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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 114 / 282
DT2216 DB18020
small molecule | CAS: 2365172-42-3

Deskripsi belum tersedia.

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DTP-348 DB12741
small molecule | CAS: 1383370-92-0

Dtp348 has been used in trials studying the treatment of Solid Tumors and Head and Neck Neoplasms.

Target Protein:
Carbonic anhydrase 9
Waktu Paruh-
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DTS-201 DB06071
small molecule

DTS-201 is a prodrug of doxorubicin, a widely used anti-cancer drug that Diatos intends to develop for the treatment of various solid tumors. It is activated in the tumor environment. DTS-201 may be suitable for the treatment of many types of solid tumors, i…

Kategori:
AnthracyclinesCarbohydratesGlycosides +1
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DTx-1252 DB18086
small molecule

DTx-1252 is a siRNA therapeutic under investigation for the treatment of Charcot-Marie-Tooth Disease type 1A (CMTD1A).[L48096]

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DU125530 DB16040
small molecule | CAS: 161611-99-0

DU125530 is under investigation in clinical trial NCT01119430 (Fluoxetine Versus Fluoxetine Plus DU125530 in Major Depressive Disorder).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT1 Receptor Antagonists +4
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
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Dubermatinib DB15187
small molecule | CAS: 1341200-45-0

Dubermatinib is under investigation in clinical trial NCT03572634 (Phase 1/2 Study of TP-0903 (an Inhibitor of AXL Kinase) in Patients With Previously Treated CLL).

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Tyrosine-protein kinase receptor UFO
Waktu Paruh-
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Dulaglutide Approved DB09045
biotech | CAS: 923950-08-7

Dulaglutide, marketed by Eli Lilly as Trulicity, is a once-weekly subcutaneous glucagon-like peptide-1 (GLP-1) receptor agonist designed using recombinant DNA technology; it has been approved as an adjunct therapy to diet and exercise in the management of 2 …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +21
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhIn a pharmacokineti…
Vol. DistribusiThe apparent volume…
KlirensThe apparent popula…
Genetik -
Dulanermin DB12349
biotech | CAS: 867153-61-5

Dulanermin has been used in trials studying the treatment of Colorectal Cancer, Non-Hodgkin's Lymphoma, and Metastatic Colorectal Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +4
Waktu Paruh-
Vol. Distribusi-
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Duligotuzumab DB12142
biotech | CAS: 1314238-96-4

Duligotuzumab has been used in trials studying the treatment of Neoplasms, Colorectal Cancer, Head and Neck Cancer, and Epithelial Tumors, Malignant.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
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Duloxetine Approved DB00476
small molecule | CAS: 116539-59-4

Duloxetine is a dual serotonin and norepinephrine reuptake inhibitor.[label] It was originally discovered in 1993 and developed by Eli Lilly and Company as LY248686.[A178741] Duloxetine first received approval from the FDA in August, 2004 as Cymbalta for the …

Kategori:
Agents producing tachycardiaAnalgesicsAntidepressive Agents +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Waktu ParuhMean of 12 h with a…
Vol. DistribusiApparent Vd of 1620…
KlirensThere is a large de…
Genetik -
Dupilumab Approved DB12159
biotech | CAS: 1190264-60-8

Dupilumab is a fully human monoclonal antibody of the immunoglobulin G4 subclass that binds to the interleukin-4 (IL-4) receptor, inhibiting the receptor signaling pathways.[A180478] As an interleukin-4 receptor alpha antagonist, dupilumab inhibits the signal…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAnti-Asthmatic Agents +13
Target Protein:
Interleukin-4 receptor subunit alphaInterleukin-13Interleukin-4
Waktu ParuhThere is limited hu…
Vol. DistribusiThe estimated volum…
KlirensThere is limited da…
Genetik -
Durlobactam Approved DB16704
small molecule | CAS: 1467829-71-5

Durlobactam is a diazabicyclooctane non-beta-lactam, beta-lactamase inhibitor. It is typically given in combination with [sulbactam] to protect it from degradation by certain serine-beta-lactamases.[L47336] The combination product of durlobactam and sulbactam…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +3
Target Protein:
Beta-lactamase CTX-M
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of du…
Genetik -
Duroquinone DB01927
small molecule | CAS: 527-17-3

Deskripsi belum tersedia.

Kategori:
Quinones
Target Protein:
NAD(P)H dehydrogenase [quinone] 1
Waktu Paruh-
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Durvalumab Approved DB11714
biotech | CAS: 1428935-60-7

Durvalumab is a human immunoglobulin G1 kappa (IgG1?) monoclonal antibody and a novel immune-checkpoint inhibitor for cancer treatment.[A192789] Produced by recombinant DNA technology in Chinese Hamster Ovary (CHO) cell suspension culture,[L12621] durvalumab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntibodies +20
Target Protein:
Programmed cell death 1 ligand 1Programmed cell death protein 1
Waktu ParuhBased on baseline c…
Vol. DistribusiIn patients receivi…
KlirensClearance of durval…
Genetik -
Dusigitumab DB12363
biotech | CAS: 1204390-13-5

