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6694

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3751 (56.0%)
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Halaman 103 / 134
Plasminogen Approved DB16701
biotech | CAS: 9001-91-6

Plasminogen is a pro-enzyme (i.e. a zymogen) which is cleaved to form plasmin - also known as [fibrinolysin] - as part of the fibrinolytic pathway that breaks down fibrin blood clots.[A236035] This pathway is activated when a clot is no longer needed or to pr…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBeta-Globulins +11
Waktu ParuhThe mean half-life …
Vol. DistribusiThe mean steady-sta…
KlirensThe clearance of Ry…
Genetik -
Platanus occidentalis pollen Approved DB10392
biotech

Platanus occidentalis pollen is the pollen of the Platanus occidentalis plant. Platanus occidentalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Platensimycin DB08407
small molecule | CAS: 835876-32-9

Deskripsi belum tersedia.

Kategori:
3-Oxoacyl-(Acyl-Carrier-Protein) SynthaseAcids, CarbocyclicAmides +10
Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Platinum DB12257
small molecule | CAS: 7440-06-4

Platinum is under investigation for the treatment of Metastatic Breast Cancer, Non-small Cell Lung Cancer, Gastric Large Cell Neuroendocrine Carcinoma, Colorectal Large Cell Neuroendocrine Carcinoma, and Pancreatic Large Cell Neuroendocrine Carcinoma, among o…

Kategori:
Antineoplastic AgentsChlorine CompoundsCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plazomicin Approved DB12615
small molecule | CAS: 1154757-24-0

Developed by Achaogen biopharmaceuticals, plazomicin is a next-generation aminoglycoside synthetically derived from [DB12604]. The structure of plazomicin was established via appending hydroxylaminobutyric acid to [DB12604] at position 1 and 2-hydroxyethyl gr…

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +12
Target Protein:
rRNA methyltransferase 2, mitochondrial30S ribosomal protein S1130S ribosomal protein S14
Waktu ParuhThe mean (±SD) half…
Vol. DistribusiThe mean (±SD) volu…
KlirensFollowing administr…
Genetik -
Plecanatide Approved DB13170
small molecule | CAS: 467426-54-6

Plecanatide is a drug approved in January 2017 by the FDA for the treatment of chronic idiopathic constipation (CIC). It should not be used in children less than six years of age, and should be avoided in patients six years to 18 years of age

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +12
Target Protein:
Guanylyl cyclase CGuanylate cyclase soluble subunit alpha-2
Waktu Paruhhalf-life (t½) cann…
Vol. DistribusiConcentrations of p…
KlirensNo excretion studie…
Genetik -
Plerixafor Approved DB06809
small molecule | CAS: 110078-46-1

Plerixafor is a small-molecule inhibitor of C-X-C chemokine receptor type 4 (CXCR4) that acts as a hematopoietic stem cell mobilizer.[A7117,L45678] It is used to stimulate the release of stem cells from the bone marrow into the blood in patients with non-Hodg…

Kategori:
Adjuvants, ImmunologicAminesAnti-HIV Agents +9
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhPlerixafor has a di…
Vol. DistribusiPlerixafor has an a…
KlirensPlerixafor has a to…
Genetik -
Plicamycin Approved DB06810
small molecule | CAS: 18378-89-7

Plicamycin is an antineoplastic antibiotic produced by Streptomyces plicatus. It has been used in the treatment of testicular cancer, Paget's disease of bone, and, rarely, the management of hypercalcemia. The manufacturer discontinued plicamycin in 2000.

