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6694

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4518 (67.5%)
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3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 110 / 134
Rindopepimut DB05374
small molecule | CAS: 1108208-65-6

Rindopepimut (CDX-110) is an injectable peptide cancer vaccine which targets a mutant protein called EGFRvIII present in about 25% to 30% of glioblastoma cases. The vaccine consists of the EGFRv3-specific peptide (a 13-amino acid mutant vIII epitope) conjugat…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalBiological Products +2
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rintatolimod DB16425
biotech | CAS: 38640-92-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsBase Pair Mismatch +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rinucumab DB16313
biotech | CAS: 1569263-06-4

Rinucumab is under investigation in clinical trial NCT02418754 (Study of Intravitreal REGN2176-3 in Participants With Neovascular ("Wet") Age-related Macular Degeneration (AMD)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Riociguat Approved DB08931
small molecule | CAS: 625115-55-1

Riociguat is a soluble guanylate cyclase (sGC) agonist approved in the USA, Europe and several other regions for patients with group I PAH (pulmonary arterial hypertension) in WHO FC II or III; and for the treatment of patients with inoperable CTEPH (chronic …

Kategori:
Antihypertensive AgentsAntihypertensives for Pulmonary Arterial HypertensionBCRP/ABCG2 Substrates +11
Target Protein:
Retinal guanylyl cyclase 1Guanylate cyclase soluble subunit alpha-2
Waktu ParuhAbout 12 hours in p…
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
Ripasudil DB13165
small molecule | CAS: 223645-67-8

Ripasudil, as hydrochloride hydrate (K-115), is a specifc Rho-associated coiled-coil containing protein kinase (ROCK) inhibitor used for the treatment of glaucoma and ocular hypertension. It was first approved for treatment in Japan in September 2014. This me…

Kategori:
AmidesAntiglaucoma Preparations and MioticsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Rho-associated protein kinase 1Rho-associated protein kinase 2
Waktu ParuhThe half life of Ri…
Vol. Distribusi-
KlirensRipasudil has a ren…
Genetik -
Ripertamab DB16314
biotech | CAS: 2249927-04-4

Ripertamab is under investigation in clinical trial NCT02772822 (A Study Comparing the Efficiency and Safety of S-chop(cyclophosphamide, Hydroxydaunomycin, Oncovin, and Prednisone) Versus R-CHOP in Untreated Cd20(cluster of Differentiation Antigen 20)-positiv…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ripretinib Approved DB14840
small molecule | CAS: 1442472-39-0

Ripretinib is a kinase inhibitor used for the treatment of advanced gastrointestinal stromal tumor (GIST) that has not adequately responded to other kinase inhibitors such as [sunitinib] and [imatinib]. Ripretinib, also known as Qinlock, is manufactured by De…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Mast/stem cell growth factor receptor KitPlatelet-derived growth factor receptor betaAngiopoietin-1 receptor +3
Waktu ParuhThe average half-li…
Vol. DistribusiThe mean volume of …
KlirensThe mean apparent c…
Genetik -
Risdiplam Approved DB15305
small molecule | CAS: 1825352-65-5

Risdiplam is an orally bioavailable mRNA splicing modifier used for the treatment of spinal muscular atrophy (SMA).[L12615] It increases systemic SMN protein concentrations by improving the efficiency of _SMN2_ gene transcription. This mechanism of action is …

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +11
Waktu ParuhThe terminal elimin…
Vol. DistribusiFollowing oral admi…
KlirensFor a 14.9kg patien…
Genetik -
Risedronic acid Approved DB00884
small molecule | CAS: 105462-24-6

Risedronic acid is a third generation bisphosphonate that is used for the treatment of some forms of osteoperosis and Paget's disease[FDA Label][A959,A203111]. It functions by preventing resorption of bone[FDA Label][A959].

