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14361

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Halaman 114 / 288
Eculizumab Approved DB01257
biotech | CAS: 219685-50-4

Eculizumab is a monoclonal antibody that targets complement protein C5.[L6919,A2245] Binding to this protein prevents the activation of a complement terminal complex, which is used to treat a number of autoimmune conditions.[L6919,A2245,A2246] Eculizumab w…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Complement C5
Waktu ParuhThe half life of ec…
Vol. DistribusiThe volume of distr…
KlirensPharmacokinetic pro…
Genetik -
Edaravone Approved DB12243
small molecule | CAS: 89-25-8

Edaravone is a free radical scavenger and neuroprotective agent with antioxidant properties.[A254257] It has three tautomers.[A19140] Edaravone works to scavenge reactive oxygen species, which have been implicated in neurological disorders, such as amyotrophi…

Kategori:
AntioxidantsCentral Nervous System AgentsCompounds used in a research, industrial, or household setting +14
Target Protein:
Apoptosis regulator Bcl-2
Waktu ParuhThe mean terminal e…
Vol. DistribusiAfter intravenous a…
KlirensFollowing intraveno…
Genetik -
Edasalonexent DB15010
small molecule | CAS: 1204317-86-1

Edasalonexent is under investigation in clinical trial NCT01511900 (A Multiple Ascending Dose Study of CAT-1004 in Patients With Type 2 Diabetes).

Kategori:
AmidesEicosanoidsFatty Acids +3
Target Protein:
Nuclear factor NF-kappa-B p105 subunitTranscription factor RelBNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edecesertib DB18917
small molecule | CAS: 2408839-73-4

Edecesertib is under investigation in clinical trial NCT05629208 (Study of Edecesertib in Participants With Cutaneous Lupus Erythematosus (CLE)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 62-33-9

Edetate calcium disodium is a metal ion chelator used to reduce blood concentrations and depot stores of lead from the body.[L12774] It is on the World Health Organization Model List of Essential Medicines.[A204173] Edetate calcium disodium was granted FDA…

Kategori:
AcetatesAcids, AcyclicAmines +26
Target Protein:
LeadIronManganese cation
Waktu ParuhThe half life of ed…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 14025-15-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edetate disodium anhydrous Approved DB14600
small molecule | CAS: 139-33-3

Edetate disodium anhydrous is a polyvalent chelating agent used to treat hypercalcemia and digitalis toxicity associated ventricular arrhythmias.[A204275]

Kategori:
Calcium BinderCalcium Chelating ActivityCalcium Chelating Agents +8
Target Protein:
LeadIronManganese cation
Waktu Paruh-
Vol. DistribusiData regarding the …
KlirensThe mean clearance …
Genetik -
Edetic acid Approved DB00974
small molecule | CAS: 60-00-4

A chelating agent (chelating agents) that sequesters a variety of polyvalent cations. It is used in pharmaceutical manufacturing and as a food additive.

Kategori:
AcetatesAcids, AcyclicAmines +19
Target Protein:
LeadIronManganese cation
Waktu ParuhThe half life of ed…
Vol. Distribusi-
Klirens-
Genetik -
EDI-200 DB18188
biotech

EDI-200 is a fusion protein consisting of human immunoglobim G1 constant region Fc region fused to the human receptor binding domain of ectodysplasin-A1.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Proteins +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EDIT-101 DB18687
biotech

EDIT-101 is a recombinant adeno-associated virus pseudotyped with serotype 5 viral capsid encoding CRISPR/Cas9 (clustered regularly interspaced short palindromic repeats associated protein 9) gene editing constructs.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EDIT-301 DB18645
biotech

EDIT-301 is an investigational cell therapy consisting of autologous CD34+ hematopoietic stem and progenitor cells edited by CRISPR/CAS12a at the gamma globin gene (HBG1 and HBG2).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edivoxetine DB09184
small molecule | CAS: 1194508-25-2

Edivoxetine is a drug which acts as a selective norepinephrine reuptake inhibitor and is currently under development by Eli Lilly for attention-deficit hyperactivity disorder (ADHD) and as an antidepressant treatment. Edivoxetine failed to be approved for maj…

Kategori:
Adrenergic Uptake InhibitorsAlcoholsAntidepressive Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edobacomab DB17779
biotech | CAS: 141410-98-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edodekin alfa DB15631
biotech | CAS: 187348-17-0

Edodekin alfa is under investigation in clinical trial NCT01468896 (Cetuximab and Recombinant Interleukin-12 in Treating Patients With Squamous Cell Carcinoma of the Head and Neck That Is Recurrent, Metastatic, or Cannot Be Removed by Surgery).

