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12560

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9109 (72.5%)
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12560 (100.0%)

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Halaman 103 / 252
biotech | CAS: 2417199-08-5

Englumafusp alfa is under investigation in clinical trial NCT04077723 (A Study to Evaluate the Safety, Pharmacokinetics and Preliminary Anti-tumor Activity of Englumafusp Alfa in Combination With Obinutuzumab and in Combination With Glofitamab Following a Pre…

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Enibarcimab DB16730
biotech | CAS: 2305638-98-4

Enibarcimab is under investigation in clinical trial NCT03989531 (Adrecizumab in Cardiogenic Shock).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
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Enibomal DB13229
small molecule | CAS: 125-55-3

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics, GeneralNervous System +2
Waktu Paruh-
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Eniluracil DB03516
small molecule | CAS: 59989-18-3

Eniluracil, which was previously under development by GlaxoSmithKline (GSK), is being developed by Adherex to enhance the therapeutic value and effectiveness of 5-fluorouracil (5-FU), one of the world’s most widely-used oncology agents. 5-FU is widely used i…

Kategori:
Enzyme InhibitorsPyrimidinesPyrimidinones
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Aldehyde oxidaseXanthine dehydrogenase/oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enisoprost DB19319
small molecule | CAS: 81026-63-3

Deskripsi belum tersedia.

Kategori:
Anti-Ulcer AgentsAutacoidsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
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Enitociclib DB17297
small molecule | CAS: 1610408-97-3

Deskripsi belum tersedia.

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ENMD-1198 DB05959
small molecule | CAS: 864668-87-1

Deskripsi belum tersedia.

Kategori:
EstranesFused-Ring CompoundsSteroids
Target Protein:
Hypoxia-inducible factor 1-alphaTumor necrosis factor receptor superfamily member 11ASignal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENMD-981693 DB16891
small molecule | CAS: 934353-76-1

Deskripsi belum tersedia.

Kategori:
Protein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Enmetazobactam Approved DB18716
small molecule | CAS: 1001404-83-6

Enmetazobactam is a penicillanic acid sulfone extended-spectrum beta (?)-lactamase (ESBL) inhibitor.[A263266] Because ESBL enzymes can hydrolyze important antibiotics such as penicillins, broad-spectrum cephalosporins and monobactams, ESBL-producing bacteria …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +7
Target Protein:
Extended-spectrum beta-lactamase PER-1Beta-lactamase
Waktu ParuhThe mean (SD) half-…
Vol. DistribusiMean (SD) steady st…
KlirensThe mean (SD) clear…
Genetik -
Enoblituzumab DB15017
biotech | CAS: 1353485-38-7

Enoblituzumab is under investigation in clinical trial NCT02982941 (Enoblituzumab (MGA271) in Children With B7-H3-expressing Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enobosarm DB12078
small molecule | CAS: 841205-47-8

Enobosarm has been used in trials studying the treatment of Stress Urinary Incontinence and Triple Negative Breast Cancer.

Kategori:
AmidesAminesAniline Compounds
Waktu Paruh-
Vol. Distribusi-
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Enokizumab DB05555
biotech | CAS: 909875-08-7

A humanized immunoglobulin G1k anti-interleukin-9 mAb.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Enoxacin Approved DB00467
small molecule | CAS: 74011-58-8

A broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-betaDNA gyrase subunit ADNA topoisomerase 4 subunit A +1
Waktu ParuhPlasma half-life is…
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Enoxaparin Approved DB01225
small molecule | CAS: 9005-49-6

Enoxaparin is a common low-molecular-weight heparin (LMWH) used in the prevention and management of various thromboembolic disorders. Initially approved by the FDA in 1993, it is administered by a subcutaneous or intravenous injection and marketed by several …

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +7
Target Protein:
Antithrombin-IIICoagulation factor XProthrombin
Waktu ParuhThe half-life of en…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Enoxolone DB13089
small molecule | CAS: 471-53-4

Enoxolone (glycyrrhetic acid) has been investigated for the basic science of Apparent Mineralocorticoid Excess (AME).

Kategori:
Anti-Inflammatory AgentsCicatrizantsDermatologicals +4
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enpatoran DB16501
small molecule | CAS: 2101938-42-3

Enpatoran (M5049) was under investigation in clinical trials for various conditions. It was investigated for systemic lupus erythematosus and cutaneous lupus erythematosus in completed trials (NCT04647708 and NCT05162586) and in a recruiting trial (NCT0554032…

Kategori:
Experimental Unapproved Treatments for COVID-19
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Enprostil DB13824
small molecule | CAS: 73121-56-9

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsAutacoids +12
Waktu Paruh-
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Enrasentan DB06460
small molecule | CAS: 167256-08-8

Deskripsi belum tersedia.

