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2279

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Halaman 11 / 46
biotech | CAS: 372075-36-0

Cintredekin besudotox has been developed as a specific tumor-targeting agent, which is administered by positive-pressure convection-enhanced delivery (CED) directly to brain tissue at risk for residual infiltrating glioblastoma multiforme (GBM) after tumor re…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +6
Target Protein:
Interleukin-13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cipaglucosidase alfa Approved DB16708
biotech | CAS: 2359727-71-0

Cipaglucosidase alfa (ATB200) is a novel recombinant human acid alpha-glucosidase (GAA) investigated for the treatment of patients with Pompe disease, a rare inherited metabolic disorder characterized by a deficiency in GAA.[A232955] Other types of enzyme rep…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +1
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe mean volume of …
KlirensCoadministration of…
Genetik -
Ciprofloxacin Approved DB00537
small molecule | CAS: 85721-33-1

Ciprofloxacin is a second generation fluoroquinolone that has spawned many derivative antibiotics.[A178870] It is formulated for oral, intravenous, intratympanic, ophthalmic, and otic administration for a number of bacterial infections.[L6469,L6472,L6475,L647…

Kategori:
4-QuinolonesAgents Causing Muscle ToxicityAnti-Bacterial Agents +38
Target Protein:
DNA topoisomerase 4 subunit ADNA gyrase subunit BThymidylate synthase +10
Waktu ParuhThe average half li…
Vol. DistribusiCirpofloxacin follw…
KlirensThe average renal c…
Genetik -
Cisapride Approved DB00604
small molecule | CAS: 81098-60-4

In many countries (including Canada) cisapride has been either withdrawn or has had its indications limited due to reports about long QT syndrome due to cisapride, which predisposes to arrhythmias. The FDA issued a warning letter regarding this risk to health…

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmides +36
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 2A +1
Waktu Paruh6-12 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 945228-49-9

VB6-845 is a humanized antibody fragment targeting EpCAM fused with the deimmunized form of the cytotoxin Bouganin and is designed for systemic use against metastatic cancer. VB6-845 has demonstrated effective cancer cell killing properties in pre-clinical te…

Target Protein:
Epithelial cell adhesion molecule
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Citicoline Approved DB12153
small molecule | CAS: 987-78-0

Citicoline is a donor of choline in biosynthesis of choline-containing phosphoglycerides. It has been investigated for the treatment, supportive care, and diagnosis of Mania, Stroke, Hypomania, Cocaine Abuse, and Bipolar Disorder, among others.

Kategori:
AminesCentral Nervous System AgentsCytidine Diphosphate +13
Target Protein:
LicC protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cixutumumab DB12250
biotech | CAS: 947687-12-9

Cixutumumab has been used in trials studying the treatment of Lung Cancer, Malignant Neoplasm, Leukemia, Mast-Cell, Non-Small-Cell Lung Carcinoma, and Adenocarcinoma of the Prostate. Cixutumumab is a highly specific recombinant human monoclonal antibody wi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Insulin-like growth factor 1 receptor
Waktu Paruh148 h (3 mg/kg dose…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2145123-44-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clesrovimab DB18877
biotech | CAS: 2429913-18-6

Clesrovimab is under investigation in clinical trial NCT04938830 (Clesrovimab (MK-1654) in Infants and Children at Increased Risk for Severe Respiratory Syncytial Virus (RSV) Disease (MK-1654-007)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clomethiazole DB06470
small molecule | CAS: 533-45-9

Clomethiazole is a well-established ?-aminobutyric acid (GABAA)-mimetic drug. It is a sedative and hypnotic that is widely used in treating and preventing symptoms of acute alcohol withdrawal. It is a drug which is structurally related to thiamine (vitamin B1…

Kategori:
AnticonvulsantsCentral Nervous System AgentsCentral Nervous System Depressants +17
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clomipramine Approved DB01242
small molecule | CAS: 303-49-1

Clomipramine, the 3-chloro analog of imipramine, is a dibenzazepine-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-de…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +45
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2B +3
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhFollowing oral admi…
Vol. Distribusi~ 17 L/kg (range: 9…
Klirens-
Genetik 9 Varian
Clorindione DB13275
small molecule | CAS: 1146-99-2

Clorindione is a vitamin K antagonist, which may be useful to decrease prothrombin levels in humans.

