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11778

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8554 (72.6%)
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6383 (54.2%)
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11778 (100.0%)

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Halaman 108 / 236
Fusarium graminearum Approved DB13907
biotech

Fusarium graminearum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Fusicoccin DB01780
small molecule | CAS: 20108-30-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesMycotoxins
Target Protein:
14-3-3 protein epsilon
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Fusidic acid Approved DB02703
small molecule | CAS: 6990-06-3

An antibiotic isolated from the fermentation broth of Fusidium coccineum. (From Merck Index, 11th ed) It acts by inhibiting translocation during protein synthesis. It is often used topically in creams and eyedrops but is available in systemic formulations inc…

Kategori:
Agents Causing Muscle ToxicityAnti-Bacterial AgentsAnti-Infective Agents +35
Target Protein:
Elongation factor GChloramphenicol acetyltransferaseChloramphenicol acetyltransferase 3
Waktu ParuhApproximately 5 to …
Vol. Distribusi-
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Genetik -
Futibatinib Approved DB15149
small molecule | CAS: 1448169-71-8

Futibatinib is an inhibitor of Fibroblast Growth Factor receptor (FGFR), which comprises a group of receptor tyrosine kinases that play a key role in cell proliferation, differentiation, migration, and survival. FGFR was investigated in oncology as a therapeu…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +10
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +1
Waktu ParuhThe mean (CV%) elim…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Futuximab DB15262
biotech | CAS: 1310460-85-5

Futuximab is under investigation in clinical trial NCT01955473 (Japanese Phase 1 Trial of Sym004 in Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Genetik -
G100 DB17244
biotech

Deskripsi belum tersedia.

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G17DT Immunogen DB04914
biotech

G17DT Immunogen is a vaccine that neutralizes gastrin-17, a hormone required for the growth of a number of cancers of the gastrointestinal tract. It is in phase III trials for advanced pancreatic cancer as a monotherapy and in combination with gemcitabine. It…

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +10
Waktu Paruh-
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G207 DB05827
biotech

G207 is cancer-killing viruses, so-called oncolytic viruses, for the treatment of various forms of cancer developed by MediGene AG. These viruses are specific herpes simplex viruses, or HSVs, generally known as the cause of cold sores. MediGene uses these vir…

Waktu Paruh-
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G305 DB17292
biotech

G305 is a [recombinant NY-ESO-1 protein] plus glucopyranosyl lipid A (GLA) in a stable emulsion (SE). G305 is an active component of CMB305 along with [LV305].[L47346]

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Gabaculine DB02054
small molecule | CAS: 87980-11-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins +2
Target Protein:
Ornithine aminotransferase, mitochondrialGlutamate-1-semialdehyde 2,1-aminomutase
Waktu Paruh-
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Genetik -
Gabapentin Approved DB00996
small molecule | CAS: 60142-96-3

Gabapentin is a structural analogue of the inhibitory neurotransmitter gamma-aminobutyric acid ([GABA]) that was first approved for use in the United States in 1993.[L8717] It was originally developed as a novel anti-epileptic for the treatment of certain typ…

Kategori:
Acids, AcyclicAcids, CarbocyclicAmines +24
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1Gamma-aminobutyric acid type B receptor subunit 2Gamma-aminobutyric acid type B receptor subunit 1 +5
Waktu ParuhThe elimination t<s…
Vol. DistribusiThe apparent volume…
KlirensBoth the plasma cle…
Genetik -
Gabapentin enacarbil Approved DB08872
small molecule | CAS: 478296-72-9

Gabapentin enacarbil is marketed under the name Horizant. It is a prodrug of gabapentin, and indicated in adults for the treatment of Restless Legs Syndrome (RLS) and postherpetic neuralgia (PHN).

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +6
Target Protein:
Sodium-dependent multivitamin transporterVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent calcium channel subunit alpha-2/delta-2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance of …
Genetik -
Gaboxadol DB06554
small molecule | CAS: 64603-91-4

Gaboxadol also known as 4,5,6,7-tetrahydroisoxazolo(5,4-c)pyridin-3-ol (THIP) is an experimental sleep aid drug developed by Lundbeck and Merck, who reported increased deep sleep without the reinforcing effects of benzodiazepines. Development of Gaboxadol was…

Kategori:
AnalgesicsAnestheticsAnticonvulsants +8
Target Protein:
Gamma-aminobutyric acid receptor subunit delta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gadobenic acid Approved DB00743
small molecule | CAS: 113662-23-0

