Hasil Filter

15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (15718)

Halaman 113 / 315
Dexelvucitabine DB12470
small molecule | CAS: 134379-77-4

Dexelvucitabine has been used in trials studying the treatment of HIV Infections and Human Immunodeficiency Virus.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +13
Target Protein:
Reverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexepicatechin DB19253
small molecule | CAS: 35323-91-2

Dexepicatechin is under investigation in clinical trial NCT02964377 (Plus Epicatechin Duchenne Muscular Dystrophy in Non-ambulatory Adolescents).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexetimide DB08997
small molecule | CAS: 21888-98-2

A muscarinic antagonist that has been used to treat neuroleptic-induced parkinsonism. Benzetimide is the (-)-enantimorph of dexetimide.

Kategori:
Agents producing tachycardiaAnti-Dyskinesia AgentsAnti-Parkinson Drugs +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexfenfluramine Approved DB01191
small molecule | CAS: 3239-44-9

Dexfenfluramine, also marketed under the name Redux, is a serotoninergic anorectic drug. For a fairly limited time during the middle of the nineties, the US FDA had approved it for use in managing weight loss. However, following multiple concerns about the ca…

Kategori:
Alimentary Tract and MetabolismAminesAntidepressive Agents +17
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 2C
Waktu Paruh17-20 hours
Vol. Distribusi-
Klirens-
Genetik -
Dexfosfoserine DB04522
small molecule | CAS: 407-41-0

The phosphoric acid ester of serine.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +1
Target Protein:
3-phosphoinositide-dependent protein kinase 1Glycogen phosphorylase, muscle formProtein kinase C theta type +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexibuprofen Approved DB09213
small molecule | CAS: 51146-56-6

Dexibuprofen, S(+)-ibuprofen, is a non-steroidal anti-inflammatory drug (NSAID). It is a pharmacologically effective enantiomer of racemic ibuprofen that differs in physicochemical properties. It is proposed to be more pharmacologically active and tolerable w…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Apoptosis regulator Bcl-2 +9
Waktu ParuhOral tablets contai…
Vol. DistribusiFor more informatio…
KlirensFor more informatio…
Genetik -
small molecule | CAS: 1620401-56-0

Dexisometheptene mucate is under investigation in clinical trial NCT02423408 (Safety and Efficacy Study of TNX-201 Capsules for Treatment of Single Tension-type Headache).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexketoprofen Approved DB09214
small molecule | CAS: 22161-81-5

Dexketoprofen is a non-steroidal anti-inflammatory drug. It is available in the various countries in Europe, Asia and Latin America. It has analgesic, antipyretic and anti-inflammatory properties [L1298].

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +23
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh1.65 h [L1299]
Vol. Distribusi<0.25 L/kg [L1299]
KlirensMainly cleared via …
Genetik -
Dexlansoprazole Approved DB05351
small molecule | CAS: 138530-94-6

Dexlansoprazole is a new-generation proton pump inhibitor (PPI) used for the management of symptoms associated with gastroesophageal reflux disease (GERD) and erosive esophagitis. Dexlansoprazole is the R-enantiomer of [DB00448], which is composed of a racemi…

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcid ReducersAlimentary Tract and Metabolism +20
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit betaN(G),N(G)-dimethylarginine dimethylaminohydrolase 1
Waktu ParuhDexlansoprazole is …
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik -
Dexloxiglumide DB04856
small molecule | CAS: 119817-90-2

Dexloxiglumide is a selective cholecystokinin type A (CCKA) receptor antagonist in phase III testing by Rottapharm in Europe only, as U.S. trials have been discontinued. As the D-isomer of loxiglumide, it retains all pharmacological properties of loxiglumide …

Kategori:
Acids, AcyclicCytochrome P-450 CYP2B6 SubstratesCytochrome P-450 CYP2C9 Inhibitors +12
Target Protein:
Gastrin/cholecystokinin type B receptorCholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexmecamylamine DB11807
small molecule | CAS: 107538-05-6

Dexmecamylamine has been used in trials studying the basic science and treatment of Patients, Depression, Drug Abuse, Pharmacokinetics, and Renal Impairment, among others.

Kategori:
Autonomic Ganglionic BlockerDecreased Autonomic Ganglionic Activity
Target Protein:
Neuronal acetylcholine receptor subunit beta-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexmedetomidine Approved DB00633
small molecule | CAS: 113775-47-6

An agonist of receptors, adrenergic alpha-2 that is used in veterinary medicine for its analgesic and sedative properties. It is the racemate of dexmedetomidine.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +28
Target Protein:
Alpha-2A adrenergic receptor
Waktu Paruh2 hours
Vol. Distribusi* 118 L
Klirens* 39 L/h [Healthy v…
Genetik -
Dexmethylphenidate Approved DB06701
small molecule | CAS: 40431-64-9