Kategori:
AnticoagulantsBlood and Blood Forming OrgansIndenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clove oil Approved DB11338
biotech | CAS: 8000-34-8

Clove oil is obtained by extraction from the dried flower buds of the clove plant. Traditionally, it has been used as a flavouring spice in foods, or as a fragrance. It is also found in topical analgesics. Clove oil has shown to exert some antimicrobial activ…

Kategori:
Biological ProductsComplex MixturesDrugs that are Mainly Renally Excreted +3
Target Protein:
Vascular cell adhesion protein 1C-X-C motif chemokine 10Collagen alpha-1(I) chain +1
Waktu ParuhIn a pharmacokineti…
Vol. Distribusi-
Klirens-
Genetik -
Cloxazolam DB01553
small molecule | CAS: 24166-13-0

Cloxazolam is a benzodiazepine with anxiolytic, sedative/hypnotic, muscle relaxant, and antiepileptic effects. It is marketed in the Argentina, Australia, Portugal, Belgium, Switzerland, Luxembourg, Germany, Taiwan and Japan -- mainly for anti-anxiety. The us…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +4
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh65 hours
Vol. Distribusi-
Klirens-
Genetik -
CN-201 DB18726
biotech

CN-201 is a humanized anti-CD3/CD19 bispecific antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 181054-95-5

Recombinant Coagulation Factor IX is a purified Factor IX glycoprotein produced by recombinant DNA technology. It has a primary amino acid sequence that is identical to the Ala148 allelic form of human factor IX, and has structural and functional characterist…

Kategori:
Blood Coagulation FactorsHemostaticsIncreased Coagulation Activity
Target Protein:
Coagulation factor XCoagulation factor XICoagulation factor VII +4
Waktu Paruh18.8 ± 5.4 hours
Vol. Distribusi-
Klirens8.62 ± 1.7
Genetik -
Coagulation Factor IX Human Approved DB13152
biotech | CAS: 181054-95-5

Factor IX (or Christmas factor) is one of the serine proteases of the coagulation system; it belongs to peptidase family S1. Deficiency of this protein causes hemophilia B.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor XCoagulation factor XICoagulation factor VII +4
Waktu Paruh18.8 ± 5.4 hours.
Vol. Distribusi-
Klirens8.62 ± 1.7.
Genetik -
Coagulation factor VII human Approved DB13150
biotech

Coagulation factor VII is human serine protease type enzyme that is involved in the extrinsic coagulation cascade which results in blood clotting.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +8
Target Protein:
Tissue factorCoagulation factor XCoagulation factor IX
Waktu Paruh5 h
Vol. Distribusi45 ml/kg
Klirens7.4 ml/kgh
Genetik -
biotech | CAS: 102786-61-8

Recombinant human coagulation Factor VIIa (rFVIIa), intended for promoting hemostasis by activating the extrinsic pathway of the coagulation cascade. NovoSeven is a vitamin K-dependent glycoprotein consisting of 406 amino acid residues. Cloned and expressed i…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +15
Target Protein:
Coagulation factor XTissue factor
Waktu Paruh-
Vol. Distribusi* 121 ± 30 mL/kg [a…
Klirens* 33 - 37 mL/h x kg…
Genetik -
Coagulation factor X human Approved DB13148
biotech

Coagulation Factor X (Human), is a plasma-derived human blood coagulation factor is used by adults and children (aged 12 years and above) with hereditary Factor X deficiency. However its use is limited in the perioperative setting for the management of bleedi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
biotech | CAS: 9013-55-2

Coagulation factor XIa is under investigation in clinical trial NCT01701947 (HEMOLEVEN® Expanded Access Program Prevention of Surgical/Postpartum Hemorrhage Severe Inherited Factor XI Deficiency).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coagulin-B DB17703
biotech

Coagulin-B is an adeno-associated viral vector expressing human blood-coagulation Factor IX.[A259038, A259043] It was previously investigated for the treatment of hemophilia; however, the manufacturing company discontinued the Phase I trial in 2004, halting i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobalt Approved DB14574
small molecule | CAS: 7440-48-4

A trace element that is a component of vitamin B12. It has the atomic symbol Co, atomic number 27, and atomic weight 58.93. It is used in nuclear weapons, alloys, and pigments. Deficiency in animals leads to anemia; its excess in humans can lead to erythrocyt…

Kategori:
Cell-mediated ImmunityDiet, Food, and NutritionElements +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobicistat Approved DB09065
small molecule | CAS: 1004316-88-4

Cobicistat, marketed under the name Tybost (formerly GS-9350), indicated for treating infection with human immunodeficiency virus (HIV). Although it does not have any anti-HIV activity, cobicistat acts as a pharmacokinetic enhancer by inhibiting cytochrome P4…