Kategori:
Endothelin Receptor AntagonistsIndenes
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu Paruh-
Vol. Distribusi-
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Enrofloxacin DB11404
small molecule | CAS: 93106-60-6

Enrofloxacin is an antibiotic agent from the fluoroquinolone family produced by the Bayer Corporation. Enrofloxacin is approved by the FDA for its veterinary use. Due to the identification of fluoroquinolone-resistant strains of _Campylobacter_, in September …

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Ensartinib DB14860
small molecule | CAS: 1370651-20-9

Ensartinib is under investigation in clinical trial NCT03420508 (Treating Patients With Melanoma and ALK Alterations With Ensartinib).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
ALK tyrosine kinase receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensifentrine Approved DB16157
small molecule | CAS: 1884461-72-6

Ensifentrine is a first-in-class, selective dual inhibitor of the phosphodiesterase 3 (PDE3) and phosphodiesterase 4 (PDE4) enzymes.[L50903] On June 26, 2024, the FDA announced the approval of an inhaled product of ensifentrine for the treatment of chronic o…

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP2D6 Substrates +6
Target Protein:
Phosphodiesterase 3Phosphodiesterase 4
Waktu ParuhFollowing twice-dai…
Vol. DistribusiApparent central an…
Klirens-
Genetik -
Ensitrelvir DB18834
small molecule | CAS: 2647530-73-0

Ensitrelvir is under investigation in clinical trial NCT05605093 (Strategies and Treatments for Respiratory Infections & Viral Emergencies (STRIVE): Shionogi Protease Inhibitor (Ensitrelvir)).

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +5
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Ensituximab DB12342
biotech | CAS: 1092658-06-4

Ensituximab has been used in trials studying the treatment of Pancreatic Cancer, Adult, Metastatic Colorectal Cancer, and Metastatic Pancreatic Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Ensovibep DB19078
biotech | CAS: 2451126-06-8

Ensovibep is under investigation in clinical trial NCT04501978 (ACTIV-3: Therapeutics for Inpatients With COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
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Ensulizole Approved DB11115
small molecule | CAS: 27503-81-7

Ensulizole, also known as 2-phenylbenzimidazole-5-sulfonic acid, is a water-soluble sunscreen agent that absorbs strongly at UV-B wavelengths. It is commonly found in cosmetic products and sunscreen formulas in combination with other UV filter compounds due t…

Kategori:
AcidsAcids, NoncarboxylicHeterocyclic Compounds, Fused-Ring +3
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Entacapone Approved DB00494
small molecule | CAS: 130929-57-6

Entacapone is a selective, reversible catechol-O-methyl transferase (COMT) inhibitor for the treatment of Parkinson's disease. It is a member of the class of nitrocatechols. When administered concomittantly with levodopa and a decarboxylase inhibitor (e.g., c…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBenzene Derivatives +11
Target Protein:
Catechol O-methyltransferase
Waktu Paruh0.4-0.7 hour
Vol. Distribusi* 20 L
Klirens* 850 mL/min
Genetik -
Entecavir Approved DB00442
small molecule | CAS: 142217-69-4

Entecavir is an oral antiviral drug used in the treatment of hepatitis B infection. It is marketed under the trade name Baraclude (BMS). Entecavir is a guanine analogue that inhibits all three steps in the viral replication process, and the manufacturer cl…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
DNA
Waktu ParuhAfter reaching peak…
Vol. Distribusi-
Klirens* renal cl=383.2 +/…
Genetik -
biotech

Deskripsi belum tersedia.

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Entolimod DB12304
biotech | CAS: 951628-22-1

Entolimod has been used in trials studying the treatment of Mucositis, Tongue Cancer, Colorectal Cancer, Stage IVA Verrucous Carcinoma of the Larynx, and Stage IVB Verrucous Carcinoma of the Larynx, among others.

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
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Entrectinib Approved DB11986
small molecule | CAS: 1108743-60-7

Entrectinib is a tropomyosin receptor tyrosine kinase (TRK) TRKA, TRKB, TRKC, proto-oncogene tyrosine-protein kinase ROS1, and anaplastic lymphoma kinase (ALK) inhibitor.[L8081] It was approved by the FDA in August 2019 for use in the treatment of ROS1-positi…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
ALK tyrosine kinase receptorHigh affinity nerve growth factor receptorNT-3 growth factor receptor +4
Waktu ParuhEntrectinib has a h…
Vol. DistribusiEntrectinib has an …
KlirensThe apparent cleara…
Genetik -
Envafolimab DB15769
biotech | CAS: 2102192-68-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Programmed cell death 1 ligand 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enzacamene Approved DB11219
small molecule | CAS: 36861-47-9

Commonly known as 4-methylbenzylidene-camphor (4-MBC), enzacamene is a camphor derivative and an organic chemical UV-B filter. It is used in cosmetic products such as sunscreen to provide skin protection against UV rays. While its effects on the human reprodu…

Kategori:
Bicyclic MonoterpenesBornanesBridged-Ring Compounds +5
Target Protein:
Progesterone receptorAndrogen receptorEstrogen receptor beta +1
Waktu ParuhThe half life of en…
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Enzalutamide Approved DB08899
small molecule | CAS: 915087-33-1

Enzalutamide is an androgen receptor (AR) inhibitor for the treatment of castration-resistant prostate cancer (CRPC), both metastatic and non-metastatic.[L40639] It is a second-generation antiandrogen agent that the FDA approved on August 31, 2012.[L40639, A2…

