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14361

Total database: 17430
Struktur (SMILES)
9916 (69.0%)
Target
7893 (55.0%)
Genomik
112 (0.8%)
Referensi
14361 (100.0%)

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Hasil Pencarian (14361)

Halaman 108 / 288
Difluocortolone Approved DB09095
small molecule | CAS: 2607-06-9

Difluocortolone is a potent topical corticosteroid. It is commonly used in dermatology for the reduction of inflammation and itching. It was submitted to the FDA in July 1984 by the pharmaceutical company Schering AG.[L1082]

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +24
Target Protein:
Annexin A3Glucocorticoid receptor
Waktu ParuhThe half-life of di…
Vol. DistribusiLess of 1% of the a…
KlirensDiflucortolone gets…
Genetik -
small molecule | CAS: 15845-96-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Difluprednate Approved DB06781
small molecule | CAS: 23674-86-4

Difluprednate is a topical corticosteroid indicated for the treatment of infammation and pain associated with ocular surgery. It is a butyrate ester of 6(?), 9(?)-difluoro prednisolone acetate. Difluprednate is abbreviated DFBA, or difluoroprednisolone butyra…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +17
Target Protein:
Glucocorticoid receptorAnnexin A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Digitoxin Approved DB01396
small molecule | CAS: 71-63-6

A cardiac glycoside sometimes used in place of digoxin. It has a longer half-life than digoxin; toxic effects, which are similar to those of digoxin, are longer lasting. (From Martindale, The Extra Pharmacopoeia, 30th ed, p665)

Kategori:
Antiarrhythmic agentsCarbohydratesCardanolides +21
Target Protein:
Sodium/potassium-transporting ATPase subunit beta-2Sodium/potassium-transporting ATPase subunit beta-3Sodium/potassium-transporting ATPase subunit alpha-1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Digoxin Approved DB00390
small molecule | CAS: 20830-75-5

Digoxin is one of the oldest cardiovascular medications used today.[A178225] It is a common agent used to manage atrial fibrillation and the symptoms of heart failure.[A178234] Digoxin is classified as a cardiac glycoside and was initially approved by the FDA…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +28
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-2Sodium/potassium-transporting ATPase subunit alpha-3Sodium/potassium-transporting ATPase subunit beta-1 +4
Waktu ParuhDigoxin has a half-…
Vol. DistribusiThis drug is widely…
KlirensThe clearance of di…
Genetik -
Digoxin Immune Fab (Ovine) Approved DB00076
biotech

Digoxin Immune Fab is a sheep antibody (26-10) FAB fragment from sheep immunized with the digoxin derivative Digoxindicarboxymethylamine. It is used as an antidote for overdose of digoxin.

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesBlood Proteins +6
Target Protein:
Digoxin
Waktu Paruh15-20 hrs
Vol. Distribusi* 0.3 L/kg [DigiFab…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
mRNA-capping enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 97067-70-4

Dihematoporphyrin ether is under investigation in clinical trial NCT00118222 (High Light and Low Light Dose PDT in Glioma).

Kategori:
Antineoplastic AgentsBiological FactorsDermatologicals +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1783-84-2

A 20-carbon-chain fatty acid, unsaturated at positions 8, 11, and 14. It differs from arachidonic acid, 5,8,11,14-eicosatetraenoic acid, only at position 5.

Kategori:
Dietary SupplementsEicosanoidsFatty Acids +3
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydralazine Approved DB12945
small molecule | CAS: 484-23-1

Dihydralazine is under investigation in clinical trial NCT00311974 (The Effect of Dihydralazine on Kidney Function and Hormones in Healthy Individuals).

Kategori:
Antihypertensive AgentsArteriolar Smooth Muscle, Agents Acting OnCardiovascular Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydrexidine DB12890
small molecule | CAS: 123039-93-0

Dihydrexidine has been used in trials studying the treatment of SPD, Cocaine-Related Disorders, and Schizotypal Personality Disorder.

Kategori:
Dopamine AgentsDopamine AgonistsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
D(1A) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 959343-20-5

Deskripsi belum tersedia.

Kategori:
Anticholinergic AgentsNicotinic Antagonists
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydro-alpha-ergocryptine Approved DB11274
small molecule | CAS: 25447-66-9

Alpha-dihydroergocryptine is usually referred to the mixture of the alpha and beta dihydroergocryptine. These two compounds are differentiated in the position of a methyl group. This structural difference is due to a proteinogenic amino acid replacement from …

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates
Target Protein:
5-hydroxytryptamine receptor 75-hydroxytryptamine receptor 2BD(2) dopamine receptor +2
Waktu ParuhAlpha-dihydroergocr…
Vol. DistribusiIn preclinical stud…
KlirensIn preclinical stud…
Genetik -
Dihydrocapsiate DB15398
small molecule | CAS: 205687-03-2

Dihydrocapsiate is under investigation in clinical trial NCT00999297 (Effect of 4-week Dihydrocapsiate Ingestion on Resting Metabolic Rate).

