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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
Referensi
11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 111 / 236
Glyburide Approved DB01016
small molecule | CAS: 10238-21-8

Glyburide is a second generation sulfonylurea used to treat patients with diabetes mellitus type II.[L8123] It is typically given to patients who cannot be managed with the standard first line therapy, [metformin].[L8123] Glyburide stimulates insulin secretio…

Kategori:
Alimentary Tract and MetabolismAmidesBCRP/ABCG2 Substrates +28
Target Protein:
ATP-binding cassette sub-family C member 8Sulfonylurea receptor 1, Kir6.2ATP-binding cassette sub-family C member 9 +6
Waktu ParuhElderly patients ha…
Vol. DistribusiElderly patients ha…
KlirensElderly patients ha…
Genetik -
Glycerin Approved DB09462
small molecule | CAS: 56-81-5

A trihydroxy sugar alcohol that is an intermediate in carbohydrate and lipid metabolism.

Kategori:
AlcoholsAlimentary Tract and MetabolismBasic Ointments and Protectants +21
Target Protein:
Peroxisome proliferator-activated receptor deltaGroup IIE secretory phospholipase A2Inositol-3-phosphate synthase 1 +11
Waktu Paruh30 - 45 minutes
Vol. DistribusiGlycerin is distrib…
Klirens-
Genetik -
Glycerol phenylbutyrate Approved DB08909
small molecule | CAS: 611168-24-2

Glycerol phenylbutyrate is a nitrogen-binding agent. Chemically, it is a triglyceride in which three molecules of phenylbutyrate are linked to a glycerol backbone. FDA approved on February 1, 2013.

Kategori:
Acids, CarbocyclicAlcoholsAlimentary Tract and Metabolism +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 614-33-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 27215-38-9

Deskripsi belum tersedia.

Kategori:
Cariostatic AgentsCompounds used in a research, industrial, or household settingFatty Acids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glyceryl monocaprylate Approved DB19362
small molecule | CAS: 26402-26-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsLipids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 31566-31-1

Glycerol monostearate, commonly known as GMS, is the glycerol ester of stearic acid . It is commonly used as an emulsifier in foods.

Kategori:
Lipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycinamide DB03636
small molecule | CAS: 598-41-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Neutrophil collagenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsNucleic Acids, Nucleotides, and Nucleosides +1
Target Protein:
Phosphoribosylglycinamide formyltransferase 2Phosphoribosylglycinamide formyltransferaseTrifunctional purine biosynthetic protein adenosine-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycine Approved DB00145
small molecule | CAS: 56-40-6

A non-essential amino acid. It is found primarily in gelatin and silk fibroin and used therapeutically as a nutrient. It is also a fast inhibitory neurotransmitter.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBlood and Blood Forming Organs +7
Target Protein:
Glutamate receptor ionotropic, NMDA 2A2-amino-3-ketobutyrate coenzyme A ligase, mitochondrial5-aminolevulinate synthase, non-specific, mitochondrial +22
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 640-79-9

A bile salt formed in the liver from chenodeoxycholate and glycine, usually as the sodium salt. It acts as a detergent to solubilize fats for absorption and is itself absorbed. It is a cholagogue and choleretic. [PubChem]

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBile Acids and Salts +12
Target Protein:
7-alpha-hydroxysteroid dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 475-31-0

The glycine conjugate of cholic acid. It acts as a detergent to solubilize fats for absorption and is itself absorbed.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBile Acids and Salts +11
Target Protein:
Gastrotropin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycocyamine DB02751
small molecule | CAS: 352-97-6

Deskripsi belum tersedia.

Kategori:
Affinity LabelsAmino AcidsAmino Acids, Peptides, and Proteins +3
Target Protein:
Guanidinoacetate N-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycol salicylate Approved DB11323
small molecule | CAS: 87-28-5

Glycol salicylate, also known as _2-hydroxyethyl salicylate_, is a benzoate ester formed from the condensation of the carboxy group of salicylic acid with one of the hydroxy groups of ethylene glycol. It is found as an active ingredient and topical analgesic …

Kategori:
Acids, CarbocyclicAnti-Inflammatory AgentsAnti-Inflammatory Agents, Non-Steroidal +5
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhThe serum half-life…
Vol. Distribusi-
Klirens-
Genetik -
GlycoPEG-GCSF DB06022
biotech

GlycoPEG-GCSF is a long-acting GlycoPEGylated granulocyte colony stimulating factor for the treatment of chemotherapy-induced neutropenia.

