Hasil Filter

6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (6694)

Halaman 109 / 134
Resveratrol DB02709
small molecule | CAS: 501-36-0

Resveratrol (3,5,4'-trihydroxystilbene) is a polyphenolic phytoalexin. It is a stilbenoid, a derivate of stilbene, and is produced in plants with the help of the enzyme stilbene synthase. It exists as cis-(Z) and trans-(E) isomers. The trans- form can undergo…

Kategori:
Angiogenesis InhibitorsAnticarcinogenic AgentsAntioxidants +33
Target Protein:
NAD-dependent protein deacetylase sirtuin-1Ribosyldihydronicotinamide dehydrogenase [quinone]Casein kinase II subunit alpha +23
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Retaspimycin DB05626
small molecule | CAS: 857402-23-4

Deskripsi belum tersedia.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Retatrutide DB18993
biotech | CAS: 2381089-83-2

Retatrutide is under investigation in clinical trial NCT06354660 (Effect of Retatrutide Compared With Placebo in Adult Participants With Type 2 Diabetes and Inadequate Glycemic Control With Diet and Exercise Alone (TRANSCEND-T2D-1)).

Kategori:
Amino Acids, Peptides, and ProteinsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Reteplase Approved DB00015
biotech | CAS: 133652-38-7

Human tissue plasminogen activator, purified, glycosylated, 355 residues purified from CHO cells. Retavase is considered a "third-generation" thrombolytic agent, genetically engineered to retain and delete certain portions of human tPA. Retavase is a deletion…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +17
Target Protein:
PlasminogenFibrinogen alpha chainPlasminogen activator inhibitor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Retifanlimab Approved DB15766
biotech | CAS: 2079108-44-2

Retifanlimab is a humanized IgG4 kappa monoclonal antibody that binds to the programmed death receptor-1 (PD-1), blocking PD-1 interaction with its ligands, programmed death-ligand 1 (PD-L1) and programmed death-ligand 2 (PD-L2). By blocking the PD-1/PD-L1/2 …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +11
Target Protein:
Programmed cell death protein 1
Waktu ParuhAt steady-state, re…
Vol. DistribusiAt steady-state, re…
KlirensFollowing the first…
Genetik -
small molecule | CAS: 74193-17-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2395839-91-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Revefenacin Approved DB11855
small molecule | CAS: 864750-70-9

Revefenacin is a novel biphenyl carbamate tertiary amine agent that belongs to the family of the long-acting muscarinic antagonists (LAMA). The labile primary amide in the structure produces a "soft-drug" site that allows rapid systemic clearance and minimizi…

Kategori:
AmidesAnticholinergic AgentsBCRP/ABCG2 Substrates +9
Target Protein:
Muscarinic acetylcholine receptor
Waktu ParuhThe apparent termin…
Vol. DistribusiAfter intravenous a…
KlirensThe renal clearance…
Genetik -
biotech | CAS: 1446198-96-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Reviparin Approved DB09259
small molecule | CAS: 9041-08-1

Reviparin is a low molecular weight heparin which seems to have a better safety profile than unfractionated heparin.[A32019] It is prepared from porcine intestinal mucosa by nitrous acid depolymerization. Reviparin has a molecular weight of 3.9 kDa.[A32021] I…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Revumenib Approved DB18515
small molecule | CAS: 2169919-21-3

Abnormal gene rearrangements at chromosome locus 11q23, called KMT2A rearrangements or translocations, are present in 5%-10% of patients with acute leukemias and are the sole genetic aberration found in the majority of infant acute lymphoblastic leukemia case…

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +17
Target Protein:
Menin
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe the geometric m…
KlirensFollowing oral admi…
Genetik -
RGX-111 DB17632
biotech

RGX-111 is an adeno-associated virus vector AAV9 designed to deliver the ?-L-iduronidase (IDUA) gene. Developed by REGENXBIO Inc., it was investigated for the treatment of mucopolysaccharidosis Type I (MPS I).[L46666]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RGX-121 DB17681
biotech

RGX-121 is designed to use the NAV AAV9 vector to deliver the human iduronate-2-sulfatase gene to the central nervous system.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RGX-181 DB17942
biotech

RGX-181 consists of an adeno-associated virus serotype 9 (AAV9) vector designed to deliver the soluble lysosomal enzyme tripeptidyl peptidase I (TPP1) gene. Developed by REGENXBIO, it is being investigated for the treatment of late-infantile neuronal ceroid l…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RGX-501 DB17639
biotech

