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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 106 / 282
Depemokimab DB18846
biotech | CAS: 2243274-14-6

Depemokimab is under investigation in clinical trial NCT05274750 (Efficacy and Safety of Depemokimab (GSK3511294) in Participants With Chronic Rhinosinusitis With Nasal Polyps).

Waktu Paruh-
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Depreotide DB11628
small molecule | CAS: 161982-62-3

Depreotide is an ingredient in the EMA-withdrawn product NeoSpect.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
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Depulfavirine DB18890
small molecule | CAS: 867365-76-2

Depulfavirine is under investigation in clinical trial NCT05204394 (Study to Evaluate Efficacy and Safety of Switching to VM-1500A-LAI + 2nrtis From the 1st Line Standard of Care Therapy).

Waktu Paruh-
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Dequalinium Approved DB04209
small molecule | CAS: 6707-58-0

Dequalinium is an antibacterial agent with multi-targeted actions. It also possesses antifungal, antiparasitic, antiviral, anticancer, and neuroprotective properties.[A249255] It is a quaternary ammonium compound,[L42190] as it consists of an amphipathic cati…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAnti-Infective Agents, Local +10
Target Protein:
Small conductance calcium-activated potassium channel protein 1Cyclic nucleotide-gated channel alpha-2Small conductance calcium-activated potassium channel protein 2 +10
Waktu ParuhThere is no informa…
Vol. DistribusiThere is no informa…
KlirensThere is no informa…
Genetik -
Deracoxib DB11395
small molecule | CAS: 169590-41-4

Deracoxib is a non-steroidal anti-inflammatory drug of the coxib class, used in veterinary medicine to treat osteoarthritis in dogs. It is sold in tablets, which have added beefy flavour to increase palatability. Deramaxx received FDA approval in August 2002 …

Kategori:
AmidesAnalgesicsAnalgesics, Non-Narcotic +11
Waktu Paruh-
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Deramciclane DB06512
small molecule | CAS: 120444-71-5

Deramciclane (EGIS-3886) is used for the treatment of a number of anxiety disorders. Deramciclane differs from other anti anxiety medications in that it is not a benzodiazepine and so has a different structure and target. It antagonizes 5-HT2A receptors, agon…

Kategori:
Anti-Anxiety AgentsAnticonvulsantsAntidepressive Agents +17
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Derazantinib DB14889
small molecule | CAS: 1234356-69-4

Derazantinib is under investigation in clinical trial NCT03230318 (Derazantinib in Subjects With FGFR2 Gene Fusion Positive Inoperable or Advanced Intrahepatic Cholangiocarcinoma).

Kategori:
AminesHeterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 1
Waktu Paruh-
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Derenofylline DB12446
small molecule | CAS: 251945-92-3

Derenofylline has been used in trials studying the treatment of Congestive Heart Failure and Acute Decompensated Heart Failure; Renal Dysfunction.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aklanonic acid methyl ester cyclase AcmA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 24967-94-0

Deskripsi belum tersedia.

Kategori:
AnticoagulantsBlood and Blood Forming OrgansCarbohydrates +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dersalazine DB06251
small molecule | CAS: 188913-58-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +5
Target Protein:
Platelet-activating factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dersimelagon DB18007
small molecule | CAS: 1835256-48-8

Deskripsi belum tersedia.

Target Protein:
Melanocyte-stimulating hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 130525-62-1

Deskripsi belum tersedia.

Target Protein:
Neuraminidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desaspidin DB13567
small molecule | CAS: 114-43-2

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnticestodalsAntiparasitic Agents +2
Waktu Paruh-
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Klirens-
Genetik -
Descartes-30 DB16361
biotech

Descartes-30 is an RNA-engineered off-the-shelf allogeneic mesenchymal stem cell (MSC) product developed by Cartesian Therapeutics.[L27531] The RNA-engineering is performed with Cartesian Therapeutics’ proprietary RNA Armory which is a platform that activates…

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Deserpidine Approved DB01089
small molecule | CAS: 131-01-1

Deserpidine is an ester alkaloid drug isolated from Rauwolfia canescens (family Apocynaceae) with antipsychotic and antihypertensive properties that has been used for the control of high blood pressure and for the relief of psychotic behavior.

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +8
Target Protein:
Synaptic vesicular amine transporterAngiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desfesoterodine DB15578
small molecule | CAS: 207679-81-0

Desfesoterodine is a metabolite of [tolterodine].

Kategori:
Drugs for Urinary Frequency and IncontinenceGenito Urinary System and Sex HormonesUrologicals
Waktu Paruh-
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Desflurane Approved DB01189
small molecule | CAS: 57041-67-5

Desflurane, or I-653, a a volatile anesthetic that is more rapidly cleared and less metabolized than previous inhaled anesthetics such as [methoxyflurane], [sevoflurane], [enflurane], or [isoflurane].[A226390,A39015,A226893]. It was developed in the late 1980…

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +14
Target Protein:
GABA(A) ReceptorGlycine receptor subunit alpha-1Glutamate receptor 1 +4
Waktu ParuhDesflurane has a te…
Vol. DistribusiDesflurane has a me…
KlirensA 26 g dose of desf…
Genetik -
Desidustat DB16135
small molecule | CAS: 1616690-16-4

Desidustat is under investigation in clinical trial NCT04012957 (Desidustat in the Treatment of Anemia in CKD).

