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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 114 / 236
GSK-923295 DB06097
small molecule

GSK-923295 is a small-molecule inhibitor of the mitotic kinesin centromere-associated protein E (CENP-E), and the third novel drug candidate to arise from Cytokinetics' broad strategic alliance with GlaxoSmithKline (GSK). GSK-923295 demonstrated a broad spect…

Target Protein:
Centromere-associated protein E
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK-945237 DB15345
small molecule | CAS: 944406-54-6

GSK-945237 is under investigation in clinical trial NCT01039610 (A Single Center Four Part Study in Healthy Adult Subjects to Evaluate: the Safety, Tolerability and Pharmacokinetics of a Single Oral Dose and Repeat Escalating Oral Doses of GSK945237; the Effe…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK159797 DB05043
small molecule

GSK159797 ('797) is an inhaled, longer-acting Beta2 agonist developed for the treatment of respiratory disease such as asthma and COPD.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
GSK2245035 DB16076
small molecule | CAS: 1207629-49-9

GSK2245035 is under investigation in clinical trial NCT02833974 (Effect of the GSK2245035 on the Allergen-induced Asthmatic Response).

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK2256098 DB16106
small molecule | CAS: 1224887-10-8

GSK2256098 is under investigation in clinical trial NCT02523014 (Vismodegib and FAK Inhibitor GSK2256098 in Treating Patients With Progressive Meningiomas).

Kategori:
AminesHydroxy AcidsHydroxylamines +1
Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GSK2798745 DB16033
small molecule | CAS: 1419609-94-1

GSK2798745 is under investigation in clinical trial NCT03372603 (A Study to Assess the Effectiveness and Side Effects of GSK2798745 in Participants With Chronic Cough).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GsMtx-4 DB17861
biotech

GsMtx-4 is a peptide found in tarantula venom that inhibits mechanosensitive ion channel (MSC) activity.

Kategori:
Amino Acids, Peptides, and ProteinsArthropod VenomsBiological Factors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GT-AS DB17883
biotech

GT-AS recombinant adeno-associated virus serotype 9 vector containing the transgene UBE3A encoding for ubiquitin protein ligase E3A/E6-AP.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
GTA002 DB17187
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
GTP-506 DB17682
biotech

GTP-506 is a gene therapy formed by two vectors, a nuclease vector targeting gene editing in the well-characterized PCSK9 gene locus and a therapeutic donor vector that inserts the OTC gene to provide the desired genetic correction.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
GTS-21 DB05708
small molecule | CAS: 148372-04-7

GTS-21 (also known as DMBX-A), is a novel, small-molecule, orally active and selective alpha-7 nicotinic acetylcholine (nACh) receptor agonist that has demonstrated memory and cognition enhancement activity in human clinical trials. Athenagen licensed the exc…

Kategori:
Benzene DerivativesCholinergic AgentsCholinergic Agonists +5
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GTX-102 DB16981
biotech

GTX-102 is an antisense oligonucleotide designed to target and inhibit the expression of UBE3A-AS. It is being investigated for the treatment of Angelman Syndrome.[L46772]

Kategori:
Antisense Oligonucleotide Specific to the Antisense Transcript of UBE3A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GTX-758 DB14969
small molecule | CAS: 938067-78-8

GTX-758 is under investigation in clinical trial NCT01420861 (GTx-758 on Serum Prostate-specific Antigen (PSA) in Men With Castrate Resistant Prostate Cancer).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guaifenesin Approved DB00874
small molecule | CAS: 93-14-1

Guaifenesin possesses a storied history, having been originally formally approved by the US FDA in 1952 and continues to be one of very few - if not perhaps the only drug that is readily available and used as an expectorant [F4525]. Since that time the agent …

Kategori:
Benzene DerivativesCatecholsCough and Cold Preparations +6
Target Protein:
NMDA receptor
Waktu ParuhThe half-life in pl…
Vol. DistribusiThe geometric mean …
KlirensThe mean clearance …
Genetik -
Guanabenz Approved DB00629
small molecule | CAS: 5051-62-7

An alpha-2 selective adrenergic agonist used as an antihypertensive agent. [PubChem]

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +11
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu Paruh6 hours.
Vol. Distribusi-
Klirens-
Genetik -
Guanazodine DB13604
small molecule | CAS: 32059-15-7

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanethidine Approved DB01170
small molecule | CAS: 55-65-2

An antihypertensive agent that acts by inhibiting selectively transmission in post-ganglionic adrenergic nerves. It is believed to act mainly by preventing the release of norepinephrine at nerve endings and causes depletion of norepinephrine in peripheral sym…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAmidines +16
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh1.5 days
Vol. Distribusi-
Klirens* Renal cl=56 ml/min
Genetik -
Guanfacine Approved DB01018
small molecule | CAS: 29110-47-2

Guanfacine, or BS 100-141,[A189838,A189841] is a selective alpha-A2 adrenergic receptor agonist initially indicated for the treatment of hypertension[L11274] but is now indicated as an extended release tablet for the treatment of ADHD.[L11277] Guanfacine was …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +26
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu ParuhGuanfacine has a ha…
Vol. DistribusiGuanfacine has a vo…
KlirensGuanfacine has a to…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Trypsin-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 77482-44-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic Acids
Target Protein:
Carboxypeptidase D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanine DB02377
small molecule | CAS: 73-40-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPurinesPurinones +1
Target Protein:
GTP cyclohydrolase 1Purine nucleoside phosphorylasePurine nucleoside phosphorylase 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanoclor DB13779
small molecule | CAS: 5001-32-1

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanosine DB02857
small molecule | CAS: 118-00-3