RGX-501 is an adeno-associated virus vector 8 (AAV8)-mediated gene therapy that delivers a functional copy of the human low-density lipoprotein receptor (LDLR) gene to liver cells. It is being investigated for the treatment of homozygous familial hypercholest…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rhamnetin DB16772
small molecule | CAS: 90-19-7

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rhein DB13174
small molecule | CAS: 478-43-3

Rhein is an anthraquinone metabolite of rheinanthrone and senna glycoside is present in many medicinal plants including Rheum palmatum, Cassia tora, Polygonum multiflorum, and Aloe barbadensis [A19247]. It is known to have hepatoprotective, nephroprotective, …

Kategori:
AnthracenesCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +10
Target Protein:
Heat shock protein HSP 90-alphaOxysterols receptor LXR-alphaOxysterols receptor LXR-beta +2
Waktu Paruh4-10h [A19300].
Vol. Distribusi15-60L [A19300].
KlirensTotal CL is 1.5 L/h…
Genetik -
Rheinanthrone DB13175
small molecule | CAS: 480-09-1

Rheinanthrone is the active metabolite of senna glycoside [DB11365] known for its laxative effect [A19235]. It is commonly produced by plants of the Rheum species [L772].

Kategori:
Anthracenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rhGAD65 DB04963
biotech

rhGAD65 (recombinant human glutamic acid decarboxylase) is a vaccine being developed to treat insulin dependent type 1 diabetes.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rhMBL DB05237
biotech

rhMBL is a protein therapeutic being developed by Enzon for the prevention and treatment of severe infections in individuals with low levels of Mannose-Binding Lectin (MBL). Over 10 percent of the general population is estimated to be MBL-deficient. Natural M…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 104114-27-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rhodamine 6G DB03825
small molecule | CAS: 989-38-8

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsColoring AgentsCompounds used in a research, industrial, or household setting +7
Target Protein:
HTH-type transcriptional regulator QacRMultidrug efflux pump subunit AcrB
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rhodotorula mucilaginosa Approved DB10701
biotech

Rhodotorula mucilaginosa is a fungus which can provoke allergic reactions. Rhodotorula mucilaginosa is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rhThrombin Approved DB04923
biotech | CAS: 1270043-60-1

rhThrombin (recombinant human thrombin) is being developed by ZymoGenetics, Inc. as a general aid to achieving hemostasis during surgery. ZymoGenetics is developing rhThrombin, a recombinant form of human thrombin that is not derived from animal or human bloo…

Waktu ParuhApproximately 15 ho…
Vol. Distribusi-
Klirens-
Genetik -
Ribavirin Approved DB00811
small molecule | CAS: 36791-04-5

Producing a broad-spectrum activity against several RNA and DNA viruses, Ribavirin is a synthetic guanosine nucleoside and antiviral agent that interferes with the synthesis of viral mRNA. It is primarily indicated for use in treating hepatitis C and viral he…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntimetabolites +13
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1RNA-directed RNA polymerase LGenome polyprotein +2
Gen Terkait:
IFNL3
Waktu ParuhThe terminal half-l…
Vol. DistribusiRibavirin displays …
KlirensThe total apparent …
Genetik 1 Varian
small molecule | CAS: 1352921-29-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ribaxamase DB16311
biotech | CAS: 1792207-66-9

Ribaxamase is under investigation in clinical trial NCT02563106 (A Study of SYN-004 for the Prevention of c.diff in Patients With a LRTI).

Kategori:
AmidohydrolasesAmino Acids, Peptides, and ProteinsEnzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ribociclib Approved DB11730
small molecule | CAS: 1211441-98-3

Ribociclib is a selective cyclin-dependent kinase inhibitor, a class of drugs that help slow the progression of cancer by inhibiting two proteins called cyclin-dependent kinase 4 and 6 (CDK4/6). These proteins, when over-activated, can enable cancer cells to …

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhAt steady-state in …
Vol. DistribusiAt steady-state, th…
KlirensAt steady-state in …
Genetik -
Riboflavin Approved DB00140
small molecule | CAS: 83-88-5

Nutritional factor found in milk, eggs, malted barley, liver, kidney, heart, and leafy vegetables. The richest natural source is yeast. It occurs in the free form only in the retina of the eye, in whey, and in urine; its principal forms in tissues and cells a…