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
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Desirudin Approved DB11095
biotech | CAS: 120993-53-5

Desirudin is a direct inhibitor of human thrombin. It has a protein structure that is similar to that of hirudin, the naturally occurring anticoagulant present in the peripharyngeal glands in the medicinal leech, Hirudo medicinalis. Hirudin is a single polype…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Waktu Paruh~2 hours.
Vol. Distribusi0.25 L/kg.
Klirens1.5 to 2.7 mL/min/k…
Genetik -
Deslanoside Approved DB01078
small molecule | CAS: 17598-65-1

Deacetyllanatoside C. A cardiotonic glycoside from the leaves of Digitalis lanata.

Kategori:
Antiarrhythmic agentsCarbohydratesCardanolides +13
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh36 hours
Vol. Distribusi-
Klirens-
Genetik -
Desloratadine Approved DB00967
small molecule | CAS: 100643-71-8

Desloratadine is a second generation, tricyclic antihistamine that which has a selective and peripheral H1-antagonist action. It is the active descarboethoxy metabolite of loratidine (a second generation histamine). Desloratidine has a long-lasting effect and…

Kategori:
Anticholinergic AgentsAntihistamines for Systemic UseBenzocycloheptenes +13
Target Protein:
Histamine H1 receptor
Waktu ParuhDesloratadine has a…
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Desmeninol DB15832
small molecule | CAS: 583-91-5

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +2
Waktu Paruh-
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Desmopressin Approved DB00035
small molecule | CAS: 16679-58-6

Desmopressin (dDAVP), a synthetic analogue of 8-arginine vasopressin (ADH), is an antidiuretic peptide drug modified by deamination of 1-cysteine and substitution of 8-L-arginine by 8-D-arginine. ADH is an endogenous pituitary hormone that has a crucial role …

Kategori:
Agents that produce hypertensionAmino Acids, Peptides, and ProteinsAntidiuretic Agents +27
Target Protein:
Oxytocin receptorVasopressin V2 receptorVasopressin V1a receptor +1
Waktu ParuhFollowing an intran…
Vol. DistribusiThe distribution vo…
Klirens-
Genetik -
Desmoteplase DB04925
biotech | CAS: 145137-38-8

Desmoteplase is a chemical in the saliva of vampire bats. It activates plasminogen to the serine protease, plasmin. Plasmin acts by breaking down fibrin blood clots. When a vampire bat bites its victim, it secretes an enzyme that prevents the blood from clott…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBlood Proteins +13
Target Protein:
Plasminogen
Waktu Paruh-
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Desogestrel Approved DB00304
small molecule | CAS: 54024-22-5

Desogestrel, a prodrug, is a third generation progestogen[A176315] and hence, a member of the gonane family which was largely used in Europe before being approved in the US and Canada.[A176339] It was firstly generated from a study that showed that 11-beta an…

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +25
Target Protein:
Progesterone receptorEstrogen receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe apparent volume…
KlirensThe metabolic clear…
Genetik -
Desomorphine DB01531
small molecule | CAS: 427-00-9

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desonide Approved DB01260
small molecule | CAS: 638-94-8

A nonfluorinated corticosteroid anti-inflammatory agent used topically for dermatoses.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +18
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desoximetasone Approved DB00547
small molecule | CAS: 382-67-2

A topical anti-inflammatory glucocorticoid used in dermatoses, skin allergies, psoriasis, etc.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +14
Target Protein:
Estrogen-related receptor gammaGlucocorticoid receptorSteroid hormone receptor ERR2 +1
Waktu ParuhThe half-life of th…
Vol. Distribusi-
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Desoxycorticosterone acetate Approved DB06780
small molecule | CAS: 56-47-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Mineralocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desoxycortone DB15972
small molecule | CAS: 64-85-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids for Systemic Use +11
Waktu Paruh-
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Klirens-
Genetik -
Desoxyribonuclease Approved DB09551
biotech | CAS: 9003-98-9

Desoxyribonuclease is a crystalline enzyme that aids in the digestion of the thymus nucleic acid. The mechanism of action of the enzyme involves the splitting of thymus nucleic acid into fragments approaching the size of tetranucleotides without the release o…

Kategori:
Blood and Blood Forming OrgansDeoxyribonucleasesEnzymes +3
Waktu Paruh-
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Genetik -
small molecule | CAS: 5863-40-1

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Chloramphenicol acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 101485-50-1

Deskripsi belum tersedia.

Target Protein:
Desvancosaminyl-vancomycin vancosaminetransferasedTDP-epi-vancosaminyltransferase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Desvenlafaxine Approved DB06700
small molecule | CAS: 93413-62-8

Desvenlafaxine (O-desmethylvenlafaxine) is the 0-demetyhlated active metabolite of [venlafaxine]. Like its parent drug, desvenlafaxine is also an antidepressant belonging to the class of serotonin-norepinephrine reuptake inhibitor (SNRI) class.[A261266,A26126…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlcohols +40
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe steady-state vo…
KlirensFollowing the admin…
Genetik -
Dethiobiotin DB03775
small molecule | CAS: 533-48-2

Deskripsi belum tersedia.

