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6694

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4518 (67.5%)
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3751 (56.0%)
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Halaman 108 / 134
RCT1100 DB18830
biotech

RCT1100 is an investigational mRNA-based therapeutic that aims to treat primary ciliary dyskinesia caused by pathogenic mutations in DNAI1.[L50788]

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RDP58 DB06566
small molecule

RDP58 (NH2-arg-norleucine (nle)-nle-arg-nle-nle-nle-gly-tyr-CONH2) (Sangstat Corp., Fremont, California) is a novel synthetic peptide that inhibits early signal transduction pathways for the expression of inflammatory cytokines.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +3
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Rebeccamycin DB14729
small molecule | CAS: 93908-02-2

Rebeccamycin is a weak topoisomerase I inhibitor isolated from _Nocardia sp_.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
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Recaticimab DB19302
biotech | CAS: 2361290-85-7

Recaticimab is under investigation in clinical trial NCT06467617 (Adebrelimab Plus Chemo and Recaticimab Perioperative Treatment for Resectable NSCLC).

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biotech

Receptor binding domain SARS-CoV-2 Hepatitis B surface antigen virus-like particle vaccine (RBD SARS-CoV-2 HBsAg VLP vaccine), is a virus-like particle vaccine candidate where the RBD antigen is conjugated to the hepatitis B surface antigen[A226593]. Virus-li…

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Recifercept DB17899
biotech | CAS: 2226238-09-9

Deskripsi belum tersedia.

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Recilisib DB18310
small molecule | CAS: 334969-03-8

Deskripsi belum tersedia.

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biotech

Alpha 1-antitrypsin is a glycoprotein primarily produced by hepatocytes, and to a lesser extent, immune system cells. Recombinant alpha 1-antitrypsin (rAAT) is produced from yeast, which unlike commercially available forms of plasma-derived AAT, eliminates th…

Target Protein:
Alpha-1-antitrypsin
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biotech

B38-CAP is structured as a carboxypeptidase and derived from _Paenibacillus sp._ The molecule, an Angiotensin Converting Enzyme 2 (ACE2)-like enzyme, shares structural similarities to the mammalian ACE2. B38-CAP is an ACE2-like enzyme which decreases angioten…

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biotech

Deskripsi belum tersedia.

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biotech

Recombinant CD40-ligand is under investigation in clinical trial NCT00053391 (Vaccine Therapy in Treating Patients With Stage III or Stage IV Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +8
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biotech

Deskripsi belum tersedia.

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biotech

The Recombinant SARS-CoV-2 Vaccine was created by inserting genes of the SARS-CoV-2 spike protein’s receptor-binding domain into a baculovirus expression system[F4738, A226853]. In pre-clinical trial testing on mice, rabbits, and non-human primates, the candi…

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biotech

Recombinant stabilized RSV B prefusion F antigen is one component of a bivalent respiratory syncytial virus (RSV) vaccine called Abrysvo. The vaccine comprises two antigens - the other being [recombinant stabilized RSV A prefusion F antigen] - which have been…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
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biotech

Recombinant stabilized RSV B prefusion F antigen is one component of a bivalent respiratory syncytial virus (RSV) vaccine called Abrysvo. The vaccine comprises two antigens - the other being [recombinant stabilized RSV A prefusion F antigen] - which have been…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
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Redasemtide DB19121
biotech | CAS: 1606186-88-2

Redasemtide is under investigation in clinical trial NCT05953480 (A Phase 2b, Randomized, Double-blind Study of Redasemtide (S-005151) in Adult Participants With Acute Ischemic Stroke).

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Regorafenib Approved DB08896
small molecule | CAS: 755037-03-7

Regorafenib is an orally-administered inhibitor of multiple kinases. It is used for the treatment of metastatic colorectal cancer, advanced gastrointestinal stromal tumours, and hepatocellular carcinoma. FDA approved on September 27, 2012. Approved use of Reg…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +31
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +15
Waktu ParuhRegorafenib, 160 mg…
Vol. DistribusiRegorafenib undergo…
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Regramostim DB05386
biotech | CAS: 127757-91-9