Kategori:
Alimentary Tract and MetabolismBiological FactorsCoenzymes +14
Target Protein:
Riboflavin kinaseRiboflavin synthaseFlavin reductase (NADPH)
Waktu Paruh66-84 minutes
Vol. Distribusi-
Klirens-
Genetik -
Ribostamycin Approved DB03615
small molecule | CAS: 25546-65-0

Ribostamycin is an aminoglycoside antibiotic[A187166] isolated from _Streptomyces ribosidificus_[A187178] listed as one of the World Health Organization's critically important antimicrobials.[L9071]

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
Target Protein:
30S ribosomal protein S12Protein disulfide-isomeraseAminoglycoside N(6')-acetyltransferase type 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rice bran oil Approved DB11293
biotech

Rice bran oil is extracted from the hard outer brown layer of rice after chaff (rice husk) used for high-temperature cooking methods such as deep frying and stir frying. It contains monosaturated fatty acids, polyunsaturated fatty acids, and saturated fatty a…

Kategori:
Biological ProductsComplex MixturesDietary Fats +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ricinoleic acid DB02955
small molecule | CAS: 141-22-0

Deskripsi belum tersedia.

Kategori:
Biological ProductsFatsFats, Unsaturated +6
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ricolinostat DB12376
small molecule | CAS: 1316214-52-4

Ricolinostat is under investigation for the treatment of Breast Carcinoma and Metastatic Breast Cancer.

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ridinilazole DB15308
small molecule | CAS: 308362-25-6

Ridinilazole is under investigation in clinical trial NCT02092935 (A Study of SMT19969 Compared With Vancomycin for the Treatment of Clostridium Difficile-Associated Diarrhoea (CDAD)).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rifabutin Approved DB00615
small molecule | CAS: 72559-06-9

A broad-spectrum antibiotic that is being used as prophylaxis against disseminated Mycobacterium avium complex infection in HIV-positive patients.

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +27
Target Protein:
DNA-directed RNA polymerase subunit alphaDNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta' +2
Waktu Paruh45 (± 17) ho…
Vol. Distribusi-
Klirens* 0.69 +/- 0.32 L/h…
Genetik -
Rifalazil DB04934
small molecule | CAS: 129791-92-0

Rifalazil is a derivative of the antibiotic rifamycin. It is being investigated by ActivBiotics for the treatment of various bacterial infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics, Antitubercular +7
Target Protein:
DNA-directed RNA polymerase subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rifampin Approved DB01045
small molecule | CAS: 13292-46-1

Rifampin, also known as rifampicin, is a broad-spectrum antimicrobial [A263748] that was first discovered in 1965 [A263753] and clinically used in 1968.[A263768] Rifampin is used to treat tuberculosis and works by inhibiting the microbial DNA-dependent RNA po…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +55
Target Protein:
DNA-directed RNA polymerase subunit betaNuclear receptor subfamily 1 group I member 2
Waktu ParuhIn healthy adults, …
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Rifamycin Approved DB11753
small molecule | CAS: 6998-60-3

Rifamycin is the prime member of the rifamycin family which are represented by drugs that are a product of fermentation from the gram-positive bacterium _Amycolatopsis mediterranei_, also known as _Streptomyces mediterranei_. The parent compound of rifamycin …

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +49
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'DNA-directed RNA polymerase subunit beta +2
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik -
Rifapentine Approved DB01201
small molecule | CAS: 61379-65-5

Rifapentine is an antibiotic drug used in the treatment of tuberculosis. It inhibits DNA-dependent RNA polymerase activity in susceptible cells. Specifically, it interacts with bacterial RNA polymerase but does not inhibit the mammalian enzyme.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics, Antitubercular +24
Target Protein:
DNA-directed RNA polymerase subunit beta'
Waktu Paruh-
Vol. Distribusi* 70.2 ± 9.1 L
Klirens* Apparent Oral cl=…
Genetik -
Rifasutenizol DB18981
small molecule | CAS: 1001314-13-1

Rifasutenizol is under investigation in clinical trial NCT05857163 (Efficacy and Safety of Rifasutenizol (TNP 2198) in Participants With H. Pylori Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rifaximin Approved DB01220
small molecule | CAS: 80621-81-4

Rifaximin is a semisynthetic, rifamycin-based non-systemic antibiotic, meaning that the drug will not pass the gastrointestinal wall into the circulation as is common for other types of orally administered antibiotics. It has multiple indications and is used …