Kategori:
Agents Causing Muscle ToxicityBisphosphonatesBone Density Conservation Agents +9
Target Protein:
HydroxylapatiteFarnesyl pyrophosphate synthase
Waktu ParuhThe initial half li…
Vol. Distribusi13.8 L/kg[FDA Label…
KlirensMean renal clearanc…
Genetik -
Ritivixibat DB18030
small molecule | CAS: 2460667-52-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ritlecitinib Approved DB14924
small molecule | CAS: 1792180-81-4

Ritlecitinib (PF-06651600) is a highly selective inhibitor of Janus kinase 3 (JAK3) and the tyrosine kinase expressed in hepatocellular carcinoma (TEC) kinase family. In June 2023, it was approved by the FDA for the treatment of severe alopecia areata in adul…

Kategori:
Antineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +16
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase TecTyrosine-protein kinase ITK/TSK +3
Waktu ParuhRitlecitinib has a …
Vol. DistribusiRitlecitinib is pre…
KlirensRitlecitinib is pre…
Genetik -
Ritobegron DB12080
small molecule | CAS: 255734-04-4

Ritobegron is under investigation in clinical trial NCT02256735 (Study to Investigate the Effect of KUC 7483 CL on the QT/QTc Interval of the ECG in Comparison to Placebo and Moxifloxacin in Healthy Male and Female Volunteers).

Kategori:
Acids, AcyclicAdrenergic AgentsAdrenergic Agonists +15
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ritonavir Approved DB00503
small molecule | CAS: 155213-67-5

Ritonavir is an HIV protease inhibitor that interferes with the reproductive cycle of HIV. Although it was initially developed as an independent antiviral agent, it has been shown to possess advantageous properties in combination regimens with low-dose ritona…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAnti-HIV Agents +69
Target Protein:
Gag-Pol polyproteinPol polyproteinNuclear receptor subfamily 1 group I member 2
Waktu ParuhThe approximate hal…
Vol. DistribusiThe estimated volum…
KlirensThe apparent oral c…
Genetik -
Rivipansel DB12778
small molecule | CAS: 927881-99-0

Rivipansel has been used in trials studying the other, basic science, and treatment of Pain Crisis, Renal impairment, Anemia, Sickle Cell, Sickle Cell Disease, and Sickle Cell Disorders, among others.

Kategori:
CarbohydratesGlycoconjugatesLipids
Target Protein:
E-selectinL-selectinP-selectin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ro 12-7310 DB08455
small molecule | CAS: 65316-65-6

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-6870810 DB15151
small molecule | CAS: 1349719-98-7

RO-6870810 is under investigation in clinical trial NCT02308761 (A Study of RO6870810/TEN-010 in Participants With Acute Myeloid Leukemia and Myelodysplastic Syndrome).

Kategori:
Sulfur CompoundsThiazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO7284755 DB17527
biotech

RO7284755 is an investigational cancer drug: it is a PD-1-targeted IL-2 variant antibody fusion protein. RO7284755 is under investigation in clinical trial NCT04303858 (A Study to Evaluate Safety and Anti-tumor Activity of RO7284755 Alone or in Combination Wi…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO7296682 DB17531
biotech

RO7296682 is a monoclonal antibody against CD25 (IL-2R alpha) expressed on tumour-infiltrating regulatory T (T<sub>reg</sub>) cells. RO7296682 is under investigation in clinical trial NCT04642365 (A Study to Evaluate the Safety and Tolerability of RO7296682 i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO7300490 DB17535
biotech

RO7300490 is an investigational Fibroblast Activation Protein-? (FAP) targeted CD40 agonist. RO7300490 is under investigation in clinical trial NCT04857138 (A Study to Evaluate Safety, Pharmacokinetics and Anti-tumor Activity of RO7300490, as Single Agent or …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Robenacoxib DB11455
small molecule | CAS: 220991-32-2

Robenacoxib is a non-steroidal anti-inflammatory drug used in veterinary medicine for the relief of pain and inflammation in cats and dogs.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +6
Target Protein:
Cyclooxygenase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Robenidine DB11542
small molecule | CAS: 25875-51-8

Robenidine is identified as a coccidiostat drug, which slows both the growth and reproductive cycles of coccidian parasites. Robenidine is used to control coccidiosis, a lethal infection in poultry which has shown a significant economic burden. Despite the av…

Kategori:
AmidinesAnti-Infective AgentsAntiparasitic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Robinia pseudoacacia pollen Approved DB10474
biotech

Robinia pseudoacacia pollen is the pollen of the Robinia pseudoacacia plant. Robinia pseudoacacia pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocaglamide DB15495
small molecule | CAS: 84573-16-0

Rocaglamide, also referred to as rocaglamide-A, is the eponymous member of a class of anti-cancer phytochemicals known as rocaglamides.[A186760] Rocaglamides are secondary metabolites of the plant genus _Aglaia_, and extracts of the plant have traditionally b…

