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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Halaman 112 / 315
Descartes-30 DB16361
biotech

Descartes-30 is an RNA-engineered off-the-shelf allogeneic mesenchymal stem cell (MSC) product developed by Cartesian Therapeutics.[L27531] The RNA-engineering is performed with Cartesian Therapeutics’ proprietary RNA Armory which is a platform that activates…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deserpidine Approved DB01089
small molecule | CAS: 131-01-1

Deserpidine is an ester alkaloid drug isolated from Rauwolfia canescens (family Apocynaceae) with antipsychotic and antihypertensive properties that has been used for the control of high blood pressure and for the relief of psychotic behavior.

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +8
Target Protein:
Synaptic vesicular amine transporterAngiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desfesoterodine DB15578
small molecule | CAS: 207679-81-0

Desfesoterodine is a metabolite of [tolterodine].

Kategori:
Drugs for Urinary Frequency and IncontinenceGenito Urinary System and Sex HormonesUrologicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desflurane Approved DB01189
small molecule | CAS: 57041-67-5

Desflurane, or I-653, a a volatile anesthetic that is more rapidly cleared and less metabolized than previous inhaled anesthetics such as [methoxyflurane], [sevoflurane], [enflurane], or [isoflurane].[A226390,A39015,A226893]. It was developed in the late 1980…

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +14
Target Protein:
GABA(A) ReceptorGlycine receptor subunit alpha-1Glutamate receptor 1 +4
Waktu ParuhDesflurane has a te…
Vol. DistribusiDesflurane has a me…
KlirensA 26 g dose of desf…
Genetik -
Desidustat DB16135
small molecule | CAS: 1616690-16-4

Desidustat is under investigation in clinical trial NCT04012957 (Desidustat in the Treatment of Anemia in CKD).

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desipramine Approved DB01151
small molecule | CAS: 50-47-5

Desipramine hydrochloride is a dibenzazepine-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individuals, de…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +52
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +14
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +4
Waktu Paruh7-60+ hours; 70% el…
Vol. Distribusi-
Klirens-
Genetik 7 Varian
Desirudin Approved DB11095
biotech | CAS: 120993-53-5

Desirudin is a direct inhibitor of human thrombin. It has a protein structure that is similar to that of hirudin, the naturally occurring anticoagulant present in the peripharyngeal glands in the medicinal leech, Hirudo medicinalis. Hirudin is a single polype…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Waktu Paruh~2 hours.
Vol. Distribusi0.25 L/kg.
Klirens1.5 to 2.7 mL/min/k…
Genetik -
Deslanoside Approved DB01078
small molecule | CAS: 17598-65-1

Deacetyllanatoside C. A cardiotonic glycoside from the leaves of Digitalis lanata.

Kategori:
Antiarrhythmic agentsCarbohydratesCardanolides +13
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh36 hours
Vol. Distribusi-
Klirens-
Genetik -
Desloratadine Approved DB00967
small molecule | CAS: 100643-71-8

Desloratadine is a second generation, tricyclic antihistamine that which has a selective and peripheral H1-antagonist action. It is the active descarboethoxy metabolite of loratidine (a second generation histamine). Desloratidine has a long-lasting effect and…

Kategori:
Anticholinergic AgentsAntihistamines for Systemic UseBenzocycloheptenes +13
Target Protein:
Histamine H1 receptor
Waktu ParuhDesloratadine has a…
Vol. Distribusi-
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Genetik -
Deslorelin DB11510
small molecule | CAS: 57773-65-6

Deslorelin acetate is an injectable gonadotropin releasing hormone super-agonist also known as an LHRH agonist. It stops the production of sex hormones.

Kategori:
Adrenal Cortex HormonesAlcohol Dehydrogenase, antagonists & inhibitorsAmino Acids, Peptides, and Proteins +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desmeninol DB15832
small molecule | CAS: 583-91-5

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13147-09-6

Desmethylprodine, a derivative of meperidine, is an opioid analgesic with the potency of morphine. It has been listed as a Schedule I controlled drug in the United States, and thus is not used clinically. It is known to be a designer drug, synthesized in 1977…

Kategori:
Isonipecotic AcidsPiperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 87857-41-8

Desmethylsertraline is a metabolite of sertraline.

