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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 104 / 252
EPI-589 DB16041
small molecule | CAS: 1147883-03-1

EPI-589 is under investigation in clinical trial NCT02460679 (Safety and Biomarker Study of EPI-589 in Participants With Amyotrophic Lateral Sclerosis (ALS)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epibatidine DB07720
small molecule | CAS: 140111-52-0

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticCentral Nervous System Agents +6
Target Protein:
CHRNA7-FAM7A fusion proteinNeuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit beta-2 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epicaptopril DB02032
small molecule | CAS: 63250-36-2

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAmino AcidsAmino Acids, Cyclic +6
Target Protein:
Metallo-beta-lactamase L1Beta-lactamaseOrganic hydroperoxide resistance protein, putative +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epicept NP-1 DB05492
small molecule

EpiCept NP-1 is a prescription topical analgesic cream designed to provide effective, long-term relief from the pain of peripheral neuropathies. Peripheral neuropathies are medical conditions caused by damage to the nerves in the peripheral nervous system. Th…

Target Protein:
Mu-type opioid receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2B +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epicriptine Approved DB11275
small molecule | CAS: 88660-47-3

Epicriptine is also known as beta-dihydroergocryptine presents a molecular formula of 9,10 alpha-dihydro-13'-epi-b-ergocryptine. Together with the alpha-dihydroergocryptine, it represents one-third of the ergoloid mesylate mixture. Epicriptine differs from th…

Kategori:
AlkaloidsDopamine Agonists
Target Protein:
Dopamine receptor
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 25615-05-8

Epigallo Catechin Gallate is under investigation in clinical trial NCT00799890 (Sunphenon in Progressive Forms of Multiple Sclerosis).

Kategori:
BenzopyransChromansChromones +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 970-74-1

Deskripsi belum tersedia.

Kategori:
BenzopyransChromansChromones +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 989-51-5

Epigallocatechin gallate has been investigated for the treatment of Hypertension and Diabetic Nephropathy.

Kategori:
Anticarcinogenic AgentsAntimutagenic AgentsAntineoplastic Agents +13
Target Protein:
Fatty acid synthaseSignal transducer and activator of transcription 3Gag-Pol polyprotein +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epinastine Approved DB00751
small molecule | CAS: 80012-43-7

Epinastine is used for the prevention of itching associated with allergic conjunctivitis. It has a multi-action effect that inhibits the allergic response in 3 ways: 1. stabilizes mast cells by preventing mast cell degranulation to control the allergic respon…

Kategori:
Acid ReducersAntidepressive AgentsCentral Nervous System Depressants +27
Target Protein:
Histamine H1 receptorHistamine H2 receptorAlpha-1A adrenergic receptor +3
Waktu Paruh12 hours
Vol. Distribusi-
Klirens* 56 L/hr [patients…
Genetik -
Epinephrine Approved DB00668
small molecule | CAS: 51-43-4

Epinephrine, also known as _adrenaline_, is a hormone and neurotransmitter and produced by the adrenal glands that can also be used as a drug due to its various important functions. Though it has long been used in the treatment of hypersensitivity reactions, …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +52
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorBeta-1 adrenergic receptor +5
Waktu ParuhThe plasma half-lif…
Vol. Distribusi-
KlirensIntravenous injecti…
Genetik -
Epirizole DB08991
small molecule | CAS: 18694-40-1

Epirizole is an oral nonsteroidal anti-inflammatory drug (NSAID) used for muscle and joint pain.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epirubicin Approved DB00445
small molecule | CAS: 56420-45-2

An anthracycline which is the 4'-epi-isomer of doxorubicin. The compound exerts its antitumor effects by interference with the synthesis and function of DNA.

