Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprodisate DB06405
small molecule | CAS: 21668-77-9

Eprodisate slows the decline of renal function in AA amyloidosis.

Kategori:
AcidsAcids, NoncarboxylicAlkanes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprosartan Approved DB00876
small molecule | CAS: 133040-01-4

Eprosartan is an angiotensin II receptor antagonist used to treat hypertension. It performs 2 actions on the renin angiotensin system. By preventing the binding of angiotensin II to AT1, vascular smooth muscle relaxes and vasodilation occurs. By inhibiting no…

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +13
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhThe terminal elimin…
Vol. Distribusi-
Klirens-
Genetik -
Eprotirome DB05035
small molecule | CAS: 355129-15-6

Eprotirome which is a compound with promising properties for treatment of obesity and dyslipidemia. Eprotirome increases the body’s energy consumption and reduces body weight and markedly reduces blood lipids and blood glucose.

Kategori:
AmidesAminesAniline Compounds
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprozinol DB13395
small molecule | CAS: 32665-36-4

Deskripsi belum tersedia.

Kategori:
Drugs for Obstructive Airway Diseases
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 944130-77-2

Eptacog alfa pegol (activated) has been used in trials studying the prevention and treatment of Haemophilia A, Haemophilia B, Congenital Bleeding Disorder, Haemophilia B With Inhibitors, and Haemophilia A With Inhibitors.

Kategori:
Pegylated agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eptifibatide Approved DB00063
biotech | CAS: 188627-80-7

Synthetic cyclic hexapeptide that binds to platelet receptor glycoprotein and inhibits platelet aggregation. Derived from venom of the Southeastern pygmy rattlesnake (Sistrurus miliarus barbouri), eptifibatide is a cyclic heptapeptide that belongs to the clas…

Kategori:
Amino Acids, Peptides, and ProteinsAntiplatelet agentsBlood and Blood Forming Organs +5
Target Protein:
Integrin beta-3Integrin alpha-IIbVoltage-dependent N-type calcium channel
Waktu ParuhApproximately 2.5 h…
Vol. Distribusi-
Klirens* 55 mL/kg/h [patie…
Genetik -
Eptinezumab Approved DB14040
biotech | CAS: 1644539-04-7

Eptinezumab is a fully-humanized IgG1 antibody manufactured using yeast (_Pichia pastoris_) and developed by Lundbeck Seattle Biopharmaceuticals.[L12318] Eptinezumab has been specifically designed to bind to both alpha and beta forms of the human calcitonin g…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +12
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe central volume …
KlirensThe apparent cleara…
Genetik -
Eptotermin alfa Approved DB11631
biotech | CAS: 129805-33-0

A bone morphogenetic protein that is widely expressed during EMBRYONIC DEVELOPMENT. It is both a potent osteogenic factor and a specific regulator of nephrogenesis. Eptotermin alfa is an ingredient in the EMA-withdrawn product Osigraft.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBone Morphogenetic Proteins +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EQ101 DB17396
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equilenin DB03515
small molecule | CAS: 517-09-9

Equilenin is an estrogenic steroid produced by horses. It has a total of five double bonds in the A- and B-ring. High concentration of equilenin is found in the urine of pregnant mares.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesCytochrome P-450 CYP3A Substrates +12
Target Protein:
Steroid Delta-isomeraseSteroid Delta-isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equilin DB02187
small molecule | CAS: 474-86-2

An estrogenic steroid produced by horses. It has a total of four double bonds in the A- and B-ring. High concentration of equilin is found in the urine of pregnant mares.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesCytochrome P-450 CYP3A Substrates +12
Target Protein:
17-beta-hydroxysteroid dehydrogenase type 1Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Equine Botulinum Neurotoxin A Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype A. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
BoNT/A
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin B Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype B. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type B
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin C Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype C. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type C1
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin D Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype D. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type D
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin E Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype E. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type E
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin F Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype F. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type F
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin G Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype G. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type G
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
Equine collagen DB16613
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equisetum arvense top Approved DB14349
biotech

Equisetum arvense top is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equol DB11674
small molecule | CAS: 531-95-3

Equol has been used in trials studying the treatment of Breast Cancer.

Kategori:
BenzopyransChromonesEstrogens +7
Target Protein:
Estrogen receptor betaSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ER-176 C-11 DB19181
small molecule | CAS: 1623028-18-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eragidomide DB19242
small molecule | CAS: 1860875-51-9

Eragidomide is under investigation in clinical trial NCT04297124 (A Study to Evaluate the Metabolism and Excretion of [14C]-CC-90009 in Healthy Male Subjects).

