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13591

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13591 (100.0%)

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Halaman 111 / 272
biotech | CAS: 2049067-94-7

Efavaleukin alfa is a fusion protein consisting of interleukin mutein fused to the C-terminus of an immunoglobulin G Fc domain by way of a G4S linker. It is under investigation in clinical trial NCT03422627 (Safety and Efficacy of AMG 592 in Subjects With Ste…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efavirenz Approved DB00625
small molecule | CAS: 154598-52-4

Efavirenz (brand names Sustiva® and Stocrin®) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) and is used as part of highly active antiretroviral therapy (HAART) for the treatment of a human immunodeficiency virus (HIV) type 1. For HIV infectio…

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiinfectives for Systemic Use +52
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Gen Terkait:
CYP2B6
Waktu Paruh40-55 hours
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Efbemalenograstim alfa Approved DB18704
biotech | CAS: 2200269-79-8

Efbemalenograstim alfa is a long-acting recombinant fusion protein of granulocyte-colony stimulating factor (G-CSF) due to the addition of the Fc portion of human IgG2, allowing for once-per-cycle administration.[L48852,A262167] As endogenous G-CSF mediates t…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsColony-Stimulating Factors +2
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Efgartigimod alfa Approved DB15270
biotech | CAS: 1821402-21-4

Myasthenia gravis (MG) is an autoimmune disorder characterized by significant muscle weakness - particularly in the eye, throat, and extremities - caused by autoantibodies attacking the neuromuscular junction.[A243759] The production of IgG autoantibodies aga…

Kategori:
AntibodiesAntineoplastic and Immunomodulating AgentsGlobulins +6
Target Protein:
IgG receptor FcRn large subunit p51
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Efinaconazole Approved DB09040
small molecule | CAS: 164650-44-6

Efinaconazole is a 14 alpha-demethylase inhibitor indicated in the treatment of fungal infection of the nail, known as onychomycosis. It was approved for use in Canada and the USA in 2014 and is marketed by Valeant Pharmaceuticals North America LLC under the …

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +4
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylase
Waktu Paruh29.9 hours in healt…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2026634-47-7

Efineptakin alfa (also known as NT-I7) is a long-acting human interleukin-7 (IL-7) fusion protein that promotes T-cell development, contributing to the immune response. Compared to endogenous IL-7, NT-I7 is more stable and potent, has a longer half-life, and …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efinopegdutide DB15077
biotech | CAS: 2055640-93-0

Efinopegdutide is under investigation in clinical trial NCT03606057 (A Study to Investigate the Effect of JNJ-64565111 on Cardiac Repolarization (Corrected QT Interval) Compared With Placebo in Healthy Adults: a Thorough ECG Study Employing Placebo, JNJ-64565…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1635395-27-5

Efizonerimod alfa is under investigation in clinical trial NCT02221960 (A Phase 1 Study to Evaluate MEDI6383 Alone and in Combination With MEDI4736 in Adult Subjects With Select Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eflapegrastim Approved DB15001
biotech | CAS: 1384099-30-2

Febrile neutropenia (FN), defined as the co-occurrence of fever (temperature > 38 ?C) and severe neutropenia (ANC < 500 cells/mm<sup>3</sup>), is a potential side effect of myelosuppressive chemotherapy in which the patient develops an infection during a peri…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +20
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhIn patients with br…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ef…
Genetik -
biotech

Eflepedocokin alfa is a recombinant IL-22-Fc fusion protein manufactured in Chinese hamster ovary cells that is composed of 2 human interleukin 22 (IL-22) molecules linked to an immunoglobulin constant region (IgG2-Fc).[A225706, L27661] It is being developed …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eflornithine Approved DB06243
small molecule | CAS: 70052-12-9

Eflornithine is an irreversible ornithine decarboxylase inhibitor originally developed as a treatment for human African trypanosomiasis.[A262829] Further research has also implicated ornithine decarboxylase in other conditions like facial hirsutism and cancer…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAmino AcidsAmino Acids, Basic +15
Target Protein:
Ornithine decarboxylase
Waktu ParuhThe terminal plasma…
Vol. DistribusiEflornithine volume…
KlirensThe clearance (CL/F…
Genetik -
Efloxate DB13333
small molecule | CAS: 119-41-5

Deskripsi belum tersedia.

