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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 107 / 272
Disopyramide Approved DB00280
small molecule | CAS: 3737-09-5

A class I anti-arrhythmic agent (one that interferes directly with the depolarization of the cardiac membrane and thus serves as a membrane-stabilizing agent) with a depressant action on the heart similar to that of guanidine. It also possesses some anticholi…

Kategori:
Agents producing tachycardiaAntiarrhythmic agentsAntiarrhythmics, Class I +21
Target Protein:
Sodium channel protein type 5 subunit alphaMuscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +5
Waktu Paruh6.7 hours (range 4-…
Vol. Distribusi-
Klirens-
Genetik -
Disperse Blue 106 Approved DB14203
small molecule | CAS: 68516-81-4

Disperse Blue 106 is used in allergenic testing.

Kategori:
AllergensAntigensBiological Factors +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Distearyldimonium Approved DB14143
small molecule | CAS: 14357-21-2

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAminesAmmonium Compounds +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Distigmine DB13694
small molecule | CAS: 17299-00-2

Distigmine is a parasympathomimetic agent with a longer duration of action and enhanced drug accumulation compared to [DB00545] and [DB01400]. It is an anticholinergic drug and long-acting reversible carbamate cholinesterase inhibitor that binds directly and …

Kategori:
Cholinergic AgentsCholinesterase InhibitorsEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disufenton DB17298
small molecule | CAS: 168021-77-0

Deskripsi belum tersedia.

Kategori:
AntioxidantsArylsulfonatesArylsulfonic Acids +9
Target Protein:
Extracellular sulfatase Sulf-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dithiazanine DB11516
small molecule | CAS: 7187-55-5

Dithiazanine is a highly potent anthelmintic, introduced in 1959 for the treatment of strongyloid worms and whipworms. However, its use is severely limited due to its toxicity. Dithiazanine iodide was associated with eight fatal cases of severe acidosis and s…

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6892-68-8

A compound that, along with its isomer, Cleland's reagent (dithiothreitol), is used for the protection of sulfhydryl groups against oxidation to disulfides and for the reduction of disulfides to sulfhydryl groups. [PubChem]

Kategori:
AlcoholsCarbohydratesCompounds used in a research, industrial, or household setting +6
Target Protein:
Listeriolysin regulatory protein6,7-dimethyl-8-ribityllumazine synthaseThymidine kinase, cytosolic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dithiopyr DB15230
small molecule | CAS: 97886-45-8

Dithiopyr is under investigation in clinical trial NCT01236781 (Comparison of Full-Field Digital Mammography With Digital Breast Tomography for Screening Call-Back Rates).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ditiocarb zinc Approved DB14193
small molecule | CAS: 14324-55-1

Ditiocarb zinc, also known as Diethyldithiocarbamic acid zinc salt, is a known chelator for copper and zinc. It also a dermatological sensitizer and allergen. Sensitivity to ditiocarb zinc may be identified with a clinical patch test.

Kategori:
Acids, AcyclicAdjuvants, ImmunologicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical Use +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Divarasib DB17488
small molecule | CAS: 2417987-45-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Divozilimab DB18878
biotech | CAS: 2254061-60-2

Divozilimab is under investigation in clinical trial NCT05730699 (Efficacy and Safety of Divozilimab in Patients With Neuromyelitis Optica Spectrum Disorders (AQUARELLE)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dixanthogen DB13712
small molecule | CAS: 502-55-6

Deskripsi belum tersedia.

Kategori:
AnionsAntiparasitic Products, Insecticides and RepellentsEctoparasiticides, Incl. Scabicides +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dixyrazine DB13784
small molecule | CAS: 2470-73-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAntiemetics +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha-Tocopherol Approved DB14476
small molecule | CAS: 10191-41-0

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18656-38-7

A synthetic phospholipid used in liposomes and lipid bilayers for the study of biological membranes. It is used in commercial drug preparations to solubilize drugs for injection [A32711]

Kategori:
Compounds used in a research, industrial, or household settingGlycerophosphatesGlycerophospholipids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61361-72-6

DL-dimyristoylphosphatidylglycerol is a phospholipid used in commercially available pharmaceutical preparations to solubilize drugs for injection.

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-Methylephedrine Approved DB11278
small molecule | CAS: 1201-56-5

Methylephedrine is a sympathomimetic amine that appears in various over-the-counter cough and cold medications throughout the world [L2838], [L2839], [L2840]. The abuse of methylephedrine-containing medications has been reported in Japan. Methylephedrine is n…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +10
Target Protein:
Beta-1 adrenergic receptorAlpha-2A adrenergic receptorAlpha adrenergic receptor +1
Waktu Paruh3-6 hours (Ephedrin…
Vol. DistribusiEphedrine: 2.5-3.0 …
Klirens-
Genetik -
DM-1157 DB18600
small molecule | CAS: 1239953-66-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DMP-777 DB18488
small molecule | CAS: 157341-41-8

DMP-777 is a selective inhibitor of polymorphonuclear leukocyte (PMN) elastase.