Kategori:
AnthracyclinesAntibiotics, AntineoplasticAntineoplastic Agents +15
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plitidepsin DB04977
small molecule | CAS: 137219-37-5

Aplidine is a peptide found in tunicates which shows promise in shrinking tumors in pancreatic, stomach, bladder, and prostate cancers. The specific marine organism is _Aplidium albicans_. Aplidine is also of interest as a potential treatment for some leukemi…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Palmitoyl-protein thioesterase 1Elongation factor 1-alpha 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PLN-74809 DB16515
small molecule

PLN-74809 is a small-molecule that dually inhibits both ?<sub>v</sub>?<sub>6</sub> and ?<sub>v</sub>?<sub>1</sub> to treat both idiopathic pulmonary fibrosis (IPF) and primary sclerosing cholangitis (PSC)[L31693]. The compound was granted orphan drug designat…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Integrin alpha-VIntegrin beta-1Integrin beta-6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plozalizumab DB12520
biotech | CAS: 1610761-46-0

Plozalizumab has been investigated for the treatment of Atherosclerosis. Plozalizumab, a novel humanized monoclonal antibody, specifically targets CCR2 chemokine receptors found on the surface of certain white blood cells including macrophages and monocytes. …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PLX51107 DB17543
small molecule | CAS: 1627929-55-8

PLX51107 is a potent and selective inhibitor of the bromodomain and extraterminal (BET) protein family.[A257246,A257251] PLX51107 is under investigation in clinical trial NCT04022785 (PLX51107 and Azacitidine in Treating Patients With Acute Myeloid Leukemia o…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PMX-205 DB17938
small molecule | CAS: 514814-49-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesReceptor, Anaphylatoxin C5a, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PNT001 DB18375
biotech

PNT001 is a humanized IgG4 S228P monoclonal antibody targeting the cis conformation of the phosphorylated Thr231-Pro232 motif in tau.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pociredir DB18070
small molecule | CAS: 2490676-18-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Podofilox Approved DB01179
small molecule | CAS: 518-28-5

A lignan found in podophyllin resin from the roots of podophyllum plants. It is a potent spindle poison, toxic if taken internally, and has been used as a cathartic. It is very irritating to skin and mucous membranes, has keratolytic actions, has been used to…

Kategori:
Antimitotic AgentsAntineoplastic Agents, PhytogenicAntiviral Agents +11
Target Protein:
DNA topoisomerase 2-betaTubulin alpha-4A chainTubulin beta chain +1
Waktu Paruh1.0 to 4.5 hours.
Vol. Distribusi-
Klirens-
Genetik -
Podophyllin Approved DB09094
small molecule | CAS: 9000-55-9

Podophyllin is a resin extracted from the roots of _Podophyllum peltatum_ (American mandrake) and _Podophyllum emodi_, which contains numerous compounds, amongst which is podophyllin (as well as the drug [podophyllotoxin]). Podophyllin is the principal active…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicBiological Products +11
Waktu ParuhNo data available.
Vol. DistribusiNo data available.
KlirensNo data available.
Genetik -
Polaprezinc DB09221
small molecule | CAS: 107667-60-7

Polaprezinc is a chelated form of zinc and L-carnosine. It is a zinc-related medicine approved for the first time in Japan, which has been clinically used to treat gastric ulcers [L1307, L1308]. It was determined that polaprezinc may be effective in pressure…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Ulcer AgentsDipeptides +10
Target Protein:
Tumor necrosis factorInterleukin-6Interleukin-3 +5
Waktu ParuhThe half-life of po…
Vol. Distribusi-
Klirens-
Genetik -
Polatuzumab vedotin Approved DB12240
biotech | CAS: 1313206-42-6

Polatuzumab vedotin is a CD79b-directed antibody-drug conjugate that delivers monomethyl auristatin E (MMAE), an anti-mitotic agent, to cancer cells.[L6658] The drug consists of three components - a humanized immunoglobulin G1 (IgG1) monoclonal antibody speci…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +22
Target Protein:
B-cell antigen receptor complex-associated protein beta chain
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe estimated centr…
KlirensThe predicted clear…
Genetik -
Poliglusam DB11234
small molecule | CAS: 9012-76-4