Regramostim (GM-CSF) is a differentially glycosylated factor produced mainly by activated T cells and macrophages. Endothelial cells and fibroblasts can also produce GM-CSF after exposure to TNF-?, IL-1, IL-2 and IFN-?. GM-CSF is found associated with extrace…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +10
Target Protein:
Granulocyte-macrophage colony-stimulating factor receptor subunit alphaGM-CSF receptor alpha subunit
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small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase Chk1
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Relamorelin DB12678
small molecule | CAS: 661472-41-9

Relamorelin has been investigated for the treatment and basic science of Gastroparesis, Gastric Motility, Diabetes Mellitus, Parkinson's Disease, and Chronic Constipation, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Relatlimab Approved DB14851
biotech | CAS: 1673516-98-7

Relatlimab is a human IgG4 monoclonal antibody and novel immune checkpoint inhibitor that targets lymphocyte activation gene-3 (LAG-3).[A246165,L41265] It was the first commercially developed anti-LAG-3 antibody, entering clinical trials in 2013,[A246155] and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Lymphocyte activation gene 3 protein
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensAt steady-state, th…
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Relebactam Approved DB12377
small molecule | CAS: 1174018-99-5

Relebactam is a diazabicyclooctane beta-lactamase inhibitor, similar in structure to [avibactam].[A181195,A181207] It includes a piperidine ring which reduces export from bacterial cells by producing a positive charge.[A181207] It is currently available in a …

Kategori:
Antibacterials for Systemic UseAntiinfectives for Systemic UseAza Compounds +6
Target Protein:
Beta-lactamaseBeta-lactamase TEMBeta-lactamase SHV-1 +3
Waktu ParuhRelebactam has a ha…
Vol. DistribusiRelebactam has a vo…
KlirensRelebactam has a re…
Genetik -
biotech

Deskripsi belum tersedia.

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Reloxaliase DB15560
biotech | CAS: 202011-67-4

Reloxaliase is a crystalline formulation of oxalate decarboxylase derived from _Bacillus Subtilis_. Reloxaliase is under investigation in clinical trial NCT03456830 (Evaluate ALLN-177 in Patients With Enteric Hyperoxaluria).

Kategori:
Carbon-Carbon LyasesEnzymesEnzymes and Coenzymes +1
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Reloxiliase DB17653
biotech

Reloxiliase is a first-in-class, oral crystalline formulation of the oxalate-specific, microbial enzyme oxalate decarboxylase. It is being investigated for the treatment of hyperoxaluria.[A258823]

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Reltecimod DB16687
small molecule | CAS: 1447799-33-8

Reltecimod is under investigation in clinical trial NCT02469857 (Phase III Efficacy and Safety Study of AB103 in the Treatment of Patients With Necrotizing Soft Tissue Infections).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Differentiation +7
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Relugolix Approved DB11853
small molecule | CAS: 737789-87-6

Relugolix is a gonadotropin-releasing hormone (GnRH) receptor antagonist used in the treatment of several hormone-responsive conditions. It was first approved in Japan in 2019, under the brand name Relumina, for the symptomatic treatment of uterine fibroids,[…

Kategori:
AmidesAnti-Gonadotropin-Releasing HormonesAntiandrogens +30
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe average effecti…
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KlirensThe average renal c…
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Remdesivir Approved DB14761
small molecule | CAS: 1809249-37-3

Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) is the causative agent of coronavirus disease 2019 (COVID-19), which is a respiratory disease that is capable of progressing to viral pneumonia and acute respiratory distress syndrome (ARDS); COVID-…

Kategori:
Adenine NucleotidesAmino AcidsAmino Acids, Peptides, and Proteins +37
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1abReplicase polyprotein 1ab +1
Waktu ParuhRemdesivir has an e…
Vol. DistribusiData regarding the …
KlirensData regarding the …
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Remestemcel-L Approved DB13973
biotech

Remestemcel-L is a third-party, off-the-shelf suspension of ex-vivo cultured adult human mesenchymal stem cells intended for intravenous infusion. The mesenchymal stem cells are derived from the bone marrow of unrelated and human leukocyte antigen (HLA)–unmat…

Kategori:
Anti-Infective AgentsAnti-Inflammatory AgentsAntiviral Agents +6
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Remifentanil Approved DB00899
small molecule | CAS: 132875-61-7

