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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 106 / 236
Flurbiprofen Approved DB00712
small molecule | CAS: 5104-49-4

Flurbiprofen, a propionic acid derivative, is a nonsteroidal anti-inflammatory agent (NSAIA) with antipyretic and analgesic activity. Oral formulations of flurbiprofen may be used for the symptomatic treatment of rheumatoid arthritis, osteoarthritis and ankly…

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +37
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhR-flurbiprofen, 4.7…
Vol. Distribusi* 14 L [Normal Heal…
Klirens-
Genetik -
small molecule | CAS: 91503-79-6

Flurbiprofen axetil is under investigation in clinical trial NCT02043366 (Effect of Butorphanol Combined With Flurbiprofen Axetil on Preventing Hyperalgesia Induced by Remifentanil in Patients).

Kategori:
Acids, AcyclicAnalgesicsAnalgesics, Non-Narcotic +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 863887-89-2

Flurpiridaz F-18 is a radioactive diagnostic drug indicated for positron emission tomography (PET) myocardial perfusion imaging (MPI), which is an imaging process used in patients with known or suspected coronary artery disease (CAD).[A264519] Flurpiridaz F-1…

Kategori:
Fluorine RadioisotopesRadioactive Diagnostic Agent
Target Protein:
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13
Waktu ParuhFluorine-18 has a h…
Vol. DistribusiFlurpiridaz F-18 di…
Klirens-
Genetik -
Flutamide Approved DB00499
small molecule | CAS: 13311-84-7

An antiandrogen with about the same potency as cyproterone in rodent and canine species.

Kategori:
AmidesAminesAndrogen Receptor Antagonists +19
Target Protein:
Androgen receptorAryl hydrocarbon receptorNuclear receptor subfamily 1 group I member 2
Waktu ParuhThe plasma half-lif…
Vol. Distribusi-
Klirens-
Genetik -
Flutemetamol DB15058
small molecule | CAS: 637003-10-2

Flutemetamol is under investigation in clinical trial NCT02353949 (Investigating the Clinical Consequences of Flutemetamol-PET-scanning).

Kategori:
AminesCompounds used in a research, industrial, or household settingContrast Media +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flutemetamol (18F) Approved DB09151
small molecule | CAS: 765922-62-1

Flutemetamol (18F) is a PET scanning radiopharmaceutical containing the radionuclide fluorine-18. It is indicated for Positron Emission Tomography (PET) imaging of the brain to estimate ? amyloid neuritic plaque density in adult patients with cognitive impair…

Kategori:
AminesCentral Nervous SystemCompounds used in a research, industrial, or household setting +11
Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluticasone Approved DB13867
small molecule | CAS: 90566-53-3

Fluticasone is a synthetic glucocorticoid available as 2 esters, [DB08906] and [DB00588][F4355,F4358,F4361,F4364][FDA Label]. These drugs are available as inhalers, nasal, sprays, and topical treatments for various inflammatory indications[F4355,F4358,F4361,F…

Kategori:
Adrenal Cortex HormonesAndrostadienesAndrostanes +42
Target Protein:
Glucocorticoid receptorProgesterone receptorCytosolic phospholipase A2 +1
Waktu Paruh15.1 hours for intr…
Vol. Distribusi608L at steady stat…
Klirens57.8L/h for [DB0890…
Genetik -
Fluticasone furoate Approved DB08906
small molecule | CAS: 397864-44-7

Fluticasone furoate is a synthetic glucocorticoid available as an inhaler and nasal spray for various inflammatory indications[FDA Label][F4364]. Fluticasone furoate was first approved in 2007[L5965].

Kategori:
Adrenal Cortex HormonesAgents to Treat Airway DiseaseAndrostanes +32
Target Protein:
Glucocorticoid receptorProgesterone receptorMineralocorticoid receptor
Waktu ParuhFollowing repeat-do…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Fluticasone propionate Approved DB00588
small molecule | CAS: 80474-14-2

Fluticasone propionate is a synthetic glucocorticoid[F4355,F4358][FDA Label]. These drugs are available as inhalers, nasal, sprays, and topical treatments for various inflammatory indications[F4355,F4358][FDA Label]. Fluticasone propionate was first approved …

Kategori:
Adrenal Cortex HormonesAdrenalsAgents to Treat Airway Disease +35
Target Protein:
Glucocorticoid receptorProgesterone receptorCytosolic phospholipase A2 +1
Waktu Paruh7.8 hours for intra…
Vol. DistribusiThe volume of distr…
Klirens1093mL/min for flut…
Genetik -
small molecule | CAS: 1274863-98-7