Poliglusam, or chitosan, is a linear polysaccharide consisting of D-glucosamine and N-acetyl-D-glucosamine. Naturally-occuring poliglusam is found in the cell walls of fungi, soil and sediments where it is produced from degradation of chitin induced by certai…

Kategori:
Anticholesteremic AgentsBiocompatible MaterialsBiopolymers +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Poliovirus type 1 antigen is a suspension of poliovirus Type 1 (Mahoney) used in the active immunization of infants (as young as 6 weeks of age), children, and adults for the prevention of poliomyelitis caused by poliovirus Type 1. The vaccine contains purifi…

Kategori:
Actively Acquired ImmunityInactivated Poliovirus Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Poliovirus type 2 antigen is a suspension of poliovirus Type 2 (MEF-1) used in the active immunization of infants (as young as 6 weeks of age), children, and adults for the prevention of poliomyelitis caused by poliovirus Type 2. The vaccine contains purified…

Kategori:
Actively Acquired ImmunityInactivated Poliovirus Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Poliovirus type 3 antigen is a suspension of poliovirus Type 3 (Saukett) used in the active immunization of infants (as young as 6 weeks of age), children, and adults for the prevention of poliomyelitis caused by poliovirus Type 3. The vaccine contains purifi…

Kategori:
Actively Acquired ImmunityInactivated Poliovirus Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Poloxamer 188 Approved DB11333
small molecule | CAS: 691397-13-4

Poloxamer 188 (P188) is a nonionic block linear copolymer that exhibits rheologic, anti-thrombotic, anti-inflammatory, and cytoprotective activities in various tissue injury models [A33121]. Composed of two hydrophilic side-chains attached to a hydrophobic ce…

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +9
Waktu ParuhIn humans, P188 has…
Vol. DistribusiThe volume of distr…
KlirensFollowing a 48-hour…
Genetik -
small molecule | CAS: 26811-96-1

Poly(lactic acid) is under investigation in clinical trial NCT00126308 (Facial Lipoatrophy Trial: Immediate Versus Deferred Injections of Poly-L-Lactic Acid for HIV Facial Lipoatrophy).

Kategori:
Dental ImplantsMacromolecular SubstancesPolymers
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Polycarbophil DB09311
small molecule | CAS: 9003-97-8

Polycarbophil calcium is a synthetic polymer manufactured from the cross-linking of polyacrylic acid with divinyl glycol and a calcium counter-ion. Polycarbophil calcium is a stool stabilizer used to treat constipation. This drug may also be used to help rel…

Kategori:
AntidiarrhealsBulk-Forming LaxativesCompounds used in a research, industrial, or household setting +6
Waktu ParuhCalcium polycarboph…
Vol. DistribusiCalcium polycarboph…
KlirensCalcium polycarboph…
Genetik -
Polydatin Approved DB11263
small molecule | CAS: 27208-80-6

Polydatin, or Piceid, is a natural precursor and glycoside form of resveratrol with a monocrystalline structure. While it is isolated from the bark of *Picea sitchensis* or *Polygonum cuspidatum*, polydatin may be detected in grape, peanut, hop cones, red win…

Kategori:
Benzene DerivativesBenzylidene CompoundsCarbohydrates +3
Target Protein:
Pyruvate kinase PKM
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Polyestradiol phosphate Approved DB09369
small molecule | CAS: 28014-46-2

Polymeric phosphoric acid ester of estradiol.

