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14361

Total database: 17430
Struktur (SMILES)
9916 (69.0%)
Target
7893 (55.0%)
Genomik
112 (0.8%)
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14361 (100.0%)

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Hasil Pencarian (14361)

Halaman 113 / 288
Duloxetine Approved DB00476
small molecule | CAS: 116539-59-4

Duloxetine is a dual serotonin and norepinephrine reuptake inhibitor.[label] It was originally discovered in 1993 and developed by Eli Lilly and Company as LY248686.[A178741] Duloxetine first received approval from the FDA in August, 2004 as Cymbalta for the …

Kategori:
Agents producing tachycardiaAnalgesicsAntidepressive Agents +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Waktu ParuhMean of 12 h with a…
Vol. DistribusiApparent Vd of 1620…
KlirensThere is a large de…
Genetik -
Dupilumab Approved DB12159
biotech | CAS: 1190264-60-8

Dupilumab is a fully human monoclonal antibody of the immunoglobulin G4 subclass that binds to the interleukin-4 (IL-4) receptor, inhibiting the receptor signaling pathways.[A180478] As an interleukin-4 receptor alpha antagonist, dupilumab inhibits the signal…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAnti-Asthmatic Agents +13
Target Protein:
Interleukin-4 receptor subunit alphaInterleukin-13Interleukin-4
Waktu ParuhThere is limited hu…
Vol. DistribusiThe estimated volum…
KlirensThere is limited da…
Genetik -
Durlobactam Approved DB16704
small molecule | CAS: 1467829-71-5

Durlobactam is a diazabicyclooctane non-beta-lactam, beta-lactamase inhibitor. It is typically given in combination with [sulbactam] to protect it from degradation by certain serine-beta-lactamases.[L47336] The combination product of durlobactam and sulbactam…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +3
Target Protein:
Beta-lactamase CTX-M
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of du…
Genetik -
Durvalumab Approved DB11714
biotech | CAS: 1428935-60-7

Durvalumab is a human immunoglobulin G1 kappa (IgG1?) monoclonal antibody and a novel immune-checkpoint inhibitor for cancer treatment.[A192789] Produced by recombinant DNA technology in Chinese Hamster Ovary (CHO) cell suspension culture,[L12621] durvalumab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntibodies +20
Target Protein:
Programmed cell death 1 ligand 1Programmed cell death protein 1
Waktu ParuhBased on baseline c…
Vol. DistribusiIn patients receivi…
KlirensClearance of durval…
Genetik -
Dusigitumab DB12363
biotech | CAS: 1204390-13-5

Dusigitumab has been used in trials studying the treatment of Cancer, Advanced Solid Malignancies, Unresectable or Metastatic Hepatocellular Carcinoma (HCC), and Hormone-sensitive, HER-2 Negative Metastatic Breast Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dusquetide DB11879
small molecule | CAS: 931395-42-5

Dusquetide has been used in trials studying the treatment of Oral Mucositis.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dutasteride Approved DB01126
small molecule | CAS: 164656-23-9

Dutasteride is an oral synthetic 4-azasteroid commonly marketed under the trade name Avodart. It is a novel dual 5?-reductase inhibitor that works by blocking both isoforms of 5?-reductase enzymes in a potent, selective, and irreversible manner.[A1909] Type I…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +14
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 1Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 2
Waktu ParuhThe terminal elimin…
Vol. DistribusiDutasteride display…
KlirensIn a study of healt…
Genetik -
Dutogliptin DB11723
small molecule | CAS: 852329-66-9

Dutogliptin has been investigated for the treatment of Diabetes Mellitus, Type II.

Kategori:
AcidsAcids, NoncarboxylicAgents causing angioedema +3
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh10-13 hours
Vol. Distribusi-
Klirens-
Genetik -
Duvakitug DB19444
biotech | CAS: 2750005-84-4

Duvakitug is under investigation in clinical trial NCT05668013 (A Study to Evaluate the Long-term Effect of TEV-48574 in Moderate to Severe Ulcerative Colitis or Crohn's Disease).