Kategori:
Acids, AcyclicAnti-HIV AgentsAnti-Infective Agents +29
Target Protein:
Cytochrome P450 3A4Cytochrome P450 3A5Cytochrome P450 3A7
Waktu ParuhThe terminal plasma…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61789-40-0

Cocamidopropyl betaine is a mixture of closely related organic compounds derived from coconut oil and dimethylaminopropylamine that typically acts as an amphoteric surfactant in cosmetics and personal care products. It is a zwitterionic ammonium compound and …

Kategori:
AminesCompounds used in a research, industrial, or household settingOnium Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cocarboxylase Approved DB01987
small molecule | CAS: 136-08-3

The coenzyme form of Vitamin B1 present in many animal tissues. It is a required intermediate in the pyruvate dehydrogenase complex and the ketoglutarate dehydrogenase complex.

Kategori:
CoenzymesEnzymes and CoenzymesMicronutrients +5
Target Protein:
RNAAcetolactate synthase, catabolicPyruvate dehydrogenase E1 component +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cofirasersen DB19037
biotech | CAS: 2247669-96-9

Cofirasersen is under investigation in clinical trial NCT04441788 (A Study to Assess the Safety, Tolerability, and Efficacy of ION-827359 in Participants With Mild to Moderate Chronic Obstructive Pulmonary Disease (COPD) With Chronic Bronchitis (CB)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Col-Treg DB18451
biotech

Col-Treg is an autologous T-cell therapy comprising type I regulatory T-cells specific for human type II collagen.[A261635]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1269764-99-9

Coltuximab ravtansine (SAR3419) targets CD19 and is being investigated for the treatment of acute lymphoblastic leukemia (ALL).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +16
Target Protein:
B-lymphocyte antigen CD19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Conestat alfa Approved DB09228
biotech | CAS: 80295-38-1

C1 Esterase Inhibitor (Recombinant) is a recombinant analogue of endogenous complement component-1 esterase inhibitor (rhC1INH), purified from the milk of transgenic rabbits. The primary function of endogenous C1INH is to regulate the activation of the comple…

Kategori:
Amino Acids, Peptides, and ProteinsAngioedemas, Hereditary, drug therapyBlood and Blood Forming Organs +16
Target Protein:
Complement C1r subcomponentComplement C1s subcomponentPlasma kallikrein +4
Waktu Paruh-
Vol. Distribusi-
KlirensClearance was found…
Genetik -
Conjugated estrogens Approved DB00286
small molecule | CAS: 12126-59-9

The conjugated estrogens are noncrystalline mixtures of purified female sex hormones obtained either by its isolation from the urine of pregnant mares or by synthetic generation from vegetal material. Both of these products are later conjugated to natrium sul…

Kategori:
Agents causing angioedemaBCRP/ABCG2 SubstratesCOMT Substrates +26
Target Protein:
Estrogen receptor betaEstrogen receptor
Waktu ParuhThe median half-lif…
Vol. DistribusiThe physiological d…
KlirensThe reported normal…
Genetik -
Copper Approved DB09130
small molecule | CAS: 7440-50-8

Copper is a transition metal and a trace element in the body. It is important to the function of many enzymes including cytochrome c oxidase, monoamine oxidase and superoxide dismutase [FDA Label]. Copper is commonly used in contraceptive intrauterine devices…

Kategori:
Copper-containing Intrauterine DeviceDecreased Embryonic ImplantationDecreased Sperm Motility +12
Target Protein:
Amyloid-beta precursor proteinAdenosylhomocysteinaseHistone H2B type 1-C/E/F/G/I +143
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Copper gluconate Approved DB11246
small molecule | CAS: 527-09-3

Copper gluconate is a copper salt of D-gluconic acid that displays a light blue to bluish-green color. It is prepared by the reaction of gluconic acid solutions with cupric oxide or basic cupric carbonate. According to the good manufacturing or feeding practi…

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Copper oxodotreotide Cu-64 Approved DB15873
small molecule | CAS: 1426155-87-4

Copper Cu 64 dotatate is a newly approved Cu labeled somatostatin analog and has several advantages over <sup>68</sup>Ga-labeled somatostatin analogs for positron emission tomography (PET).[A220348] Copper Cu 64 dotatate has a longer half-life and can be prod…

Kategori:
Amino Acids, Peptides, and ProteinsCopper RadioisotopesPeptides +4
Target Protein:
Somatostatin receptor type 2
Waktu ParuhThe half-life of Co…
Vol. Distribusi-
Klirens-
Genetik -
Coprelotamab DB16380
biotech | CAS: 2348469-84-9