Kategori:
BenzopyransCardiac TherapyChromones +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1953227-87-6

Efmarodocokin alfa is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1644543-31-6

Efmitermant alfa, a locally-acting GDF/activin ligand trap, is under investigation in clinical trial NCT03124459 (Study of ACE-083 in Patients With Charcot-marie-tooth Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efmoroctocog alfa Approved DB11607
biotech | CAS: 1270012-79-7

Efmoroctocog alfa is a fully recombinant factor VIII-Fc fusion protein (rFVIIIFc) with an extended half-life compared with conventional factor VIII (FVIII) preparations, including recombinant FVIII (rFVIII) products such as [DB13999][A31551]. It is an antihem…

Kategori:
HemostaticsHuman Antihemophilic Factors
Target Protein:
von Willebrand factor
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Efocipegtrutide DB18194
biotech | CAS: 2513399-19-2

Efocipegtrutide is a long-acting, monomeric peptide triple agonist.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efonidipine DB09235
small molecule | CAS: 111011-63-3

Efonidipine is a calcium channel blocker of the _dihydropyridine class_, commercialized by Shionogi & Co. (Japan). Initially, it was marketed in 1995 under the trade name, _Landel_. The drug has been shown to block T-type in addition to L-type calcium channel…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +22
Target Protein:
Voltage gated L-type calcium channelVoltage-dependent calcium channelVoltage-dependent T-type calcium channel +4
Waktu ParuhThe peak plasma con…
Vol. Distribusi-
Klirens-
Genetik -
Efpeglenatide DB15650
biotech | CAS: 1296200-77-5

Efpeglenatide is under investigation in clinical trial NCT03713684 (Efficacy and Safety of Efpeglenatide Versus Placebo in Patients With Type 2 Diabetes Mellitus Inadequately Controlled With Basal Insulin Alone or in Combination With Oral Antidiabetic Drug(s)…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +2
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efruxifermin DB19012
biotech | CAS: 2375240-92-7

Efruxifermin is under investigation in clinical trial NCT06215716 (A Study Evaluating Efruxifermin in Subjects With Non-cirrhotic Nonalcoholic Steatohepatitis (Nash)/metabolic Dysfunction-associated Steatohepatitis (MASH) and Fibrosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1800476-36-1

Eftilagimod alfa is under investigation in clinical trial NCT02614833 (IMP321 (Eftilagimod Alpha) as Adjunctive to a Standard Chemotherapy Paclitaxel Metastatic Breast Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Differentiation +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eftrenonacog alfa Approved DB11608
biotech | CAS: 1270012-74-2

Eftrenonacog alfa is a long-acting recombinant fusion protein used in the treatment of hemophilia B. It is comprised of a single molecule of human factor IX (FIX) covalently linked to the constant region (Fc) domain of human IgG1 via recombinant DNA technolog…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +15
Target Protein:
IgG receptor FcRn large subunit p51
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Efzofitimod DB16453
biotech

Efzofitimod (ATYR1923) is a fusion protein comprised of the immuno-modulatory domain of histidyl tRNA synthetase fused to the FC region of a human antibody. It is a selective modulator of neuropilin-2 that downregulates the innate and adaptive immune response…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Neuropilin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Egaptivon pegol DB05202
biotech | CAS: 934868-74-3

Egaptivon pegol, formerly known as ARC1779, is a therapeutic aptamer antagonist of the A1 domain of von Willebrand Factor (vWF), the ligand for receptor glycoprotein 1b on platelets. Egaptivon pegol is being investigated for the treatment of thrombotic thromb…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +2
Target Protein:
von Willebrand factorPlatelet glycoprotein Ib alpha chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EGEN-001 DB05953
small molecule

EGEN-001 is a novel non-viral vector consisting of a plasmid DNA encoding the human gene for interleukin 12 (IL-12) and a biocompatible, biodegradable delivery polymer with potential antineoplastic activity.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Egg phospholipids Approved DB14233
biotech | CAS: 93685-90-6

Egg phospholipids are primarily a mixture of naturally occurring phospholipids which are isolated from the egg yolk. Egg phospholipids are available as an intravenous fat emulsion indicated as a source of calories for patients requiring parenteral nutrition.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Egg yolk Approved DB10530
biotech

Egg yolk allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EGT-201 DB17648
biotech