Waktu Paruh-
Vol. Distribusi-
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Duvelisib Approved DB11952
small molecule | CAS: 1201438-56-3

Duvelisib, also known as IPI-145 and INK-1197, is a small-molecule inhibitor of phosphoinositide-3 kinases that was designed initially to prove that simultaneous inhibition of the isoforms delta and gamma can produce a broad adaptative and innate immune cell …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +10
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe reported half-l…
Vol. DistribusiThe volume of distr…
KlirensDuvelisib clearance…
Genetik -
Duvoglustat DB03206
small molecule | CAS: 19130-96-2

An alpha-glucosidase inhibitor with antiviral action. Derivatives of deoxynojirimycin may have anti-HIV activity.

Kategori:
AlkaloidsAmino SugarsAnti-Infective Agents +7
Target Protein:
Maltase-glucoamylaseLysosomal alpha-glucosidaseNeutral alpha-glucosidase AB +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Duvortuxizumab DB15211
biotech | CAS: 1831098-91-9

Duvortuxizumab is under investigation in clinical trial NCT02743546 (Study of the Safety, Pharmacokinetics, Pharmacodynamics, and Efficacy of Duvortuxizumab (JNJ-64052781) Plus Ibrutinib in Lymphoma).

Waktu Paruh-
Vol. Distribusi-
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Dyclonine Approved DB00645
small molecule | CAS: 586-60-7

Dyclonine is an oral anaesthetic found in Sucrets, an over the counter throat lozenge. It may also be found in some Cepacol sore throat spray products.

Kategori:
AnestheticsAnesthetics, LocalCentral Nervous System Agents +6
Target Protein:
Sodium channel protein type 10 subunit alphaSodium channel protein type 5 subunit alpha
Waktu ParuhApproximately 30 to…
Vol. Distribusi-
Klirens-
Genetik -
Dydrogesterone Approved DB00378
small molecule | CAS: 152-62-5

A synthetic progestational hormone with no androgenic or estrogenic properties. Unlike many other progestational compounds, dydrogesterone produces no increase in temperature and does not inhibit ovulation.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Target Protein:
Progesterone receptor
Waktu ParuhDydrogesterone: 5-7…
Vol. Distribusi-
Klirens-
Genetik -
DYN-101 DB17921
biotech

DYN-101 is an antisense product candidate designed to reduce the expression of dynamin 2 protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dynasore DB15964
small molecule | CAS: 304448-55-3

Deskripsi belum tersedia.

Kategori:
Dynamins, antagonists & inhibitorsHydrazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DYNE-251 DB18130
biotech

DYNE-251 is a phosphorodiamidate morpholino oligomer (PMO) conjugated to a fragment antibody (Fab) that binds to the transferrin receptor 1 (TfR1). It is being investigated for the treatment of Duchenne muscular dystrophy (DMD) in patients who are amenable to…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dynorphin DB16146
small molecule | CAS: 80448-90-4

Dynorphin is under investigation in clinical trial NCT00000244 (Effects of Dynorphin 1-13 on Heroin Addiction - 1).

Kategori:
Amino Acids, Peptides, and ProteinsNerve Tissue ProteinsNeuropeptides +4
Target Protein:
Kappa-type opioid receptorMu-type opioid receptorDelta-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dyphylline Approved DB00651
small molecule | CAS: 479-18-5

Dyphylline is a theophylline derivative with broncho- and vasodilator properties. It is typically used in the management of asthma, cardiac dyspnea, and bronchitis.

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +13
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B5'-nucleotidase3',5'-cyclic-AMP phosphodiesterase 4A +4
Waktu Paruh2 hours (range 1.8 …
Vol. Distribusi-
Klirens-
Genetik -
E-2012 DB05171
small molecule | CAS: 870843-42-8

E-2012 is a gamma secretase modulator that is being evaluated as a potential new treatment for Alzheimer's disease.