Kategori:
AmidesAndrogen Receptor AntagonistsAndrogen Receptor Inhibitors +35
Target Protein:
Androgen receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean (%CV) volu…
KlirensThe mean apparent c…
Genetik -
Enzalutamide d3 DB19123
small molecule | CAS: 1443331-82-5

Enzalutamide d3 is under investigation in clinical trial NCT03850795 (HC-1119 Versus Enzalutamide in Metastatic Castration-resistant Prostate Cancer (Mcrpc)).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enzastaurin DB06486
small molecule | CAS: 170364-57-5

Enzastaurin, an investigational, targeted, oral agent, will be evaluated at more than 100 sites worldwide for the treatment of relapsed glioblastoma multiforme (GBM), an aggressive and malignant form of brain cancer.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein kinase C beta typePhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformRAC-alpha serine/threonine-protein kinase +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EO-3021 DB18358
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
EP-0042 DB18120
small molecule | CAS: 1402709-93-6

Deskripsi belum tersedia.

Waktu Paruh-
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EP-2104R DB05675
biotech

EP-2104R is an imaging pharmaceutical under development for the detection of blood clots. It is the first targeted high-resolution technique designed to visualize blood clots directly. It is being developed by EPIX Pharmaceuticals, Inc.

Kategori:
Amino Acids, Peptides, and ProteinsContrast MediaElements +3
Target Protein:
Fibrinogen alpha chain
Waktu Paruh-
Vol. Distribusi-
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EP0057 DB05899
small molecule

EP0057 is a conjugate of Insert's proprietary drug delivery molecule, Cyclosert, and the potent anti-cancer compound [camptothecin].

Kategori:
AlkaloidsCarbohydratesCompounds used in a research, industrial, or household setting +5
Waktu Paruh-
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Epacadostat DB11717
small molecule | CAS: 1204669-58-8

Epacadostat has been used in trials studying the treatment of HL, Melanoma, Glioblastoma, Mucosal Melanoma, and Ovarian Carcinoma, among others.

Kategori:
AmidesAminesAntineoplastic Agents +4
Target Protein:
Indoleamine 2,3-dioxygenase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epafipase DB16158
biotech | CAS: 208576-22-1

Epafipase is under investigation in clinical trial NCT00037687 (Safety and Efficacy of Recombinant Human Platelet-activating Factor Acetylhydrolase for the Treatment of Severe Sepsis).

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Epalrestat DB15293
small molecule | CAS: 82159-09-9

Epalrestat is under investigation in clinical trial NCT03244358 (Evaluation of Epalrestat in Metastatic Triple-negative Breast Cancer).

Kategori:
Enzyme InhibitorsSulfur CompoundsThiazoles
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
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Epaminurad DB18973
small molecule | CAS: 1198153-15-9

Epaminurad is under investigation in clinical trial NCT05815901 (A Therapeutic Confirmatory Study of Epaminurad Versus Febuxostat in Gout Patients).

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Epanolol DB13757
small molecule | CAS: 86880-51-5

Epanolol is an beta blocker.

Kategori:
AcetamidesAdrenergic AgentsAdrenergic Antagonists +18
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
EPC2407 DB05189
small molecule

EPC2407 is a novel small molecule vascular disruption agent and apoptosis inducer for the treatment of patients with advanced solid tumors and lymphomas. It is intended for the treatment of advanced cancer patients with solid tumors that are well vascularized…

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
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Genetik -
Epcoritamab Approved DB16672
biotech | CAS: 2134641-34-0

Epcoritamab is an IgG1-bispecific antibody that simultaneously binds to CD3 on T-cells and CD20 on B-cells.[A259736,A258488,A259761,L46516] Epcoritamab promotes the activation and expansion of T-cells and, by being able to bind to both CD20 and CD3, it leads …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +13
Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3 epsilon chain
Waktu ParuhA full dose of epco…
Vol. DistribusiEpcoritamab has an …
KlirensA full dose of epco…
Genetik -
Epeleuton DB18100
small molecule | CAS: 1667760-39-5

Deskripsi belum tersedia.

Kategori:
Dietary FatsDietary Fats, UnsaturatedEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Epelsiban DB11934
small molecule | CAS: 872599-83-2

Epelsiban has been investigated for the treatment of Premature Ejaculation.

Kategori:
OxazinesPiperazines
Target Protein:
Oxytocin receptor
Waktu Paruh-
Vol. Distribusi-
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Ephedrine Approved DB01364
small molecule | CAS: 299-42-3

Ephedrine was first described in western literature in 1888, as a naturally occurring component of the ephedra plant, along with [pseudoephedrine].[A193698] Ephedrine acts as both a direct and indirect sympathomimetic. It is an alpha- and beta-adrenergic rece…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +39
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptorBeta-1 adrenergic receptor +2
Waktu ParuhOral ephedrine has …
Vol. DistribusiOral ephedrine has …
KlirensOral ephedrine has …
Genetik -
small molecule | CAS: 1082659-36-6

Deskripsi belum tersedia.

Waktu Paruh-
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Menampilkan 5101–5150 dari 12560
Sebelumnya Halaman 103 / 252 Berikutnya