Kategori:
Antineoplastic and Immunomodulating AgentsEndocrine TherapyEstradiol Congeners +10
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Polyethylene glycol Approved DB09287
small molecule | CAS: 25322-68-3

Polyethylene glycol (PEG) is a synthetic polymer produced via polymerization of ethylene oxide molecules to make joining units of ethylene glycol by an ether linkage.[A190975,A190978] PEGs are water-soluble polymers that can form hydrogen bonds in a ratio of …

Kategori:
AlcoholsAlimentary Tract and MetabolismCompounds used in a research, industrial, or household setting +21
Waktu ParuhFollowing a two-day…
Vol. DistribusiFollowing a two-day…
KlirensThere is limited in…
Genetik -
Polyethylene glycol 300 Approved DB11161
small molecule | CAS: 25322-68-3

Polyethylene glycol 300 (PEG 300) is a water-miscible polyether with an average molecular weight of 300 g/mol. It is a clear viscous liquid at room temperature with non-volatile, stable properties [A33116]. Polyethylene glycols are widely used in biochemistry…

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +3
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Polyethylene glycol 400 Approved DB11077
small molecule | CAS: 25322-68-3

Polyethylene glycols (PEGs) are products made of condensed ethylene oxide and water that can contain various derivatives and have various functions. Because many PEG types are hydrophilic, they are favorably used as enhancers of penetration, and used heavily …

Kategori:
AlcoholsArtificial TearsCompounds used in a research, industrial, or household setting +8
Target Protein:
Ectonucleotide pyrophosphatase/phosphodiesterase family member 1Oxidoreductase HTATIP2
Waktu ParuhGreat than 24h [L17…
Vol. Distribusi-
KlirensIn mice, lease than…
Genetik -
Polygala senega root Approved DB14749
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 31961-54-3

Deskripsi belum tersedia.

Kategori:
AmidinesFlocculation
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Polymyxin B Approved DB00781
biotech | CAS: 1404-26-8

Polymyxin B was discovered in the 1940s[A176429]. They are basic polypeptides of about eight amino acids and have cationic detergent action on cell membranes[A176426]. Polymyxin B is used for infections with gram-negative organisms, but may be neurotoxic and …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnti-Bacterial Agents +19
Target Protein:
Bacterial outer membraneDihydropteroate synthase
Waktu ParuhIn one study the ha…
Vol. Distribusi1 compartment model…
Klirens1 compartment model…
Genetik -
small molecule | CAS: 81859-24-7

Polyquaternium-10 is a quaternized hydroxyethyl cellulose and a polycationic polymer. It is commonly found in cosmetics and personal care products to mainly reduce static electricity and form films.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Polysorbate 20 Approved DB11178
small molecule | CAS: 9005-64-5

Polysorbate 20 is a polysorbate-type nonionic surfactant used in many commercial, household and pharmaceutical products. It is composed of 20 repeated units of polyethylene glycol via ethoxylation. Polysorbate 20 is a wetting agent in food products, as well a…

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Polysorbate 80 Approved DB11063
small molecule | CAS: 9005-65-6

Polysorbate, a substance formulated by the reaction of sorbitan fatty acid ester (a nonionic surfactant) with ethylene oxide, is used in many foreign countries, including the U.S. and the EU, where it acts as an emulsifier, a solubilizer in many foods, includ…

Kategori:
AlcoholsArtificial TearsCompounds used in a research, industrial, or household setting +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Polyvalent antigen-KLH conjugate vaccine is a multivalent cancer vaccine comprised of the five tumor-associated antigens (TAAs) globo H, GM2 ganglioside, Tn-MUC1, TF, and sTn conjugated with the immunoadjuvant keyhole limpet hemocyanin (KLH). It is under inve…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Polyvinyl alcohol Approved DB11060
small molecule | CAS: 9002-89-5

Polyvinyl alcohol is a water-soluble synthetic polymer obtained by polymerization of vinyl alcohol. It has varying roles in commercial and industrial applications such as papermaking, textiles, and printing. Polyvinyl alcohol is found in ophthalmic solutions …

Kategori:
AlcoholsAlkenesArtificial Tears +8
Waktu ParuhWhen injected intra…
Vol. DistribusiThis drug does not …
Klirens-
Genetik -
Ponatinib Approved DB08901
small molecule | CAS: 943319-70-8