Kategori:
Amyloid Precursor Protein SecretasesEnzyme InhibitorsGamma Secretase Inhibitors and Modulators
Target Protein:
Gamma-secretase subunit APH-1BNicastrinPresenilin-1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
E-6005 DB12776
small molecule | CAS: 947620-48-6

E6005 has been used in trials studying the treatment of Atopic Dermatitis.

Kategori:
Acids, CarbocyclicAntipruriticsHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
E-6201 DB11687
small molecule | CAS: 603987-35-5

E6201 has been investigated for the treatment of Chronic Plaque Psoriasis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
E1v1.11 DB18363
biotech

E1v1.11 is an antisense oligonucleotide targeting the _SMN2_ gene which is under investigation for the treatment of spinal muscular atrophy (SMA).[L48196]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
E59 DB18372
biotech

E59 is a humanized IgG1 low affinity allergic reactivity inhibiting (LARI) monoclonal antibody. It was developed by Sixal Inc.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EA-230 DB19114
small molecule | CAS: 503844-09-5

EA-230 is under investigation in clinical trial NCT03145220 (Immunomodulation of EA-230 Following On-pump Coronary Artery Bypass Grafting (CABG)).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EA-2353 DB18506
small molecule

EA-2353 is a small molecule inhibitor of kinase mediators of the Wnt pathway.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EB003 DB18362
biotech

EB003 is a CRISPR-based sequence-specific antimicrobial (SSAM) targeted against shiga toxin-producing _E. coli_.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
EB05 DB16477
biotech | CAS: 2641646-59-3

EB05, in combination with standard of care (SOC), is being investigated in clinical trial NCT04401475 to evaluate its safety and efficacy in adult hospitalized patients with COVID-19 and ARDS.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Ebola virus vaccine is a vaccine used to prevent Ebola virus disease caused by _Zaire ebolavirus_ in adults, prevent outbreaks, and reduce the extent of the virus spreading in case of outbreaks.[L10854] Ebola virus disease, formerly known as Ebola hemorrhagic…

Kategori:
ImmunizationImmunologic FactorsVaccines +1
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Ebopiprant DB16147
small molecule | CAS: 2005486-31-5

Ebopiprant is under investigation in clinical trial NCT03369262 (Poc Study of OBE022 in Threatened Preterm Labour).

Kategori:
Sulfur CompoundsThiazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ebselen DB12610
small molecule | CAS: 60940-34-3

Ebselen has been investigated for the treatment and basic science of Meniere's Disease, Type 2 Diabetes Mellitus, and Type 1 Diabetes Mellitus.

Kategori:
Agents that produce hypertensionAnalgesicsAnalgesics, Non-Narcotic +17
Target Protein:
AlbuminLysine-specific demethylase 4ABifunctional epoxide hydrolase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ebvaciclib DB18967
small molecule | CAS: 2185857-97-8

Ebvaciclib is under investigation in clinical trial NCT03519178 (A Study of PF-06873600 in People With Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EC-0652 DB15340
small molecule | CAS: 1025066-50-5

EC-0652 is under investigation in clinical trial NCT02202447 (Phase 1 of EC1169 In Patients With Recurrent MCRPC).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ecabet DB05265
small molecule | CAS: 33159-27-2

Ecabet is a prescription eye drop for the treatment of dry eye syndrome. Ecabet represents a new class of molecules that increases the quantity and quality of mucin produced by conjunctival goblet cells and corneal epithelia. Mucin is a glycoprotein component…

Kategori:
Anti-Infective AgentsAnti-Ulcer AgentsAnticarcinogenic Agents +10
Target Protein:
Urease subunit alphaNADPH oxidase organizer 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ecallantide Approved DB05311
biotech | CAS: 460738-38-9

Ecallantide is a potent and selective human plasma kallikrein inhibitor that is indicated for the symptomatic treatment of hereditary angioedema. Ecallantide is a recombinant 60-amino-acid protein produced in _Pichia pastoris_ yeast cells that contains three …

