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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 109 / 236
small molecule | CAS: 53861-57-7

Deskripsi belum tersedia.

Kategori:
1-Carboxyglutamic AcidAcids, AcyclicAmino Acids +5
Target Protein:
ProthrombinCoagulation factor IXCoagulation factor X +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseGlutathione S-transferase Mu 4High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A
Waktu Paruh-
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Genetik -
Gamolenic acid Approved DB13854
small molecule | CAS: 506-26-3

Gamolenic acid, or gamma-linolenic acid (?-Linolenic acid) or GLA, is an essential fatty acid (EFA) comprised of 18 carbon atoms with three double bonds [F27] that is most commonly found in human milk and other botanical sources [A32848]. It is an omega-6 pol…

Kategori:
Agents that reduce seizure thresholdDermatologicalsFatty Acids +5
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Ganaplacide DB16173
small molecule | CAS: 1261113-96-5

Ganaplacide is under investigation in clinical trial NCT03167242 (Efficacy and Safety of KAF156 in Combination With LUM-SDF in Adults and Children With Uncomplicated Plasmodium Falciparum Malaria).

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Ganaxolone Approved DB05087
small molecule | CAS: 38398-32-2

Ganaxolone is the 3?-methylated synthetic analog of [allopregnanolone],[L41130] a metabolite of [progesterone].[A3197] Ganaxolone belongs to a class of compounds referred to as neurosteroids.[A3197] Endogenous neurosteroids, which comprise certain metabolites…

Kategori:
AnticonvulsantsCentral Nervous System DepressantsCytochrome P-450 CYP2B6 Substrates +14
Target Protein:
GABA(A) Receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiBoth ganaxolone and…
Klirens-
Genetik -
Gancotamab DB14784
biotech | CAS: 1509928-00-0

Gancotamab is under investigation in clinical trial NCT02213744 (MM-302 Plus Trastuzumab vs. Chemotherapy of Physician's Choice Plus Trastuzumab in HER2-Positive Locally Advanced/Metastatic Breast Cancer Patients).

Kategori:
Amino Acids, Peptides, and ProteinsAnthracyclinesAntibodies +16
Waktu Paruh-
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Genetik -
Gandotinib DB13040
small molecule | CAS: 1229236-86-5

Gandotinib has been used in trials studying the treatment of Myelofibrosis, Polycythemia Vera, Primary Myelofibrosis, Thrombocythemia, Essential, and Myeloproliferative Disorders, among others.

Kategori:
Janus Kinase 2, antagonists & inhibitorsJanus Kinases, antagonists & inhibitors
Target Protein:
Tyrosine-protein kinase JAK2
Waktu Paruh-
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Ganetespib DB12047
small molecule | CAS: 888216-25-9

Ganetespib is under investigation for the treatment of BREAST CANCER, Small Cell Lung Cancer, Acute Myeloid Leukaemia, and Myelodysplastic Syndrome.

Kategori:
HSP90 Heat-Shock Proteins, antagonists & inhibitors
Waktu Paruh-
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Genetik -
Ganglioside GM1 DB16948
small molecule | CAS: 116950-37-9

Deskripsi belum tersedia.

Waktu Paruh-
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Ganirelix Approved DB06785
small molecule | CAS: 124904-93-4

Ganirelix is a synthetic decapeptide and a competitive gonadotropin-releasing hormone (GnRH) antagonist. Derived from endogenous GnRH, ganirelix has amino acid substitutions. Ganirelix is indicated for controlled ovarian hyperstimulation in assisted reproduct…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Gonadotropin-Releasing HormonesDecreased GnRH Secretion +16
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean (SD) volum…
KlirensClearance following…
Genetik -
Ganitumab DB12205
biotech | CAS: 905703-97-1

Ganitumab has been used in trials studying the treatment of Colon Cancer, Rectal Cancer, Breast Cancer, Breast Tumors, and Breast Neoplasms, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Ganstigmine DB06525
small molecule | CAS: 457075-21-7

Ganstigmine is an orally active, geneserine derived, carbamate-based acetylcholinesterase inhibitor developed for the treatment of Alzheimer's disease.

Kategori:
Acids, AcyclicCarbamates
Target Protein:
Acetylcholinesterase
Waktu Paruh-
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Genetik -
Gantacurium DB05710
small molecule | CAS: 758669-50-0

Gantacurium chloride is a new, investigational, non-depolarizing ultra-short acting neuromuscular blocker. It is being developed by Avera Pharmaceuticals.

