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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 109 / 252
Ezogabine Approved DB04953
small molecule | CAS: 150812-12-7

Ezogabine (D23129) is a close structural analog of the centrally acting analgesic flupitrine. It is a neuronal potassium channel opener being developed as a first-in-class antiepileptic drug (AED) and is currently being studied in Phase 3 trials as an adjunct…

Kategori:
Acids, AcyclicAminesAniline Compounds +15
Target Protein:
Potassium voltage-gated channel subfamily KQT member 3Potassium voltage-gated channel subfamily KQT member 2Potassium voltage-gated channel subfamily KQT member 4 +1
Waktu ParuhTerminal half-life …
Vol. Distribusi8.7 L/kg
Klirens0.58 - 0.76 L/h·kg.…
Genetik -
Ezurpimtrostat DB16458
small molecule | CAS: 1914148-72-3

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ezutromid DB12888
small molecule | CAS: 945531-77-1

Ezutromid has been investigated for the treatment of Muscular Dystrophy, Duchenne.

Kategori:
Heterocyclic Compounds, Fused-RingMuscular Dystrophy, Duchenne
Target Protein:
Utrophin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
F-15599 DB16936
small molecule | CAS: 635323-95-4

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNeurotransmitter Agents +3
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 78-96-6

Deskripsi belum tersedia.

Target Protein:
Glutamate mutase sigma subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
F6-734 DB17444
biotech

F6-734 is a bispecific monoclonal antibody with affinity for anticarcinoembryonic antigen (CEA) and anti-diethylenetriamine pentaacetic acid (DTPA) (hMN-14 × m734).[A255217,A255222]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fabomotizole DB13623
small molecule | CAS: 173352-21-1

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsNervous System +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Facinicline DB05586
small molecule | CAS: 677306-35-3

Deskripsi belum tersedia.

Kategori:
Bridged-Ring CompoundsHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Factor XIII (human) Approved DB12909
biotech | CAS: 9013-56-3

Factor XIII (human) is a heat-treated, lyophilized concentrate of coagulation factor XIII, an endogenous enzyme responsible for the crosslinking of fibrin and an essential component of the coagulation cascade [FDA Label]. For people with congenital deficiency…

Kategori:
AcyltransferasesAmino Acids, Peptides, and ProteinsAminoacyltransferases +14
Waktu Paruh6.6 ±2.29 days [FDA…
Vol. DistribusiVss = 51.1 mL/kg (v…
Klirens0.25 ±0.09 mL/hr/kg…
Genetik -
Fagrocorat DB14676
small molecule | CAS: 1044535-52-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fagus grandifolia pollen Approved DB10350
biotech

Fagus grandifolia pollen is the pollen of the Fagus grandifolia plant. Fagus grandifolia pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Faldaprevir DB11808
small molecule | CAS: 801283-95-4

Faldaprevir has been investigated for the treatment of Chronic Hepatitis C.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Branched-Chain +16
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Falimarev DB17333
biotech | CAS: 685563-14-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fallypride DB15167
small molecule | CAS: 166173-78-0

Fallypride is under investigation in clinical trial NCT02310360 (Striatal and Extra-striatal Dopamine Release in Response to Food in Healthy Humans).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fallypride F-18 DB19254
small molecule | CAS: 166173-82-6

Fallypride F-18 is under investigation in clinical trial NCT00846040 (Reduced Carbohydrate Versus Fat in Obese Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Famitinib DB11741
small molecule | CAS: 1044040-56-3

Famitinib has been used in trials studying the treatment of Colorectal Cancer, Renal Cell Cancer, Colorectal Cancer Recurrent, Colorectal Cancer Metastatic, and Metastatic Renal Cell Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-RingReceptor Protein-Tyrosine Kinases, antagonists & inhibitors
Target Protein:
Platelet-derived growth factor receptor alphaReceptor-type tyrosine-protein kinase FLT3Mast/stem cell growth factor receptor Kit +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Famotidine Approved DB00927
small molecule | CAS: 76824-35-6

Famotidine is a competitive histamine-2 (H<sub>2</sub>) receptor antagonist that works to inhibit gastric acid secretion. It is commonly used in gastrointestinal conditions related to acid secretion, such as gastric ulcers and gastroesophageal reflux disease …

Kategori:
Acid ReducersAlimentary Tract and MetabolismAnti-Ulcer Agents +20
Target Protein:
Histamine H2 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensRenal clearance is …
Genetik -
Famphur DB11408
small molecule | CAS: 52-85-7