Kategori:
Agents that reduce seizure thresholdAminesNaphthalenes +1
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desmopressin Approved DB00035
small molecule | CAS: 16679-58-6

Desmopressin (dDAVP), a synthetic analogue of 8-arginine vasopressin (ADH), is an antidiuretic peptide drug modified by deamination of 1-cysteine and substitution of 8-L-arginine by 8-D-arginine. ADH is an endogenous pituitary hormone that has a crucial role …

Kategori:
Agents that produce hypertensionAmino Acids, Peptides, and ProteinsAntidiuretic Agents +27
Target Protein:
Oxytocin receptorVasopressin V2 receptorVasopressin V1a receptor +1
Waktu ParuhFollowing an intran…
Vol. DistribusiThe distribution vo…
Klirens-
Genetik -
Desmoteplase DB04925
biotech | CAS: 145137-38-8

Desmoteplase is a chemical in the saliva of vampire bats. It activates plasminogen to the serine protease, plasmin. Plasmin acts by breaking down fibrin blood clots. When a vampire bat bites its victim, it secretes an enzyme that prevents the blood from clott…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBlood Proteins +13
Target Protein:
Plasminogen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desogestrel Approved DB00304
small molecule | CAS: 54024-22-5

Desogestrel, a prodrug, is a third generation progestogen[A176315] and hence, a member of the gonane family which was largely used in Europe before being approved in the US and Canada.[A176339] It was firstly generated from a study that showed that 11-beta an…

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +25
Target Protein:
Progesterone receptorEstrogen receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe apparent volume…
KlirensThe metabolic clear…
Genetik -
Desomorphine DB01531
small molecule | CAS: 427-00-9

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desonide Approved DB01260
small molecule | CAS: 638-94-8

A nonfluorinated corticosteroid anti-inflammatory agent used topically for dermatoses.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +18
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 94087-98-6

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Desoximetasone Approved DB00547
small molecule | CAS: 382-67-2

A topical anti-inflammatory glucocorticoid used in dermatoses, skin allergies, psoriasis, etc.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +14
Target Protein:
Estrogen-related receptor gammaGlucocorticoid receptorSteroid hormone receptor ERR2 +1
Waktu ParuhThe half-life of th…
Vol. Distribusi-
Klirens-
Genetik -
Desoxycorticosterone acetate Approved DB06780
small molecule | CAS: 56-47-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Mineralocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 808-48-0

Desoxycorticosterone pivalate is a mineralocorticoid hormone and an analog of desoxycorticosterone. It is white, odorless, and stable in air. It is practically insoluble in water, sparingly soluble in acetone, slightly soluble in methanol, ether and vegetable…

Kategori:
Adrenal Cortex HormonesCorticosteroidsCytochrome P-450 CYP3A Substrates +10
Target Protein:
Mineralocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desoxycortone DB15972
small molecule | CAS: 64-85-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids for Systemic Use +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desoxyribonuclease Approved DB09551
biotech | CAS: 9003-98-9

Desoxyribonuclease is a crystalline enzyme that aids in the digestion of the thymus nucleic acid. The mechanism of action of the enzyme involves the splitting of thymus nucleic acid into fragments approaching the size of tetranucleotides without the release o…

Kategori:
Blood and Blood Forming OrgansDeoxyribonucleasesEnzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 5863-40-1

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Chloramphenicol acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 101485-50-1

Deskripsi belum tersedia.