Kategori:
CoenzymesEnzymes and CoenzymesImidazoles +4
Target Protein:
ATP-dependent dethiobiotin synthetase BioDATP-dependent dethiobiotin synthetase BioD 1Biotin synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Detomidine DB11556
small molecule | CAS: 76631-46-4

Detomidine is an ?2-adrenergic agonist that is used as a horse sedative. Normally, it is administered in the salt form, detomidine hydrochloride. This drug is prescribed by veterinarians and is marketed as _Dormosedan_. Currently, it is only approved by the F…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deucravacitinib Approved DB16650
small molecule | CAS: 1609392-27-9

Deucravacitinib is a novel oral selective tyrosine kinase 2 (TYK2) inhibitor. Unlike other Janus kinase 1/2/3 inhibitors that bind to the conserved active domain of these non-receptor tyrosine kinases, deucravacitinib binds to the regulatory domain of TYK2 wi…

Kategori:
Antineoplastic and Immunomodulating AgentsBCRP/ABCG2 InhibitorsBCRP/ABCG2 Substrates +17
Target Protein:
Non-receptor tyrosine-protein kinase TYK2
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik -
Deucrictibant DB18303
small molecule | CAS: 2340111-58-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1079043-55-2

Deudextromethorphan is under investigation in clinical trial NCT02153502 (Efficacy, Safety, and Tolerability Study of AVP-786 as an Adjunctive Therapy in Patients With Major Depressive Disorder With an Inadequate Response to Antidepressant Treatment).

Target Protein:
Sodium-dependent serotonin transporterSigma non-opioid intracellular receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deudomperidone DB19055
small molecule | CAS: 2121525-08-2

Deudomperidone is under investigation in clinical trial NCT05832151 (A Study to Evaluate the Efficacy and Safety of CIN-102 (Deudomperidone) in Adults With Diabetic Gastroparesis).

Kategori:
Acids, CarbocyclicBenzene DerivativesPharmaceutical Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1404475-07-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Deupirfenidone DB19056
small molecule | CAS: 1093951-85-9

Deupirfenidone is under investigation in clinical trial NCT05321420 (LYT-100 in Patients With Idiopathic Pulmonary Fibrosis (IPF)).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deuruxolitinib DB18847
small molecule | CAS: 1513883-39-0

Deuruxolitinib is a deuterated form of [ruxolitinib] that selectively inhibits Janus kinases (JAK) JAK1 and JAK2. Deuteration allows the drug to circumvent extensive oxidative metabolism around the cyclopentyl ring, which increases the duration of the pharmac…

Kategori:
BCRP/ABCG2 InhibitorsBCRP/ABCG2 SubstratesBile Salt Export Pump Inhibitors +12
Target Protein:
Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK1Non-receptor tyrosine-protein kinase TYK2
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
Klirens-
Genetik -
Deutarserine DB19057
small molecule | CAS: 103292-62-2

Deutarserine is under investigation in clinical trial NCT04158687 (A Phase 2 Study to Evaluate the Safety and Efficacy of CTP-692 as an Adjunctive Treatment in Adults With Schizophrenia).

Waktu Paruh-
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Genetik -
Deuterium oxide DB19251
small molecule | CAS: 7789-20-0

Deskripsi belum tersedia.

Kategori:
AlkaliesAnionsAntineoplastic Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deutetrabenazine Approved DB12161
small molecule | CAS: 1392826-25-3

Deutetrabenazine is a novel, highly selective vesicular monoamine transporter 2 (VMAT2) inhibitor indicated for the management of chorea associated with Huntington’s disease. It is a hexahydro-dimethoxybenzoquinolizine derivative and a deuterated [DB04844] [A…

Kategori:
Cytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2D6 SubstratesCytochrome P-450 CYP3A Substrates +11
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhThe half-life of to…
Vol. DistribusiThe median volume o…
KlirensIn patients with Hu…
Genetik -
Deutivacaftor DB15141
small molecule | CAS: 1413431-07-8

Deutivacaftor is under investigation in clinical trial NCT03227471 (A Study of VX-445 in Healthy Subjects and Subjects With Cystic Fibrosis).

Waktu Paruh-
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Genetik -
biotech | CAS: 2143580-11-2

Devafidugene civaparvovec is an investigational _in vivo_ genome editing product. It uses proprietary zinc finger nucleases (ZFN) that insert a functional copy of the alpha-L-iduronidase (IDUA) enzyme. Developed by Sangamo Therapeutics, Inc., devafidugene civ…

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Devimistat DB12109
small molecule | CAS: 95809-78-2

Devimistat (CPI-613) has been used in trials studying the treatment of Cancer, Lymphoma, Solid Tumors, Advanced Cancer, and Pancreatic Cancer, among others.

Kategori:
Acids, AcyclicAnionsElectrolytes +5
Target Protein:
2-oxoglutarate dehydrogenase complex component E1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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