Remifentanil (marketed by Abbott as Ultiva) is a potent ultra short-acting synthetic opioid given to patients during surgery for pain relief and adjunctive to an anaesthetic. Remifentanil is a specific mu-type-opioid receptor agonist which means it reduces sy…

Kategori:
Acids, AcyclicAgents producing tachycardiaAgents that produce hypertension +24
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh1-20 minutes
Vol. Distribusi* 350 mL/kg * 452 …
Klirens* 40 mL/min/kg [you…
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Remikiren DB00212
small molecule | CAS: 126222-34-2

Remikiren is an orally active, high specificity renin inhibitor.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAntihypertensive AgentsCardiovascular Agents +3
Target Protein:
Renin
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small molecule | CAS: 442201-24-3

Remogliflozin etabonate has been used in trials studying the treatment and basic science of Type 2 Diabetes Mellitus and Diabetes Mellitus, Type 2.

Kategori:
Blood Glucose Lowering AgentsCarbohydratesGlycosides +1
Target Protein:
Sodium/glucose cotransporter 2Probable glucose sensor protein SLC5A4
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Remoxipride Approved DB00409
small molecule | CAS: 80125-14-0

Remoxipride is an atypical antipsychotic agent that is specific for dopamine D<sub>2</sub> receptors.[A215422] It gained approval in the UK in 1989 but was withdrawn in 1993 after it was found to be associated with an increased incidence of aplastic anemia.[A…

Kategori:
Acids, CarbocyclicAmidesAntipsychotic Agents +21
Target Protein:
D(2) dopamine receptorD(4) dopamine receptorD(3) dopamine receptor +2
Waktu ParuhThe half life of re…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
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Remternetug DB18994
biotech | CAS: 2571940-41-3

Remternetug is under investigation in clinical trial NCT05463731 (A Study of Remternetug (LY3372993) in Participants With Alzheimer's Disease (TRAILRUNNER-ALZ 1)).

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Repaglinide Approved DB00912
small molecule | CAS: 135062-02-1

Repaglinide is an oral antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). It belongs to the meglitinide class of short-acting insulin secretagogues, which act by binding to ? cells of the pancreas to stimulate i…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBlood Glucose Lowering Agents +14
Target Protein:
ATP-binding cassette sub-family C member 9ATP-binding cassette sub-family C member 8Histamine H1 receptor +1
Waktu Paruh1 hour
Vol. Distribusi31 L following IV a…
Klirens33-38 L/hour follow…
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Repotrectinib Approved DB16826
small molecule | CAS: 1802220-02-5

Repotrectinib is a next-generation tyrosine kinase inhibitor (TKI) specifically designed to address resistance in the treatment of non-small cell lung cancer (NSCLC), specifically due to mutations in the ROS1 gene.[A262056] ROS1 mutations are one of the defin…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +28
Target Protein:
Proto-oncogene tyrosine-protein kinase ROSHigh affinity nerve growth factor receptorBDNF/NT-3 growth factors receptor +1
Waktu ParuhThe repotrectinib m…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
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Reproterol DB12846
small molecule | CAS: 54063-54-6

Reproterol has been used in trials studying the treatment of Asthma, Exercise-Induced.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +25
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biotech | CAS: 2085240-27-1

AT132 is under investigation in clinical trial NCT03199469 (Gene Transfer Clinical Study in X-linked Myotubular Myopathy).

Kategori:
Adeno-associated Viral Vector Therapies
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Rescinnamine Approved DB01180
small molecule | CAS: 24815-24-5

Rescinnamine is an angiotensin-converting enzyme inhibitor used as an antihypertensive drug. It is an alkaloid obtained from _Rauwolfia serpentina_ and other species of _Rauwolfia_.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +11
Target Protein:
Angiotensin-converting enzyme
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Reserpine Approved DB00206
small molecule | CAS: 50-55-5

An alkaloid found in the roots of Rauwolfia serpentina and R. vomitoria. Reserpine inhibits the uptake of norepinephrine into storage vesicles resulting in depletion of catecholamines and serotonin from central and peripheral axon terminals. It has been used …

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAlkaloids +37
Target Protein:
Synaptic vesicular amine transporterChromaffin granule amine transporterBaculoviral IAP repeat-containing protein 5
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Resiniferatoxin DB06515
small molecule | CAS: 57444-62-9

Resiniferatoxin (RTX) is a naturally occurring, ultrapotent capsaicin analog that activates the vanilloid receptor in a subpopulation of primary afferent sensory neurons involved in nociception (the transmission of physiological pain).