Target Protein:
Desvancosaminyl-vancomycin vancosaminetransferasedTDP-epi-vancosaminyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desvenlafaxine Approved DB06700
small molecule | CAS: 93413-62-8

Desvenlafaxine (O-desmethylvenlafaxine) is the 0-demetyhlated active metabolite of [venlafaxine]. Like its parent drug, desvenlafaxine is also an antidepressant belonging to the class of serotonin-norepinephrine reuptake inhibitor (SNRI) class.[A261266,A26126…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlcohols +40
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe steady-state vo…
KlirensFollowing the admin…
Genetik -
Detomidine DB11556
small molecule | CAS: 76631-46-4

Detomidine is an ?2-adrenergic agonist that is used as a horse sedative. Normally, it is administered in the salt form, detomidine hydrochloride. This drug is prescribed by veterinarians and is marketed as _Dormosedan_. Currently, it is only approved by the F…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deucravacitinib Approved DB16650
small molecule | CAS: 1609392-27-9

Deucravacitinib is a novel oral selective tyrosine kinase 2 (TYK2) inhibitor. Unlike other Janus kinase 1/2/3 inhibitors that bind to the conserved active domain of these non-receptor tyrosine kinases, deucravacitinib binds to the regulatory domain of TYK2 wi…

Kategori:
Antineoplastic and Immunomodulating AgentsBCRP/ABCG2 InhibitorsBCRP/ABCG2 Substrates +17
Target Protein:
Non-receptor tyrosine-protein kinase TYK2
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik -
Deucrictibant DB18303
small molecule | CAS: 2340111-58-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1079043-55-2

Deudextromethorphan is under investigation in clinical trial NCT02153502 (Efficacy, Safety, and Tolerability Study of AVP-786 as an Adjunctive Therapy in Patients With Major Depressive Disorder With an Inadequate Response to Antidepressant Treatment).

Target Protein:
Sodium-dependent serotonin transporterSigma non-opioid intracellular receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deudomperidone DB19055
small molecule | CAS: 2121525-08-2

Deudomperidone is under investigation in clinical trial NCT05832151 (A Study to Evaluate the Efficacy and Safety of CIN-102 (Deudomperidone) in Adults With Diabetic Gastroparesis).

Kategori:
Acids, CarbocyclicBenzene DerivativesPharmaceutical Preparations
Waktu Paruh-
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Genetik -
small molecule | CAS: 1404475-07-5

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Deupirfenidone DB19056
small molecule | CAS: 1093951-85-9

Deupirfenidone is under investigation in clinical trial NCT05321420 (LYT-100 in Patients With Idiopathic Pulmonary Fibrosis (IPF)).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deuruxolitinib DB18847
small molecule | CAS: 1513883-39-0

Deuruxolitinib is a deuterated form of [ruxolitinib] that selectively inhibits Janus kinases (JAK) JAK1 and JAK2. Deuteration allows the drug to circumvent extensive oxidative metabolism around the cyclopentyl ring, which increases the duration of the pharmac…

Kategori:
BCRP/ABCG2 InhibitorsBCRP/ABCG2 SubstratesBile Salt Export Pump Inhibitors +12
Target Protein:
Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK1Non-receptor tyrosine-protein kinase TYK2
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
Klirens-
Genetik -
Deutarserine DB19057
small molecule | CAS: 103292-62-2

Deutarserine is under investigation in clinical trial NCT04158687 (A Phase 2 Study to Evaluate the Safety and Efficacy of CTP-692 as an Adjunctive Treatment in Adults With Schizophrenia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deuterium oxide DB19251
small molecule | CAS: 7789-20-0

Deskripsi belum tersedia.

Kategori:
AlkaliesAnionsAntineoplastic Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deutetrabenazine Approved DB12161
small molecule | CAS: 1392826-25-3

Deutetrabenazine is a novel, highly selective vesicular monoamine transporter 2 (VMAT2) inhibitor indicated for the management of chorea associated with Huntington’s disease. It is a hexahydro-dimethoxybenzoquinolizine derivative and a deuterated [DB04844] [A…

Kategori:
Cytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2D6 SubstratesCytochrome P-450 CYP3A Substrates +11
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhThe half-life of to…
Vol. DistribusiThe median volume o…
KlirensIn patients with Hu…
Genetik -
Deutivacaftor DB15141
small molecule | CAS: 1413431-07-8

Deutivacaftor is under investigation in clinical trial NCT03227471 (A Study of VX-445 in Healthy Subjects and Subjects With Cystic Fibrosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2143580-11-2

Devafidugene civaparvovec is an investigational _in vivo_ genome editing product. It uses proprietary zinc finger nucleases (ZFN) that insert a functional copy of the alpha-L-iduronidase (IDUA) enzyme. Developed by Sangamo Therapeutics, Inc., devafidugene civ…

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Devimistat DB12109
small molecule | CAS: 95809-78-2

Devimistat (CPI-613) has been used in trials studying the treatment of Cancer, Lymphoma, Solid Tumors, Advanced Cancer, and Pancreatic Cancer, among others.