EGT-201 is an adeno-associated viral vector serotype 9 (AAV9) vector-based gene therapy consisting of the alpha-N-acetyglucosaminidase (NAGLU) transgene. Developed by Esteve Pharmaceuticals, it is being investigated for Sanfilippo syndrome type B.[L45939]

Waktu Paruh-
Vol. Distribusi-
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Genetik -
EGT-301 DB17649
biotech

EGT-301 is a gene therapy being investigated for Hunter Syndrome. It consists of an adeno-associated viral vector serotype 9 (AAV9) containing the human Iduronate-2-sulfatase (I2S) transgene designed to restore I2S functional deficiency in patients with Hunte…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EHP-102 DB16933
small molecule | CAS: 1807652-43-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elacestrant Approved DB06374
small molecule | CAS: 722533-56-4

Elacestrant is a non-steroidal small molecule and an estrogen receptor (ER) antagonist.[A256838,L44918] In January 2023, it was approved by the FDA for the treatment of ER-positive, HER2-negative, ESR1-mutated advanced or metastatic breast cancer.[L44918,L449…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Estrogen receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiElacestrant has an …
KlirensElacestrant has an …
Genetik -
Elacridar DB04881
small molecule | CAS: 143664-11-3

Elacridar (GW120918) is an oral bioenhancer that targets multiple drug resistance in tumors. In many cases, the appearance of multidrug resistance in cancer is due to a change in expression of protein inhibitors. As of August 2007 elacridar was not listed on …

Kategori:
BCRP/ABCG2 InhibitorsBenzocycloheptenesDrug Resistance, Multiple +3
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eladocagene exuparvovec Approved DB16780
biotech | CAS: 2098615-91-7

Eladocagene exuparvovec is a recombinant adeno-associated virus-2 (AAV2)-based gene therapy that expresses human aromatic L-amino acid decarboxylase (AADC), and it is used to treat AADC deficiency, a fatal and rare genetic disorder that causes severe disabili…

Kategori:
Adeno-associated Viral Vector TherapiesAlimentary Tract and MetabolismEnzymes +2
Waktu ParuhNot available.
Vol. DistribusiThe biodistribution…
KlirensNot available.
Genetik -
Elafibranor Approved DB05187
small molecule | CAS: 923978-27-2

Elafibranor is a dual peroxisome proliferator-activated receptor (PPAR) ? and ?/? agonist [A263833] that works to inhibit bile acid synthesis.[L50768] On June 10, 2024, elafibranor was granted accelerated approval by the FDA for the treatment of primary bilia…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBCRP/ABCG2 Inhibitors +21
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor gamma
Waktu ParuhFollowing a single …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent t…
Genetik -
Elagolix Approved DB11979
small molecule | CAS: 834153-87-6

Elagolix has been used in trials studying the basic science and treatment of Endometriosis, Folliculogenesis, Uterine Fibroids, Heavy Uterine Bleeding, and Heavy Menstrual Bleeding. As of 24 July 2018, however, the U.S. Food and Drug Administration (FDA) appr…

Kategori:
Anti-Gonadotropin-Releasing HormonesAntigonadotropins and Similar AgentsCytochrome P-450 CYP2C19 Inhibitors +16
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe terminal phase …
Vol. DistribusiThe apparent volume…
KlirensThe oral clearance …
Genetik -
Elaidamide DB03784
small molecule | CAS: 4303-70-2

Deskripsi belum tersedia.

Target Protein:
Phospholipase A2, membrane associated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elamipretide DB11981
small molecule | CAS: 736992-21-5

Elamipretide has been used in trials studying the treatment of Leber's Hereditary Optic Neuropathy.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elapegademase Approved DB14712
biotech | CAS: 1709806-75-6

Elapegademase is a PEGylated recombinant adenosine deaminase. It can be defined molecularly as a genetically modified bovine adenosine deaminase with a modification in cysteine 74 for serine and with about 13 methoxy polyethylene glycol chains bound via carbo…

Kategori:
Adenosine Deaminase InhibitorsAdjuvants, ImmunologicAmino Acids, Peptides, and Proteins +12
Target Protein:
Adenosine
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Elastin (human) DB15364
biotech | CAS: 9007-58-3

Elastin (human) is under investigation in clinical trial NCT01466413 (Two Formulations of ELAPR Compared to Restylane® Vital Light Following Repeat Implants in the Upper Arm Dermis).