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +17
Target Protein:
DNA topoisomerase 2-betaDNADNA topoisomerase 2-alpha
Waktu ParuhHalf-lives for the …
Vol. Distribusi* 21 ± 2 L/kg [60 m…
Klirens* 65 +/- 8 L/hour […
Genetik -
Epitestosterone DB07768
small molecule | CAS: 481-30-1

Epitestosterone is the 17-alpha isomer of testosterone, derived from pregnenolone via the delta5-steroid pathway, and via 5-androstene-3-beta,17-alpha-diol. Epitestosterone acts as an antiandrogen in various target tissues. The ratio between testosterone/epit…

Kategori:
AndrostanesAndrostenesAndrostenols +7
Target Protein:
Aldo-keto reductase family 1 member C1Aldo-keto reductase family 1 member C2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epitizide DB13989
small molecule | CAS: 1764-85-8

Epitizide is an agent, commonly found in combination [triamterene], used to produce diuresis.

Kategori:
DiureticsLow-Ceiling Diuretics and Potassium-Sparing AgentsSodium Chloride Symporter Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EpiVacCorona DB16439
biotech

EpiVacCorona Vaccine, developed by the Vektor State Research Center of Virology and Biotechnology in Russia, is based on peptide-antigens that facilitate immunity to the SARS-CoV-2 virus[L30608]. It is currently being tested in Phase I/II clinical trials for …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eplivanserin DB12177
small molecule | CAS: 130579-75-8

Eplivanserin has been used in trials studying the treatment of Sleep, Insomnia, Chronic Pain, Fibromyalgia, and Primary Insomnia, among others.

Kategori:
Antidepressive AgentsBenzene DerivativesCardiovascular Agents +8
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eplontersen Approved DB16199
biotech | CAS: 1637600-16-8

Eplontersen is a transthyretin-directed antisense oligonucleotide with 3 covalently linked e N-acetyl galactosamine residues for hepatic delivery. It was previously investigated as a potential treatment for hereditary transthyretin-mediated amyloidosis.[A2629…

Kategori:
Antisense OligonucleotidesNervous SystemNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Transthyretin mRNA
Waktu ParuhThe terminal elimin…
Vol. DistribusiEplontersen is expe…
KlirensThe clearance was e…
Genetik -
Epoetin beta DB19434
biotech | CAS: 122312-54-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epoetin delta Approved DB11624
biotech | CAS: 261356-80-3

Epoetin Delta is an ingredient in the EMA-withdrawn product Dynepo.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epofolate DB12266
small molecule | CAS: 958646-17-8

Epofolate has been used in trials studying the treatment of Advanced Solid Tumors. Epofolate (BMS-753493) is a folate conjugate of the epothilone analog BMS-748285 that was designed to selectively target folate receptor expressing cancer cells. In Phase I/IIa…

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsCytochrome P-450 CYP3A Inhibitors +9
Target Protein:
Folate receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epoprostenol Approved DB01240
small molecule | CAS: 35121-78-9

A prostaglandin that is a powerful vasodilator and inhibits platelet aggregation. It is biosynthesized enzymatically from prostaglandin endoperoxides in human vascular tissue. The sodium salt has been also used to treat primary pulmonary hypertension.

Kategori:
AnticoagulantsAntihypertensive AgentsAntiplatelet agents +19
Target Protein:
Prostacyclin synthaseP2Y purinoceptor 12Prostacyclin receptor
Waktu ParuhThe in vitro half-l…
Vol. Distribusi* 357 mL/kg
Klirens-
Genetik -
Epothilone D DB01873
small molecule | CAS: 189453-10-9

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntimitotic AgentsAntineoplastic Agents +9
Target Protein:
Tubulin beta chainTubulin beta-1 chainTubulin beta-4B chain +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epratuzumab DB04958
biotech | CAS: 205923-57-5

Epratuzumab is a humanized monoclonal antibody derived from the murine IG2a monoclonal antibody, LL2 (EPB-2). This agent may subsequently be well matched for use in oncology and the treatment of inflammatory autoimmune disorders, such as lupus.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
B-cell receptor CD22
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprenetapopt DB11684
small molecule | CAS: 5291-32-7

Eprenetapopt has been used in trials studying the treatment of Prostatic Neoplasms, Hematologic Neoplasms, and Platinum Sensitive Recurrent High-grade Serous Ovarian Cancer With Mutated p53.

Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprinomectin DB11405
small molecule | CAS: 123997-26-2

Deskripsi belum tersedia.

Kategori:
AgrochemicalsAnthelminticsAnti-Bacterial Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprodisate DB06405
small molecule | CAS: 21668-77-9

Eprodisate slows the decline of renal function in AA amyloidosis.

Kategori:
AcidsAcids, NoncarboxylicAlkanes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprosartan Approved DB00876
small molecule | CAS: 133040-01-4

Eprosartan is an angiotensin II receptor antagonist used to treat hypertension. It performs 2 actions on the renin angiotensin system. By preventing the binding of angiotensin II to AT1, vascular smooth muscle relaxes and vasodilation occurs. By inhibiting no…

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +13
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhThe terminal elimin…
Vol. Distribusi-
Klirens-
Genetik -
Eprotirome DB05035
small molecule | CAS: 355129-15-6

Eprotirome which is a compound with promising properties for treatment of obesity and dyslipidemia. Eprotirome increases the body’s energy consumption and reduces body weight and markedly reduces blood lipids and blood glucose.

Kategori:
AmidesAminesAniline Compounds
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eprozinol DB13395
small molecule | CAS: 32665-36-4

Deskripsi belum tersedia.

Kategori:
Drugs for Obstructive Airway Diseases
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eptinezumab Approved DB14040
biotech | CAS: 1644539-04-7

Eptinezumab is a fully-humanized IgG1 antibody manufactured using yeast (_Pichia pastoris_) and developed by Lundbeck Seattle Biopharmaceuticals.[L12318] Eptinezumab has been specifically designed to bind to both alpha and beta forms of the human calcitonin g…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +12
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe central volume …
KlirensThe apparent cleara…
Genetik -
Eptotermin alfa Approved DB11631
biotech | CAS: 129805-33-0

A bone morphogenetic protein that is widely expressed during EMBRYONIC DEVELOPMENT. It is both a potent osteogenic factor and a specific regulator of nephrogenesis. Eptotermin alfa is an ingredient in the EMA-withdrawn product Osigraft.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBone Morphogenetic Proteins +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equilenin DB03515
small molecule | CAS: 517-09-9

Equilenin is an estrogenic steroid produced by horses. It has a total of five double bonds in the A- and B-ring. High concentration of equilenin is found in the urine of pregnant mares.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesCytochrome P-450 CYP3A Substrates +12
Target Protein:
Steroid Delta-isomeraseSteroid Delta-isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equilin DB02187
small molecule | CAS: 474-86-2

An estrogenic steroid produced by horses. It has a total of four double bonds in the A- and B-ring. High concentration of equilin is found in the urine of pregnant mares.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesCytochrome P-450 CYP3A Substrates +12
Target Protein:
17-beta-hydroxysteroid dehydrogenase type 1Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equol DB11674
small molecule | CAS: 531-95-3

Equol has been used in trials studying the treatment of Breast Cancer.

Kategori:
BenzopyransChromonesEstrogens +7
Target Protein:
Estrogen receptor betaSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ER2001 DB18165
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eragidomide DB19242
small molecule | CAS: 1860875-51-9

Eragidomide is under investigation in clinical trial NCT04297124 (A Study to Evaluate the Metabolism and Excretion of [14C]-CC-90009 in Healthy Male Subjects).

Kategori:
AcetatesAcids, AcyclicAmides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eravacycline Approved DB12329
small molecule | CAS: 1207283-85-9

Eravacycline, known as _Xerava_ by Tetraphase Pharmaceuticals, is a fully synthetic fluorocycline antibiotic of the tetracycline class with activity against clinically significant gram-negative, gram-positive aerobic, and facultative bacteria. This includes m…

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +6
Target Protein:
30S ribosomal protein S4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe volume of distr…
Klirens17.82 L/min (standa…
Genetik -
ERB-196 DB06875
small molecule | CAS: 550997-55-2

Deskripsi belum tersedia.