Kategori:
AzetinesEnzyme InhibitorsPancreatic Elastase, antagonists & inhibitors
Target Protein:
Neutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DNL343 DB18678
small molecule | CAS: 2278265-85-1

DNL343 is under investigation in clinical trial NCT05842941 (HEALEY ALS Platform Trial - Regimen G DNL343).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Dobesilic acid DB13529
small molecule | CAS: 88-46-0

Deskripsi belum tersedia.

Kategori:
Antivaricose TherapyArylsulfonatesArylsulfonic Acids +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dobutamine Approved DB00841
small molecule | CAS: 34368-04-2

A beta-1 agonist catecholamine that has cardiac stimulant action without evoking vasoconstriction or tachycardia. It is proposed as a cardiotonic after myocardial infarction or open heart surgery.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +28
Target Protein:
Alpha-1 adrenergic receptorsBeta-1 adrenergic receptorBeta-2 adrenergic receptor +1
Waktu Paruh2 minutes
Vol. Distribusi-
Klirens-
Genetik -
Docaravimab DB17802
biotech | CAS: 2247196-23-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Docarpamine DB18046
small molecule | CAS: 74639-40-0

Deskripsi belum tersedia.

Kategori:
AminesBenzene DerivativesBiogenic Amines +8
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 177021-00-0

Deskripsi belum tersedia.

Kategori:
AnticoagulantsCarbohydratesExperimental Unapproved Treatments for COVID-19 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doconexent Approved DB03756
small molecule | CAS: 6217-54-5

A mixture of fish oil and primrose oil, doconexent is used as a high-docosahexaenoic acid (DHA) supplement. DHA is a 22 carbon chain with 6 cis double bonds with anti-inflammatory effects. It can be biosythesized from alpha-linolenic acid or commercially manu…

Kategori:
Cytochrome P-450 CYP2C9 InhibitorsCytochrome P-450 CYP2C9 Inhibitors (strength unknown)Cytochrome P-450 CYP2C9 Substrates +11
Target Protein:
Peroxisome proliferator-activated receptor alphaProstaglandin G/H synthase 1Prostaglandin G/H synthase 2 +6
Waktu ParuhApproximately 20 ho…
Vol. DistribusiDHA is the most abu…
Klirens-
Genetik -
Docosanol Approved DB00632
small molecule | CAS: 661-19-8

Docosanol is a drug used for topical treatment for recurrent herpes simplex labialis episodes (episodes of cold sores or fever blisters). A saturated 22-carbon aliphatic alcohol, docosanol exhibits antiviral activity against many lipid enveloped viruses inclu…

Kategori:
AlcoholsAnti-Infective AgentsAntiviral Agents +2
Target Protein:
Envelope glycoprotein GP350Envelope glycoprotein GP340
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Docusate Approved DB11089
small molecule | CAS: 10041-19-7

Docusate, or dioctyl sulfosuccinate, is a stool softener indicated for the treatment of constipation[A32201]. Docusate acts by increasing the amount of water the stool absorbs in the gut, making the stool softer and easier to pass [L1801]. Docusate can be ora…

Kategori:
Alimentary Tract and MetabolismDrugs for ConstipationEnemas +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dodecyl sulfate DB03967
small molecule | CAS: 151-41-7

Deskripsi belum tersedia.

Kategori:
AlcoholsAlkanesulfonatesAlkanesulfonic Acids +8
Target Protein:
Lysozyme CLipid A palmitoyltransferase PagP
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Retinoic acid receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dodecyl-Coa DB03264
small molecule

Deskripsi belum tersedia.

Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 3Fatty acid metabolism regulator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1643-20-5

Deskripsi belum tersedia.

Kategori:
AminesCompounds used in a research, industrial, or household settingDetergents +3
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialReaction center protein L chainReaction center protein M chain +47
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dolasetron Approved DB00757
small molecule | CAS: 115956-12-2

Dolasetron is an antinauseant and antiemetic agent indicated for the prevention of nausea and vomiting associated with moderately-emetogenic cancer chemotherapy and for the prevention of postoperative nausea and vomiting. Dolasetron is a highly specific and s…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +21
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh8.1 hours
Vol. Distribusi* 5.8 L/kg [adults]
Klirens* Apparent cl=9.4 m…
Genetik -
Dolastatin 10 DB12730
small molecule | CAS: 110417-88-4

Dolastatin 10 has been used in trials studying the treatment of Sarcoma, Leukemia, Lymphoma, Liver Cancer, and Kidney Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntimitotic AgentsAntineoplastic Agents +4
Target Protein:
Tubulin beta-2A chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dolcanatide DB13112
biotech | CAS: 1092457-65-2

Dolcanatide has been investigated in Exposure.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme ActivatorsGastrointestinal Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dolutegravir Approved DB08930
small molecule | CAS: 1051375-16-6

