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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
Referensi
11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 106 / 236
Fradafiban DB06472
small molecule | CAS: 148396-36-5

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesPlatelet Glycoprotein GPIIb-IIIa Complex, antagonists & inhibitors
Target Protein:
Integrin alpha-IIbIntegrin beta-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frankincense DB16592
biotech

Deskripsi belum tersedia.

Kategori:
Biological ProductsBiopolymersComplex Mixtures +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fremanezumab Approved DB14041
biotech | CAS: 1655501-53-3

Fremanezumab is a humanized monoclonal antibody targeted against human calcitonin gene-related peptide (CGRP) for the prevention of migraine headaches.[L11749] It was developed by Teva Pharmaceuticals USA and approved by the FDA in September 2018.[L11779] Alo…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +12
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhThe mean half-life …
Vol. DistribusiFremanezumab has an…
KlirensThe apparent cleara…
Genetik -
Fresolimumab DB12396
biotech | CAS: 948564-73-6

Fresolimumab has been used in trials studying the treatment of Primary Brain Tumors, Metastatic Breast Cancer, Diffuse Systemic Sclerosis, Pleural Malignant Mesothelioma, and Primary Focal Segmental Glomerulosclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frexalimab DB18926
biotech | CAS: 2515463-86-0

Frexalimab is under investigation in clinical trial NCT06141486 (Efficacy and Safety Study of Frexalimab (SAR441344) in Adults With Nonrelapsing Secondary Progressive Multiple Sclerosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Friulimicin B DB06087
small molecule | CAS: 239802-15-4

Friulimicin B is a naturally occurring antibiotic produced by a micro-organism, *Actinoplanes friuliensis*. It shows strong cidal activity against a number of Gram-positive pathogens which commonly cause serious infections in hospital patients and which are b…

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Froniglutide DB16178
biotech | CAS: 1417579-81-7

Glymera is under investigation in clinical trial NCT01658501 (Phase 2b Multicenter, Randomized, Double-blind, Placebo- and Active-controlled, Parallel-group Study to Assess the PD Response and Safety of Three Dose Levels of (PB1023) Injection Following 20 Wee…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frovocimab DB15089
biotech | CAS: 1643672-70-1

Frovocimab is under investigation in clinical trial NCT01671085 (A Study of LY3015014 in Healthy Participants With High Cholesterol).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glucosamine-6-phosphate deaminase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 643-13-0

Deskripsi belum tersedia.

Kategori:
CarbohydratesHexosephosphatesSugar Phosphates
Target Protein:
Fructose-1,6-bisphosphatase 1Fructose-1,6-bisphosphatase isozyme 26-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frunexian DB18771
small molecule | CAS: 1803270-60-1

Deskripsi belum tersedia.

Kategori:
AmidesAminesPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fruquintinib Approved DB11679
small molecule | CAS: 1194506-26-7

Fruquintinib is a novel small-molecule anti-VEGFR that targets VEGFR-1,-2, and -3 to inhibit angiogenesis. Tumor angiogenesis is one of the most critical biological processes for increasing oxygen and nutrient supply to cancer cells, and the VEGF/VEGFR pathwa…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +10
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3
Waktu ParuhThe fruquintinib's …
Vol. DistribusiThe mean (SD) appar…
KlirensThe apparent cleara…
Genetik -
FT-1101 DB17553
small molecule | CAS: 1776060-36-6

FT-1101 is a novel Bromodomain and Extra-Terminal motif (BET) inhibitor.[A257301] FT-1101 is under investigation in clinical trial NCT02543879 (Study of a Novel BET Inhibitor FT-1101 in Patients With Relapsed or Refractory Hematologic Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FT516 DB15732
biotech

FT516 is an investigational and engineered off-the-shelf natural killer (NK) cell therapy originating from induced pluripotent stem cells (iPSC). This compound expresses a high-affinity 158V, CD16 (hnCD16) Fc receptor that has an enhanced binding ability to t…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucitol DB03815
small molecule | CAS: 13074-06-1

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydrates
Target Protein:
L-fucose isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucose DB15236
small molecule | CAS: 2438-80-4

Fucose is under investigation in clinical trial NCT03354533 (Study of ORL-1F (L-fucose) in Patients With Leukocyte Adhesion Deficiency Type II).