Kategori:
Estrogen Receptor beta, agonistsNaphthalenes
Target Protein:
Estrogen receptor betaNuclear receptor coactivator 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erbumine DB18019
small molecule | CAS: 1919888-06-4

Deskripsi belum tersedia.

Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erdafitinib Approved DB12147
small molecule | CAS: 1346242-81-6

In early April of 2019, the US FDA approved Janssen Pharmaceutical Companies' brand name Balversa (erdafitinib) as the first-ever fibroblast growth factor receptor (FGFR) kinase inhibitor indicated for patients with locally advanced or metastatic urothelial c…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C9 Substrates +25
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +7
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe mean total appa…
Genetik -
Erdosteine Approved DB05057
small molecule | CAS: 84611-23-4

Erdosteine is a drug that causes a breakdown of mucus, also known as a _mucolytic_ agent. It is a _thiol_ derivative produced for the clinical management of chronic obstructive bronchitis, in addition to infective exacerbations of chronic bronchitis. This dru…

Kategori:
AcetatesAcids, AcyclicCough and Cold Preparations +4
Target Protein:
Chymotrypsin-like elastase family member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erenumab Approved DB14039
biotech | CAS: 1582205-90-0

Erenumab (AMG-334) (INN; trade name Aimovig) is a human monoclonal antibody designed specifically to bind and antagonize the calcitonin gene-related peptide receptor (CGRPR) as a means to prevent migraines. Aimovig, as released and marketed by Novartis and Am…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhErenumab exhibits n…
Vol. DistribusiAfter a single 140 …
KlirensCertain studies sho…
Genetik -
Ergidina DB18565
biotech

Ergidina is a recombinant human minibody against complement component C5 fused with RGD-motif.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ergocalciferol Approved DB00153
small molecule | CAS: 50-14-6

Ergocalciferol is an inactivated vitamin D analog.[A177526] It is synthesized by some plants in the presence of UVB light.[T577] The production of ergocalciferol was prompted by the identification of dietary deficiency, more specifically vitamin D, as the mai…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCalcium-Regulating Hormones and Agents +11
Target Protein:
Vitamin D3 receptorVoltage-dependent calcium channel
Waktu ParuhErgocalciferol can …
Vol. DistribusiThe amount of circu…
KlirensThere are no formal…
Genetik -
Ergoloid mesylate Approved DB01049
small molecule | CAS: 8067-24-1

Ergoloid Mesylate is an equiproportional preparation of three different ergotamantriones: dihydroergocornine, dihydroergocristine, and dihydroergocryptine.[A32912] All these components are produced by the fungus _Claviceps purpurea_ and are all derivatives of…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +24
Target Protein:
Dopamine receptorAlpha adrenergic receptorBeta adrenergic receptor +1
Waktu ParuhThe reported plasma…
Vol. DistribusiThe volume of distr…
KlirensTo know more about …
Genetik -
Ergometrine Approved DB01253
small molecule | CAS: 60-79-7

An ergot alkaloid with uterine and vascular smooth muscle contractile properties.

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +20
Target Protein:
Alpha-1A adrenergic receptorD(2) dopamine receptor
Waktu Paruht<sub>1/2 &alpha;</…
Vol. Distribusi-
Klirens-
Genetik -
Ergosterol Approved DB04038
small molecule | CAS: 57-87-4

A steroid of interest both because its biosynthesis in FUNGI is a target of ANTIFUNGAL AGENTS, notably AZOLES, and because when it is present in SKIN of animals, ULTRAVIOLET RAYS break a bond to result in ERGOCALCIFEROL.

Kategori:
CholestanesCholestenesDiet, Food, and Nutrition +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ergotamine Approved DB00696
small molecule | CAS: 113-15-5

A vasoconstrictor found in ergot of Central Europe. It is an alpha-1 selective adrenergic agonist and is commonly used in the treatment of migraine disorders.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +39
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 2A +11
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Eribaxaban DB06920
small molecule | CAS: 536748-46-6

Deskripsi belum tersedia.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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