Dolutegravir is an HIV-1 integrase inhibitor that blocks the strand transfer step of the integration of the viral genome into the host cell (INSTI).[A7514] The effect of this drug has no homology in human host cells, which gives it excellent tolerability and …

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +20
Target Protein:
Gag-Pol polyproteinIntegrase
Gen Terkait:
UGT1A1 UGT1A1 UGT1A1
Waktu ParuhThe half-life of do…
Vol. DistribusiThe administration …
KlirensThe apparent cleara…
Genetik 3 Varian
Domagrozumab DB15083
biotech | CAS: 1629605-31-7

Domagrozumab is under investigation in clinical trial NCT01616277 (A Phase 1 Study To Evaluate The Safety And Tolerability Of PF-06252616 In Healthy Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domatinostat DB17521
small molecule | CAS: 910462-43-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domiodol DB13768
small molecule | CAS: 61869-07-6

Deskripsi belum tersedia.

Kategori:
Cough and Cold PreparationsDioxolesExpectorants
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domiphen Approved DB11594
small molecule | CAS: 13900-14-6

Domiphen bromide is a quaternary ammonium compound that is predominantly employed as a topically administered antiseptic agent.

Kategori:
Alimentary Tract and MetabolismAminesAmmonium Compounds +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2382896-04-8

Domofenogene zalfaparvovec, formerly known as BMN-307, is an investigational AAV5-phenylalanine hydroxylase (PAH) gene therapy developed by BioMarin Pharmaceutical.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domperidone Approved DB01184
small molecule | CAS: 57808-66-9

A specific blocker of dopamine receptors. It speeds gastrointestinal peristalsis, causes prolactin release, and is used as antiemetic and tool in the study of dopaminergic mechanisms.

Kategori:
Alimentary Tract and MetabolismAntiemeticsAutonomic Agents +25
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
Waktu Paruh7 hours
Vol. Distribusi-
Klirens-
Genetik -
Domvanalimab DB18848
biotech | CAS: 2368219-35-4

Domvanalimab is under investigation in clinical trial NCT05502237 (Zimberelimab and Domvanalimab in Combination With Chemotherapy Versus Pembrolizumab With Chemotherapy in Patients With Untreated Metastatic Non-small Cell Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Donanemab Approved DB16647
biotech | CAS: 1931944-80-7

Donanemab is a humanized immunoglobulin gamma 1 (IgG1) monoclonal antibody directed against insoluble N-truncated pyroglutamate amyloid beta (A?), [L50978] which is found in the brain amyloid plaques that contribute to the pathophysiology of Alzheimer's Disea…

Kategori:
Alzheimer Disease, drug therapyAmino Acids, Peptides, and ProteinsAmyloid Beta-directed Antibodies +11
Target Protein:
Beta amyloid plaque
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe central volume …
KlirensThe clearance is ab…
Genetik -
Donepezil Approved DB00843
small molecule | CAS: 120014-06-4

In 2016, the global burden of dementia was estimated to be 43.8 million, demonstrating a significant increase from a global prevalence of 20.2 million in 1990.[A182411] Donepezil, also known as Aricept, is a piperidine derivative acetylcholinesterase inhibito…

Kategori:
Anti-Dementia DrugsBCRP/ABCG2 SubstratesBradycardia-Causing Agents +20
Target Protein:
Acetylcholinesterase5-hydroxytryptamine receptor 2ACholinesterase +5
Gen Terkait:
CYP2D6
Waktu ParuhThe average elimina…
Vol. DistribusiThe volume of distr…
KlirensAccording to the FD…
Genetik 1 Varian
Donidalorsen DB18751
biotech | CAS: 2304692-48-4

Donidalorsen is under investigation in clinical trial NCT05392114 to assess the long-term safety and efficacy of donidalorsen in the prophylactic treatment of hereditary angioedema (HAE)

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Donislecel Approved DB17961
biotech

Donislecel is the first allogeneic pancreatic islet cellular from deceased donor pancreatic cells used for the treatment of adult type 1 diabetes with unsuccessful control of glycated hemoglobin, despite intensive diabetes management and treatments.[L47166,L4…

Kategori:
Cellular and Gene TherapyDrugs Used in Diabetes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dopamine Approved DB00988
small molecule | CAS: 51-61-6

One of the catecholamine neurotransmitters in the brain. It is derived from tyrosine and is the precursor to norepinephrine and epinephrine. Dopamine is a major transmitter in the extrapyramidal system of the brain, and important in regulating movement. A fa…

Kategori:
Adrenergic and Dopaminergic AgentsAgents producing tachycardiaAgents that produce hypertension +26
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(1B) dopamine receptor +13
Waktu Paruh2 minutes
Vol. Distribusi-
Klirens-
Genetik -
Dopastatin DB16144
small molecule | CAS: 868562-36-1

Dopastatin is under investigation in clinical trial NCT04335357 (TBR-760 in Adult Patients With Non-functioning Pituitary Adenomas).

Kategori:
AminesAmino Acids, Peptides, and ProteinsBenzene Derivatives +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5301–5350 dari 13591
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