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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 111 / 134
Rosoxacin Approved DB00817
small molecule | CAS: 40034-42-2

Rosoxacin is a quinolone derivative antibiotic for the treatment of bacterial infection of respiratory tract, urinary tract, GI, CNS and immuno compromised patients. Rosoxacin is known to be effective against penicillin resistant strains and is a single dose …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +9
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA gyrase subunit B +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Rosuvastatin Approved DB01098
small molecule | CAS: 287714-41-4

Rosuvastatin, also known as the brand name product Crestor, is a lipid-lowering drug that belongs to the statin class of medications, which are used to lower the risk of cardiovascular disease and manage elevated lipid levels by inhibiting the endogenous prod…

Kategori:
Agents Causing Muscle ToxicityAlimentary Tract and MetabolismAmides +32
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-L
Gen Terkait:
KIF6 HMGCR ABCG2
Waktu ParuhThe elimination hal…
Vol. DistribusiRosuvastatin underg…
Klirens-
Genetik 3 Varian
Rotavirus vaccine Approved DB10276
biotech

Rotavirus commonly infects children and infants causing severe diarrhea and vomiting leading to potentially fatal dehydration.[L1117] Two rotavirus vaccines are available for the prevention of rotavirus gastroenteritis, Rotateq and Rotarix. Rotateq is a live …

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBiological Products +6
Waktu ParuhThe median duration…
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Genetik -
Rotenone DB11457
small molecule | CAS: 83-79-4

Rotenone is an isoflavone compound that naturally occurs in the jicama vine plant as well as many Fabaceae plants. It has broad spectrum insecticide and pesticide activity and is also toxic to fish.

Kategori:
AgrochemicalsBenzopyransChromones +10
Waktu Paruh-
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Rotigaptide DB13067
small molecule | CAS: 355151-12-1

Rotigaptide is under investigation for the basic science of Heart Disease and Vascular Disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
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Genetik -
Rotigotine Approved DB05271
small molecule | CAS: 99755-59-6

Rotigotine (Neupro) is a non-ergoline dopamine agonist indicated for the treatment of Parkinson's disease (PD) and restless legs syndrome (RLS) in Europe and the United States. It is formulated as a once-daily transdermal patch which provides a slow and const…

Kategori:
Agents that produce hypertensionAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +23
Target Protein:
D(3) dopamine receptorD(4) dopamine receptorD(2) dopamine receptor +4
Waktu ParuhAfter removal of th…
Vol. DistribusiThe weight normaliz…
Klirens-
Genetik -
Rovaleucel DB18691
biotech

Rovaleucel is an EBV-specific autologous T-cell therapy under investigation for the treatment of EBV-positive cancers.

Waktu Paruh-
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Roxadustat Approved DB04847
small molecule | CAS: 808118-40-3

Roxadustat is a first-in-class hypoxia-inducible factor prolyl hydroxylase inhibitor used to treat anemia associated with chronic kidney disease. It works by reducing the breakdown of the hypoxia-inducible factor (HIF), which is a transcription factor that st…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntianemic Preparations +10
Target Protein:
Egl nine homolog 1Prolyl hydroxylase EGLN2Prolyl hydroxylase EGLN3
Waktu ParuhThe mean effective …
Vol. DistribusiThe blood-to-plasma…
KlirensThe apparent total …
Genetik -
Roxarsone DB11458
small molecule | CAS: 121-19-7

Roxarsone is an organoarsenic molecule added to poultry feed. The addition of this compound to poultry feed improves weight gain and feed efficiency as well as prevent the growth of coccidian parasites. The drug is also approved in the United States for use i…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 78628-28-1

Roxatidine acetate is a specific and competitive H2 receptor antagonist. It is currently approved in South Africa under the tradename Roxit.

Kategori:
Acid ReducersAlimentary Tract and MetabolismAnti-Ulcer Agents +8
Target Protein:
Histamine H2 receptor
Waktu Paruh5-6 hours
Vol. Distribusi-
Klirens-
Genetik -
Roxithromycin Approved DB00778
small molecule | CAS: 80214-83-1

Roxithromycin is a semi-synthethic macrolide antibiotic that is structurally and pharmacologically similar to [erythromycin], [azithromycin], or [clarithromycin]. It was shown to be more effective against certain Gram-negative bacteria, particularly _Legionel…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +19
Target Protein:
50S ribosomal protein L10ATP-dependent translocase ABCB1
Waktu Paruh12 hours
Vol. Distribusi-
Klirens-
Genetik -
Rozanolixizumab Approved DB14919
biotech | CAS: 1584645-37-3

Rozanolixizumab is a humanized high-affinity anti-human neonatal Fc receptor (FcRn) monoclonal antibody (IgG4P) targeting the immunoglobulin G (IgG). Rozonolixizumab itself is an IgG4P, an inactive isotype, to reduce the likelihood of unwanted chain exchange.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
IgG receptor FcRn large subunit p51
Waktu Paruh-
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Rozibafusp Alfa DB19233
biotech | CAS: 2143449-47-0

