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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 111 / 282
Diphenhydramine Approved DB01075
small molecule | CAS: 58-73-1

Diphenhydramine - perhaps known most commonly as its brand name formulation Benadryl - is a first-generation H1 receptor antihistamine that is used extensively for the treatment of seasonal allergies, insect bites and stings, and rashes [L5263, L5266, L5269, …

Kategori:
Agents producing tachycardiaAminesAminoalkyl Ethers +41
Target Protein:
Histamine N-methyltransferaseHistamine H1 receptorMuscarinic acetylcholine receptor M2
Waktu ParuhThe elimination hal…
Vol. DistribusiDiphenhydramine is …
KlirensValues for plasma c…
Genetik -
Diphenidol Approved DB01231
small molecule | CAS: 972-02-1

Diphenidol is an antiemetic agent used in the treatment of vomiting and vertigo. Diphenidol overdose may result in serious toxicity in children.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAntiemetics +6
Target Protein:
Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1 +1
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
Diphenoxylate Approved DB01081
small molecule | CAS: 915-30-0

A meperidine congener used as an antidiarrheal, usually in combination with atropine. At high doses, it acts like morphine. Its unesterified metabolite difenoxin has similar properties and is used similarly. It has little or no analgesic activity. This medica…

Kategori:
Alimentary Tract and MetabolismAnalgesicsAntidiarrheals +11
Target Protein:
Mu-type opioid receptorDelta-type opioid receptor
Waktu Paruh12-14 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 117-34-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicPhenylacetates
Target Protein:
Cathepsin B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 244-54-2

An NADPH oxidase 2 (NOX2) inhibitor.[A252987]

Kategori:
Blood Glucose Lowering AgentsEnzyme InhibitorsNitric Oxide Synthase, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diphenylguanidine Approved DB14191
small molecule | CAS: 102-06-7

Diphenylguanidine is a complexing agent used in the detection of metals and organic bases and used as an accelerator in the vulcanization of rubber. It is found in some rubber products. It is also a dermatological sensitizer and allergen. Sensitivity to di…

Kategori:
AmidinesCell-mediated ImmunityIncreased Histamine Release +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Diphenylpyraline Approved DB01146
small molecule | CAS: 147-20-6

Diphenylpyraline is an antihistamine. Antihistamines used in the treatment of allergy act by competing with histamine for H 1-receptor sites on effector cells. Antihistamines prevent, but do not reverse, responses mediated by histamine alone. Antihistamines a…

Kategori:
Aminoalkyl EthersAntihistamines for Systemic UseHistamine Antagonists +1
Target Protein:
Histamine H1 receptorSodium-dependent dopamine transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diphthamide DB03223
small molecule | CAS: 75645-22-6

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins
Target Protein:
Elongation factor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 499-83-2

Deskripsi belum tersedia.

Kategori:
Chelating AgentsCompounds used in a research, industrial, or household settingEnzyme Inhibitors +3
Target Protein:
4-hydroxy-tetrahydrodipicolinate reductase4-hydroxy-tetrahydrodipicolinate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dipivefrin Approved DB00449
small molecule | CAS: 52365-63-6

Dipivefrin is a prodrug of adrenaline, which is used to treat glaucoma. It is available as ophthalmic solution (eye drops).

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +24
Target Protein:
Beta-1 adrenergic receptorAlpha-1A adrenergic receptorAlpha-2A adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dipotassium phosphate Approved DB09414
small molecule | CAS: 7758-11-4

Dipotassium phosphate (K2HPO4) is a highly water-soluble salt often used as a fertilizer and food additive as a source of phosphorus and potassium as well as a buffering agent.

Kategori:
AcidsAcids, NoncarboxylicAnions +14
Waktu ParuhIn healthy children…
Vol. DistribusiDistribution is lar…
KlirensPhosphates are rapi…
Genetik -
Dipraglurant DB12733
small molecule | CAS: 872363-17-2

Dipraglurant has been used in trials studying the treatment of Parkinson's Disease. It is a metabotropic glutamate receptor 5 (mGluR5) negative allosteric modulator (NAM).

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 63065-88-3

Dipropyl-4-hydroxytryptamine is the 4-hydroxyl analog of dipropyltryptamine (DPT). Dipropyl-4-hydroxytryptamine was first synthesized by Alexander Shulgin. This agent and its properties haven't been fully elucidated.

Waktu Paruh-
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Genetik -
small molecule | CAS: 25265-71-8

Deskripsi belum tersedia.