Guanosine is a nucleoside comprising guanine attached to a ribose (ribofuranose) ring via a ?-N9-glycosidic bond. Guanosine can be phosphorylated to become GMP (guanosine monophosphate), cGMP (cyclic guanosine monophosphate), GDP (guanosine diphosphate) and G…

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
DNA polymerase catalytic subunitDNA polymerase catalytic subunitPurine nucleoside phosphorylase +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 117-68-0

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
RibonucleaseBifunctional protein PyrR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 33503-72-9

Guanosine tetraphosphate is a guanine nucleotide containing four phosphate groups. Two phosphate groups are esterified to the sugar moiety in the 5' position and the other two in the 2' or 3' position. This nucleotide serves as a messenger to turn off the syn…

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseXanthine phosphoribosyltransferaseGTPase Obg
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 38557-85-6

Deskripsi belum tersedia.

Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 130-50-7

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
GDP-mannose 4,6 dehydratase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 85-32-5

Guanosine 5'-monophosphate. A guanine nucleotide containing one phosphate group esterified to the sugar moiety and found widely in nature. [PubChem]

Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseDNA polymerase catalytic subunitDNA polymerase catalytic subunit +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 86-01-1

Guanosine 5'-(tetrahydrogen triphosphate). A guanine nucleotide containing three phosphate groups esterified to the sugar moiety. [PubChem]

Target Protein:
GTP cyclohydrolase 1Genome polyproteinRNA-directed RNA polymerase +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanoxabenz DB13410
small molecule | CAS: 24047-25-4

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanoxan Approved DB13211
small molecule | CAS: 2165-19-7

Guanoxan is an antihypertensive agent similar in its mechanism of action to guanethidine; may cause liver damage. Guanoxan was approved in the UK but was withdrawn from the market due to hepatotoxicity.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gusacitinib DB15670
small molecule | CAS: 1425381-60-7

Gusacitinib is under investigation in clinical trial NCT02550678 (A Study of the Efficacy and Safety of ASN-002 in Adult Patients With Low-risk Nodular Basal Cell Carcinoma).

Kategori:
Nitriles
Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guselkumab Approved DB11834
biotech | CAS: 1350289-85-8

Guselkumab is a human immunoglobulin G1 lambda (IgG1?) monoclonal antibody that selectively blocks interleukin-23. IL-23 is an inflammatory cytokine that activates the CD4+ T-helper (Th17) cell pathway to mediate the inflammatory cascade that induces psoriati…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Interleukin-23 subunit alpha
Waktu ParuhMean half-life of g…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik -
Gusperimus DB12692
small molecule | CAS: 98629-43-7

Gusperimus has been used in trials studying the treatment of Lupus Nephritis, Wegeners Granulomatosis, and Wegener's Granulomatosis.

Kategori:
AmidinesAntibiotics, AntineoplasticAntineoplastic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GVAX DB17276
biotech

GVAX is a granulocyte-macrophage colony-stimulating factor (GM-CSF) gene-transfected tumor cell vaccine.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW 468816 DB05417
small molecule

GW 468816 is glycine receptor antagonist. It is designed to aid abstinence in people who have just quit smoking, delaying the time to relapse. It was undergoing phase II trials since December 2003.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glycine receptor subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW 597599 DB05418
small molecule

GW 597599, a neurokinin-1 (NK1) receptor antagonist is currently in phase II trials for chemotherapy-induced vomiting; functional dyspepsia; depression and anxiety.

Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-274150 DB12237
small molecule | CAS: 210354-22-6

GW274150 has been used in trials studying the treatment and prevention of Asthma, Migraine, Migraine Disorders, and Arthritis, Rheumatoid.

Kategori:
AnionsElectrolytesHydrogen Sulfide +3
Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-3965 DB03791
small molecule | CAS: 405911-09-3

GW-3965 is a liver X receptor ligand.

Kategori:
Acids, CarbocyclicAminesBenzene Derivatives +2
Target Protein:
Oxysterols receptor LXR-betaOxysterols receptor LXR-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-468816 DB15099
small molecule | CAS: 476689-77-7

GW-468816 is under investigation in clinical trial NCT00218465 (Effectiveness of GW468816, an NMDA Glycine Site Antagonist, for Prevention of Relapse to Smoking).

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-493838 DB12760
small molecule | CAS: 253124-46-8

GW493838 has been used in trials studying the treatment of Neuropathic Pain.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-559090 DB06508
small molecule | CAS: 278598-52-0

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Integrin alpha-5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-590735 DB07215
small molecule | CAS: 343321-96-0

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Nuclear receptor coactivator 1Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-813893 DB07278
small molecule | CAS: 478644-12-1

Deskripsi belum tersedia.

Kategori:
AmidesAnticoagulantsAntithrombins +8
Target Protein:
Coagulation factor XProthrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-870086 DB12322
small molecule | CAS: 827319-43-7

GW870086X has been investigated for the treatment of ASTHMA.

Kategori:
Fused-Ring Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW810781 DB16032
small molecule | CAS: 280571-30-4

GW810781 is under investigation in clinical trial NCT00046332 (A Study Comparing 4 Doses of GW810781 Versus Placebo in Hiv-infected Patients).

Kategori:
Anti-HIV Agents
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW842166 DB11903
small molecule | CAS: 666260-75-9

GW842166X has been used in trials studying the treatment of Pain, Analgesia, Inflammation, Osteoarthritis, and Pain, Inflammatory, among others.

Kategori:
Agents producing tachycardiaCannabinoid Receptor AgonistsCannabinoids and similars +1
Target Protein:
Cannabinoid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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