Flutriciclamide F-18 is under investigation in clinical trial NCT02350426 (A Study to Assess Inflammation in Rheumatoid Arthritis Using Molecular Imaging Techniques).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flutrimazole DB13425
small molecule | CAS: 119006-77-8

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluvastatin Approved DB01095
small molecule | CAS: 93957-54-1

Fluvastatin is an antilipemic agent that competitively inhibits hydroxymethylglutaryl-coenzyme A (HMG-CoA) reductase. HMG-CoA reductase catalyzes the conversion of HMG-CoA to mevalonic acid, the rate-limiting step in cholesterol biosynthesis. Fluvastatin belo…

Kategori:
Agents Causing Muscle ToxicityCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +35
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseHistone deacetylase 2
Waktu Paruh3 hours
Vol. Distribusi* 0.35 L/kg
Klirens* 0.8 L/h/kg * 107…
Genetik -
Fluvoxamine Approved DB00176
small molecule | CAS: 54739-18-3

Fluvoxamine is an antidepressant which functions pharmacologically as a selective serotonin reuptake inhibitor. Though it is in the same class as other SSRI drugs, it is most often used to treat obsessive-compulsive disorder. Fluvoxamine has been in use in c…

Kategori:
AminesAnti-Anxiety AgentsAntidepressive Agents +44
Target Protein:
Sodium-dependent serotonin transporterVoltage-gated inwardly rectifying potassium channel KCNH2
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +3
Waktu Paruh15.6 hours [FDA Lab…
Vol. Distribusi* 25 L/kg [FDA Labe…
Klirens-
Genetik 6 Varian
Fluzoparib DB15637
small molecule | CAS: 1358715-18-0

Fluzoparib is under investigation in clinical trial NCT03863860 (A Trial of Maintenance Treatment With Fluzoparib Versus Placebo in Relapsed Ovarian Cancer Patients).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsPoly(ADP-ribose) Polymerase Inhibitors +1
Target Protein:
Poly [ADP-ribose] polymerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FLX475 DB15570
small molecule

FLX475 is a small molecule CCR4 antagonist being investigated for the treatment of cancer.[L9875]

Target Protein:
C-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FN-1501 DB17383
small molecule | CAS: 1429515-59-2

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 2Receptor-type tyrosine-protein kinase FLT3Cyclin-dependent kinase 4 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fobrepodacin DB18409
small molecule | CAS: 1384984-31-9

Deskripsi belum tersedia.

Target Protein:
DNA gyrase subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Folic acid Approved DB00158
small molecule | CAS: 59-30-3

Folic acid, also known as folate or Vitamin B9, is a member of the B vitamin family and an essential cofactor for enzymes involved in DNA and RNA synthesis. More specifically, folic acid is required by the body for the synthesis of purines, pyrimidines, and m…

Kategori:
Antianemic PreparationsAutacoidsBCRP/ABCG2 Substrates +19
Target Protein:
Proton-coupled folate transporterReduced folate transporterFolate receptor gamma +2
Waktu Paruh-
Vol. DistribusiTetrahydrofolic aci…
Klirens-
Genetik -
Folitixorin DB17113
small molecule | CAS: 3432-99-3

Deskripsi belum tersedia.

Kategori:
CoenzymesEnzymes and CoenzymesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Follitropin Approved DB00066
biotech | CAS: 146479-72-3

Follitropin is a human follicle stimulating hormone (FSH) preparation of recombinant DNA origin, which consists of two non-covalently linked, non-identical glycoproteins designated as the alpha- and beta- subunits. The alpha- and beta- subunits have 92 and 11…

Kategori:
Amino Acids, Peptides, and ProteinsFollicle Stimulating HormoneGenito Urinary System and Sex Hormones +12
Target Protein:
Follicle-stimulating hormone receptor
Waktu ParuhCirculation half li…
Vol. Distribusi* 8 L [female subje…
Klirens* 0.01 1*h-1kg-1 [E…
Genetik -
Fomepizole Approved DB01213
small molecule | CAS: 7554-65-6

Fomepizole is used as an antidote in confirmed or suspected methanol or ethylene glycol poisoning. Fomepizole is a competitive inhibitor of alcohol dehydrogenase, the enzyme that catalyzes the initial steps in the metabolism of ethylene glycol and methanol to…

Kategori:
AntidotesCompounds used in a research, industrial, or household settingCytochrome P-450 CYP2A6 Inhibitors +13
Target Protein:
Alcohol dehydrogenase 1AAll-trans-retinol dehydrogenase [NAD(+)] ADH1BAlcohol dehydrogenase 1C +1
Waktu ParuhThe plasma half-lif…
Vol. Distribusi* 0.6 to 1.02 L/kg
Klirens-
Genetik -
Fomivirsen Approved DB06759
biotech | CAS: 144245-52-3