Coprelotamab is under investigation in clinical trial NCT04170595 (Clinical Study of Recombinant Anti-her2 Humanized Monoclonal Antibody for Injection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coramitug DB19411
biotech | CAS: 2626841-92-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CoronaVac DB15806
biotech

CoronaVac, previously known as PiCoVacc, is a SARS-CoV-2 purified, inactivated, and adsorbed vaccine candidate developed by SinoVac Biotech Corporation[A219758]. It was developed by propagating the SARS-CoV-2 CN2 strain inside Vero Cells and inactivating it w…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Corticorelin DB05394
small molecule | CAS: 86784-80-7

Corticotropin-releasing factor is studied in the treatment of brain cancer. It is made naturally by the hypothalamus (a part of the brain) and can also be made in the laboratory. Human corticotropin-releasing factor may help reduce symptoms caused by edema (s…

Kategori:
Amino Acids, Peptides, and ProteinsCorticotropin-Releasing HormoneDiagnostic Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 121249-14-7

Corticorelin, available commercially as corticorelin ovine triflutate (tradename Acthrel), is a synthetic form of the peptide human corticotropin-releasing hormone (hCRH), a potent stimulator of adrenocorticotropic hormone (ACTH) release from the anterior pit…

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsHormones +9
Target Protein:
Corticotropin-releasing factor receptor 1Corticotropin-releasing factor receptor 2
Waktu ParuhPlasma half-lives f…
Vol. DistribusiThe mean volume of …
Klirens95 ± 11 L/m2/day
Genetik -
Corticosterone DB04652
small molecule | CAS: 50-22-6

An adrenocortical steroid that has modest but significant activities as a mineralocorticoid and a glucocorticoid. (From Goodman and Gilman&#39;s The Pharmacological Basis of Therapeutics, 8th ed, p1437)

Kategori:
11-HydroxycorticosteroidsAdrenal Cortex HormonesAnti-Inflammatory Agents +11
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1Glucocorticoid receptorNuclear receptor coactivator 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cosfroviximab DB17774
biotech | CAS: 1792982-57-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2246424-95-1

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector TherapiesAmino Acids, Peptides, and ProteinsGenetic Phenomena +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CoVac-1 DB16429
biotech

Sponsored by the University Hospital Tuebingen in Germany, CoVac-1 is a multi-peptide COVID-19 vaccine candidate created from HLA class I and HLA-DR T-cell epitopes of the S-protein[A226588]. It is being investigated in the clinical trial NCT04546841 (Safety …

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Through analysis of potential immunogenic targets of the SARS-Cov2 genome, a synthetic ‘minigene’ was developed using domains of viral structural proteins and a polyprotein protease. Specifically, the COVID-19 infection relies on the binding of the Spike prot…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Dendritic cells (DCs) can be derived and differentiated from peripheral blood mononuclear cells in the presence of specific cytokines and growth factors. These cells are then loaded with antigens produced by a virus or tumor cell and administered as a vaccine…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CPGJ602 DB17485
biotech

CPGJ602 is a recombinant anti-EGFR human-mouse chimeric monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CPI-006 DB16488
biotech | CAS: 2451856-97-4

CPI-006 was investigated in clinical trials NCT03454451, NCT04464395, and NCT04734873 to evaluate its safety and efficacy. NCT03454451 focused on advanced cancers (e.g., non-small cell lung cancer, renal cell cancer, colorectal cancer). NCT04464395 and NCT047…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CR002 DB05139
biotech

CR002 is a novel investigational fully human monoclonal antibody that blocks the activity of excess platelet-derived growth factor-D (PDGF-D), a target shown to play a role in kidney inflammation. This is a novel therapeutic approach to treat kidney inflammat…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Platelet-derived growth factor D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Crefmirlimab DB17577
biotech | CAS: 2611099-93-3

Crefmirlimab is an anti-human CD8 probe targeting the CD8 antigen, for the diagnosis of various cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cresol Approved DB11143
small molecule | CAS: 1319-77-3

Cresol is a hydroxytoluene that can be extracted naturally from coal tar or made synthetically. Pure cresol is a mixture of ortho-, meta-, and para- isomers. Cresols are precursors or synthetic intermediates to various other compounds and materials, including…

Kategori:
Benzene DerivativesDrugs that are Mainly Renally ExcretedPhenols +1
Waktu ParuhThere does not appe…
Vol. DistribusiOne study determine…
KlirensAs colonic microbia…
Genetik -
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