Gadobenic acid, usually available in the salt form gadobenate dimeglumine, is a linear MRI gadolinium-based contrast agent (GBCA) used primarily for MR imaging of the liver.[A263086] It differs from other GBCAs due to the benzene ring that confers weak protei…

Kategori:
AlcoholsAmino SugarsCarbohydrates +14
Target Protein:
Albumin
Waktu ParuhGadobenate ion has …
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
Gadobutrol Approved DB06703
small molecule | CAS: 770691-21-9

Gadobutrol is a second-generation extracellular non-ionic macrocyclic GBCA (gadolinium-based contrast agent) used in magnetic resonance imaging (MRI) in adults and children older than 2 years of age. Due to its physicochemical properties, gadobutrol is formu…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +5
Waktu ParuhFor adult patients,…
Vol. DistribusiIn children aged 2 …
KlirensIn healthy subjects…
Genetik -
Gadofosveset trisodium Approved DB06705
small molecule | CAS: 193901-90-5

Gadofosveset trisodium is an intravenous contrast agent used with magnetic resonance angiography(MRA), which is a non-invasive way of imaging blood vessels. The agent allows for the vascular system to be imaged more clearly by the MRA. In this way, gadofosves…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +11
Target Protein:
Albumin
Waktu Paruh18.5 hours
Vol. Distribusi48 ± 16 mL/kg
Klirens6.57 ± 0.97 mL/h/kg…
Genetik -
Gadolinium Approved DB12091
small molecule | CAS: 7440-54-2

Gadolinium is under investigation in Hypertension, ACUTE KIDNEY INJURY, and Chronic Kidney Disease. Gadolinium has been investigated for the basic science of CAD, Multiple Sclerosis, and Coronary Artery Disease.

Kategori:
Anti-Inflammatory AgentsCompounds used in a research, industrial, or household settingContrast Media +5
Waktu Paruh-
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Genetik -
small molecule | CAS: 22541-19-1

Deskripsi belum tersedia.

Kategori:
Gadolinium-based Contrast AgentMagnetic Resonance Contrast Activity
Waktu Paruh-
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Genetik -
Gadopentetic acid Approved DB00789
small molecule | CAS: 80529-93-7

A complex of gadolinium with a chelating agent, diethylenetriamine penta-acetic acid (DTPA see pentetic acid), that is given to enhance the image in cranial and spinal MRIs. (From Martindale, The Extra Pharmacopoeia, 30th ed, p706)

Kategori:
AcetatesAcids, AcyclicAmines +12
Target Protein:
6-phosphogluconate dehydrogenase, decarboxylating
Waktu ParuhDistribution half l…
Vol. Distribusi* 266 ± 43 mL/kg
Klirens* 1.94 +/- 0.28 mL/…
Genetik -
Gadopiclenol Approved DB17084
small molecule | CAS: 933983-75-6

Gadopiclenol is a gadolinium-based contrast agent (GBCA) based on a pyclen macrocyclic structure. It is indicated for use with magnetic resonance imaging (MRI) to detect and visualize lesions with abnormal vascularity in the central nervous system and the bod…

Kategori:
Contrast MediaDiagnostic Uses of ChemicalsGadolinium-based Contrast Agent +5
Waktu ParuhGadopiclenol has a …
Vol. DistribusiAt steady state, th…
KlirensGadopiclenol has a …
Genetik -
Gadoteric acid Approved DB09132
small molecule | CAS: 72573-82-1

Gadoteric acid, commonly used in the salt form gadoterate meglumine, is a macrocyclic, ionic gadolinium-based contrast agent (GBCA).[A263131] It is composed of the organic acid DOTA (1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid) used for its chel…

Kategori:
AlcoholsAmino SugarsCarbohydrates +12
Waktu ParuhFollowing an intrav…
Vol. DistribusiThe volume of distr…
KlirensIn healthy subjects…
Genetik -
Gadoteridol Approved DB00597
small molecule | CAS: 120066-54-8

Gadoteridol is a macrocyclic nonionic gadolinium that provides contrast enhancement of the brain, spine, and surrounding tissues, resulting in improved visualization (compared with unenhanced MRI) of lesions with abnormal vascularity or those thought to disru…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +10
Waktu ParuhThe elimination hal…
Vol. DistribusiThe plasma distribu…
KlirensThe renal and plasm…
Genetik -
Galactose Approved DB11735
small molecule | CAS: 59-23-4

