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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 107 / 236
Fosigotifator DB19409
small molecule | CAS: 2415715-84-1

Fosigotifator is under investigation in clinical trial NCT05757141 (An Open-label Exploratory Study of ABBV-CLS-7262 Subjects With Vanishing White Matter Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosinopril Approved DB00492
small molecule | CAS: 98048-97-6

Fosinopril is a phosphinic acid-containing ester prodrug that belongs to the angiotensin-converting enzyme (ACE) inhibitor class of medications. It is rapidly hydrolyzed to fosinoprilat, its principle active metabolite. Fosinoprilat inhibits ACE, the enzyme r…

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +17
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh12 hours
Vol. Distribusi-
Klirens* 26 - 39 mL/min [h…
Genetik -
Fosinoprilat DB14207
small molecule | CAS: 95399-71-6

Fosinoprilat is the active phosphinic acid metabolite of prodrug [fosinopril], which is activated by esterases in vivo. It binds zinc with phosphinic acid group.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foslevodopa Approved DB16683
small molecule | CAS: 97321-87-4

Foslevodopa is under investigation in clinical trial NCT04750226 (Study to Assess Adverse Events and Change in Disease Activity of 24-hour Continuous Subcutaneous Infusion of ABBV-951 in Adult Participants With Advanced Parkinson's Disease).

Kategori:
Anti-Parkinson DrugsDopa and Dopa DerivativesDopamine Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foslinanib DB16172
small molecule | CAS: 1256037-60-1

Foslinanib is under investigation in clinical trial NCT03600233 (Study of CVM-1118 for Patients With Advanced Neuroendocrine Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosmanogepix DB15183
small molecule | CAS: 2091769-17-2

Fosmanogepix is under investigation in clinical trial NCT03604705 (An Efficacy and Safety Study of APX001 in Non-Neutropenic Patients With Candidemia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosnetupitant Approved DB14019
small molecule | CAS: 1703748-89-3

In April 2018, the U.S. Food and Drug Administration (FDA) and the Swiss company Helsinn approved the intravenous formulation of AKYNZEO® (NEPA, a fixed antiemetic combination of fosnetupitant, 235mg, and palonosetron, 0.25mg) as an alternative treatment opti…

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Inhibitors +6
Target Protein:
Substance-P receptor
Waktu ParuhNetupitant is elimi…
Vol. DistribusiThe mean SD volume …
KlirensNetupitant has a me…
Genetik -
Fospropofol Approved DB06716
small molecule | CAS: 258516-89-1

Fospropofol is a water soluble prodrug and is converted to propofol in the liver. Fospropofol is a short acting hypnotic/sedative/anesthetic agent. Unlike propofol, does not cause injection-site pain as it is unable to activate TRPA1. FDA approved in December…

Kategori:
Agents that reduce seizure thresholdAnestheticsAnesthetics, General +5
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit beta-3
Waktu ParuhWhen given to a pat…
Vol. DistribusiFospropofol = 0.33±…
KlirensTotal body clearanc…
Genetik -
Fosravuconazole DB15204
small molecule | CAS: 351227-64-0

Fosravuconazole is under investigation in clinical trial NCT03378661 (BENDITA BEnznidazole New Doses Improved Treatment and Associations).

Kategori:
Antifungals for Dermatological UseAntifungals for Systemic UseDermatologicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fostamatinib Approved DB12010
small molecule | CAS: 901119-35-5

Fostamatinib has been investigated for the treatment and basic science of Rheumatoid Arthritis and Immune Thrombocytopenic Purpura (ITP). It was approved on April 17, 2018, under the trade name Tavalisse for use in ITP [L2644, FDA Label]. Fostamatinib has als…

Kategori:
AminesBCRP/ABCG2 InhibitorsBlood and Blood Forming Organs +17
Target Protein:
Tyrosine-protein kinase SYKAdenosine receptor A3Synaptic vesicular amine transporter +297
Waktu ParuhR406 has a half-lif…
Vol. DistribusiR406 has an apparen…
KlirensR406 has an apparen…
Genetik -
Fostemsavir Approved DB11796
small molecule | CAS: 864953-29-7

Fostemsavir is the phosphonooxymethyl prodrug of temsavir, a novel HIV-1 attachment inhibitor.[L14867] It binds to and inhibits the activity of gp120, a subunit within the HIV-1 gp160 envelope glycoprotein that facilitates the attachment of HIV-1 to host cell…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +18
Target Protein:
Envelope glycoprotein gp160
Waktu ParuhThe half-life of te…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Fotemustine DB04106
small molecule | CAS: 92118-27-9

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAmidesAntineoplastic Agents +3
Target Protein:
Thioredoxin reductase 1, cytoplasmic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FOV 2501 DB17886
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 141790-23-0

Fozivudine Tidoxil has been used in trials studying the treatment of HIV Infections.