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA-directed RNA polymerase subunit betaNuclear receptor subfamily 1 group I member 2
Waktu ParuhApproximately 6 hou…
Vol. Distribusi-
Klirens-
Genetik -
Rigosertib DB12146
small molecule | CAS: 592542-59-1

Rigosertib has been used in trials studying the treatment and basic science of MDS, RAEB, Cancer, Hepatoma, and Neoplasms, among others.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +3
Target Protein:
Serine/threonine-protein kinase PLK1Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rilapladib DB05119
small molecule | CAS: 412950-08-4

Rilapladib is the third genomics-derived small molecule drug arising from the Human Genome Sciences-GlaxoSmithKline collaboration to enter clinical development. It is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor. Lp-PLA2 is an enzyme associat…

Kategori:
AcetatesAcids, AcyclicAmides +2
Target Protein:
Thymidine kinase, cytosolicPhospholipase A2Platelet-activating factor acetylhydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rilematovir DB15672
small molecule | CAS: 1383450-81-4

Rilematovir is under investigation in clinical trial NCT04056611 (Effects of JNJ-53718678 in Adult and Adolescent Participants Who Had a Hematopoietic Stem Cell Transplantation and Who Are Infected With Respiratory Syncytial Virus (RSV)).

Kategori:
Heterocyclic Compounds, Fused-RingImidazoles
Target Protein:
Fusion glycoprotein F0
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rilonacept Approved DB06372
biotech | CAS: 501081-76-1

Rilonacept is a dimeric fusion protein consisting of portions of IL-1R and the IL-1R accessory protein linked to the Fc portion of immunoglobulin G1. Rilonacept functions as an interleukin 1 inhibitor and is used in the treatment of CAPS, also known as cryopy…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +9
Target Protein:
Interleukin-1 betaInterleukin-1 alphaInterleukin-1 receptor antagonist protein
Waktu Paruh8.6 days
Vol. Distribusi-
Klirens-
Genetik -
Rilpivirine Approved DB08864
small molecule | CAS: 500287-72-9

Rilpivirine is non-nucleoside reverse transcriptase inhibitor (NNRTI) which is used for the treatment of HIV-1 infections in treatment-naive patients.[A31328] It is a diarylpyrimidine derivative.[A31329] The internal conformational flexibility of rilpivirine …

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +43
Target Protein:
Reverse transcriptase/RNaseHSodium channel protein type 10 subunit alphaGag-Pol polyprotein +1
Waktu ParuhRilpivirine has a t…
Vol. DistribusiIn HIV-1 patients, …
KlirensIn HIV-1 patients, …
Genetik -
Riltozinameran Approved DB17095
biotech | CAS: 2749948-25-0

The Omicron variant of SARS-CoV-2 is a variant of concern that was first reported in November 2021.[L43922] It tends to cause less severe disease but is significantly more virulent than both the original virus and earlier variants (e.g. Delta).[L43917] As of …

Kategori:
COVID-19 VaccinesmRNA VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rimiducid DB04974
small molecule | CAS: 195514-63-7

Rimiducid is a lipid-permeable tacrolimus analogue and a protein dimerizer. It was designed to overcome limitations of current cellular immunotherapies used for cancer and other blood disorders by enhancing the control of the immune cell activity and function…

Kategori:
Cross-Linking Reagents
Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1ASerine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rimonabant Approved DB06155
small molecule | CAS: 168273-06-1

Rimonabant is an anorectic anti-obesity drug produced and marketed by Sanofi-Aventis. It is an inverse agonist for the cannabinoid receptor CB1. Its main avenue of effect is reduction in appetite. Rimonabant is the first selective CB1 receptor blocker to be a…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Obesity Agents +12
Target Protein:
Cannabinoid receptor 1G-protein coupled receptor 55
Waktu Paruh6 to 9 days with no…
Vol. Distribusi-
Klirens-
Genetik -
Rimtuzalcap DB16733
small molecule | CAS: 2167246-24-2

Rimtuzalcap is a novel modulator of small-conductance calcium-activated potassium channels that is under investigation for the treatment of essential tremor.[L38414]

Target Protein:
Small conductance calcium-activated potassium channel protein 1Small conductance calcium-activated potassium channel protein 2Small conductance calcium-activated potassium channel protein 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5401–5450 dari 6694
Sebelumnya Halaman 109 / 134 Berikutnya