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAngiogenesis Inhibitors +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edonerpic DB05938
small molecule | CAS: 519187-23-6

Edonerpic is a neurotrophic agent intended for the treatment of Alzheimer's disease which is under phase I clinical trial.

Kategori:
Acids, AcyclicDicarboxylic AcidsSulfur Compounds
Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edotecarin DB04882
small molecule | CAS: 174402-32-5

Edotecarin is a novel, non-camptothecin, DNA topoisomerase I inhibitor. It is member of the class of compounds called indolocarbazoles.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Target Protein:
DNA topoisomerase 1
Waktu Paruh20 to 25 hours
Vol. Distribusi-
Klirens-
Genetik -
Edotreotide DB17969
small molecule | CAS: 204318-14-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edotreotide gallium Ga-68 Approved DB15494
small molecule | CAS: 2101630-92-4

Edotreotide gallium Ga-68 is an 8 amino acid peptide bound to the chelator 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid (DOTA).[L8603] Edotreotide gallium Ga-68 is indicated for localizing somatostatin receptor positive neuroendocrine tumors by po…

Kategori:
Diagnostic RadiopharmaceuticalsGallium RadioisotopesRadiopharmaceuticals +1
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 5Somatostatin receptor type 3 +1
Waktu ParuhEdotreotide gallium…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
small molecule | CAS: 322407-70-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edoxaban Approved DB09075
small molecule | CAS: 480449-70-5

Edoxaban is a member of the Novel Oral Anti-Coagulants (NOACs) class of drugs, and is a rapidly acting, oral, selective factor Xa inhibitor. By inhibiting factor Xa, a key protein in the coagulation cascade, edoxaban prevents the stepwise amplification of pro…

Kategori:
AnticoagulantsAntithrombinsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor X
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe steady state vo…
Klirens22 L/hr
Genetik -
Edoxudine Approved DB13421
small molecule | CAS: 15176-29-1

Edoxudine is a deoxythymidine analog with activity against herpes simplex virus. It is a potent and selective inhibitor of herpes simplex virus type 1 and 2. The obtained product is an antiviral ointment.[L2407] The activity of edoxudine against herpes simple…

Kategori:
Anti-Infective AgentsAntiviral AgentsDeoxyribonucleosides +5
Target Protein:
Thymidine kinase, cytosolicDNA polymerase
Waktu ParuhIn preclinical tria…
Vol. DistribusiThis pharmacokineti…
KlirensThe plasma clearanc…
Genetik -
EDP1815 DB16486
biotech

EDP1815, was investigated in several clinical trials (NCT05066373, NCT05439941, NCT05682222, NCT03733353, NCT04603027, NCT04488575, NCT05121480, NCT04393246) to evaluate its safety and efficacy in conditions such as gastrointestinal behavior, atopic dermatiti…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edralbrutinib DB18095
small molecule | CAS: 1858206-58-2

Edralbrutinib is an orally available small molecule inhibitor of Bruton's tyrosine kinase.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edratide DB15272
small molecule | CAS: 433922-67-9

Edratide is under investigation in clinical trial NCT00203151 (A Study to Evaluate the Tolerability, Safety and Effectiveness of Edratide in the Treatment of Lupus).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Edrophonium Approved DB01010
small molecule | CAS: 312-48-1

A rapid-onset, short-acting cholinesterase inhibitor used in cardiac arrhythmias and in the diagnosis of myasthenia gravis. It has also been used as an antidote to curare principles.