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Prohibitin 1Transcription factor RelBNuclear factor NF-kappa-B p100 subunit +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocatinlimab DB18809
biotech | CAS: 2431972-52-8

Rocatinlimab is a subcutaneously administered anti-OX40 antibody developed for the treatment of moderate-to-severe atopic dermatitis. In clinical trials, it has shown significant efficacy and safety compared to a placebo. The drug works by targeting the OX40 …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Tumor necrosis factor receptor superfamily member 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocbrutinib DB19445
small molecule | CAS: 2485861-07-0

Rocbrutinib is under investigation in clinical trial NCT05716087 (A Study of Rocbrutinib in Participants With Relapse or Refractory Mantle Cell Lymphoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rociletinib DB11907
small molecule | CAS: 1374640-70-6

Rociletinib has been used in trials studying the treatment and prevention of Nonsmall Cell Lung Cancer, Non-small Cell Lung Cancer, and Locally Advanced or Metastatic Non-small Cell Lung Cancer.

Kategori:
Acids, AcyclicAcrylatesAmides +4
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rociverine DB13581
small molecule | CAS: 53716-44-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +9
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocuronium Approved DB00728
small molecule | CAS: 143558-00-3

Rocuronium (rapid onset-curonium) is a desacetoxy analogue of vecuronium with a more rapid onset of action. It is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia, to facilitate endotracheal intubation and t…

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +16
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M25-hydroxytryptamine receptor 3A
Waktu ParuhThe rapid distribut…
Vol. Distribusi* 0.3 L/kg [3 to <1…
Klirens* 0.25 L/kg/hr [Adu…
Genetik -
Rodatristat DB18478
small molecule | CAS: 1673568-73-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1673571-51-1

Deskripsi belum tersedia.

Target Protein:
Tryptophan 5-hydroxylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rofecoxib Approved DB00533
small molecule | CAS: 162011-90-7

Rofecoxib is used for the treatment of osteoarthritis, rheumatoid arthritis, acute pain in adults, and primary dysmenorrhea, as well as acute treatment of migraine attacks with or without auras. Rofecoxib is a solid. This compound belongs to the stilbenes. Th…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +29
Target Protein:
Prostaglandin G/H synthase 2Elastin
Waktu Paruh17 hours
Vol. Distribusi-
Klirens-
Genetik -
Roflumilast Approved DB01656
small molecule | CAS: 162401-32-3

Roflumilast is a highly selective phosphodiesterase-4 (PDE4) inhibitor.[A251385] PDE4 is a major cyclic-3',5?-adenosinemonophosphate (cyclic AMP, cAMP)-metabolizing enzyme [L37564] expressed on nearly all immune and pro-inflammatory cells, in addition to stru…

Kategori:
Acids, CarbocyclicAgents to Treat Airway DiseaseAmides +17
Target Protein:
cAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4)
Waktu ParuhFollowing oral admi…
Vol. DistribusiFollowing a single …
KlirensPlasma clearance of…
Genetik -
Rokitamycin DB13409
small molecule | CAS: 74014-51-0

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolapitant Approved DB09291
small molecule | CAS: 552292-08-7

Rolapitant is a potent, highly selective, long-acting Neurokinin-1 (NK-1) receptor antagonist approved for the prevention of delayed chemotherapy-induced nausea and vomiting (CINV) in adults. Delayed-phase CINV typically occurs >24 hours after chemotherapy tr…

Kategori:
Alimentary Tract and MetabolismAntiemetics and AntinauseantsBCRP/ABCG2 Inhibitors +11
Target Protein:
Substance-P receptor
Waktu ParuhMean terminal half …
Vol. Distribusi460 L
Klirens0.96 L/hour
Genetik -
Rolicyclidine DB01549
small molecule | CAS: 2201-39-0

Rolicyclidine (PCPy) is classified as a dissociative anesthetic agent. It also has hallucinogenic and sedative properties. Because of its pharmacodynamic similarity to the drug phencyclidine (PCP), rolicyclidine was added to the Schedule I list of illegal dr…

Kategori:
Piperidines
Target Protein:
Glutamate receptor ionotropic, NMDA 3AD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolitetracycline Approved DB01301
small molecule | CAS: 751-97-3

A pyrrolidinylmethyl tetracycline.