Kategori:
AlkaloidsAlkenesAlkynes +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydrocodeine Approved DB01551
small molecule | CAS: 125-28-0

Dihydrocodeine is an opioid analgesic used as an alternative or adjunct to codeine to treat moderate to severe pain, severe dyspnea, and cough. It is semi-synthetic, and was developed in Germany in 1908 during an international search to find a more effect…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +19
Target Protein:
Mu-type opioid receptor
Waktu Paruh4h
Vol. DistribusiThe disposition of …
KlirensPlasma clearance is…
Genetik -
Dihydroergocornine Approved DB11273
small molecule | CAS: 25447-65-8

Dihydroergocornine is one of the dihydrogenated ergot compounds that present very large hypotensive effects.[A32962] It is an artificial derivative of the crude extract of ergot and later purified, ergocornine.[A32964] The formation of dihydroergocornine impl…

Kategori:
Agents that produce hypertensionAlkaloidsCytochrome P-450 CYP3A Substrates +10
Target Protein:
Serotonin ReceptorsBeta adrenergic receptorAlpha adrenergic receptor
Waktu ParuhTo know more about …
Vol. DistribusiTo know more about …
KlirensNo pharmacokinetic …
Genetik -
Dihydroergocristine Approved DB13345
small molecule | CAS: 17479-19-5

Dihydroergocristine is part of the ergoloid mixture products.[L2637] It is a semisynthetic ergot alkaloid and thus, it is characterized by a structural skeleton formed by an alkaloid ergoline.[A32879] To know more about ergoloid mixtures, please visit [DB0104…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAgents that produce hypertension +13
Target Protein:
Serotonin ReceptorsAlpha-2C adrenergic receptorBeta adrenergic receptor +2
Waktu ParuhThe half-life of di…
Vol. DistribusiDihydroergocristine…
KlirensDihydroergocristine…
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAlkaloidsAnti-Parkinson Drugs +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydroergotamine Approved DB00320
small molecule | CAS: 511-12-6

A 9,10alpha-dihydro derivative of [ergotamine]. Dihydroergotamine is used as an abortive therapy for migraines.[L38469] Its use has largely been supplanted by triptans in current therapy due to the class's greater selectivity and more favourable side effect p…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +37
Target Protein:
5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1F +13
Waktu ParuhDHE exhibits a biph…
Vol. DistribusiDHE has a steady-st…
KlirensThe total clearance…
Genetik -
small molecule | CAS: 14357-76-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 29505-79-1

Deskripsi belum tersedia.

Target Protein:
L-xylulose reductasePhosphate-binding protein PstS
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 462-20-4

Deskripsi belum tersedia.

Kategori:
AntioxidantsBiological FactorsCoenzymes +7
Target Protein:
Glycine cleavage system H protein, mitochondrialDihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, mitochondrial[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydromorphine DB01565
small molecule | CAS: 509-60-4

A semisynthetic analgesic used in the study of narcotic receptors. It has abuse potential. [PubChem]

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +12
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 27200-12-0

Dihydromyricetin is under investigation in clinical trial NCT03606694 (Effect of Dihydromirycetin on Glycemic Control, Insulin Sensitivity and Insulin Secretion in Type 2 Diabetes Mellitus).

Kategori:
BenzopyransChromonesFlavonoids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydrostreptomycin Approved DB11512
small molecule | CAS: 128-46-1

Dihydrostreptomycin is an aminoglycoside antibiotic. In humans, the use of dihydrostreptomycin has been associated with ototoxicity. The FDA withdrew its approval for the use of all drug products containing dihydrostreptomycin sulfate.[L43942]

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydrotachysterol Approved DB01070
small molecule | CAS: 67-96-9

A vitamin D that can be regarded as a reduction product of vitamin D2.

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCholestanes +14
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydrouracil DB01849
small molecule | CAS: 504-07-4

Deskripsi belum tersedia.

Kategori:
PyrimidinesPyrimidinones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydrouridine DB17822
small molecule | CAS: 5627-05-4

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 96-26-4

A ketotriose compound. Its addition to blood preservation solutions results in better maintenance of 2,3-diphosphoglycerate levels during storage. It is readily phosphorylated to dihydroxyacetone phosphate by triokinase in erythrocytes. In combination with na…

Kategori:
CarbohydratesKetosesMonosaccharides +1
Target Protein:
Dihydroxyacetone kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 57-04-5

Dihydroxyacetone phosphate is an important intermediate in lipid biosynthesis and in glycolysis. Dihydroxyacetone phosphate has been investigated for the treatment of Lymphoma, Large-Cell, Diffuse.

Kategori:
CarbohydratesSugar Phosphates
Target Protein:
Fructose-bisphosphate aldolase ATriosephosphate isomeraseFructose-bisphosphate aldolase B +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 19309-14-9

Cardamonin (also known as Dihydroxymethoxychalcone), as shown by the increasing number of publications, has received growing attention from the scientific community due to the expectations toward its benefits to human health. Cardamonin's name comes from the …

Kategori:
BenzopyransChromonesFlavonoids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 162870-29-3

Deskripsi belum tersedia.