Kategori:
NeurotoxinsTerpenes
Target Protein:
Transient receptor potential cation channel subfamily V member 1
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Resiquimod DB06530
small molecule | CAS: 144875-48-9

A substance being studied in the treatment of some types of skin cancer. When put on the skin, resiquimod causes some immune cells to make certain chemicals that may help them kill tumor cells. It is also being studied to find out if adding it to a tumor vacc…

Kategori:
Immunologic FactorsImmunomodulatory AgentsToll-Like Receptor Agonists
Target Protein:
Toll-like receptor 7Toll-like receptor 8
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Reslizumab Approved DB06602
biotech | CAS: 241473-69-8

Reslizumab is a humanized interleukin-5 (IL-5) antagonist monoclonal antibody (IgG4 kappa) that is produced by recombinant DNA technology in murine myeloma non-secreting 0 (NS0) cells. IL-5 is a pro-inflammatory cytokine that is responsible for the growth and…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntibodies +12
Target Protein:
Interleukin-5
Waktu ParuhThe half-life is ap…
Vol. DistribusiThe approximate vol…
KlirensReslizumab clearanc…
Genetik -
Resmetirom Approved DB12914
small molecule | CAS: 920509-32-6

Resmetirom is a thyroid hormone receptor-beta (THR-beta) agonist. On March 14, 2024, it was approved by the FDA as the first treatment of liver fibrosis due to noncirrhotic non-alcoholic steatohepatitis (NASH), which is a form of non-alcoholic fatty liver dis…

Kategori:
BCRP/ABCG2 InhibitorsBCRP/ABCG2 SubstratesBSEP/ABCB11 Inhibitors +15
Target Protein:
Thyroid hormone receptor beta
Waktu ParuhThe median terminal…
Vol. DistribusiResmetirom apparent…
KlirensThe steady state ap…
Genetik -
Resminostat DB12392
small molecule | CAS: 864814-88-0

Resminostat has been used in trials studying the treatment of Sezary Syndrome, Mycosis fungoides, Hodgkin's Lymphoma, Hepatocellular Carcinoma, and Lymphoma, T-Cell, Cutaneous, among others.

Kategori:
AmidesAminesHydroxy Acids +3
Target Protein:
Histone deacetylase 1
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Resolvin E1 DB13105
small molecule | CAS: 552830-51-0

Resolvin E1 (RX 10001) is under investigation in clinical trial NCT00941018 (Single and Multiple Ascending Oral Dose Study of Resolvin E1 in Healthy Volunteers).

Kategori:
Dietary FatsDietary Fats, UnsaturatedEicosanoids +7
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Resorcinol Approved DB11085
small molecule | CAS: 108-46-3

Resorcinol is a 1,3-isomer (or meta-isomer) of benzenediol with the formula C6H4(OH)2. It is used as an antiseptic and disinfectant in topical pharmaceutical products in the treatment of skin disorders and infections such as acne, seborrheic dermatitis, eczem…

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseAnti-Infective Agents +8
Target Protein:
Carbonic anhydrase 12Carbonic anhydrase 2Carbonic anhydrase 14 +2
Waktu ParuhSpecific data regar…
Vol. DistribusiSpecific data regar…
KlirensSpecific data regar…
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Resorcinol monoacetate Approved DB15480
small molecule | CAS: 102-29-4

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesPhenols
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RESP301 DB16497
small molecule

RESP301 was under investigation in clinical trials for various conditions. It was studied in community patients at risk of viral infections, including SARS-CoV-2, in a terminated trial (NCT04858451) and adults with rifampicin-susceptible pulmonary tuberculosi…

Kategori:
Experimental Unapproved Treatments for COVID-19
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biotech

Arexvy (respiratory syncytial virus vaccine, adjuvanted) is an adjuvanted vaccine developed by GlaxoSmithKline Biologicals. It comprises lyophilized recombinant respiratory syncytial virus glycoprotein F (RSVPreF3) stabilized in pre-fusion conformation as the…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
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