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
30S ribosomal protein S916S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romifidine DB11543
small molecule | CAS: 65896-16-4

Romifidine is a veterinary drug utilized as a sedative primarily in large animals, most frequently horses. It is also used less commonly in a wide variety of other animal species. This drug's chemical structure closely resembles that of clonidine, however, ro…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romilkimab DB16318
biotech | CAS: 1399584-78-1

Romilkimab is under investigation in clinical trial NCT02345070 (Efficacy and Safety of SAR156597 in the Treatment of Idiopathic Pulmonary Fibrosis).

Target Protein:
Interleukin-13Interleukin-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romiplostim Approved DB05332
biotech | CAS: 267639-76-9

Romiplostim is a thrombopoiesis stimulating dimer Fc-peptide fusion protein (peptibody) to increase platelet production through activation of the thrombopoietin receptor. The peptibody molecule has two identical single-chain subunits, each one is made up of 2…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +17
Target Protein:
Thrombopoietin receptor
Waktu ParuhImmune thrombocytop…
Vol. DistribusiIn healthy voluntee…
Klirens-
Genetik -
Romosozumab Approved DB11866
biotech | CAS: 909395-70-6

Romosozumab is a humanized monoclonal antibody indicated for the treatment of osteoperosis in postmenopausal women at high risk of fracture and patients who have failed in other treatments or are intolerant to other osteoperosis therapies[L9554]. Romosozumab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Sclerostin
Waktu Paruh12.8 days[L9554].
Vol. Distribusi3.92L[L9554].
Klirens0.38mL/hr/kg[L9554].
Genetik -
Ronacaleret DB05255
small molecule | CAS: 753449-67-1

Ronacaleret is a calcium-sensing receptor antagonist.

Kategori:
Acids, CarbocyclicIndenes
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roniciclib DB12974
small molecule | CAS: 1223498-69-8

Roniciclib has been investigated for the treatment of Small Cell Lung Carcinoma.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ropivacaine Approved DB00296
small molecule | CAS: 84057-95-4

Ropivacaine is an aminoamide local anesthetic drug marketed by AstraZeneca under the trade name Naropin. It exists as a racemate of its S- and R-enantiomers, although the marketed form is supplied only as the purified S-enantiomer.[L42140]

Kategori:
AmidesAminesAnesthetics +19
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu ParuhThe mean terminal h…
Vol. DistribusiFollowing intravasc…
KlirensFollowing intraveno…
Genetik -
Ropsacitinib DB18709
small molecule | CAS: 2127109-84-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roquinimex DB11366
small molecule | CAS: 84088-42-6

Roquinimex is a derivative of quinoline that presents immunostimulant properties. Its effects are suggested to increase the activity of NK cells and macrophage cytotoxicity. Additionally, roquinimex is known to inhibit angiogenesis and to decrease the synthes…

Kategori:
Adjuvants, ImmunologicAngiogenesis InhibitorsAngiogenesis Modulating Agents +7
Target Protein:
Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosemary DB14272
biotech

Rosemary is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosemary oil Approved DB14689
biotech | CAS: 8000-25-7

Deskripsi belum tersedia.

Kategori:
Biological ProductsLipidsOils +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosiglitazone Approved DB00412
small molecule | CAS: 122320-73-4

Rosiglitazone is an anti-diabetic drug in the thiazolidinedione class of drugs. It is marketed by the pharmaceutical company GlaxoSmithKline as a stand-alone drug (Avandia) and in combination with metformin (Avandamet) or with glimepiride (Avandaryl). Like ot…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsBSEP/ABCB11 Substrates +33
Target Protein:
Peroxisome proliferator-activated receptor gammaLong-chain-fatty-acid--CoA ligase 4Peroxisome proliferator-activated receptor alpha +4
Waktu Paruh3-4 hours (single o…
Vol. Distribusi* 17.6 L [oral volu…
Klirens* Oral clearance (C…
Genetik -
Rosin Approved DB11165
biotech | CAS: 8050-09-7

Rosin is a solid form of resin obtained from pines and other plants, mostly conifers. It is prepared from heating fresh liquid resin to vaporize the volatile liquid terpene components. Rosin is used in various commercial and industrial applications, including…

Kategori:
Biological ProductsBiopolymersCell-mediated Immunity +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rosmarinic acid DB16865
small molecule | CAS: 20283-92-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAldehyde Reductase, antagonists & inhibitorsAnalgesics +22
Target Protein:
TyrosinaseInduced myeloid leukemia cell differentiation protein Mcl-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5451–5500 dari 6694
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