Kategori:
AminesAntidotesCholinergic Agents +10
Target Protein:
CholinesteraseAcetylcholinesterase
Waktu ParuhDistribution half-l…
Vol. Distribusi* 1.6±0.4 L/kg [Adu…
Klirens* 6.8 +/- 2. mL/kg/…
Genetik -
EF-022 DB17768
biotech

EF-022 is a modified version of vitamin D binding protein macrophage activator, with potential antineoplastic and anti-angiogenic activities.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efalizumab Approved DB00095
biotech | CAS: 214745-43-4

Humanized IgG1 kappa isotype monoclonal antibody that binds to human CD11a. Efalizumab has a molecular weight of approximately 150 kilodaltons and is produced in a Chinese hamster ovary mammalian cell expression system in a nutrient medium containing the anti…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Integrin alpha-XIntegrin alpha-L
Waktu Paruh5 days
Vol. Distribusi-
Klirens-
Genetik -
Efanesoctocog alfa Approved DB16662
biotech | CAS: 2252477-42-0

Efanesoctocog alfa (BIVV001) is a recombinant factor VIII (FVIII) analogue fusion protein used for the routine prophylaxis, perioperative management of bleeding and on-demand treatment and control of bleeding episodes in patients with hemophilia A.[L45379] Th…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
Target Protein:
Coagulation factor IXCoagulation factor XLow-density lipoprotein receptor-related protein 2 +1
Waktu ParuhEfanesoctocog alfa …
Vol. DistribusiEfanesoctocog alfa …
KlirensEfanesoctocog alfa …
Genetik -
Efaproxiral DB08486
small molecule | CAS: 131179-95-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAminesAntineoplastic Agents +9
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efatutazone DB11894
small molecule | CAS: 223132-37-4

Efatutazone has been used in trials studying the treatment of Lymphoma, Liposarcoma, Solid Tumors, Multiple Myeloma, and Recurrent Thyroid Cancer, among others.

Kategori:
Antineoplastic AgentsPPAR gamma, antagonists & inhibitorsSulfur Compounds +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2049067-94-7

Efavaleukin alfa is a fusion protein consisting of interleukin mutein fused to the C-terminus of an immunoglobulin G Fc domain by way of a G4S linker. It is under investigation in clinical trial NCT03422627 (Safety and Efficacy of AMG 592 in Subjects With Ste…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efavirenz Approved DB00625
small molecule | CAS: 154598-52-4

Efavirenz (brand names Sustiva® and Stocrin®) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) and is used as part of highly active antiretroviral therapy (HAART) for the treatment of a human immunodeficiency virus (HIV) type 1. For HIV infectio…

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiinfectives for Systemic Use +52
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Gen Terkait:
CYP2B6
Waktu Paruh40-55 hours
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Efbemalenograstim alfa Approved DB18704
biotech | CAS: 2200269-79-8

Efbemalenograstim alfa is a long-acting recombinant fusion protein of granulocyte-colony stimulating factor (G-CSF) due to the addition of the Fc portion of human IgG2, allowing for once-per-cycle administration.[L48852,A262167] As endogenous G-CSF mediates t…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsColony-Stimulating Factors +2
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Efepoetin alfa DB19197
biotech | CAS: 1905452-78-9

Efepoetin alfa is under investigation in clinical trial NCT04155125 (A Study of Efepoetin Alfa in Treating Anaemia Associated With Chronic Kidney Diseases Patient).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efgartigimod alfa Approved DB15270
biotech | CAS: 1821402-21-4

Myasthenia gravis (MG) is an autoimmune disorder characterized by significant muscle weakness - particularly in the eye, throat, and extremities - caused by autoantibodies attacking the neuromuscular junction.[A243759] The production of IgG autoantibodies aga…

Kategori:
AntibodiesAntineoplastic and Immunomodulating AgentsGlobulins +6
Target Protein:
IgG receptor FcRn large subunit p51
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Efinaconazole Approved DB09040
small molecule | CAS: 164650-44-6

Efinaconazole is a 14 alpha-demethylase inhibitor indicated in the treatment of fungal infection of the nail, known as onychomycosis. It was approved for use in Canada and the USA in 2014 and is marketed by Valeant Pharmaceuticals North America LLC under the …

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +4
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylase
Waktu Paruh29.9 hours in healt…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2026634-47-7

Efineptakin alfa (also known as NT-I7) is a long-acting human interleukin-7 (IL-7) fusion protein that promotes T-cell development, contributing to the immune response. Compared to endogenous IL-7, NT-I7 is more stable and potent, has a longer half-life, and …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efinopegdutide DB15077
biotech | CAS: 2055640-93-0