Kategori:
Anticholinergic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Neuronal acetylcholine receptor subunit alpha-3
Waktu Paruh3.09±0.21 minutes
Vol. Distribusi-
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Genetik -
Gantenerumab DB12034
biotech | CAS: 1043556-46-2

Alzheimer's disease (AD) is the most common cause of dementia in elderly patients, with classical histopathological hallmarks including extracellular amyloid-beta (A?) plaques and intraneuronal neurofibrillary tangles (NFTs). As the classical view of AD patho…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhGantenerumab admini…
Vol. Distribusi-
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Genetik -
Garenoxacin DB06160
small molecule | CAS: 194804-75-6

Garenoxacin, a quinolone antibiotic, is being investigated for the treatment of gram-positive and gram-negative bacterial infections.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garetosmab DB16379
biotech | CAS: 2097125-54-5

Fibrodysplasia ossificans progressiva (FOP) is a rare autosomal dominant disorder of episodic, progressive heterotropic ossification. FOP is characterized by episodic inflammatory episodes, which may be precipitated by trauma, including immunizations and mino…

Target Protein:
Inhibin beta A chain
Waktu Paruh-
Vol. DistribusiGaretosmab had a st…
KlirensWhen administered a…
Genetik -
Garivulimab DB16670
biotech | CAS: 2342597-81-1

Garivulimab is under investigation in clinical trial NCT03379259 (Study of BGB-A333 Alone and in Combination With Tislelizumab in Advanced Solid Tumors).

Waktu Paruh-
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Garlic oil DB15989
biotech | CAS: 8000-78-0

Deskripsi belum tersedia.

Kategori:
AlkenesAnionsAnticarcinogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gartisertib DB18770
small molecule | CAS: 1613191-99-3

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
biotech | CAS: 100040-31-1

Gastric inhibitory polypeptide is under investigation in clinical trial NCT03081676 (The Effect of GIP and GLP-1 on Insulin and Glucagon Secretion in Patients With HNF1A-diabetes Treated With or Without Sulphonylurea).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsGastrointestinal Agents +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Gatifloxacin Approved DB01044
small molecule | CAS: 112811-59-3

Gatifloxacin is an antibiotic agent and a member of the fourth-generation fluoroquinolone family. It works by inhibiting the bacterial enzymes DNA gyrase and topoisomerase IV. It was first introduced by Bristol-Myers Squibb in 1999 under the brand name Tequin…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh7-14 hours
Vol. Distribusi-
Klirens-
Genetik -
Gatipotuzumab DB18861
biotech | CAS: 1264737-26-9

Gatipotuzumab is under investigation in clinical trial NCT01899599 (Pankomab-gex™ Versus Placebo as Maintenance Therapy in Advanced Ovarian Cancer).

Waktu Paruh-
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Gatralimab DB16528
biotech | CAS: 1826020-80-7

Gatralimab is under investigation in clinical trial NCT02389452 (Study of Safety and Efficacy of 6 Ml Synvisc-one (Hylan G-F 20) in Indian Patients With Symptomatic Osteoarthritis of Knee(s) After Initial and Repeat Treatment).

Waktu Paruh-
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Genetik -
Gavestinel DB06741
small molecule | CAS: 153436-22-7

Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Gavestinel displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites and is o…

Kategori:
Excitatory Amino Acid AgentsExcitatory Amino Acid AntagonistsGlycine Agents +5
Target Protein:
Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2Glycine receptor subunit alpha-3 +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Gavocabtagene autoleucel is a novel cell therapy consisting of autologous genetically engineered T cells expressing a single-domain antibody that recognizes human Mesothelin, fused to the CD3-epsilon subunit which, upon expression, is incorporated into the en…

Waktu Paruh-
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Gavorestat DB16707
small molecule | CAS: 2170729-29-8

Gavorestat is under investigation in clinical trial NCT04902781 (Clinical Benefit, Safety, PK and PD Study of AT-007 in Pediatric Subjects With Classic Galactosemia).

Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Gaxilose Approved DB12767
small molecule | CAS: 14087-31-1

Gaxilose has been used in trials studying the diagnostic of Lactose Intolerance.

Kategori:
CarbohydratesOligosaccharidesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GB-115 DB19204
small molecule | CAS: 678996-63-9

GB-115 is under investigation in clinical trial NCT05586789 (A Study of the Efficacy and Safety of Ranquilon Tablets in Patients With Anxiety in Neurasthenia and Adjustment Disorders).