Rozibafusp Alfa is under investigation in clinical trial NCT04058028 (Efficacy and Safety of AMG 570 in Subjects With Active Systemic Lupus Erythematosus (SLE)).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
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Rozrolimupab DB05209
biotech | CAS: 909402-77-3

Rozrolimupab is a recombinant polyclonal antibody consisting of 25 different anti-Rhesus D (RhD) antibodies to replace existing anti-RhD hyperimmune immunoglobulins for the treatment of Idiopathic Thrombocytopenic Purpura (ITP) and the prevention of Hemolytic…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Target Protein:
Rhesus blood group D antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RP-72 DB17156
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
RP-A501 DB17647
biotech

RP-A501 is a gene therapy product consisting of a recombinant adeno-associated virus serotype 9 (rAAV9) capsid containing the human LAMP2B transgene (AAV9:LAMP2B), which encodes lysosome-associated membrane protein 2 (LAMP-2). It is being investigated for Dan…

Waktu Paruh-
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RP-A601 DB18339
biotech

RP-A601 is an adeno-associated virus serotype rhesus 10 vector expressing the human galactocerebrosidase (GALC) gene

Waktu Paruh-
Vol. Distribusi-
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Genetik -
RR001 DB17369
biotech

RR001 is an investigational gene therapy consisting of autologous human adipose perivascular stromal cells genetically modified to secrete soluble tumour necrosis factor-related apoptosis-inducing ligand (AD-PC sTRAIL).[L44276]

Waktu Paruh-
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RRx-001 DB12060
small molecule | CAS: 925206-65-1

RRx-001 has been used in trials studying the treatment of Lymphomas, Brain Metastases, Cholangiocarcinoma, Colorectal Neoplasms, and Malignant Solid Tumor, among others.

Kategori:
AzetinesCarbon Radioisotopes
Waktu Paruh-
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Genetik -
rsPSMA Vaccine Approved DB06361
biotech

Prostate-specific membrane antigen (PSMA) is an ?100 kDa transmembrane glycoprotein that is abundantly and preferentially expressed in prostate cancer, including recurrent and hormone-refractory cases. rsPSMA Vaccine is a subunit vaccine based on a novel rsPS…

Waktu Paruh-
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RST-001 DB17843
biotech

RST-001 is a non-replicating recombinant adeno-associated virus vector containing a fragment of the gene encoding channel rhodopsin-2 protein.

Waktu Paruh-
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RTP-801i DB06048
biotech

RTP-801i is an siRNA drug candidate designed to inhibit the expression of the hypoxia-inducible gene RTP801. The proposed primary indication for RTP-801i is the treatment of patients with neovascular (wet) Age-related Macular Degeneration (AMD or ARMD).

Kategori:
Antisense Elements (Genetics)Nucleic AcidsNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
DNA damage-inducible transcript 4 protein
Waktu Paruh-
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Genetik -
RU82197 DB03268
small molecule

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
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Genetik -
RU85053 DB03712
small molecule

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rubella virus vaccine Approved DB10317
biotech

Rubella virus vaccine is a live attenuated virus vaccine for active immunization against rubella (German measles) that is subcutaneously administered. It is prepared from RA 27/3 strain of live attenuated rubella virus. Rubella is a common childhood disease, …

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseLive Attenuated Rubella Virus Vaccine +5
Waktu Paruh-
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Genetik -
Rubitecan DB06159
small molecule | CAS: 91421-42-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ruboxistaurin DB11829
small molecule | CAS: 169939-94-0

Ruboxistaurin has been investigated for the basic science of Type 2 Diabetes Mellitus and Type 1 Diabetes Mellitus.

Kategori:
Acids, AcyclicDicarboxylic AcidsEnzyme Inhibitors +4
Target Protein:
Peptide deformylase, mitochondrialProtein kinase C beta type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rufloxacin DB13772
small molecule | CAS: 101363-10-4

Rufloxacin is a quinolone antibiotic. [A31894]

Kategori:
4-QuinolonesAnti-Bacterial AgentsAntibacterials for Systemic Use +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rugonersen DB18662
biotech | CAS: 2591587-57-2

Rugonersen is a locked nucleic acid antisense oligonucleotide under investigation for the treatment of Angelman Syndrome.

Waktu Paruh-
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Rulonilimab DB18922
biotech | CAS: 2417124-95-7

Rulonilimab is under investigation in clinical trial NCT05408221 (The Efficacy and Safety of Rulonilimab in Combination With Lenvatinib in Hepatocellular Carcinoma).