Fomivirsen is a antisense 21 mer phosphorothioate oligonucleotide. It is an antiviral agent that was used in the treatment of cytomegalovirus retinitis (CMV) in immunocompromised patients, including those with AIDS. As a complementary nucleotide to the messen…

Kategori:
Anti-Infective AgentsAntisense Elements (Genetics)Antisense Oligonucleotides +13
Target Protein:
30 kDa immediate-early protein 245 kDa immediate-early protein 2
Waktu ParuhIntravitreal drug c…
Vol. DistribusiPreclinical studies…
KlirensClearance from reti…
Genetik -
Fonadelpar DB16169
small molecule | CAS: 515138-06-4

Fonadelpar is under investigation in clinical trial NCT03527212 (A Study to Assess the Safety and Effectiveness of SJP-0035 for the Treatment of Patients With Dry Eye Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foralumab DB16170
biotech | CAS: 946415-64-1

Foralumab is under investigation in clinical trial NCT03291249 (Assessment of the Safety of Foralumab, an Oral Anti-cd3 Antibody, in Patients With NASH and T2DM).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2248111-37-5

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Foreskin fibroblast-like stromal cells (FDSCs) are progenitors isolated from human tissue that can differentiate into various cell types [A32660]. Also known as Dermagraft, this device is a cryopreserved human fibroblast-derived dermal substitute. Composed…

Kategori:
Allogeneic Cultured Cell Scaffold
Target Protein:
Vascular endothelial growth factor receptor 1Interleukin-6Interleukin-1 receptor type 1 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Skin, the largest organ of the human body, plays the main role in protecting the body from mechanical damage. It is composed of epidermal, dermal and hypodermal layers. The barrier function of the skin owed to its avascular epidermal layer, which is made main…

Kategori:
Allogeneic Cultured Cell Scaffold
Target Protein:
Fibroblast growth factor 1Epidermal growth factor receptorGranulocyte-macrophage colony-stimulating factor receptor subunit alpha +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foretinib DB12307
small molecule | CAS: 849217-64-7

Foretinib has been used in trials studying the treatment of Cancer, Breast Cancer, Carcinoma, Renal Cell, Recurrent Breast Cancer, and Neoplasms, Head and Neck, among others. Foretinib is an orally available small molecule compound designed to target multiple…

Kategori:
AmidesAminesAniline Compounds +3
Target Protein:
Hepatocyte growth factor receptorVascular endothelial growth factor receptor 2Hepatocyte growth factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Forigerimod DB12490
biotech | CAS: 497156-60-2

Forigerimod is under investigation for the treatment of Lupus Erythematosus, Systemic.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesRibonucleoprotein, U1 Small Nuclear
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Forimtamig DB19015
biotech | CAS: 2649379-96-2

Forimtamig is under investigation in clinical trial NCT06055075 (A Study Evaluating Safety, Tolerability, and Clinical Activity of Forimtamig-based Treatment Combinations in Participants With Relapsed or Refractory Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formaldehyde Approved DB03843
small molecule | CAS: 50-00-0

A highly reactive aldehyde gas formed by oxidation or incomplete combustion of hydrocarbons. In solution, it has a wide range of uses: in the manufacture of resins and textiles, as a disinfectant, and as a laboratory fixative or preservative. Formaldehyde sol…

Kategori:
AldehydesAnti-Infective AgentsAnti-Infective Agents, Local +7
Target Protein:
Transient receptor potential cation channel subfamily A member 1Hematopoietic stem cellsD-alanyl-D-alanine carboxypeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formebolone DB01569
small molecule | CAS: 2454-11-7

Formebolone, a derivative of androstane, is an anabolic androgenic steroid. It is on the list of substances prohibited by the Word Anti-Doping Agency, and is regularly screened for in athletes.[A14416] It is also classified by the US Drug Enforcement Administ…

Kategori:
AndrostanesAndrostenesAndrostenols +3
Target Protein:
11-beta-hydroxysteroid dehydrogenase type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formestane Approved DB08905
small molecule | CAS: 566-48-3

Formestane was the first selective, type I, steroidal aromatase inhibitor used in the treatment of estrogen-receptor positive breast cancer in post-menopausal women. Formestane suppresses estrogen production from anabolic steroids or prohormones. Formestane i…

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +23
Target Protein:
Aromatase
Waktu ParuhTerminal plasma eli…
Vol. DistribusiVd = 1.8 L/kg; wide…
KlirensPlasma clearance is…
Genetik -
Formocortal DB13664
small molecule | CAS: 2825-60-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formononetin DB15335
small molecule | CAS: 485-72-3

Formononetin is under investigation in clinical trial NCT02174666 (Isoflavone Treatment for Postmenopausal Osteopenia.).