Galactose has been used in trials studying the treatment and diagnosis of Hepatitis C, Hepatic Cancer, Wilsons Disease, Diabetic Macular Oedema, and Focal Segmental Glomerulosclerosis, among others. There are even proposals for its use in accelerating senesce…

Kategori:
CarbohydratesContrast MediaDiagnostic Agents +4
Waktu ParuhReadily accessible …
Vol. DistribusiIt has been documen…
KlirensIn subjects with no…
Genetik -
Galantamine Approved DB00674
small molecule | CAS: 357-70-0

Galantamine is a tertiary alkaloid and reversible, competitive inhibitor of the acetylcholinesterase (AChE) enzyme, which is a widely studied therapeutic target used in the treatment of Alzheimer's disease.[A1018] First characterized in the early 1950s, galan…

Kategori:
AlkaloidsAmaryllidaceae AlkaloidsAnti-Dementia Drugs +22
Target Protein:
AcetylcholinesteraseNeuronal acetylcholine receptor subunit alpha-7Muscle nicotinic acetylcholine receptor +1
Waktu ParuhGalantamine has a t…
Vol. DistribusiThe mean volume of …
KlirensThe renal clearance…
Genetik -
Galcanezumab Approved DB14042
biotech | CAS: 1578199-75-3

Galcanezumab is a humanized monoclonal antibody developed by Eli Lilly and Company against human calcitonin gene-related peptide (CGRP).[A33105] Although several small-molecule CGRP receptor antagonists have been developed, humanized monoclonal antibodies lik…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +15
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhBetween 1 and 600 m…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
GALE-301 DB17262
biotech

GALE-301 is an investigational cancer immunotherapy. It is made up of E39, an immunogenic peptide derived from the folate binding protein (FBP), and an immune adjuvant, granulocyte macrophage-colony stimulating factor (GM-CSF).[A254696,L44166,L44171]

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GALE-302 DB17962
biotech

Deskripsi belum tersedia.

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Galegenimab DB18860
biotech | CAS: 2403683-24-7

Galegenimab is under investigation in clinical trial NCT03972709 (A Study Assessing the Safety, Tolerability, and Efficacy of Galegenimab (FHTR2163) in Participants With Geographic Atrophy Secondary to Age-related Macular Degeneration (AMD)).

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Galicaftor DB14894
small molecule | CAS: 1918143-53-9

Galicaftor is under investigation in clinical trial NCT03540524 (A Study Looking at the Safety, Tolerability and Efficacy of the Combination of the Study Drugs GLPG2451 and GLPG2222 With or Without GLPG2737 in Patients With Cystic Fibrosis.).

Kategori:
Acids, CarbocyclicBenzene DerivativesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Galidesivir DB11676
small molecule | CAS: 249503-25-1

Galidesivir is an adenosine analogue that has been investigated for use against Zaire Ebolavirus.[A191451] In animal studies, galidesivir was effective in increasing the survival rates from infections caused by various pathogens, including Ebola, Marburg, Yel…

Kategori:
Anti-Infective AgentsAntiviral AgentsCarbohydrates +9
Target Protein:
RNA-directed RNA polymerase L
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Galinpepimut-S DB17271
biotech

Deskripsi belum tersedia.

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Galiximab DB04901
biotech | CAS: 357613-77-5

Galiximab is a chimeric monoclonal antibody which is used as an immunosuppressive drug.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +7
Target Protein:
T-lymphocyte activation antigen CD80
Waktu Paruh13 to 24 days
Vol. Distribusi-
Klirens-
Genetik -
Gallamine DB13584
small molecule | CAS: 153-76-4

Deskripsi belum tersedia.