Kategori:
CarbohydratesDeoxy Sugars
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucoxanthin DB15462
small molecule | CAS: 3351-86-8

Fucoxanthin is under investigation in clinical trial NCT03613740 (Effect of Fucoxanthin on the Components of the Metabolic Syndrome, Insulin Sensitivity and Insulin Secretion). Fucoxanthin isis a marine carotenoid mainly found in brown algae, giving them a br…

Kategori:
AlkenesBiological FactorsCarotenoids +7
Target Protein:
NF-kappa-B inhibitor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fulvestrant Approved DB00947
small molecule | CAS: 129453-61-8

Fulvestrant is a drug treatment of hormone receptor (HR)-positive metastatic breast cancer in post-menopausal women with disease progression following anti-estrogen therapy. It is an estrogen receptor antagonist with no agonist effects, which works both by do…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +20
Target Protein:
Estrogen receptor
Waktu Paruh40 days
Vol. Distribusi* 3 to 5 L/kg
Klirens-
Genetik -
Fumagillin DB02640
small molecule | CAS: 23110-15-8

Deskripsi belum tersedia.

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAnti-Infective Agents +10
Target Protein:
Methionine aminopeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fumaric acid DB01677
small molecule | CAS: 110-17-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntipsoriaticsAntipsoriatics for Topical Use +2
Target Protein:
Interferon gammaMalate dehydrogenaseFumarate reductase flavoprotein subunit +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Funapide DB11769
small molecule | CAS: 1259933-16-8

Funapide has been used in trials studying the treatment of Pharmacokinetics, Postherpetic Neuralgia, and Osteoarthritis of the Knee.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Sodium channel protein type 9 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaltadone DB16567
small molecule | CAS: 139-91-3

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryFurans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaprofen DB06499
small molecule | CAS: 67700-30-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazidin DB13475
small molecule | CAS: 1672-88-4

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazolidone DB00614
small molecule | CAS: 67-45-8

A nitrofuran derivative with antiprotozoal and antibacterial activity. Furazolidone binds bacterial DNA which leads to the gradual inhibition of monoamine oxidase. (From Martindale, The Extra Pharmacopoeia, 30th ed, p514)

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Infective Agents +20
Target Protein:
DNA
Waktu Paruh10 minutes
Vol. Distribusi-
Klirens-
Genetik -
Furethidine DB01464
small molecule | CAS: 2385-81-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furfural DB16856
small molecule | CAS: 98-01-1

Deskripsi belum tersedia.

Kategori:
AldehydesFurans
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furosemide Approved DB00695
small molecule | CAS: 54-31-9

Furosemide is a potent loop diuretic that acts on the kidneys to ultimately increase water loss from the body. It is an anthranilic acid derivative.[L7958] Furosemide is used for edema secondary to various clinical conditions, such as congestive heart failure…

Kategori:
Acids, CarbocyclicAmidesAmines +30
Target Protein:
Solute carrier family 12 member 1Carbonic anhydrase 2G-protein coupled receptor 35
Waktu ParuhThe half-life from …
Vol. DistribusiThe volume of distr…
KlirensFollowing intraveno…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fursultiamine Approved DB08966
small molecule | CAS: 804-30-8

Compound used for therapy of thiamine deficiency. It has also been suggested for several non-deficiency disorders but has not yet proven useful. Fursultiamine is a vitamin B1 derivative.

Kategori:
MicronutrientsPyrimidinesSulfur Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furvina DB16547
small molecule | CAS: 189935-72-6

Furvina (G1) is an antimicrobial agent active against Gram-positive and Gram-negative bacteria, yeasts, and filamentous fungi. Furvina is marketed in Cuba as Dermofural®, an ointment containing G1 as the only active principle ingredient. It is used to treat d…

Kategori:
AlkenesAnti-Infective AgentsHydrocarbons, Acyclic
Target Protein:
30S ribosomal protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusafungine Approved DB08965
small molecule | CAS: 1393-87-9

Fusafungine is an antibiotic from Fusarium lateririum, and is used for the treatment of respiratory infections.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusarium compactum Approved DB10698
biotech

Fusarium compactum is a fungus which can provoke allergic reactions. Fusarium compactum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusarium oxysporum Approved DB10806
biotech

Fusarium oxysporum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusidic acid Approved DB02703
small molecule | CAS: 6990-06-3

An antibiotic isolated from the fermentation broth of Fusidium coccineum. (From Merck Index, 11th ed) It acts by inhibiting translocation during protein synthesis. It is often used topically in creams and eyedrops but is available in systemic formulations inc…

Kategori:
Agents Causing Muscle ToxicityAnti-Bacterial AgentsAnti-Infective Agents +35
Target Protein:
Elongation factor GChloramphenicol acetyltransferaseChloramphenicol acetyltransferase 3
Waktu ParuhApproximately 5 to …
Vol. Distribusi-
Klirens-
Genetik -
Futibatinib Approved DB15149
small molecule | CAS: 1448169-71-8