Kategori:
Pegylated agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycopyrronium Approved DB00986
small molecule | CAS: 740028-90-4

Glycopyrronium, also known as NVA237 or glycopyrrolate, is a racemic mixture of two enantiomers.[L33110] They are both quaternary ammonium compounds and long acting muscarinic antagonists.[L33110] It is one of the most commonly prescribed anticholinergic medi…

Kategori:
Adjuvants, AnesthesiaAdrenergics, InhalantsAgents producing tachycardia +30
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe half life after…
Vol. DistribusiThe mean volume of …
KlirensA 6 µg/kg intraveno…
Genetik -
Glycovir DB13106
small molecule | CAS: 131262-82-3

Glycovir has been used in trials studying the treatment of HIV Infections.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Maltase-glucoamylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
D-alanyl-D-alanine carboxypeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycyltyrosine DB15991
small molecule | CAS: 658-79-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycyrrhiza glabra Approved DB14312
biotech | CAS: 84775-66-6

Glycyrrhiza glabra is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsCell-mediated Immunity +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glycyrrhizic acid Approved DB13751
small molecule | CAS: 1405-86-3

Glycyrrhizic acid is extracted from the root of the licorice plant; _Glycyrrhiza glabra_.[F79] It is a triterpene glycoside with glycyrrhetinic acid that possesses a wide range of pharmacological and biological activities. When extracted from the plant, it ca…

Kategori:
Alimentary Tract and MetabolismAnti-Inflammatory AgentsBile and Liver Therapy +6
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1Tumor necrosis factorCaspase-3 +2
Waktu ParuhDepending on the do…
Vol. DistribusiThe apparent volume…
KlirensThe constant reabso…
Genetik -
Glymidine Approved DB01382
small molecule | CAS: 339-44-6

Glycodiazine is used with diet to lower blood glucose by increasing the secretion of insulin from pancreas and increasing the sensitivity of peripheral tissues to insulin. The mechanism of action of glycodiazine in lowering blood glucose appears to be depende…

Kategori:
Alimentary Tract and MetabolismAmidesBlood Glucose Lowering Agents +7
Target Protein:
ATP-sensitive inward rectifier potassium channel 1ATP-sensitive inward rectifier potassium channel 10ATP-binding cassette sub-family C member 8
Waktu Paruh4 hours.
Vol. Distribusi-
Klirens-
Genetik -
Glyphosate DB04539
small molecule | CAS: 1071-83-6

Deskripsi belum tersedia.

Kategori:
AgrochemicalsAmino AcidsAmino Acids, Peptides, and Proteins +9
Target Protein:
Aromatase3-phosphoshikimate 1-carboxyvinyltransferase3-phosphoshikimate 1-carboxyvinyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glypromate DB05633
small molecule | CAS: 32302-76-4

Neuren Pharmaceuticals was developing Glypromate (glycine-proline glutamate), a naturally occurring small-molecule neuroprotectant derived from IGF-1 which inhibits caspase III dependent apoptosis, for the potential treatment of neurodegenerative diseases by …

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GMA-161 DB15397
biotech | CAS: 946415-70-9

GMA-161 is under investigation in clinical trial NCT00244257 (Safety Study of GMA161 in Patients With Idiopathic Thrombocytopenic Purpura (ITP)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GMI-1359 DB18092
biotech

GMI-1359 is a small molecule, glycomimetic compound with dual inhibitory activity against E-selectin and CXCR4.[A261406]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GMK DB06661
biotech

GMK vaccine (a ganglioside conjugate vaccine coupled to keyhole limpet hemocyanin and formulated with the adjuvant QS-21) for the potential treatment of melanoma

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GO-203-2C DB15008
small molecule | CAS: 1469735-88-3

GO-203-2C is under investigation in clinical trial NCT02204085 (A Phase I/II Trial of the MUC1 Inhibitor, GO-203-2C in Patients With Relapsed or Refractory Acute Myeloid Leukemia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Go-6976 DB17029
small molecule | CAS: 136194-77-9

An inhibitor of calcium-dependent isoforms of protein kinase C.[A253002,A253007]

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingIndoles +1
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Goflikicept DB16396
biotech | CAS: 2416984-26-2

Goflikicept is under investigation in clinical trial NCT04380519 (Study of the Efficacy and Safety of a Single Administration of Olokizumab and RPH-104 With Standard Therapy in Patients With Severe Severe Acute Respiratory Syndrome Coronavirus 2 (Sars-cov-2) …

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Golcadomide DB18115
small molecule | CAS: 2379572-34-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 20681-14-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Goldenseal Approved DB16594
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Golidocitinib DB18057
small molecule | CAS: 2091134-68-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Golimumab Approved DB06674
biotech | CAS: 476181-74-5

Golimumab is a human IgG1? monoclonal antibody derived from immunizing genetically engineered mice with human TNF?. Golimumab binds and inhibits soluble and transmembrane human TNF?. Increased TNF? is associated with chronic inflammation. Thus golimumab is in…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +17
Target Protein:
Tumor necrosis factor
Waktu ParuhGolimumab has a lon…
Vol. DistribusiAfter IV administra…
KlirensAfter one IV dose o…
Genetik -
Golodirsen Approved DB15593
biotech | CAS: 1422959-91-8