Kategori:
AminesAnticholinergic AgentsCentral Nervous System Depressants +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gallium cation DB14524
small molecule | CAS: 22537-33-3

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Gallium chloride Ga-67 Approved DB14550
small molecule

Gallium chloride Ga-67 is the chloride salt of a gallium radioisotope which is typically complexed with [sodium citrate] to generate [gallium citrate Ga 67], which can be used to image certain cancers and inflammatory lesions.[L12705]

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Gallium citrate DB17893
small molecule | CAS: 27905-02-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicCompounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +8
Waktu Paruh-
Vol. Distribusi-
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Gallium citrate Ga-67 Approved DB06784
small molecule | CAS: 41183-64-6

Gallium citrate Ga 67 is the citrate salt of the radioisotope gallium Ga 67. Although the mechanism is unknown, gallium Ga 67 concentrates in lysosomes and is bound to a soluble intracellular protein in certain viable primary and metastatic tumors and focal s…

Kategori:
GalliumGallium RadioisotopesRadioactive Diagnostic Agent +1
Waktu Paruh78.26 hours
Vol. Distribusi-
Klirens-
Genetik -
Gallium Ga-68 gozetotide Approved DB16019
small molecule | CAS: 1906894-20-9

Gallium (Ga) 68 prostate-specific membrane antigen (PSMA)-11, or Ga-68 gozetotide, is a radiopharmaceutical agent used to identify and assess prostate-specific membrane antigen (PSMA)-positive lesions in adult men with prostate cancer during positron emission…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +14
Target Protein:
Prostate-specific antigenGlutamate carboxypeptidase 2
Waktu ParuhGallium-68 (Ga-68) …
Vol. DistribusiGa-68 PSMA-11 accum…
KlirensThere is limited in…
Genetik -
small molecule | CAS: 108560-70-9

Gallium maltolate is Titan’s novel oral agent in development for the potential treatment of chronic bacterial infections, bone disease and cancer.

Kategori:
GalliumPyrans
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gallium nitrate Approved DB05260
small molecule | CAS: 13494-90-1

Gallium nitrate is a nitrate salt of [DB14524], a heavy metal that has been used as a diagnostic agent.[A260816] Gallium nitrate is reported to possess antiresorptive and hypocalcemic effects on bone.[A17097] GANITE, a product of gallium nitrate previously us…

Kategori:
Antineoplastic AgentsBone Resorption InhibitionCalcium Resorption Inhibitor +6
Target Protein:
Interleukin-1 betaRibonucleoside-diphosphate reductase subunit M2V-type proton ATPase subunit B, brain isoform
Waktu ParuhIn phase I studies …
Vol. DistribusiIn phase I studies …
KlirensIn cancer patients …
Genetik -
Gallopamil DB12923
small molecule | CAS: 16662-47-8

Gallopamil has been used in trials studying the treatment of Asthma.

Kategori:
Agents causing hyperkalemiaAminesAntiarrhythmic agents +17
Target Protein:
Sarcoplasmic/endoplasmic reticulum calcium ATPase 2Angiotensin-converting enzymeNeprilysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Galsulfase Approved DB01279
biotech | CAS: 552858-79-4

Galsufase is a variant form of the polymorphic human enzyme N-acetylgalactosamine 4-sulfatase of recombinant DNA origin. Galsulfase is a glycoprotein with a molecular weight of approximately 56 kD. The recombinant protein is comprised of 495 amino acids and c…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsArylsulfatases +9
Target Protein:
Dermatan sulfate
Waktu Paruh9 (6 to 21) minutes…
Vol. DistribusiWeek 1: 56-323 mL/k…
Klirens-
Genetik -
Galunisertib DB11911
small molecule | CAS: 700874-72-2

Galunisertib has been used in trials studying the basic science and treatment of Glioma, Neoplasms, Solid Tumor, GLIOBLASTOMA, and Prostate Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
TGF-beta receptor type-1Transforming growth factor beta-1 proprotein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Gam-COVID-Vac DB15848
biotech

Gam-COVID-Vac was created by Gamaleya Research Institute of Epidemiology and MIcrobiology in Russia. The vaccine candidate is a heterologous COVID-19 vaccine containing two components, recombinant adenovirus type 26 (rAd26) vector and recombinant adenovirus t…

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Gambir DB14298
biotech | CAS: 8001-48-7

Gambir is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Gamithromycin DB11416
small molecule | CAS: 145435-72-9

Gamithromycin is an antibiotic used in cattle.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsLactones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 17465-86-0

Gamma cyclodextrin is under investigation in clinical trial NCT03931057 (The use of ADV6209 for Premedication in Pediatric Anesthesia).

Kategori:
CarbohydratesCyclodextrinsDextrins +4
Waktu Paruh-
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Genetik -
small molecule

Adenylic acid. Adenine nucleotide containing one phosphate group esterified to the sugar moiety in the 2&#39;-, 3&#39;-, or 5&#39;-position. [PubChem]

Target Protein:
NH(3)-dependent NAD(+) synthetaseGlycerol kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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