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Famprofazone DB16702
small molecule | CAS: 22881-35-2

Famprofazone is a nonsteroidal anti-inflammatory agent found in combination products such as ‘Gewodin’ which is marketed in Taiwan.[L34724] It is important to note that the drug is metabolized to [methamphetamine] and [amphetamine] in the body and can lead to…

Kategori:
AminesAmphetaminesAnalgesics +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Famtozinameran Approved DB17088
biotech

The Omicron variant of SARS-CoV-2 is a variant of concern that was first reported in November 2021.[L43922] It tends to cause less severe disease but is significantly more virulent than both the original virus and earlier variants (e.g. Delta).[L43917] As of …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fanapanel DB12393
small molecule | CAS: 161605-73-8

Fanapanel has been investigated for the treatment of Visual Acuity.

Kategori:
Heterocyclic Compounds, Fused-RingOrganophosphorus Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Farampator DB15012
small molecule | CAS: 211735-76-1

Farampator is under investigation in clinical trial NCT00113022 (Org 24448 to Treat Major Depression).

Kategori:
Oxazoles
Target Protein:
Glutamate receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Farglitazar DB19311
small molecule | CAS: 274687-78-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Faricimab Approved DB15303
biotech | CAS: 1607793-29-2

Retinal vascular diseases (RVDs) such as diabetic macular edema (DME), age-related macular degeneration (AMD), and retinal vein occlusion (RVO) are typically caused by retinal ischemia and subsequent neovascularization (NV).[A225985, A225990, A225995] Vascula…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Target Protein:
Vascular endothelial growth factor A, long formAngiopoietin-2
Waktu ParuhFaricimab has an es…
Vol. Distribusi-
Klirens-
Genetik -
Farletuzumab DB05595
biotech | CAS: 896723-44-7

Farletuzumab (MORAb-003) is a fully humanized monoclonal antibody against the folate receptor alpha, for the potential treatment of epithelial ovarian cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Folate receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2407465-18-1

Farletuzumab ecteribulin is under investigation in clinical trial NCT04300556 (A Study to Evaluate the Safety, Tolerability, and Efficacy of Morab-202 (Herein Referred to as Farletuzumab Ecteribulin), a Folate Receptor Alpha (Fr?)-targeting Antibody-drug Conj…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Farnesol DB02509
small molecule | CAS: 4602-84-0

A colorless liquid extracted from oils of plants such as citronella, neroli, cyclamen, and tuberose. It is an intermediate step in the biological synthesis of cholesterol from mevalonic acid in vertebrates. It has a delicate odor and is used in perfumery. (Fr…

Kategori:
AlcoholsFatty AlcoholsLipids +2
Target Protein:
Amine oxidase [flavin-containing] BBile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13058-04-3

Deskripsi belum tersedia.

Kategori:
OrganophosphatesOrganophosphorus CompoundsPotential QTc-Prolonging Agents +2
Target Protein:
Squalene synthaseProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaProtein farnesyltransferase subunit beta +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
OrganophosphatesOrganophosphorus CompoundsPotential QTc-Prolonging Agents +2
Target Protein:
Geranylgeranyl pyrophosphate synthaseMevalonate kinaseDehydrosqualene synthase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Faropenem DB12190
small molecule | CAS: 106560-14-9

Faropenem has been used in trials studying the treatment of Tuberculosis, Pulmonary Tuberculosis, and Community Acquired Pneumonia.

Kategori:
AmidesAntibacterials for Systemic UseAntiinfectives for Systemic Use +3
Target Protein:
Dihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 141702-36-5

Faropenem medoxomil is an ester prodrug derivative of the beta-lactam antibiotic [faropenem]. The prodrug form of faropenem offers dramatically improved oral bioavailability and leads to higher systemic concentrations of the drug. Faropenem medoxomil is a bro…

Kategori:
AmidesHeterocyclic Compounds, Fused-RingLactams +1
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 2BPeptidoglycan D,D-transpeptidase FtsI
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Farudodstat DB16049
small molecule | CAS: 1035688-66-4

Farudodstat (ASLAN003) is under investigation in clinical trial NCT03451084 (A Dose Optimisation Study of ASLAN003 in Acute Myeloid Leukemia).

Kategori:
AminesEnzyme InhibitorsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fasentin DB16759
small molecule | CAS: 392721-37-8

Deskripsi belum tersedia.

