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11778

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8554 (72.6%)
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6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Halaman 104 / 236
Fimepinostat DB11891
small molecule | CAS: 1339928-25-4

Fimepinostat (CUDC-907) has been used in trials studying the treatment of lymphoma, solid tumors, breast cancer, multiple myeloma, and NUT midline carcinoma, among others.

Kategori:
Antineoplastic AgentsHistone Deacetylase InhibitorsOxazines +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Finafloxacin Approved DB09047
small molecule | CAS: 209342-40-5

Finafloxacin is a fluoroquinolone antibiotic indicated in the treatment of acute otitis externa (swimmer's ear) caused by the bacteria Pseudomonas aeruginosa and Staphylococcus aureus. Finafloxacin is marketed by Novartis under the brand Xtoro™, and was appro…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Finasteride Approved DB01216
small molecule | CAS: 98319-26-7

Finasteride is a synthetic 4-azasteroid compound [L10565] and specific inhibitor of steroid Type II 5?-reductase, which is an intracellular enzyme that converts the androgen testosterone into 5?-dihydrotestosterone (DHT). It works in a similar fashion as [dut…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +22
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 2Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 1 +1
Waktu ParuhIn healthy young su…
Vol. DistribusiThe volume of distr…
KlirensIn healthy young su…
Genetik -
Finerenone Approved DB16165
small molecule | CAS: 1050477-31-0

Finerenone, or BAY 94-8862, is a mineralocorticoid receptor antagonist indicated to reduce the risk of sustained decline in glomerular filtration rate, end stage kidney disease, cardiovascular death, heart attacks, and hospitalization due to heart failure in …

Kategori:
Agents causing hyperkalemiaCytochrome P-450 CYP2C8 SubstratesCytochrome P-450 CYP3A Substrates +6
Target Protein:
Mineralocorticoid receptor
Waktu ParuhThe half life of a …
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Fingolimod Approved DB08868
small molecule | CAS: 162359-55-9

Multiple sclerosis, or MS, is a devastating inflammatory disease that often progresses and causes severe neurological, physical, and cognitive effects.[A176474] Fingolimod is a sphingosine 1-phosphate receptor modulator for the treatment of relapsing-remittin…

Kategori:
AlcoholsAminesAmino Alcohols +16
Target Protein:
D(3) dopamine receptorSphingosine kinase 1Sphingosine 1-phosphate receptor 5 +4
Waktu ParuhThe half-life of fi…
Vol. DistribusiThe volume of distr…
KlirensFingolimod blood cl…
Genetik -
FINLAY-FR-1 DB16524
biotech

FINLAY-FR-1, also known as Soberana 01, is a vaccine candidate for COVID-19 that is being led developmentally by the Finlay Vaccine Institute[L31373]. It is currently being tested in the clinical trial RPCEC00000332 (Phase I / II, randomized, controlled, adap…

Waktu Paruh-
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Fipexide DB13790
small molecule | CAS: 34161-24-5

Deskripsi belum tersedia.

Kategori:
Nervous SystemPsychoanalepticsPsychostimulants, Agents Used for ADHD and Nootropics
Waktu Paruh-
Vol. Distribusi-
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Firategrast DB12732
small molecule | CAS: 402567-16-2

Firategrast has been used in trials studying the treatment of Multiple Sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +5
Waktu Paruh-
Vol. Distribusi-
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Firazorexton DB19440
small molecule | CAS: 2274802-95-6

Firazorexton is under investigation in clinical trial NCT04096560 (A Study of TAK-994 in Adults With Type 1 and Type 2 Narcolepsy).

Waktu Paruh-
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Firocoxib DB09217
small molecule | CAS: 189954-96-9

Firocoxib is a cycooxygenase-2 (COX-2) selective non-steroidal anti-inflammatory drug. It currently approved for veterinary use in dogs and horses under the brand names Equioxx and Previcox. Firocoxib was the first COX-2 inhibitor approved by the U.S. Food an…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +6
Target Protein:
Prostaglandin G/H synthase 2
Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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Firsocostat DB16166
small molecule | CAS: 1434635-54-7

Firsocostat is under investigation in clinical trial NCT02781584 (Safety, Tolerability, and Efficacy of Selonsertib, Firsocostat, and Cilofexor in Adults With Nonalcoholic Steatohepatitis (NASH)).

Kategori:
Acids, AcyclicButyratesEnzyme Inhibitors +5
Waktu Paruh-
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Fisetin DB07795
small molecule | CAS: 528-48-3

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
Cyclin-dependent kinase 6Fatty acid synthaseCyclin homolog
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fisogatinib DB16167
small molecule | CAS: 1707289-21-1

Fisogatinib is under investigation in clinical trial NCT04194801 (A Phase Ib/ii Study of Fisogatinib(blu-554) in Subjects With Hepatocellular Carcinoma).

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Fitusiran DB15002
biotech | CAS: 1499251-18-1

Fitusiran is under investigation in clinical trial NCT02554773 (An Open-label Extension Study of an Investigational Drug, ALN-AT3SC, in Patients With Moderate or Severe Hemophilia A or B).