Dexmethylphenidate is the dextrorotary form of methylphenidate introduced in 2002[A177181]. It is a norepinephrine-dopamine reuptake inhibitor (NDRI) and thus a psychostimulant[A177193]. It is used for treatment of Attention Deficit Hyperactivity Disorder (AD…

Kategori:
Agents that produce hypertensionAntidepressive AgentsCentral Nervous System Agents +19
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu ParuhThe mean terminal h…
Vol. Distribusi2.65L/kg when admin…
Klirens0.40L/hr/kg followi…
Genetik -
Dexniguldipine DB14068
small molecule | CAS: 120054-86-6

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +10
Target Protein:
Phosphatidylcholine translocator ABCB4ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexpanthenol Approved DB09357
small molecule | CAS: 81-13-0

Dexpanthenol is an alcohol derivative of pantothenic acid, a component of the B complex vitamins and an essential component of a normally functioning epithelium. Dexpanthenol is enzymatically cleaved to form pantothenic acid, which is an essential component o…

Kategori:
AlanineAlimentary Tract and MetabolismAmino Acids +13
Waktu ParuhHalf life have not …
Vol. DistribusiDexpanthenol is rea…
Klirens-
Genetik -
Dexpramipexole DB15130
small molecule | CAS: 104632-28-2

Dexpramipexole is under investigation in clinical trial NCT01511029 (Study to Evaluate the QTC Interval in Healthy Volunteers Dosed With Dexpramipexole (QTC = Electrocardiogram (ECG) Interval Measured From the Onset of the QRS Complex to the End of the T Wave…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +12
Target Protein:
Interleukin-4Interleukin-13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexpropranolol DB03322
small molecule | CAS: 5051-22-9

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexrabeprazole DB13762
small molecule | CAS: 177795-60-7

Deskripsi belum tersedia.

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcid ReducersAlimentary Tract and Metabolism +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexrazoxane Approved DB00380
small molecule | CAS: 24584-09-6

An antimitotic agent with immunosuppressive properties. Dexrazoxane, the (+)-enantiomorph of razoxane, provides cardioprotection against anthracycline toxicity. It appears to inhibit formation of a toxic iron-anthracycline complex. [PubChem] The Food and Dru…

Kategori:
Cardiotonic AgentsCardiovascular AgentsCompounds used in a research, industrial, or household setting +12
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh2.5 hours
Vol. Distribusi* 9 to 22.6 L/m^2
Klirens* 7.88 L/h/m2 [dose…
Genetik -
Dextilidine DB16731
small molecule | CAS: 32447-90-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextran Approved DB09255
small molecule | CAS: 9004-54-0

Dextran is a polysaccharide that differs from others in that its glucose units are joined together 1:6 glucoside links. The main chain of glucose has short branches at frequent intervals which are probably joined by 1:3 and 1:4 glucoside links. The chains can…

Kategori:
AnticoagulantsBiopolymersBlood and Blood Forming Organs +16
Waktu ParuhThe elimination hal…
Vol. DistribusiThe reported volume…
Klirens-
Genetik -
Dextran 1 DB17818
small molecule

Deskripsi belum tersedia.

Kategori:
BiopolymersCarbohydratesGlucans +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextranomer DB13560
small molecule | CAS: 56087-11-7

Deskripsi belum tersedia.

Kategori:
BiopolymersCarbohydratesCicatrizants +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 142985-55-5

Deskripsi belum tersedia.

Kategori:
BiopolymersCarbohydratesDietary Carbohydrates +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextroamphetamine Approved DB01576
small molecule | CAS: 51-64-9

Dextroamphetamine is the dextrorotatory enantiomer of amphetamine[A2505]. Dextroamphetamine was approved by the FDA in 2001 for the treatment of attention deficit hyperactivity disorder[L6010,Label].

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +19
Target Protein:
Synaptic vesicular amine transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +3
Waktu Paruh11.75 hours.[Label]…
Vol. Distribusi195L.[A177247]
Klirens17L/h.[A177247]
Genetik -
Dextromethadone DB15198
small molecule | CAS: 5653-80-5

Dextromethadone is under investigation in clinical trial NCT00588640 (Study of D-Methadone in Patients With Chronic Pain).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextromethorphan Approved DB00514
small molecule | CAS: 125-71-3

Dextromethorphan is a levorphanol derivative and codeine analog commonly used as a cough suppressant and also a drug of abuse.[A215412] Although similar in structure to other opioids, it has minimal interaction with opioid receptors.[A215412] Dextromethorp…

Kategori:
AlkaloidsAnticholinergic AgentsAntidepressive Agents +37
Target Protein:
Sigma non-opioid intracellular receptor 1AromataseGlutamate receptor ionotropic, NMDA 3A +13
Gen Terkait:
CYP2D6 CYP2D6
Waktu ParuhDextromethorphan ha…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik 2 Varian
Dextromoramide DB01529
small molecule | CAS: 357-56-2