Dusigitumab has been used in trials studying the treatment of Cancer, Advanced Solid Malignancies, Unresectable or Metastatic Hepatocellular Carcinoma (HCC), and Hormone-sensitive, HER-2 Negative Metastatic Breast Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Dusquetide DB11879
small molecule | CAS: 931395-42-5

Dusquetide has been used in trials studying the treatment of Oral Mucositis.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Dutasteride Approved DB01126
small molecule | CAS: 164656-23-9

Dutasteride is an oral synthetic 4-azasteroid commonly marketed under the trade name Avodart. It is a novel dual 5?-reductase inhibitor that works by blocking both isoforms of 5?-reductase enzymes in a potent, selective, and irreversible manner.[A1909] Type I…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +14
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 1Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 2
Waktu ParuhThe terminal elimin…
Vol. DistribusiDutasteride display…
KlirensIn a study of healt…
Genetik -
Dutogliptin DB11723
small molecule | CAS: 852329-66-9

Dutogliptin has been investigated for the treatment of Diabetes Mellitus, Type II.

Kategori:
AcidsAcids, NoncarboxylicAgents causing angioedema +3
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh10-13 hours
Vol. Distribusi-
Klirens-
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Duvakitug DB19444
biotech | CAS: 2750005-84-4

Duvakitug is under investigation in clinical trial NCT05668013 (A Study to Evaluate the Long-term Effect of TEV-48574 in Moderate to Severe Ulcerative Colitis or Crohn's Disease).

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Duvelisib Approved DB11952
small molecule | CAS: 1201438-56-3

Duvelisib, also known as IPI-145 and INK-1197, is a small-molecule inhibitor of phosphoinositide-3 kinases that was designed initially to prove that simultaneous inhibition of the isoforms delta and gamma can produce a broad adaptative and innate immune cell …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +10
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe reported half-l…
Vol. DistribusiThe volume of distr…
KlirensDuvelisib clearance…
Genetik -
Duvoglustat DB03206
small molecule | CAS: 19130-96-2

An alpha-glucosidase inhibitor with antiviral action. Derivatives of deoxynojirimycin may have anti-HIV activity.

Kategori:
AlkaloidsAmino SugarsAnti-Infective Agents +7
Target Protein:
Maltase-glucoamylaseLysosomal alpha-glucosidaseNeutral alpha-glucosidase AB +6
Waktu Paruh-
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Duvortuxizumab DB15211
biotech | CAS: 1831098-91-9

Duvortuxizumab is under investigation in clinical trial NCT02743546 (Study of the Safety, Pharmacokinetics, Pharmacodynamics, and Efficacy of Duvortuxizumab (JNJ-64052781) Plus Ibrutinib in Lymphoma).

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Dyclonine Approved DB00645
small molecule | CAS: 586-60-7

Dyclonine is an oral anaesthetic found in Sucrets, an over the counter throat lozenge. It may also be found in some Cepacol sore throat spray products.

Kategori:
AnestheticsAnesthetics, LocalCentral Nervous System Agents +6
Target Protein:
Sodium channel protein type 10 subunit alphaSodium channel protein type 5 subunit alpha
Waktu ParuhApproximately 30 to…
Vol. Distribusi-
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Dydrogesterone Approved DB00378
small molecule | CAS: 152-62-5

A synthetic progestational hormone with no androgenic or estrogenic properties. Unlike many other progestational compounds, dydrogesterone produces no increase in temperature and does not inhibit ovulation.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Target Protein:
Progesterone receptor
Waktu ParuhDydrogesterone: 5-7…
Vol. Distribusi-
Klirens-
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DYN-101 DB17921
biotech

DYN-101 is an antisense product candidate designed to reduce the expression of dynamin 2 protein.

Waktu Paruh-
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Dynasore DB15964
small molecule | CAS: 304448-55-3

Deskripsi belum tersedia.

Kategori:
Dynamins, antagonists & inhibitorsHydrazines
Waktu Paruh-
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DYNE-251 DB18130
biotech

DYNE-251 is a phosphorodiamidate morpholino oligomer (PMO) conjugated to a fragment antibody (Fab) that binds to the transferrin receptor 1 (TfR1). It is being investigated for the treatment of Duchenne muscular dystrophy (DMD) in patients who are amenable to…

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Dynorphin DB16146
small molecule | CAS: 80448-90-4

Dynorphin is under investigation in clinical trial NCT00000244 (Effects of Dynorphin 1-13 on Heroin Addiction - 1).

Kategori:
Amino Acids, Peptides, and ProteinsNerve Tissue ProteinsNeuropeptides +4
Target Protein:
Kappa-type opioid receptorMu-type opioid receptorDelta-type opioid receptor
Waktu Paruh-
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Dyphylline Approved DB00651
small molecule | CAS: 479-18-5

Dyphylline is a theophylline derivative with broncho- and vasodilator properties. It is typically used in the management of asthma, cardiac dyspnea, and bronchitis.