Waktu Paruh-
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Genetik -
biotech

Rumex salicifolius var. mexicanus pollen is the pollen of the Rumex salicifolius var. mexicanus plant. Rumex salicifolius var. mexicanus pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Runcaciguat DB16700
small molecule | CAS: 1402936-61-1

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCycloparaffins
Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Rurioctocog alfa pegol Approved DB16007
biotech | CAS: 1417412-83-9

Rurioctocog alfa pegol is a pegylated recombinant human coagulation factor VIII or antihemophilic factor. Factor VIII is an essential protein involved in normal blood clotting; thus, a deficient level of functional factor VIII is associated with an elevated r…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +9
Target Protein:
von Willebrand factorCoagulation factor VIII
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Rusfertide DB17724
biotech | CAS: 1628323-80-7

Rusfertide is a hepcidin mimetic currently being developed by Protagonist Therapeutics for the treatment of polycythemia vera and beta-thalassemia.

Waktu Paruh-
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RUTI® Vaccine DB15853
biotech

The RUTI® Vaccine contains fragmented, purified and liposomed heat-inactivated Mycobacterium tuberculosis bacilli. The vaccine has demonstrated a reasonable safety profile and potent stimulation of the immune response against tuberculosis. Much like the BCG v…

Waktu Paruh-
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Genetik -
Ruxolitinib Approved DB08877
small molecule | CAS: 941678-49-5

Ruxolitinib, formerly known as INCB018424 or INC424, is an anticancer drug and a Janus kinase (JAK) inhibitor. It is a potent and selective inhibitor of JAK1 and JAK2,[A229698] which are tyrosine kinases involved in cytokine signalling and hematopoiesis.[A745…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
Urokinase plasminogen activator surface receptorTyrosine-protein kinase JAK2Tyrosine-protein kinase JAK1 +2
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensRuxolitinib clearan…
Genetik -
Ruzinurad DB19209
small molecule | CAS: 1638327-48-6

Ruzinurad is under investigation in clinical trial NCT04956432 (A Multicentre, Randomized, Double-blind, Allopurinol Controlled Study to Evaluate the Efficacy and Safety of SHR4640 in Subjects With Gout).

Kategori:
CycloparaffinsHeterocyclic Compounds, Fused-Ring
Target Protein:
Solute carrier family 22 member 12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Hydroxyacylglutathione hydrolase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Lactoylglutathione lyase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2986-20-1

S-Ethylisothiourea is a nitric oxide synthase inhibitor.

Kategori:
AmidesCardiovascular AgentsCentral Nervous System Agents +7
Target Protein:
Nitric oxide synthase, inducibleNitric oxide synthase 3Nitric oxide synthase oxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

S-hydroxycysteine is a solid. This compound belongs to the alpha amino acids and derivatives. These are amino acids in which the amino group is attached to the carbon atom immediately adjacent to the carboxylate group (alpha carbon), or a derivative thereof. …

Target Protein:
Tyrosine-protein phosphatase non-receptor type 1M-phase inducer phosphatase 2Proto-oncogene tyrosine-protein kinase Src +8
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 2922-56-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Glutathione S-transferase Mu 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 57564-91-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAnti-Infective Agents +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsGlutathione Transferase, antagonists & inhibitorsOligopeptides +1
Target Protein:
Glutathione S-transferase Mu 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1637-71-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sabarubicin DB12410
small molecule | CAS: 211100-13-9

Sabarubicin has been used in trials studying the treatment of Prostate Cancer, Testicular Germ Cell Tumor, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
AnthracyclinesCarbohydratesGlycosides +3
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sabatolimab DB16322
biotech | CAS: 2252262-24-9

Sabatolimab is under investigation in clinical trial NCT03946670 (A Study of MBG453 in Combination With Hypomethylating Agents in Subjects With IPSS-R Intermediate, High or Very High Risk Myelodysplastic Syndrome (MDS).).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Sabestomig DB19326
biotech | CAS: 2648346-74-9

Sabestomig is under investigation in clinical trial NCT05216835 (Safety and Preliminary Efficacy Assessment of AZD7789 in Patients With Relapsed or Refractory Classical Hodgkin Lymphoma).

Waktu Paruh-
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Sabirnetug DB19438
biotech | CAS: 2747959-38-0

Sabirnetug is under investigation in clinical trial NCT06335173 (A Study to Evaluate Efficacy and Safety of Intravenous Sabirnetug in Participants With Early Alzheimer's Disease (ALTITUDE-AD)).

Waktu Paruh-
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Genetik -
Sacituzumab govitecan Approved DB12893
biotech | CAS: 1491917-83-9

Metastatic triple-negative breast cancer (mTNBC) is an aggressive form of breast cancer with limited treatment options involving cytotoxic chemotherapy agents.[A193653] Targeted chemotherapy through the application of antibody-conjugated agents (ADCs) is a re…

Kategori:
AlkaloidsAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Tumor-associated calcium signal transducer 2DNA topoisomerase 1Far upstream element-binding protein 1
Waktu ParuhSacituzumab govitec…
Vol. DistribusiSacituzumab govitec…
KlirensSacituzumab govitec…
Genetik -
Menampilkan 5501–5550 dari 6694
Sebelumnya Halaman 111 / 134 Berikutnya