Efinopegdutide is under investigation in clinical trial NCT03606057 (A Study to Investigate the Effect of JNJ-64565111 on Cardiac Repolarization (Corrected QT Interval) Compared With Placebo in Healthy Adults: a Thorough ECG Study Employing Placebo, JNJ-64565…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1635395-27-5

Efizonerimod alfa is under investigation in clinical trial NCT02221960 (A Phase 1 Study to Evaluate MEDI6383 Alone and in Combination With MEDI4736 in Adult Subjects With Select Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eflapegrastim Approved DB15001
biotech | CAS: 1384099-30-2

Febrile neutropenia (FN), defined as the co-occurrence of fever (temperature > 38 ?C) and severe neutropenia (ANC < 500 cells/mm<sup>3</sup>), is a potential side effect of myelosuppressive chemotherapy in which the patient develops an infection during a peri…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +20
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhIn patients with br…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ef…
Genetik -
biotech

Eflepedocokin alfa is a recombinant IL-22-Fc fusion protein manufactured in Chinese hamster ovary cells that is composed of 2 human interleukin 22 (IL-22) molecules linked to an immunoglobulin constant region (IgG2-Fc).[A225706, L27661] It is being developed …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eflornithine Approved DB06243
small molecule | CAS: 70052-12-9

Eflornithine is an irreversible ornithine decarboxylase inhibitor originally developed as a treatment for human African trypanosomiasis.[A262829] Further research has also implicated ornithine decarboxylase in other conditions like facial hirsutism and cancer…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAmino AcidsAmino Acids, Basic +15
Target Protein:
Ornithine decarboxylase
Waktu ParuhThe terminal plasma…
Vol. DistribusiEflornithine volume…
KlirensThe clearance (CL/F…
Genetik -
biotech | CAS: 1953227-87-6

Efmarodocokin alfa is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1644543-31-6

Efmitermant alfa, a locally-acting GDF/activin ligand trap, is under investigation in clinical trial NCT03124459 (Study of ACE-083 in Patients With Charcot-marie-tooth Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efmoroctocog alfa Approved DB11607
biotech | CAS: 1270012-79-7

Efmoroctocog alfa is a fully recombinant factor VIII-Fc fusion protein (rFVIIIFc) with an extended half-life compared with conventional factor VIII (FVIII) preparations, including recombinant FVIII (rFVIII) products such as [DB13999][A31551]. It is an antihem…

Kategori:
HemostaticsHuman Antihemophilic Factors
Target Protein:
von Willebrand factor
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Efocipegtrutide DB18194
biotech | CAS: 2513399-19-2

Efocipegtrutide is a long-acting, monomeric peptide triple agonist.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efonidipine DB09235
small molecule | CAS: 111011-63-3

Efonidipine is a calcium channel blocker of the _dihydropyridine class_, commercialized by Shionogi & Co. (Japan). Initially, it was marketed in 1995 under the trade name, _Landel_. The drug has been shown to block T-type in addition to L-type calcium channel…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +22
Target Protein:
Voltage gated L-type calcium channelVoltage-dependent calcium channelVoltage-dependent T-type calcium channel +4
Waktu ParuhThe peak plasma con…
Vol. Distribusi-
Klirens-
Genetik -
Efpeglenatide DB15650
biotech | CAS: 1296200-77-5

Efpeglenatide is under investigation in clinical trial NCT03713684 (Efficacy and Safety of Efpeglenatide Versus Placebo in Patients With Type 2 Diabetes Mellitus Inadequately Controlled With Basal Insulin Alone or in Combination With Oral Antidiabetic Drug(s)…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +2
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efprezimod alfa DB16448
biotech

CD24Fc is a biological immunomodulator originally developed to address graft-versus-host disease in stem cell transplantation in leukemia patients.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efruxifermin DB19012
biotech | CAS: 2375240-92-7

Efruxifermin is under investigation in clinical trial NCT06215716 (A Study Evaluating Efruxifermin in Subjects With Non-cirrhotic Nonalcoholic Steatohepatitis (Nash)/metabolic Dysfunction-associated Steatohepatitis (MASH) and Fibrosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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