Ponatinib is a novel Bcr-Abl tyrosine kinase inhibitor that is especially effective against the T315I mutation for the treatment of chronic myeloid leukemia. FDA approved on December 14, 2012.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +23
Target Protein:
Tyrosine-protein kinase ABL1Breakpoint cluster region proteinMast/stem cell growth factor receptor Kit +12
Waktu ParuhAfter oral administ…
Vol. DistribusiAfter oral administ…
Klirens-
Genetik -
Poractant alfa Approved DB09113
biotech | CAS: 129069-19-8

Poractant alfa is a pulmonary surfactant marketed as Curosurf in the United States and Canada. It is used to treat Respiratory Distress Syndrome (RDS) in premature infants with an endogenous pulmonary surfactant deficiency. Poractant alfa is an extract of nat…

Kategori:
Alveolar Surface Tension ReductionBradycardia-Causing AgentsComplex Mixtures +6
Waktu ParuhThe half-life of po…
Vol. DistribusiNo studies on the d…
KlirensNo studies on clear…
Genetik -
Porfiromycin DB06478
small molecule | CAS: 801-52-5

Porfiromycin is a substance that is being studied in the treatment of cancer. It belongs to the family of drugs called anticancer antibiotics.

Kategori:
Antibiotics, AntineoplasticAntineoplastic AgentsAzirines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pork collagen Approved DB14100
biotech

Pork Collagen is used within MACI® (autologous cultured chondrocytes on porcine collagen membrane) as an autologous cellularized scaffold product indicated for the repair of single or multiple symptomatic, full-thickness cartilage defects of the knee with or …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Porphobilinogen DB02272
small molecule | CAS: 487-90-1

Porphobilinogen is a pyrrole involved in porphyrin metabolism. It is generated by the enzyme ALA dehydratase, and converted into hydroxymethyl bilane by the enzyme porphobilinogen deaminase.

Target Protein:
Delta-aminolevulinic acid dehydratase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Posaconazole Approved DB01263
small molecule | CAS: 171228-49-2

Posaconazole is a triazole antifungal drug that is used to treat invasive infections by Candida species and Aspergillus species in severely immunocompromised patients.

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +23
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhPosaconazole is eli…
Vol. Distribusi* 1774 L
Klirens* 32 L/hr * 51 L/h…
Genetik -
Posdinemab DB18941
biotech | CAS: 2517973-04-3

Posdinemab is under investigation in clinical trial NCT04619420 (A Study of JNJ-63733657 in Participants With Early Alzheimer's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Posoleucel DB17974
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
POT-4 DB06056
biotech

POT-4 is a peptide that specifically inhibits complement activation and is initially being developed for the treatment of age-related macular degeneration (AMD). The investigational drug was under investigation in clinical trial NCT00473928 (Safety of Intravi…

Target Protein:
Complement C3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Potassium Approved DB14500
small molecule | CAS: 7440-09-7

Potassium is an essential nutrient, like [Calcium] and [Magnesium]. It was identified as a shortfall nutrient by the 2015-2020 Advisory Committee of Dietary Guidelines for Americans.[A186928] Many conditions and diseases interfere with normal body potassium b…

Kategori:
Agents causing hyperkalemiaDiureticsElements +8
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu ParuhIn one clinical stu…
Vol. DistribusiPotassium is presen…
KlirensPotassium is freely…
Genetik -
Potassium bicarbonate Approved DB11098
small molecule | CAS: 298-14-6

Potassium bicarbonate is a white, crystalline, slightly alkaline and salty substance. It is produced by the passage of carbon dioxide through an aqueous potassium carbonate solution. It is used in medicine as an antacid.[T141] It is registered in the FDA unde…

Kategori:
Agents causing hyperkalemiaAlimentary Tract and MetabolismAnions +8
Target Protein:
Hydrogen ions
Waktu ParuhSome reports have s…
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5101–5150 dari 6694
Sebelumnya Halaman 103 / 134 Berikutnya