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +10
Target Protein:
Plasma kallikrein
Waktu ParuhFollowing subcutane…
Vol. DistribusiThe volume of distr…
KlirensPlasma clearance wa…
Genetik -
Ecamsule Approved DB09534
small molecule | CAS: 92761-26-7

Ecamsule is an organic compound which is added to many sunscreens to filter out UVA rays. It is a benzylidene camphor derivative, many of which are known for their excellent photostability. Ecamsule has been approved for use in the U.S. since 2006, but only a…

Kategori:
AcidsAcids, NoncarboxylicBicyclic Monoterpenes +12
Waktu ParuhEcamsule is not abs…
Vol. DistribusiEcamsule is intende…
KlirensEcamsule is used to…
Genetik -
Echinacea Approved DB14240
biotech

Deskripsi belum tersedia.

Kategori:
Cytochrome P-450 CYP3A InducersCytochrome P-450 CYP3A4 InducersCytochrome P-450 CYP3A4 Inducers (moderate) +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Echinacea angustifolia root Approved DB14237
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Echinacea purpurea Approved DB14239
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsAsteraceaeBiological Products +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsAsteraceaeBiological Products +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Echinacoside DB15488
small molecule | CAS: 82854-37-3

Echinacoside is a phenylethanoid glycoside isolated from _Echinacea angustifolia_ in 1950, and currently being investigated for the treatment of Parkinson's, Alzheimer's, atherosclerosis, osteoporosis, acute colitis, wound treatment, and hepatitis.[A184577] E…

Kategori:
CarbohydratesCOMT SubstratesHerbs and Natural Products
Target Protein:
Growth hormone secretagogue receptor type 1Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Echinomycin DB15582
small molecule | CAS: 512-64-1

Echinomycin is a cytotoxic polypeptide quinoxaline antibiotic isolated from _Streptomyces echinatus_ that binds to DNA and inhibits RNA synthesis.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Echothiophate Approved DB01057
small molecule | CAS: 6736-03-4

A potent, long-acting irreversible cholinesterase inhibitor used as an ocular hypertensive in the treatment of glaucoma. Occasionally used for accomodative esotropia.

Kategori:
Antiglaucoma Preparations and MioticsAutonomic AgentsCholinergic Agents +15
Target Protein:
CholinesteraseAcetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ecklonia cava DB19252
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Ecnoglutide DB19019
biotech | CAS: 2459531-73-6

Ecnoglutide is under investigation in clinical trial NCT05813795 (A Phase 3 Study to Evaluate the Efficacy of XW003 in Adults With Overweight or Obesity).

Waktu Paruh-
Vol. Distribusi-
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Econazole Approved DB01127
small molecule | CAS: 27220-47-9

A broad spectrum antimycotic with some action against Gram positive bacteria. It is used topically in dermatomycoses also orally and parenterally.

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +21
Target Protein:
Lanosterol 14-alpha demethylaseNuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ecopipam DB12273
small molecule | CAS: 112108-01-7

Ecopipam has been used in trials studying the treatment of Tourette's Syndrome, Lesch-Nyhan Disease, Pathological Gambling, and Self-injurious Behavior.

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +7
Target Protein:
D(1A) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ecraprost DB16148
small molecule | CAS: 136892-64-3

Ecraprost is under investigation in clinical trial NCT00059657 (Efficacy/safety of Ecraprost in Lipid Emulsion for Treatment of Critical Leg Ischemia Due to Peripheral Arterial Disease).

Kategori:
AutacoidsBiological FactorsEicosanoids +5
Target Protein:
Prostaglandin E2 receptor EP1 subtype
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ECT204 DB18605
biotech

ECT204 is an autologous T-cell therapy whereby T cells are genetically modified to target tumor-specific antigens.

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Ectoine DB19171
small molecule | CAS: 96702-03-3

Ectoine is under investigation in clinical trial NCT03186755 (Clinical Evaluation of Hylo-dual Versus Patanol in Children With Seasonal Allergic Conjunctivitis).

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Waktu Paruh-
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Genetik -
Menampilkan 5601–5650 dari 14361
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