Futibatinib is an inhibitor of Fibroblast Growth Factor receptor (FGFR), which comprises a group of receptor tyrosine kinases that play a key role in cell proliferation, differentiation, migration, and survival. FGFR was investigated in oncology as a therapeu…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +10
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +1
Waktu ParuhThe mean (CV%) elim…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Futuximab DB15262
biotech | CAS: 1310460-85-5

Futuximab is under investigation in clinical trial NCT01955473 (Japanese Phase 1 Trial of Sym004 in Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fx-1006A DB05352
small molecule

Fx-1006A is a small molecule compound with the potential to treat genetic disorders, such as familial amyloid cardiomyopathy (FAC) and familial amyloid polyneuropathy (FAP).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FX06 DB05685
biotech

FX06 is a naturally occurring peptide derived from the neo-N-terminus of fibrin (Bbeta(15-42)). It prevents leukocyte migration through the gap junctions of endothelial cells. FX06 has proven safe in acute and subchronic toxicological studies and recently ent…

Target Protein:
Cadherin-5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G305 DB17292
biotech

G305 is a [recombinant NY-ESO-1 protein] plus glucopyranosyl lipid A (GLA) in a stable emulsion (SE). G305 is an active component of CMB305 along with [LV305].[L47346]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G4460 DB06359
biotech

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Target Protein:
Transcriptional activator Myb
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gabapentin Approved DB00996
small molecule | CAS: 60142-96-3

Gabapentin is a structural analogue of the inhibitory neurotransmitter gamma-aminobutyric acid ([GABA]) that was first approved for use in the United States in 1993.[L8717] It was originally developed as a novel anti-epileptic for the treatment of certain typ…

Kategori:
Acids, AcyclicAcids, CarbocyclicAmines +24
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1Gamma-aminobutyric acid type B receptor subunit 2Gamma-aminobutyric acid type B receptor subunit 1 +5
Waktu ParuhThe elimination t<s…
Vol. DistribusiThe apparent volume…
KlirensBoth the plasma cle…
Genetik -
Gabapentin enacarbil Approved DB08872
small molecule | CAS: 478296-72-9

Gabapentin enacarbil is marketed under the name Horizant. It is a prodrug of gabapentin, and indicated in adults for the treatment of Restless Legs Syndrome (RLS) and postherpetic neuralgia (PHN).

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +6
Target Protein:
Sodium-dependent multivitamin transporterVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent calcium channel subunit alpha-2/delta-2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance of …
Genetik -
Gaboxadol DB06554
small molecule | CAS: 64603-91-4

Gaboxadol also known as 4,5,6,7-tetrahydroisoxazolo(5,4-c)pyridin-3-ol (THIP) is an experimental sleep aid drug developed by Lundbeck and Merck, who reported increased deep sleep without the reinforcing effects of benzodiazepines. Development of Gaboxadol was…

Kategori:
AnalgesicsAnestheticsAnticonvulsants +8
Target Protein:
Gamma-aminobutyric acid receptor subunit delta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gacyclidine DB13096
small molecule | CAS: 68134-81-6

Gacyclidine has been used in trials studying the treatment of Tinnitus.

Kategori:
Central Nervous System AgentsCompounds used in a research, industrial, or household settingCyclohexanes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gadobenic acid Approved DB00743
small molecule | CAS: 113662-23-0

Gadobenic acid, usually available in the salt form gadobenate dimeglumine, is a linear MRI gadolinium-based contrast agent (GBCA) used primarily for MR imaging of the liver.[A263086] It differs from other GBCAs due to the benzene ring that confers weak protei…

Kategori:
AlcoholsAmino SugarsCarbohydrates +14
Target Protein:
Albumin
Waktu ParuhGadobenate ion has …
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
Gadobutrol Approved DB06703
small molecule | CAS: 770691-21-9

Gadobutrol is a second-generation extracellular non-ionic macrocyclic GBCA (gadolinium-based contrast agent) used in magnetic resonance imaging (MRI) in adults and children older than 2 years of age. Due to its physicochemical properties, gadobutrol is formu…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +5
Waktu ParuhFor adult patients,…
Vol. DistribusiIn children aged 2 …
KlirensIn healthy subjects…
Genetik -
Gadodiamide Approved DB00225
small molecule | CAS: 131410-48-5

Gadodiamide is a linear, non-ionic gadolinium-based contrast agent (GBCA) that is used in magnetic resonance imaging (MRI) procedures to assist in the visualization of blood vessels.[A263086,A263091] GBCAs constitute the largest group of MR agents, and they a…

Kategori:
AcetatesAcids, AcyclicAmines +13
Waktu ParuhThe mean distributi…
Vol. DistribusiThe volume of distr…
KlirensThe renal and plasm…
Genetik -
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