Kategori:
AmidesAminesAniline Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fasinumab DB12157
biotech | CAS: 1190239-42-9

Fasinumab is a human IgG1k monoclonal antibody targeted against nerve growth factor (NGF). It is currently under investigation for the treatment osteoarthritic pain[A241045] and has demonstrated significantly greater pain relief and functional improvement as …

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Beta-nerve growth factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fasitibant DB15646
small molecule | CAS: 869939-83-3

Fasitibant is under investigation in clinical trial NCT02205814 (Fasitibant Intra-articular Injection in Patients With Symptomatic Osteoarthritis of the Knee).

Kategori:
AmidesAmino AcidsAmino Acids, Basic +9
Target Protein:
B2 bradykinin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fasoracetam DB16163
small molecule | CAS: 110958-19-5

Fasoracetam is under investigation in clinical trial NCT03609619 (PART B: Efficacy and Safety of AEVI-001 in Children and Adolescents With ADHD and Without Mglur Mutations).

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fasudil DB08162
small molecule | CAS: 103745-39-7

Fasudil has been investigated in Carotid Stenosis.

Kategori:
Antiarrhythmic agentsCalcium Channel BlockersCalcium-Regulating Hormones and Agents +12
Target Protein:
Rho-associated protein kinase 1cAMP-dependent protein kinase inhibitor alphacAMP-dependent protein kinase catalytic subunit alpha +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Favezelimab DB16729
biotech | CAS: 2231068-83-8

Favezelimab is under investigation in clinical trial NCT04626479 (Substudy 03A: A Study of Immune and Targeted Combination Therapies in Participants With First Line (1L) Renal Cell Carcinoma (MK-3475-03A)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FavId DB05249
small molecule

FavId, is an active immunotherapy that is based upon unique genetic information extracted from a patient's tumor.

Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Favipiravir Approved DB12466
small molecule | CAS: 259793-96-9

Discovered by Toyama Chemical Co., Ltd. in Japan, favipiravir is a modified pyrazine analog that was initially approved for therapeutic use in resistant cases of influenza.[A191688,A191721] The antiviral targets RNA-dependent RNA polymerase (RdRp) enzymes, wh…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +11
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'RNA-directed RNA polymerase catalytic subunit
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe recommended ora…
Genetik -
small molecule | CAS: 49564-56-9

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsMuscle RelaxantsMuscle Relaxants, Peripherally Acting Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fazirsiran DB17891
biotech | CAS: 2175009-08-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fazpilodemab DB18924
biotech | CAS: 2517935-02-1

Fazpilodemab is under investigation in clinical trial NCT04171765 (A Study to Evaluate the Efficacy, Safety, and Pharmacokinetics of BFKB8488A Compared With Placebo in Participants With Non-alcoholic Steatohepatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FB-101 DB17956
small molecule

FB-101 is a c-Abl inhibitor. Developed by 1st Biotherapeutics, it is being investigated for the treatment of neurological disorders, such as Parkinson's Disease and amyotrophic lateral sclerosis (ALS).[L47102]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FB-825 DB17598
biotech

FB-825 is an investigational humanized monoclonal antibody that targets the C?mX domain of the membrane-bound IgE (mIgE), causing a depletion of mIgE positive B-cells. It is currently being investigated for immune disorders, such as atopic dermatitis and hype…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
fb-PMT DB17394
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FCR001 DB18595
biotech

FCR001 is a somatic cell therapy product containing hematopoietic progenitor cells (HPC), Facilitating Cells (FC), and alpha beta T cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Febantel DB11409
small molecule | CAS: 58306-30-2

Deskripsi belum tersedia.

Kategori:
AmidinesAnthelminticsAnti-Infective Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Febuxostat Approved DB04854
small molecule | CAS: 144060-53-7

Febuxostat is a non-purine xanthine oxidase (XO) inhibitor.[A39743] In early 2008, febuxostat was granted marketing authorization by the European Commission for the treatment of chronic hyperuricemia and gout.[A230548] In the following year, the FDA for appro…

Kategori:
Antigout PreparationsAntirheumatic AgentsBCRP/ABCG2 Inhibitors +15
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu ParuhThe apparent mean t…
Vol. DistribusiThe apparent steady…
KlirensFollowing oral admi…
Genetik -
Fecal microbiota Approved DB17743
biotech

Fecal microbiota, given either as a rectal transplant or in an oral formulation of live spores, is an FDA-approved option to prevent the recurrence of _Clostridioides difficile_ infection (CDI) in patients given an antibacterial treatment for recurrent CDI.[A…

Kategori:
Miscellaneous Therapeutic Agents
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
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