An opioid analgesic structurally related to methadone and used in the treatment of severe pain. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1070)

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextrorphan DB14682
small molecule | CAS: 125-73-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsCentral Nervous System AgentsCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dextrose, unspecified form Approved DB09341
small molecule

Glucose is a simple sugar (monosaccharide) generated during phosynthesis involving water, carbon and sunlight in plants. It is produced in humans via hepatic gluconeogenesis and breakdown of polymeric glucose forms (glycogenolysis). It circulates in human cir…

Kategori:
Caloric AgentsCardiac FunctionCompounds used in a research, industrial, or household setting +4
Waktu ParuhThe approximate hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean metabolic …
Genetik -
Dextrothyroxine Approved DB00509
small molecule | CAS: 51-49-0

The major hormone derived from the thyroid gland. Thyroxine is synthesized via the iodination of tyrosines (monoiodotyrosine) and the coupling of iodotyrosines (diiodotyrosine) in the thyroglobulin. Thyroxine is released from thyroglobulin by proteolysis and …

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +5
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor betaThyroid peroxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexverapamil DB14063
small molecule | CAS: 38321-02-7

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAminesAntiarrhythmic agents +14
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dezamizumab DB15153
biotech | CAS: 1662664-56-3

Dezamizumab is under investigation in clinical trial NCT03417830 (Biodistribution of 89Zirconium-labelled GSK2398852 Using PET Imaging).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dezapelisib DB16137
small molecule | CAS: 1262440-25-4

Dezapelisib is under investigation in clinical trial NCT02456675 (INCB040093 and INCB040093 Combined With Itacitinib (INCB039110) in Relapsed/refractory Hodgkin Lymphoma).

Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dezocine Approved DB01209
small molecule | CAS: 53648-55-8

Dezocine is a partial opiate drug and is used for pain management. Dezocine is a very effective alternative to fentanyl when administered during outpatient laparoscopy, although is associated with an increased incidence of postoperative nausea.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +8
Target Protein:
Mu-type opioid receptorKappa-type opioid receptor
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
DF-1001 DB18231
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DFV890 DB16461
small molecule

DFV890 is under investigation in multiple clinical trials for its efficacy, safety, and tolerability across various conditions: NCT06031844 (coronary heart disease with elevated hsCRP), NCT04886258 (symptomatic knee osteoarthritis), NCT06097663 (coronary hear…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DG031 DB04929
small molecule

DG031, deCODE genetics's lead compound, is being developed for the prevention of myocardial infarction, or heart attack.

Target Protein:
Arachidonate 5-lipoxygenase-activating protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DG041 DB05027
small molecule

DG041 is a novel, first-in-class, orally-administered small molecule developmented for the prevention of arterial thrombosis and its complications. DG041, an anti-platelet compound, has shown to be a selective and potent antagonist of the EP3 receptor for p…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DG051 DB05177
small molecule

DG051 is a novel small-molecule inhibitor of leukotriene A4 hydrolase (LTA4H), the protein made by one of the genes in the leukotriene pathway that has been shown to link to risk of heart attack. DG051 is designed to decrease risk of heart attack by decreasin…

Target Protein:
Leukotriene A-4 hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1382469-39-7

Di-2-pyridylketone 4-cyclohexyl-4-methyl-3-thiosemicarbazone is under investigation in clinical trial NCT02688101 (Dose-finding and Pharmacokinetic Study of DpC, Administered Orally to Patients With Advanced Solid Tumors).

Kategori:
SemicarbazidesSemicarbazonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DI-87 DB18027
small molecule | CAS: 2107280-55-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
ADP/ATP translocase 1Bactericidal permeability-increasing protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Prosaposin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diacerein Approved DB11994
small molecule | CAS: 13739-02-1

Diacerein is a prodrug which is metabolized to rhein. It is currently approved in France for the treatment of osteoarthritis although the use of diacerein is restricted due to the side effects including severe diarrhea [L780]. Diacerein is under investigation…

Kategori:
AnthracenesAnti-Inflammatory AgentsAntiinflammatory and Antirheumatic Products +12
Target Protein:
Interleukin-1 betaOxysterols receptor LXR-alphaOxysterols receptor LXR-beta +7
Waktu Paruh4-10h [A19300].
Vol. Distribusi15-60L [A19300].
KlirensTotal CL is 1.5L/h …
Genetik -
Diacetyl benzoyl lathyrol Approved DB11260
small molecule | CAS: 218916-52-0

Diacetyl benzoyl lathyrol is an active ingredient in whitening creams. It is also reported to be a skin conditioning agent.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingPigments, Biological +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Transferon is comprised of several peptides mixed from human dialyzable leucocyte extracts and acts as an immunomodulator. It is thought to have widespread effects on the immune system, and effective in treating infections and immunological issues.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Trypsin-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5601–5650 dari 15718
Sebelumnya Halaman 113 / 315 Berikutnya