Kategori:
BenzopyransChromonesEstrogens +7
Target Protein:
Sodium/glucose cotransporter 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Formoterol Approved DB00983
small molecule | CAS: 73573-87-2

Formoterol is an inhaled beta<sub>2</sub>-agonist used in the management of COPD and asthma that was first approved for use in the United States in 2001.[L10986] It acts on bronchial smooth muscle to dilate and relax airways, and is administered as a racemic …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +29
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu ParuhThe average termina…
Vol. Distribusi-
KlirensRenal clearance of …
Genetik -
Formycin DB02281
small molecule | CAS: 6742-12-7

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
S-methyl-5'-thioadenosine phosphorylase5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Forodesine DB06185
small molecule | CAS: 209799-67-7

Forodesine is a highly potent, orally active, rationally designed PNP inhibitor that has shown activity in preclinical studies with malignant cells and clinical utility against T-cell acute lymphoblastic leukemia and cutaneous T-cell lymphoma. Additional prel…

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosamprenavir Approved DB01319
small molecule | CAS: 226700-79-4

Fosamprenavir is a prodrug of amprenavir, an inhibitor of human immunodeficiency virus (HIV) protease.

Kategori:
Acids, AcyclicAmidesAmprenavir and Prodrugs +22
Target Protein:
Pol polyproteinGag-Pol polyprotein
Waktu ParuhThe plasma eliminat…
Vol. Distribusi-
Klirens-
Genetik -
Fosaprepitant Approved DB06717
small molecule | CAS: 172673-20-0

Fosaprepitant is an intravenously administered antiemetic drug. It is a prodrug of Aprepitant. It aids in the prevention of acute and delayed nausea and vomiting associated with chemotherapy treatment.

Kategori:
AntiemeticsAprepitant and ProdrugsAutonomic Agents +24
Target Protein:
Substance-P receptor
Waktu Paruh9-13 hours
Vol. Distribusi-
Klirens-
Genetik -
Fosbretabulin DB12577
small molecule | CAS: 222030-63-9

Fosbretabulin has been investigated for the treatment of Anaplastic Thyroid Cancer.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Foscarbidopa Approved DB16171
small molecule | CAS: 1907685-81-7

Foscarbidopa is under investigation in clinical trial NCT04379050 (Extension Study to Evaluate Safety and Tolerability of 24-hour Daily Exposure of Continuous Subcutaneous Infusion of ABBV-951 in Adult Participants With Parkinson's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosciclopirox DB18772
small molecule | CAS: 1380539-06-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1951476-79-1

Fosclevudine alafenamide is under investigation in clinical trial NCT05238844 (A Study of Safety and Efficacy of ATI-2173 and Vebicorvir in Combination With Tenofovir Disoproxil Fumarate in Subjects With Chronic Hepatitis B Virus Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fosdenopterin Approved DB16628
small molecule | CAS: 150829-29-1

Molybdenum cofactor deficiency (MoCD) is an exceptionally rare autosomal recessive disorder resulting in a deficiency of three molybdenum-dependent enzymes: sulfite oxidase (SOX), xanthine dehydrogenase, and aldehyde oxidase.[A230088] Signs and symptoms begin…

Kategori:
Alimentary Tract and MetabolismBiological FactorsCyclic Pyranopterin Monophosphate +9
Target Protein:
Molybdenum cofactor biosynthesis protein 1Xanthine dehydrogenase/oxidase
Waktu ParuhThe mean half-life …
Vol. DistribusiThe volume of distr…
KlirensTotal body clearanc…
Genetik -
Fosfomycin Approved DB00828
small molecule | CAS: 23155-02-4

Fosfomycin was discovered in 1969 by scientists at the Spanish Penicillin and Antibiotics Company and is produced by _Streptomyces fradiae_.[A229338,A230348] It may also be produced synthetically and is commercially available as the disodium salt for intraven…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAnti-Infective Agents, Urinary +7
Target Protein:
UDP-N-acetylglucosamine 1-carboxyvinyltransferase
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn healthy subjects…
KlirensIn one study, the r…
Genetik -
Fosfructose DB13863
small molecule | CAS: 488-69-7

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCarbohydratesCardiac Therapy +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1562406-27-2

NUC-1031 is under investigation in clinical trial NCT03610100 (Acelarin First Line Randomised Pancreatic Study).

Kategori:
Antineoplastic AgentsCytosine NucleotidesNucleic Acids, Nucleotides, and Nucleosides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1332837-31-6

Fosifloxuridine nafalbenamide is under investigation in clinical trial NCT03428958 (A Safety Study of NUC-3373 in Combination With Standard Agents Used in Colorectal Cancer Treatment).

Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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