Kategori:
AlcoholsEthylene GlycolsGlycols
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 534-08-7

Deskripsi belum tersedia.

Kategori:
AlcoholsAntiseptics and DisinfectantsDermatologicals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diiodohydroxyquinoline Approved DB09115
small molecule | CAS: 83-73-8

Diiodohydroxyquinoline, also known as uidoquinol and iodoquinol, is a quinoline derivative that can be used in the treatment of amoebiasis. The exact mechanism of action is unknown. Iodoquinol is not currently available in any FDA-approved products.

Kategori:
AmebicidesAnti-Infective AgentsAntiparasitic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diisopromine DB13476
small molecule | CAS: 5966-41-6

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1445-75-6

Deskripsi belum tersedia.

Target Protein:
Parathion hydrolaseParathion hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Dipeptidyl peptidase 4Subtilisin BPN'Complement factor B +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dilanubicel DB18722
biotech

Dilanubicel consists of ex vivo expanded hematopoietic stem and progenitor cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dilazep DB13715
small molecule | CAS: 35898-87-4

Deskripsi belum tersedia.

Kategori:
AzepinesCardiac TherapyCardiovascular Agents +2
Target Protein:
Equilibrative nucleoside transporter 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dilmapimod DB12140
small molecule | CAS: 444606-18-2

Dilmapimod has been used in trials studying the treatment and diagnostic of Nerve Trauma, Inflammation, Pain, Neuropathic, Arthritis, Rheumatoid, and Coronary Heart Disease, among others. Dilmapimod (SB-681323) is a p38 MAP-kinase inhibitor that has potential…

Kategori:
p38 Mitogen-Activated Protein Kinases, antagonists & inhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase 14Tumor necrosis factorInterleukin-1 beta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diloxanide DB08792
small molecule | CAS: 579-38-4

Diloxanide (as [Diloxanide furoate]) is an anti-protozoal drug used in the treatment of Entamoeba histolytica and some other protozoal infections. Although it is not currently approved for use in the United States, it was approved by a CDC study in the treatm…

Kategori:
AmebicidesAnti-Infective AgentsAntiparasitic Agents +4
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Diloxanide furoate Approved DB14638
small molecule | CAS: 3736-81-0

Deskripsi belum tersedia.

Kategori:
AmebicidesAnti-Infective AgentsAntiparasitic Agents +1
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Dilpacimab DB16140
biotech | CAS: 1791420-09-1

Dilpacimab is under investigation in clinical trial NCT03368859 (A Study of ABT-165 Plus FOLFIRI vs Bevacizumab Plus FOLFIRI in Subjects With Metastatic Colorectal Cancer Previously Treated With Fluoropyrimidine, Oxaliplatin and Bevacizumab).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diltiazem Approved DB00343
small molecule | CAS: 42399-41-7

Diltiazem is a benzothiazepine derivative with antihypertensive and vasodilating properties. Approved in 1982 by the FDA, it is a member of the non-dihydropyridine calcium channel blockers drug class. It works through various mechanisms of action, but it prim…

Kategori:
Agents causing hyperkalemiaAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAntiarrhythmic agents +44
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent calcium channel gamma-1 subunit
Gen Terkait:
ADRB1
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensFollowing a single …
Genetik 1 Varian
Dimazole Approved DB13858
small molecule | CAS: 95-27-2

Dimazole (diamthazole) is an antifungal. It was withdrawn in Franch in 1972 due to neuropsychiatric reactions.

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimenhydrinate Approved DB00985
small molecule | CAS: 523-87-5

Dimehydrinate was first described in the literature in 1949,[A233120] and patented in 1950.[L32995] Early research into dimenhydrinate focused on its role as an antihistamine for urticaria; the treatment of motion sickness was an accidental discovery.[A233130…

Kategori:
AlkaloidsAminesAminoalkyl Ethers +21
Target Protein:
Histamine H1 receptor
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Dimenoxadol DB01461
small molecule | CAS: 509-78-4

Dimenoxadol is an opioid analgesic which produces typical opioid effects such as analgesia and sedation. It is structurally similar to methadone and is a benzilic acid derivative. In the United States it is classified as a Schedule I controlled drug.

Kategori:
Acids, CarbocyclicDiphenylacetic AcidsHydroxy Acids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimepheptanol DB19094
small molecule | CAS: 545-90-4

Dimepheptanol is under investigation in clinical trial NCT00218127 (Treatment of Opioid/heroin Dependence: Comparison of Three Medication Dosing Regimens).

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +5
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimercaprol Approved DB06782
small molecule | CAS: 59-52-9

Dimercaprol is a traditional chelating agent developed by British biochemists at Oxford University during World War II. It was developed as an experimental antidote against the arsenic-based poison gas Lewisite. It has been used clinically since 1949 in arsen…

Kategori:
AntidotesChelating AgentsCompounds used in a research, industrial, or household setting +7
Target Protein:
ArsenicCadmiumMercury +1
Waktu ParuhThe drug has a shor…
Vol. Distribusi-
Klirens-
Genetik -
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