Golodirsen is a morpholino antisense oligomer designed to treat about 8% of patients with Duchenne Muscular Dystrophy (DMD). This is an X-linked condition leading to progressive muscle degeneration that begins in early childhood, rendering many patients wheel…

Kategori:
Antisense Elements (Genetics)Antisense OligonucleotidesCompounds used in a research, industrial, or household setting +10
Target Protein:
Dystrophin
Waktu ParuhIn a pharmacokineti…
Vol. DistribusiThe volume of distr…
KlirensThis drug is rapidl…
Genetik -
Gonadorelin Approved DB00644
biotech | CAS: 33515-09-2

Gonadorelin is another name for gonadotropin-releasing hormone (GnRH). It is a synthetic decapeptide prepared using solid phase peptide synthesis. GnRH is responsible for the release of follicle stimulating hormone and leutinizing hormone from the anterior pi…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsDiagnostic Agents +18
Target Protein:
Gonadotropin-releasing hormone receptorPutative gonadotropin-releasing hormone II receptor
Waktu ParuhVery short, initial…
Vol. Distribusi-
Klirens-
Genetik -
Gondoic acid DB14073
small molecule | CAS: 5561-99-9

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gontivimab DB16179
biotech | CAS: 1257358-38-5

Gontivimab is under investigation in clinical trial NCT03468829 (Efficacy and Safety of ALX-0171 in Adult Hematopoietic Stem Cell Transplant (HSCT) Recipients Who Present With Respiratory Syncytial Virus (RSV) Infection).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntiviral Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gonyautoxin II DB19186
small molecule | CAS: 60508-89-6

Gonyautoxin II is under investigation in clinical trial NCT04799041 (Gonyautoxin 2/3 in the Treatment of Acute Back Pain: A Clinical Proof-of-concept Study).

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ToxinsBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gonyautoxin III DB19187
small molecule | CAS: 60537-65-7

Gonyautoxin III is currently under investigation in clinical trial (Gonyautoxin 2/?3 in the Treatment of Acute Back Pain: A Clinical Proof-of-concept Study) for the treatment of Acute Back Pain.

Kategori:
Bacterial ToxinsBiological FactorsComplex Mixtures +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Goserelin Approved DB00014
small molecule | CAS: 65807-02-5

Goserelin is a synthetic hormone. In men, it stops the production of the hormone testosterone, which may stimulate the growth of cancer cells. In women, goserelin decreases the production of the hormone estradiol (which may stimulate the growth of cancer cell…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsAntineoplastic Agents +22
Target Protein:
Lutropin-choriogonadotropic hormone receptorProgonadoliberin-1Gonadotropin-releasing hormone receptor
Waktu Paruh4-5 hours
Vol. Distribusi* 44.1 ± 13.6 L [su…
Klirens* 121 +/- 42.4 mL/m…
Genetik -
Gosogliptin DB08382
small molecule | CAS: 869490-23-3

Gosogliptin has been used in trials studying the treatment of Renal Insufficiency, Chronic.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDiabetes Mellitus, Type 2, drug therapy +1
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gosuranemab DB15376
biotech | CAS: 1788032-39-2

Gosuranemab is under investigation in clinical trial NCT02460094 (Multiple Ascending Dose Study of Intravenously Administered BMS-986168 (BIIB092) in Patients With Progressive Supranuclear Palsy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gotistobart DB19100
biotech | CAS: 2226344-78-9

Gotistobart is under investigation in clinical trial NCT05671510 (ONC-392 Versus Docetaxel in Metastatic NSCLC That Progressed on PD-1/PD-L1 Inhibitors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GP-100 antigen DB14800
biotech

GP-100 antigen is under investigation in clinical trial NCT00006385 (Vaccine Therapy With or Without Biological Therapy in Treating Patients With Metastatic Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GP2 peptide DB16180
biotech | CAS: 160790-21-6

GP2 peptide is under investigation in clinical trial NCT00524277 (Vaccine Therapy in Treating Patients With Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The gp209-2M antigen is derived from gp209, and has potential immunomodulatory and antineoplastic activities.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gpi-1046 DB01951
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GPI-1485 DB05814
small molecule | CAS: 186268-78-0

GPI 1485 is a product candidate that belongs to a class of small molecule compounds called neuroimmunophilin ligands. In preclinical experiments, neuroimmunophilin ligands have been shown to repair and regenerate damaged nerves without affecting normal, heal…

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 InhibitorsCytochrome P-450 CYP3A4 Inhibitors (strength unknown) +2
Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5501–5550 dari 11793
Sebelumnya Halaman 111 / 236 Berikutnya