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GB-13 DB18387
biotech

GB-13 is a genetically engineered recombinant protein consisting of an IL13Ra2-targeted genetically engineered mutant of IL-13 and PE4E, a derivative of Pseudomonas exotoxin A.

Waktu Paruh-
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Genetik -
GB1211 DB17499
small molecule | CAS: 1978336-95-6

GB1211 is an orally active galectin-3 (Gal-3) inhibitor.

Waktu Paruh-
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Genetik -
GBR-12783 DB17027
small molecule | CAS: 145428-33-7

A selective inhibitor of dopamine uptake.[A252997]

Kategori:
Dopamine AgentsDopamine AgonistsDopamine Uptake Inhibitors +3
Waktu Paruh-
Vol. Distribusi-
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GBR-12879 DB17028
small molecule | CAS: 67469-43-6

Deskripsi belum tersedia.

Kategori:
Piperazines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GC-24 DB03788
small molecule

Deskripsi belum tersedia.

Target Protein:
Thyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GC-373 DB15797
small molecule

GC-373 is a peptide aldehyde which is metabolized from the bisulfide adduct, [GC-376 free acid][A219031,A219036]. It is an inhibitor of M<sup>pro</sup> (otherwise known as 3CL<sup>pro</sup>), a viral encoded protease that cleaves and activates functional prot…

Kategori:
AmidesAmino AcidsAmino Acids, Branched-Chain +3
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 1417031-79-8

GC-376 is a 3C-like protease (3CL<sup>pro</sup> or M<sup>pro</sup>) inhibitor that stops the cleavage and activation of functional viral proteins required for replication and transcription in host cells[A219036]. The compound is known as a direct acting antiv…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +15
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GC5107 DB17604
biotech

GC5107 is an investigational intravenous immunoglobulin. It is marketed as IVIG-SN.

Waktu Paruh-
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GCS-100 DB17566
biotech

Deskripsi belum tersedia.

Kategori:
Carbohydrates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0134 DB17079
small molecule | CAS: 1637394-01-4

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
GDC-0152 DB12380
small molecule | CAS: 873652-48-3

GDC-0152 has been used in trials studying the treatment of Solid Cancers.

Kategori:
Cycloparaffins
Target Protein:
E3 ubiquitin-protein ligase XIAP
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GDC-0349 DB13072
small molecule | CAS: 1207360-89-1

GDC-0349 has been used in trials studying the treatment of Non-Hodgkin's Lymphoma, Solid Tumor.

Kategori:
AmidesBenzene Derivatives
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0425 DB14791
small molecule | CAS: 1627539-18-7

GDC-0425 is under investigation in clinical trial NCT01359696 (A Study Evaluating the Safety, Tolerability, and Pharmacokinetics of GDC-0425 Administered With and Without Gemcitabine in Patients With Refractory Solid Tumors or Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GDC-0810 DB12253
small molecule | CAS: 1365888-06-7

ARN-810 has been used in trials studying the basic science and treatment of Breast Cancer.

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GDC-0917 DB12336
small molecule | CAS: 1446182-94-0

CUDC-427 has been used in trials studying the treatment of LYMPHOMA and Solid Cancers.

Waktu Paruh-
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Genetik -
GDC-0927 DB14934
small molecule | CAS: 2100830-77-9

GDC-0927 is under investigation in clinical trial NCT02316509 (A Study of GDC-0927 in Postmenopausal Women With Locally Advanced or Metastatic Estrogen Receptor Positive Breast Cancer).

Waktu Paruh-
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GDC-1971 DB17487
small molecule | CAS: 2377352-49-1

Deskripsi belum tersedia.

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GDP-L-fucose DB18689
small molecule | CAS: 15839-70-0

Deskripsi belum tersedia.

Waktu Paruh-
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GE-2270A DB02975
small molecule | CAS: 134861-34-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +2
Target Protein:
Elongation factor Tu
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Gebasaxturev DB17296
biotech | CAS: 2122169-83-7

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule | CAS: 921195-93-9

GED-0507-34-Levo is under investigation in clinical trial NCT02808390 (Efficacy and Safety Study of Ged-0507-34-levo for Treatment of UC).

Kategori:
Acids, CarbocyclicAmines
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
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Genetik -
Gedatolisib DB11896
small molecule | CAS: 1197160-78-3

Gedatolisib has been used in trials studying the basic science and treatment of Neoplasm, Ovary Cancer, Breast Cancer, Advanced Cancer, and Endometrial Cancer, among others.

Kategori:
Enzyme InhibitorsOxazinesProtein Kinase Inhibitors
Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
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Genetik -
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