Kategori:
Acids, AcyclicAnionsElectrolytes +5
Target Protein:
2-oxoglutarate dehydrogenase complex component E1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexamethasone Approved DB01234
small molecule | CAS: 50-02-2

Dexamethasone, or MK-125, is a corticosteroid fluorinated at position 9 used to treat endocrine, rheumatic, collagen, dermatologic, allergic, ophthalmic, gastrointestinal, respiratory, hematologic, neoplastic, edematous, and other conditions.[L10701] Develope…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents Causing Muscle Toxicity +74
Target Protein:
Glucocorticoid receptorNuclear receptor subfamily 0 group B member 1Annexin A1 +2
Waktu ParuhThe mean terminal h…
Vol. DistribusiA 1.5mg oral dose o…
KlirensA 20mg oral tablet …
Genetik -
Dexamethasone acetate Approved DB14649
small molecule | CAS: 1177-87-3

Commonly known as decadron, dexamethasone acetate is a glucocorticosteroid previously marketed in the USA for the treatment of inflammatory respiratory, allergic, autoimmune, and other conditions.[T797,L10695,L14348] Developed in 1957, dexamethasone is struct…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsBCRP/ABCG2 Inhibitors +38
Target Protein:
Glucocorticoid receptorAnnexin A1Nitric oxide synthase, inducible +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2265-64-7

Dexamethasone isonicotinate is an anti-inflammatory, anti-allergic glucocorticoid that can be administered orally, by inhalation, topically, and parenterally. Its unintended mineralocorticoid action may cause salt and water retention.

Kategori:
Adrenal Cortex HormonesAnti-Allergic AgentsAnti-Inflammatory Agents +25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 16978-57-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsFused-Ring Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14899-36-6

Dexamethasone palmitate is under investigation in clinical trial NCT05693467 (Preemptive Co-infiltration of Dexamethasone Palmitate With Ropivacaine for Postoperative Pain in Major Spinal Surgery).

Kategori:
Fused-Ring CompoundsPregnadienesPregnadienetriols +3
Target Protein:
Steroid hormone receptor ERR1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexanabinol DB06444
small molecule | CAS: 112924-45-5

Deskripsi belum tersedia.

Kategori:
AntiemeticsAutonomic AgentsCannabinoids and similars +11
Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexbrompheniramine Approved DB00405
small molecule | CAS: 132-21-8

Dexbrompheniramine maleate is an antihistamine agent that is used for the treatment of allergic conditions, such as hay fever or urticaria.

Kategori:
Antihistamines for Systemic UseCentral Nervous System DepressantsHistamine Agents +7
Target Protein:
Histamine H1 receptor
Waktu Paruh25 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 25523-97-1

Dexchlorpheniramine is a potent S-enantiomer of chlorpheniramine. The salt form dexchlorpheniramine maleate as the active ingredient is available as a prescription drug indicated for adjunctive therapy for allergic and anaphylactic reactions. It is an antihis…

Kategori:
Agents that reduce seizure thresholdAntihistamines for Systemic UseCytochrome P-450 CYP2D6 Inhibitors +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexchlorpheniramine maleate Approved DB09555
small molecule | CAS: 2438-32-6

Dexchlorpheniramine is the S-enantiomer of chlorpheniramine which is a 1st generation anti-histamine. Dexchlorpheniramine has more pharmacological activity than the R and so is more potent than the racemic mixture.

Kategori:
Agents that reduce seizure thresholdCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +16
Target Protein:
Histamine H1 receptor
Waktu Paruh20-30 h
Vol. Distribusi321L
Klirens9.8L/h
Genetik -
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