Waktu Paruh-
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Dipyridamole Approved DB00975
small molecule | CAS: 58-32-2

A phosphodiesterase inhibitor that blocks uptake and metabolism of adenosine by erythrocytes and vascular endothelial cells. Dipyridamole also potentiates the antiaggregating action of prostacyclin. (From AMA Drug Evaluations Annual, 1994, p752)

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +17
Target Protein:
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10AcGMP-specific 3',5'-cyclic phosphodiesterase3',5'-cyclic-AMP phosphodiesterase 4A +3
Waktu Paruh40 minutes
Vol. Distribusi* 1 to 2.5 L/kg
Klirens* 2.3-3.5 mL/min/kg
Genetik -
Dipyrithione Approved DB11327
small molecule | CAS: 3696-28-4

Dipyrithione, a bactericidal and fungicidal pyrithione derivate, was formulated as Crimanex anti-dandruff shampoo, but is no longer available.[L2611] It is currently used as a pesticide, and not used in any FDA approved drug products.[A32829] Interestingl…

Target Protein:
Nitric oxide synthase, inducibleProstaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diquafosol DB15919
small molecule | CAS: 59985-21-6

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAnions +12
Target Protein:
P2Y purinoceptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diridavumab DB12607
biotech | CAS: 1393659-46-5

Cr6261 is under investigation in clinical trial NCT02016066 (A Study to Assess the Safety, Pharmacokinetics and Immunogenicity of Diridavumab in Japanese Healthy Participants).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dirithromycin DB00954
small molecule | CAS: 62013-04-1

Dirithromycin is a macrolide glycopeptide antibiotic used to treat many different types of bacterial infections, such as bronchitis, pneumonia, tonsillitis, and even skin infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +9
Target Protein:
23S ribosomal RNA
Waktu ParuhThe mean plasma hal…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2163074-23-3

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dirocaftor DB16143
small molecule | CAS: 2137932-23-9

Dirocaftor is under investigation in clinical trial NCT03251092 (Study Designed to Assess the Safety, Tolerability and PK of PTI-808 in Healthy Volunteers and in Adults With Cystic Fibrosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diroximel fumarate Approved DB14783
small molecule | CAS: 1577222-14-0

Multiple Sclerosis (MS) is a chronic, debilitating neurological disease that can lead to profound cognitive and physical symptoms, severely affecting quality of life.[A176474] It is the main cause of neurological disability not caused by trauma in the young a…

Kategori:
Acids, AcyclicAntineoplastic and Immunomodulating AgentsDicarboxylic Acids +3
Target Protein:
Neuronal acetylcholine receptor subunit alpha-10
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe apparent volume…
KlirensNo clearance inform…
Genetik -
Dirucotide DB04921
biotech | CAS: 152074-97-0

Dirucotide is a synthetically prepared peptide. In particular, the sequence prepared is a 17 amino acid chain that is identical to a section of myelin basic protein (MBP) that is found in humans. Dirucotide has been developed for the treatment of multiple scl…

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsMyelin Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 130114-83-9

Disaccharide tripeptide glycerol dipalmitoyl is under investigation in clinical trial NCT00003667 (Combination Chemotherapy and Biological Therapy in Treating Patients With High-Risk Ewing's Sarcoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2136633-23-1

Disitamab vedotin is an antibody-drug conjugate drug targeting human epidermal growth factor receptor 2 (HER2). It is currently being investigated for cancers.[A254721]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-drug Conjugates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disitertide DB12953
biotech | CAS: 272105-42-7

Disitertide has been used in trials studying the treatment of Skin Fibrosis.

Target Protein:
Transforming growth factor beta-1 proprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disomotide DB17469
biotech | CAS: 181477-43-0

Disomotide is a synthetic peptide cancer vaccine.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disopyramide Approved DB00280
small molecule | CAS: 3737-09-5

A class I anti-arrhythmic agent (one that interferes directly with the depolarization of the cardiac membrane and thus serves as a membrane-stabilizing agent) with a depressant action on the heart similar to that of guanidine. It also possesses some anticholi…

Kategori:
Agents producing tachycardiaAntiarrhythmic agentsAntiarrhythmics, Class I +21
Target Protein:
Sodium channel protein type 5 subunit alphaMuscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +5
Waktu Paruh6.7 hours (range 4-…
Vol. Distribusi-
Klirens-
Genetik -
Disperse Blue 106 Approved DB14203
small molecule | CAS: 68516-81-4

Disperse Blue 106 is used in allergenic testing.

Kategori:
AllergensAntigensBiological Factors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Distearyldimonium Approved DB14143
small molecule | CAS: 14357-21-2

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAminesAmmonium Compounds +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Distigmine DB13694
small molecule | CAS: 17299-00-2

Distigmine is a parasympathomimetic agent with a longer duration of action and enhanced drug accumulation compared to [DB00545] and [DB01400]. It is an anticholinergic drug and long-acting reversible carbamate cholinesterase inhibitor that binds directly and …

Kategori:
Cholinergic AgentsCholinesterase InhibitorsEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disufenton DB17298
small molecule | CAS: 168021-77-0

Deskripsi belum tersedia.