Kategori:
Amino SugarsAntisense Elements (Genetics)Carbohydrates +7
Waktu Paruh-
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FK-614 DB12557
small molecule | CAS: 193012-35-0

FK614 has been used in trials studying the treatment of Diabetes Mellitus.

Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
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FK-960 DB06465
small molecule | CAS: 133920-70-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
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FK352B DB06484
small molecule | CAS: 143881-08-7

FK352B is a adenosine A1 antagonist that is developed for the treatment of dialysis-induced hypotension.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
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Genetik -
Flavin adenine dinucleotide Approved DB03147
small molecule | CAS: 146-14-5

A condensation product of riboflavin and adenosine diphosphate. The coenzyme of various aerobic dehydrogenases, e.g., D-amino acid oxidase and L-amino acid oxidase. (Lehninger, Principles of Biochemistry, 1982, p972) Flavin adenine dinucleotide is approved f…

Kategori:
Adenine NucleotidesBiological FactorsCoenzymes +13
Target Protein:
Ribosyldihydronicotinamide dehydrogenase [quinone]Nitric oxide synthase 1Dihydropyrimidine dehydrogenase [NADP(+)] +83
Waktu Paruh-
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Genetik -
Flavin mononucleotide Approved DB03247
small molecule | CAS: 146-17-8

A coenzyme for a number of oxidative enzymes including NADH DEHYDROGENASE. It is the principal form in which RIBOFLAVIN is found in cells and tissues.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +11
Target Protein:
Flavin reductase (NADPH)2-Hydroxyacid oxidase 1Pyridoxine-5'-phosphate oxidase +51
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cholesterol oxidase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Flaviolin DB02521
small molecule | CAS: 479-05-0

Deskripsi belum tersedia.

Kategori:
NaphthalenesQuinones
Target Protein:
PrenyltransferaseBiflaviolin synthase CYP158A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flavone Approved DB07776
small molecule | CAS: 525-82-6

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
AromataseGamma-aminobutyric acid receptor subunit alpha-1Androgen receptor +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flax seed Approved DB10708
biotech

Flax seed allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +2
Waktu Paruh-
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Flecainide Approved DB01195
small molecule | CAS: 54143-55-4

Flecainide is a Class I anti-arrhythmic agent like [encainide] and [propafenone].[A186880] Flecainide’s development began in 1966 and was first synthesized in 1972 as an attempt to generate new anesthetics.[A186931] It is used to prevent supraventricular and …

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ic +27
Target Protein:
Sodium channel protein type 4 subunit alphaSodium channel protein type 5 subunit alphaVoltage-gated inwardly rectifying potassium channel KCNH2 +1
Waktu ParuhIn healthy subjects…
Vol. DistribusiThe average volume …
KlirensThe average clearan…
Genetik -
Fleroxacin DB04576
small molecule | CAS: 79660-72-3

Fleroxacin is a broad-spectrum antimicrobial fluoroquinolone. It strongly inhibits the DNA-supercoiling activity of DNA gyrase. Fleroxacin is not an inhibitor of CYP1A2.[A39048]

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
DNA topoisomerase 2-betaDNA gyrase subunit ADNA topoisomerase 4 subunit A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fletikumab DB12356
biotech | CAS: 1357158-22-5

Fletikumab is under investigation in clinical trial NCT01038674 (Safety and Tolerability of Anti-IL-20 in Subjects With Rheumatoid Arthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flibanserin Approved DB04908
small molecule | CAS: 167933-07-5

Flibanserin is the first drug to be approved for hypoactive sexual desire disorder (HSDD) in premenopausal women by the FDA in August 2015. It was originally developed as an antidepressant medication by Boehringer Ingelheim, but showed lack of efficacy in tri…

Kategori:
Agents that produce hypertensionAntidepressive AgentsCentral Nervous System Depressants +15
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2AD(4) dopamine receptor
Waktu Paruh?11 hours
Vol. Distribusi-
Klirens-
Genetik -
Flindokalner DB16908
small molecule | CAS: 187523-35-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Floctafenine Approved DB08976
small molecule | CAS: 23779-99-9

Floctafenine is an anti-inflammatory analgesic similar in action to aspirin. Floctafenine inhibits prostaglandin synthesis.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +14
Waktu Paruh-
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Florantyrone DB08975
small molecule | CAS: 519-95-9

Florantyrone is used in the treatment of biliary dyskinesia

Waktu Paruh-
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Florasulam DB15316
small molecule | CAS: 145701-23-1

Florasulam is under investigation in clinical trial NCT01193465 (Temperature and Humidity Among Different Anesthesia Work-station).