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +13
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B5'-nucleotidase3',5'-cyclic-AMP phosphodiesterase 4A +4
Waktu Paruh2 hours (range 1.8 …
Vol. Distribusi-
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Genetik -
E-2012 DB05171
small molecule | CAS: 870843-42-8

E-2012 is a gamma secretase modulator that is being evaluated as a potential new treatment for Alzheimer's disease.

Kategori:
Amyloid Precursor Protein SecretasesEnzyme InhibitorsGamma Secretase Inhibitors and Modulators
Target Protein:
Gamma-secretase subunit APH-1BNicastrinPresenilin-1 +2
Waktu Paruh-
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E-52862 DB16881
small molecule | CAS: 878141-96-9

Deskripsi belum tersedia.

Kategori:
OxazinesReceptors, sigma, antagonists & inhibitors
Waktu Paruh-
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E-6005 DB12776
small molecule | CAS: 947620-48-6

E6005 has been used in trials studying the treatment of Atopic Dermatitis.

Kategori:
Acids, CarbocyclicAntipruriticsHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
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E-6201 DB11687
small molecule | CAS: 603987-35-5

E6201 has been investigated for the treatment of Chronic Plaque Psoriasis.

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E-7820 DB12505
small molecule | CAS: 289483-69-8

E7820 has been investigated for the treatment of Colon Cancer and Rectal Cancer.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Integrin alpha-2
Waktu Paruh-
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E1v1.11 DB18363
biotech

E1v1.11 is an antisense oligonucleotide targeting the _SMN2_ gene which is under investigation for the treatment of spinal muscular atrophy (SMA).[L48196]

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E5531 DB06447
small molecule | CAS: 162679-36-9

E5531 is an endotoxin antagonist.

Kategori:
AntigensAntigens, BacterialBacterial Toxins +8
Target Protein:
Toll-like receptor 4
Waktu Paruh-
Vol. Distribusi-
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E59 DB18372
biotech

E59 is a humanized IgG1 low affinity allergic reactivity inhibiting (LARI) monoclonal antibody. It was developed by Sixal Inc.

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E7107 DB12508
small molecule | CAS: 630100-90-2

E7107 has been used in trials studying the treatment of Cancer.

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EA-230 DB19114
small molecule | CAS: 503844-09-5

EA-230 is under investigation in clinical trial NCT03145220 (Immunomodulation of EA-230 Following On-pump Coronary Artery Bypass Grafting (CABG)).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
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EA-2353 DB18506
small molecule

EA-2353 is a small molecule inhibitor of kinase mediators of the Wnt pathway.

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EB003 DB18362
biotech

EB003 is a CRISPR-based sequence-specific antimicrobial (SSAM) targeted against shiga toxin-producing _E. coli_.

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EB05 DB16477
biotech | CAS: 2641646-59-3

EB05, in combination with standard of care (SOC), is being investigated in clinical trial NCT04401475 to evaluate its safety and efficacy in adult hospitalized patients with COVID-19 and ARDS.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
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Ebastine Approved DB11742
small molecule | CAS: 90729-43-4

Ebastine is under investigation for the treatment of Irritable Bowel Syndrome (IBS). Ebastine has been investigated for the treatment of Urticaria.

Kategori:
Antihistamines for Systemic UseCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Eberconazole DB13656
small molecule | CAS: 128326-82-9

Deskripsi belum tersedia.

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseCycloparaffins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Ebola virus vaccine is a vaccine used to prevent Ebola virus disease caused by _Zaire ebolavirus_ in adults, prevent outbreaks, and reduce the extent of the virus spreading in case of outbreaks.[L10854] Ebola virus disease, formerly known as Ebola hemorrhagic…

Kategori:
ImmunizationImmunologic FactorsVaccines +1
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Ebopiprant DB16147
small molecule | CAS: 2005486-31-5

Ebopiprant is under investigation in clinical trial NCT03369262 (Poc Study of OBE022 in Threatened Preterm Labour).

Kategori:
Sulfur CompoundsThiazoles
Waktu Paruh-
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Ebselen DB12610
small molecule | CAS: 60940-34-3

Ebselen has been investigated for the treatment and basic science of Meniere's Disease, Type 2 Diabetes Mellitus, and Type 1 Diabetes Mellitus.

Kategori:
Agents that produce hypertensionAnalgesicsAnalgesics, Non-Narcotic +17
Target Protein:
AlbuminLysine-specific demethylase 4ABifunctional epoxide hydrolase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ebvaciclib DB18967
small molecule | CAS: 2185857-97-8

Ebvaciclib is under investigation in clinical trial NCT03519178 (A Study of PF-06873600 in People With Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EC-0652 DB15340
small molecule | CAS: 1025066-50-5

EC-0652 is under investigation in clinical trial NCT02202447 (Phase 1 of EC1169 In Patients With Recurrent MCRPC).

Waktu Paruh-
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EC-17 DB12559
small molecule | CAS: 583037-91-6

Folate Fitc has been used in trials studying the diagnostic of Ovarian Cancer.

Target Protein:
Folate receptor alpha
Waktu Paruh-
Vol. Distribusi-
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Genetik -
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