Kategori:
AntioxidantsArylsulfonatesArylsulfonic Acids +9
Target Protein:
Extracellular sulfatase Sulf-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disulfiram Approved DB00822
small molecule | CAS: 97-77-8

A carbamate derivative used as an alcohol deterrent. It is a relatively nontoxic substance when administered alone, but markedly alters the intermediary metabolism of alcohol. When alcohol is ingested after administration of disulfiram, blood acetaldehyde con…

Kategori:
Acetyl Aldehyde Dehydrogenase InhibitorsAcids, AcyclicAgents that reduce seizure threshold +26
Target Protein:
Dopamine beta-hydroxylaseAldehyde dehydrogenase family 3 member A2Aldehyde dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ditazole DB08994
small molecule | CAS: 18471-20-0

Ditazole is a non-steroidal anti-inflammatory drug (NSAID). Ditazole's analgesic and antipyretic effects are similar to phenylbutazone. Additionally, ditazole is a platelet aggregation inhibitor marketed in Spain and Portugal with trade name Ageroplas.

Kategori:
AnticoagulantsBlood and Blood Forming OrgansPlatelet Aggregation Inhibitors Excl. Heparin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dithiazanine DB11516
small molecule | CAS: 7187-55-5

Dithiazanine is a highly potent anthelmintic, introduced in 1959 for the treatment of strongyloid worms and whipworms. However, its use is severely limited due to its toxicity. Dithiazanine iodide was associated with eight fatal cases of severe acidosis and s…

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6892-68-8

A compound that, along with its isomer, Cleland's reagent (dithiothreitol), is used for the protection of sulfhydryl groups against oxidation to disulfides and for the reduction of disulfides to sulfhydryl groups. [PubChem]

Kategori:
AlcoholsCarbohydratesCompounds used in a research, industrial, or household setting +6
Target Protein:
Listeriolysin regulatory protein6,7-dimethyl-8-ribityllumazine synthaseThymidine kinase, cytosolic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dithiopyr DB15230
small molecule | CAS: 97886-45-8

Dithiopyr is under investigation in clinical trial NCT01236781 (Comparison of Full-Field Digital Mammography With Digital Breast Tomography for Screening Call-Back Rates).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ditiocarb DB02520
small molecule | CAS: 147-84-2

A chelating agent that has been used to mobilize toxic metals from the tissues of man and experimental animals. It is the main metabolite of DISULFIRAM.

Kategori:
Acids, AcyclicAdjuvants, ImmunologicAnti-Infective Agents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ditiocarb zinc Approved DB14193
small molecule | CAS: 14324-55-1

Ditiocarb zinc, also known as Diethyldithiocarbamic acid zinc salt, is a known chelator for copper and zinc. It also a dermatological sensitizer and allergen. Sensitivity to ditiocarb zinc may be identified with a clinical patch test.

Kategori:
Acids, AcyclicAdjuvants, ImmunologicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical Use +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Divarasib DB17488
small molecule | CAS: 2417987-45-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Divozilimab DB18878
biotech | CAS: 2254061-60-2

Divozilimab is under investigation in clinical trial NCT05730699 (Efficacy and Safety of Divozilimab in Patients With Neuromyelitis Optica Spectrum Disorders (AQUARELLE)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dixanthogen DB13712
small molecule | CAS: 502-55-6

Deskripsi belum tersedia.

Kategori:
AnionsAntiparasitic Products, Insecticides and RepellentsEctoparasiticides, Incl. Scabicides +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dixyrazine DB13784
small molecule | CAS: 2470-73-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAntiemetics +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha tocopheryl acetate Approved DB14477
small molecule | CAS: 52225-20-4

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18656-38-7

A synthetic phospholipid used in liposomes and lipid bilayers for the study of biological membranes. It is used in commercial drug preparations to solubilize drugs for injection [A32711]

Kategori:
Compounds used in a research, industrial, or household settingGlycerophosphatesGlycerophospholipids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61361-72-6

DL-dimyristoylphosphatidylglycerol is a phospholipid used in commercially available pharmaceutical preparations to solubilize drugs for injection.

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-Methylephedrine Approved DB11278
small molecule | CAS: 1201-56-5

Methylephedrine is a sympathomimetic amine that appears in various over-the-counter cough and cold medications throughout the world [L2838], [L2839], [L2840]. The abuse of methylephedrine-containing medications has been reported in Japan. Methylephedrine is n…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +10
Target Protein:
Beta-1 adrenergic receptorAlpha-2A adrenergic receptorAlpha adrenergic receptor +1
Waktu Paruh3-6 hours (Ephedrin…
Vol. DistribusiEphedrine: 2.5-3.0 …
Klirens-
Genetik -
DLO6002 DB05179
small molecule

DLO6002 is developed by Summit Corporation and is in phase I of clinical trials for the treatment of Parkinson's disease.

Waktu Paruh-
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Genetik -
DM-1157 DB18600
small molecule | CAS: 1239953-66-2

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Menampilkan 5501–5550 dari 14063
Sebelumnya Halaman 111 / 282 Berikutnya