Kategori:
DeoxyribonucleosidesDideoxynucleosidesNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR-234938 DB03220
small molecule | CAS: 256461-79-7

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR117016 DB02616
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR221647 DB02096
small molecule | CAS: 256461-28-6

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR230513 DB03572
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR239087 DB03370
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fradafiban DB06472
small molecule | CAS: 148396-36-5

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesPlatelet Glycoprotein GPIIb-IIIa Complex, antagonists & inhibitors
Target Protein:
Integrin alpha-IIbIntegrin beta-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frangula purshiana bark Approved DB15478
biotech | CAS: 8015-89-2

Deskripsi belum tersedia.

Kategori:
Biological ProductsCascaraLaxatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fraxinus latifolia pollen Approved DB10723
biotech

Fraxinus latifolia pollen is the pollen of the Fraxinus latifolia plant. Fraxinus latifolia pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fremanezumab Approved DB14041
biotech | CAS: 1655501-53-3

Fremanezumab is a humanized monoclonal antibody targeted against human calcitonin gene-related peptide (CGRP) for the prevention of migraine headaches.[L11749] It was developed by Teva Pharmaceuticals USA and approved by the FDA in September 2018.[L11779] Alo…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +12
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhThe mean half-life …
Vol. DistribusiFremanezumab has an…
KlirensThe apparent cleara…
Genetik -
Freneslerbart DB19080
biotech | CAS: 2453195-94-1

Freneslerbart is under investigation in clinical trial NCT04981717 (A Study to Examine the Efficacy and Safety of Anti-fel D 1 Antibodies Injections in Cat-allergic Adolescent and Adult Patients With Allergic Rhinitis Who Live With a Cat).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fresolimumab DB12396
biotech | CAS: 948564-73-6

Fresolimumab has been used in trials studying the treatment of Primary Brain Tumors, Metastatic Breast Cancer, Diffuse Systemic Sclerosis, Pleural Malignant Mesothelioma, and Primary Focal Segmental Glomerulosclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frexalimab DB18926
biotech | CAS: 2515463-86-0

Frexalimab is under investigation in clinical trial NCT06141486 (Efficacy and Safety Study of Frexalimab (SAR441344) in Adults With Nonrelapsing Secondary Progressive Multiple Sclerosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Friulimicin B DB06087
small molecule | CAS: 239802-15-4

Friulimicin B is a naturally occurring antibiotic produced by a micro-organism, *Actinoplanes friuliensis*. It shows strong cidal activity against a number of Gram-positive pathogens which commonly cause serious infections in hospital patients and which are b…

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Froniglutide DB16178
biotech | CAS: 1417579-81-7

Glymera is under investigation in clinical trial NCT01658501 (Phase 2b Multicenter, Randomized, Double-blind, Placebo- and Active-controlled, Parallel-group Study to Assess the PD Response and Safety of Three Dose Levels of (PB1023) Injection Following 20 Wee…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frovatriptan Approved DB00998
small molecule | CAS: 158747-02-5

Frovatriptan is a triptan drug developed by Vernalis for the treatment of migraine headaches, in particular those associated with menstruation. Frovatriptan causes vasoconstriction of arteries and veins that supply blood to the head.

Kategori:
Agents that produce hypertensionAminesAnalgesics +23
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B
Gen Terkait:
GNB3
Waktu Paruh26 hours
Vol. Distribusi* 4.2 L/kg [males] …
Klirens* 220 mL/min [male …
Genetik 1 Varian
Frovocimab DB15089
biotech | CAS: 1643672-70-1

Frovocimab is under investigation in clinical trial NCT01671085 (A Study of LY3015014 in Healthy Participants With High Cholesterol).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fructose Approved DB04173
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +12
Target Protein:
Maltoporin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glucosamine-6-phosphate deaminase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frunexian DB18771
small molecule | CAS: 1803270-60-1

Deskripsi belum tersedia.