Kategori:
AcetatesAcids, AcyclicAmides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eravacycline Approved DB12329
small molecule | CAS: 1207283-85-9

Eravacycline, known as _Xerava_ by Tetraphase Pharmaceuticals, is a fully synthetic fluorocycline antibiotic of the tetracycline class with activity against clinically significant gram-negative, gram-positive aerobic, and facultative bacteria. This includes m…

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +6
Target Protein:
30S ribosomal protein S4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe volume of distr…
Klirens17.82 L/min (standa…
Genetik -
Erbumine DB18019
small molecule | CAS: 1919888-06-4

Deskripsi belum tersedia.

Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ERC-1671 DB17431
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erdafitinib Approved DB12147
small molecule | CAS: 1346242-81-6

In early April of 2019, the US FDA approved Janssen Pharmaceutical Companies' brand name Balversa (erdafitinib) as the first-ever fibroblast growth factor receptor (FGFR) kinase inhibitor indicated for patients with locally advanced or metastatic urothelial c…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C9 Substrates +25
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +7
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe mean total appa…
Genetik -
Erdosteine Approved DB05057
small molecule | CAS: 84611-23-4

Erdosteine is a drug that causes a breakdown of mucus, also known as a _mucolytic_ agent. It is a _thiol_ derivative produced for the clinical management of chronic obstructive bronchitis, in addition to infective exacerbations of chronic bronchitis. This dru…

Kategori:
AcetatesAcids, AcyclicCough and Cold Preparations +4
Target Protein:
Chymotrypsin-like elastase family member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erenumab Approved DB14039
biotech | CAS: 1582205-90-0

Erenumab (AMG-334) (INN; trade name Aimovig) is a human monoclonal antibody designed specifically to bind and antagonize the calcitonin gene-related peptide receptor (CGRPR) as a means to prevent migraines. Aimovig, as released and marketed by Novartis and Am…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhErenumab exhibits n…
Vol. DistribusiAfter a single 140 …
KlirensCertain studies sho…
Genetik -
Erfonrilimab DB17446
biotech | CAS: 2367013-69-0

Erfonrilimab is a bispecific monoclonal antibody directed against both the programmed cell death-1 ligand 1 (PD-L1) and cytotoxic T-lymphocyte-associated antigen 4 (CTLA4).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ergocalciferol Approved DB00153
small molecule | CAS: 50-14-6

Ergocalciferol is an inactivated vitamin D analog.[A177526] It is synthesized by some plants in the presence of UVB light.[T577] The production of ergocalciferol was prompted by the identification of dietary deficiency, more specifically vitamin D, as the mai…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCalcium-Regulating Hormones and Agents +11
Target Protein:
Vitamin D3 receptorVoltage-dependent calcium channel
Waktu ParuhErgocalciferol can …
Vol. DistribusiThe amount of circu…
KlirensThere are no formal…
Genetik -
Ergoloid mesylate Approved DB01049
small molecule | CAS: 8067-24-1

Ergoloid Mesylate is an equiproportional preparation of three different ergotamantriones: dihydroergocornine, dihydroergocristine, and dihydroergocryptine.[A32912] All these components are produced by the fungus _Claviceps purpurea_ and are all derivatives of…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +24
Target Protein:
Dopamine receptorAlpha adrenergic receptorBeta adrenergic receptor +1
Waktu ParuhThe reported plasma…
Vol. DistribusiThe volume of distr…
KlirensTo know more about …
Genetik -
Ergometrine Approved DB01253
small molecule | CAS: 60-79-7

An ergot alkaloid with uterine and vascular smooth muscle contractile properties.

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +20
Target Protein:
Alpha-1A adrenergic receptorD(2) dopamine receptor
Waktu Paruht<sub>1/2 &alpha;</…
Vol. Distribusi-
Klirens-
Genetik -
Ergosterol Approved DB04038
small molecule | CAS: 57-87-4

A steroid of interest both because its biosynthesis in FUNGI is a target of ANTIFUNGAL AGENTS, notably AZOLES, and because when it is present in SKIN of animals, ULTRAVIOLET RAYS break a bond to result in ERGOCALCIFEROL.

Kategori:
CholestanesCholestenesDiet, Food, and Nutrition +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ergotamine Approved DB00696
small molecule | CAS: 113-15-5

A vasoconstrictor found in ergot of Central Europe. It is an alpha-1 selective adrenergic agonist and is commonly used in the treatment of migraine disorders.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +39
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 2A +11
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Ergothioneine DB17614
small molecule | CAS: 497-30-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5701–5750 dari 13591
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