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
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Florbetaben F-18 Approved DB09148
small molecule | CAS: 902143-01-5

Florbetaben is a fluorine-18 (18F)-labeled stilbene derivative used for Positron Emission Tomography (PET) imaging of the brain. It is used for the non-invasive detection of the density of ß-amyloid neuritic plaques in the brain of adult patients with cogniti…

Kategori:
AminesBenzene DerivativesBenzylidene Compounds +6
Target Protein:
Amyloid-beta precursor protein
Waktu Paruh1 hr
Vol. Distribusi-
Klirens-
Genetik -
Florbetapir F-18 Approved DB09149
small molecule | CAS: 956103-76-7

Florbetapir (18F) is a radiopharmaceutical compound containing the radionuclide fluorine-18 bound to the compound florbetapir, a molecule that binds with high affinity to beta amyloid plaque, a peptide that plays a key role in Alzheimer's Disease pathogenesis…

Kategori:
AlcoholsAminesCentral Nervous System +6
Target Protein:
Amyloid-beta precursor proteinBeta amyloid plaque
Waktu Paruh-
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Florfenicol DB11413
small molecule | CAS: 73231-34-2

Florfenicol is a fluorinated synthetic analog of thiamphenicol.

Kategori:
AlcoholsAnti-Bacterial AgentsAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1196963-74-2

Florilglutamic acid F-18 is under investigation in clinical trial NCT02370563 (PET Imaging of Intracranial Cancers With 18F-FSPG).

Waktu Paruh-
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Flortaucipir DB15033
small molecule | CAS: 1415379-56-4

Flortaucipir is under investigation in clinical trial NCT03507257 (Longitudinal Early-onset Alzheimer's Disease Study Protocol).

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +4
Target Protein:
Microtubule-associated protein tau
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flortaucipir F-18 Approved DB14914
small molecule | CAS: 1522051-90-6

Flortaucipir F-18, also known as <sup>18</sup>F-T807 and <sup>18</sup>F-AV-1451, is a small indole molecule synthesized with a radioactive fluorine isotope.[A203933] It is used as a marker in positron emission tomography (PET) imaging of patients suspected of…

Kategori:
Central Nervous SystemCompounds used in a research, industrial, or household settingContrast Media +6
Target Protein:
Microtubule-associated protein tauAmine oxidase [flavin-containing] AAmine oxidase [flavin-containing] B
Waktu ParuhFlortaucipir F-18 p…
Vol. DistribusiFlortaucipir F-18 i…
Klirens-
Genetik -
small molecule | CAS: 1565797-57-0

PMPBB3 F-18 is under investigation in clinical trial NCT04305210 (Alzheimer's Disease: Clinical Investigation and Neuroimage Studies Including 18F-PM-PBB3 and 18f-florbetapir (AV-45) PET Examination).

Waktu Paruh-
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Flosequinan Approved DB13228
small molecule | CAS: 76568-02-0

Flosequinan was approved in the USA and the UK for a year prior to being withdrawn from the market due to increased mortality in chronic heart failure patients, found in drug trials.[A174979,L43942]

Kategori:
Cardiac TherapyCardiovascular AgentsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 1010702-75-6

Deskripsi belum tersedia.

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Flotufolastat F-18 Approved DB17851
small molecule | CAS: 2639294-14-5

Flotufolastat F-18 (<sup>18</sup>F-rhPSMA-7.3) is an <sup>18</sup>F-labeled ligand that targets the prostate-specific membrane antigen (PSMA).[A259846,L46731] In patients with recurrent prostate cancer that require localized treatment, the use of <sup>18</sup…

Kategori:
Diagnostic RadiopharmaceuticalsFluorine RadioisotopesPositron Emitting Activity +1
Target Protein:
Glutamate carboxypeptidase 2
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Flovagatran DB05714
small molecule | CAS: 871576-03-3

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAmino Acids, Peptides, and Proteins +3
Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluasterone DB06250
small molecule | CAS: 112859-71-9

Has antiproliferative effects on HIV-1 and reduces HIV-1 replication.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +10
Waktu Paruh-
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Fluazuron DB15583
small molecule | CAS: 86811-58-7

Fluazuron is a benzoyl phenylurea compound.

Kategori:
AmidesBenzene Derivatives
Waktu Paruh-
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Flubendazole DB08974
small molecule | CAS: 31430-15-6

Flubendazole is an anthelmintic that is used to treat worm infection in humans. It is available OTC in Europe.

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +7
Waktu Paruh-
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Genetik -
Flubentylosin DB17769
small molecule | CAS: 1809266-03-2

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule | CAS: 1037359-47-9

Deskripsi belum tersedia.

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Fluciclatide DB14842
small molecule | CAS: 879894-00-5

Fluciclatide, an investigational radiotracer intended for PET imaging, was under investigation in clinical trials NCT00565721 and NCT01961583 to evaluate its ability to detect tumors and angiogenesis. The conditions targeted by [18F]Fluciclatide in these stud…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsEthylene Glycols +4
Waktu Paruh-
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Fluciclovine DB15237
small molecule | CAS: 222727-43-7

Fluciclovine is under investigation in clinical trial NCT03036943 (Fluciclovine (18F) Imaging of Breast Cancer).

Waktu Paruh-
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