Kategori:
AmidesAminesPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fruquintinib Approved DB11679
small molecule | CAS: 1194506-26-7

Fruquintinib is a novel small-molecule anti-VEGFR that targets VEGFR-1,-2, and -3 to inhibit angiogenesis. Tumor angiogenesis is one of the most critical biological processes for increasing oxygen and nutrient supply to cancer cells, and the VEGF/VEGFR pathwa…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +10
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3
Waktu ParuhThe fruquintinib's …
Vol. DistribusiThe mean (SD) appar…
KlirensThe apparent cleara…
Genetik -
FS-1502 DB19287
biotech

FS-1502 is an antibody-drug conjugate consisting of an anti-HER2 antibody, linker, and Monomethylauristatin F.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FT-1101 DB17553
small molecule | CAS: 1776060-36-6

FT-1101 is a novel Bromodomain and Extra-Terminal motif (BET) inhibitor.[A257301] FT-1101 is under investigation in clinical trial NCT02543879 (Study of a Novel BET Inhibitor FT-1101 in Patients With Relapsed or Refractory Hematologic Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FT516 DB15732
biotech

FT516 is an investigational and engineered off-the-shelf natural killer (NK) cell therapy originating from induced pluripotent stem cells (iPSC). This compound expresses a high-affinity 158V, CD16 (hnCD16) Fc receptor that has an enhanced binding ability to t…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucitol DB03815
small molecule | CAS: 13074-06-1

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydrates
Target Protein:
L-fucose isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucoxanthin DB15462
small molecule | CAS: 3351-86-8

Fucoxanthin is under investigation in clinical trial NCT03613740 (Effect of Fucoxanthin on the Components of the Metabolic Syndrome, Insulin Sensitivity and Insulin Secretion). Fucoxanthin isis a marine carotenoid mainly found in brown algae, giving them a br…

Kategori:
AlkenesBiological FactorsCarotenoids +7
Target Protein:
NF-kappa-B inhibitor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fulvestrant Approved DB00947
small molecule | CAS: 129453-61-8

Fulvestrant is a drug treatment of hormone receptor (HR)-positive metastatic breast cancer in post-menopausal women with disease progression following anti-estrogen therapy. It is an estrogen receptor antagonist with no agonist effects, which works both by do…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +20
Target Protein:
Estrogen receptor
Waktu Paruh40 days
Vol. Distribusi* 3 to 5 L/kg
Klirens-
Genetik -
Fumaric acid DB01677
small molecule | CAS: 110-17-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntipsoriaticsAntipsoriatics for Topical Use +2
Target Protein:
Interferon gammaMalate dehydrogenaseFumarate reductase flavoprotein subunit +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Funapide DB11769
small molecule | CAS: 1259933-16-8

Funapide has been used in trials studying the treatment of Pharmacokinetics, Postherpetic Neuralgia, and Osteoarthritis of the Knee.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Sodium channel protein type 9 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaltadone DB16567
small molecule | CAS: 139-91-3

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryFurans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaprevir DB12785
small molecule | CAS: 1435923-88-8

Furaprevir is under investigation in clinical trial NCT01523990 (A Study to Evaluate the Safety, Tolerability, and PK in Healthy Volunteers and HCV Genotype 1 Infected Patients).

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaprofen DB06499
small molecule | CAS: 67700-30-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazidin DB13475
small molecule | CAS: 1672-88-4

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazolidone DB00614
small molecule | CAS: 67-45-8

A nitrofuran derivative with antiprotozoal and antibacterial activity. Furazolidone binds bacterial DNA which leads to the gradual inhibition of monoamine oxidase. (From Martindale, The Extra Pharmacopoeia, 30th ed, p514)

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Infective Agents +20
Target Protein:
DNA
Waktu Paruh10 minutes
Vol. Distribusi-
Klirens-
Genetik -
Furosemide Approved DB00695
small molecule | CAS: 54-31-9

Furosemide is a potent loop diuretic that acts on the kidneys to ultimately increase water loss from the body. It is an anthranilic acid derivative.[L7958] Furosemide is used for edema secondary to various clinical conditions, such as congestive heart failure…

Kategori:
Acids, CarbocyclicAmidesAmines +30
Target Protein:
Solute carrier family 12 member 1Carbonic anhydrase 2G-protein coupled receptor 35
Waktu ParuhThe half-life from …
Vol. DistribusiThe volume of distr…
KlirensFollowing intraveno…
Genetik -
Furvina DB16547
small molecule | CAS: 189935-72-6

Furvina (G1) is an antimicrobial agent active against Gram-positive and Gram-negative bacteria, yeasts, and filamentous fungi. Furvina is marketed in Cuba as Dermofural®, an ointment containing G1 as the only active principle ingredient. It is used to treat d…

Kategori:
AlkenesAnti-Infective AgentsHydrocarbons, Acyclic
Target Protein:
30S ribosomal protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusafungine Approved DB08965
small molecule | CAS: 1393-87-9

Fusafungine is an antibiotic from Fusarium lateririum, and is used for the treatment of respiratory infections.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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