Kategori:
Amino Acids, Peptides, and ProteinsBiopolymersElastin +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elbasvir Approved DB11574
small molecule | CAS: 1370468-36-2

Elbasvir is a direct-acting antiviral medication used as part of combination therapy to treat chronic hepatitis C, an infectious liver disease caused by infection with hepatitis C virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine d…

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +18
Target Protein:
Nonstructural protein 5A
Waktu ParuhThe geometric mean …
Vol. DistribusiElbasvir has an est…
KlirensThe clearance of el…
Genetik -
Elcatonin DB13742
small molecule | CAS: 60731-46-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Parathyroid AgentsBone Density Conservation Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eldecalcitol DB05295
small molecule | CAS: 104121-92-8

Eldecalcitol (ED-71), a vitamin D analog, is a more potent inhibitor of bone resorption than alfacalcidol in an estrogen-deficient rat model of osteoporosis. Eldecalcitol, effectively and safely increased lumbar and hip bone mineral density (BMD) in osteopor…

Kategori:
Bone Density Conservation AgentsFused-Ring CompoundsSecosteroids +4
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eleclazine DB12394
small molecule | CAS: 1443211-72-0

Eleclazine has been used in trials studying the treatment of LQT2 Syndrome, Long QT Syndrome, Ischemic Heart Disease, Ventricular Arrhythmia, and Long QT Syndrome Type 3, among others.

Kategori:
Azepines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elenbecestat DB15391
small molecule | CAS: 1388651-30-6

Elenbecestat is under investigation in clinical trial NCT02956486 (A 24-Month Study to Evaluate the Efficacy and Safety of Elenbecestat (E2609) in Subjects With Early Alzheimer's Disease).

Target Protein:
Beta-secretase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elesclomol DB05719
small molecule | CAS: 488832-69-5

Elesclomol is a novel, injectable, drug candidate that kills cancer cells by elevating oxidative stress levels beyond a breaking point, triggering programmed cell death. In preclinical models elesclomol showed potent killing of a broad range of cancer cell ty…

Kategori:
AmidesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eletriptan Approved DB00216
small molecule | CAS: 143322-58-1

Eletriptan is a second generation triptan drug developed by Pfizer Inc for the treatment of migraine headaches.

Kategori:
Agents that produce hypertensionAminesAnalgesics +30
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1F +1
Gen Terkait:
GNB3
Waktu ParuhThe terminal elimin…
Vol. Distribusi* 138 L
Klirens* Renal cl=3.9 L/h
Genetik 1 Varian
Eleuthero Approved DB14303
biotech

Eleuthero is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAraliaceaeBiological Products +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elexacaftor Approved DB15444
small molecule | CAS: 2216712-66-0

Elexacaftor (previously VX-445) is a small molecule, next-generation corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) protein.[A187361] It received FDA approval in October 2019 in combination with [tezacaftor] and [ivacaftor] as the…

Kategori:
Cystic Fibrosis Transmembrane Conductance Regulator CorrectorsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +24
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Elezanumab DB15240
biotech | CAS: 1791416-49-3

Elezanumab is under investigation in clinical trial NCT03737812 (A Study to Assess the Safety and Efficacy of Elezanumab When Added to Standard of Care in Progressive Forms of Multiple Sclerosis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elgemtumab DB15430
biotech | CAS: 1512559-37-3

Elgemtumab is under investigation in clinical trial NCT02167854 (Open-Label Study Evaluating the Safety and Tolerability of LJM716, BYL719 and Trastuzumab in Patients With Metastatic HER2+ Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eliglustat Approved DB09039
small molecule | CAS: 491833-29-5

Eliglustat is a glucosylceramide synthase inhibitor used for the long-term treatment of type 1 Gaucher disease.[A3752,L41404] Gaucher disease is a rare genetic disorder characterized by the deficiency of acid ?-glucosidase, an enzyme that converts glucosylcer…

Kategori:
Alimentary Tract and MetabolismCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +15
Target Protein:
Ceramide glucosyltransferase
Waktu ParuhEliglustat has a te…
Vol. DistribusiIn CYP2D6 extensive…
KlirensIn healthy CYP2D6 e…
Genetik -
Menampilkan 5501–5550 dari 13591
Sebelumnya Halaman 111 / 272 Berikutnya