Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 102 / 236
small molecule | CAS: 49564-56-9

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsMuscle RelaxantsMuscle Relaxants, Peripherally Acting Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fazirsiran DB17891
biotech | CAS: 2175009-08-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fazpilodemab DB18924
biotech | CAS: 2517935-02-1

Fazpilodemab is under investigation in clinical trial NCT04171765 (A Study to Evaluate the Efficacy, Safety, and Pharmacokinetics of BFKB8488A Compared With Placebo in Participants With Non-alcoholic Steatohepatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FB-101 DB17956
small molecule

FB-101 is a c-Abl inhibitor. Developed by 1st Biotherapeutics, it is being investigated for the treatment of neurological disorders, such as Parkinson's Disease and amyotrophic lateral sclerosis (ALS).[L47102]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FB-825 DB17598
biotech

FB-825 is an investigational humanized monoclonal antibody that targets the C?mX domain of the membrane-bound IgE (mIgE), causing a depletion of mIgE positive B-cells. It is currently being investigated for immune disorders, such as atopic dermatitis and hype…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
fb-PMT DB17394
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FDL169 DB16878
small molecule | CAS: 1628416-28-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Febuxostat Approved DB04854
small molecule | CAS: 144060-53-7

Febuxostat is a non-purine xanthine oxidase (XO) inhibitor.[A39743] In early 2008, febuxostat was granted marketing authorization by the European Commission for the treatment of chronic hyperuricemia and gout.[A230548] In the following year, the FDA for appro…

Kategori:
Antigout PreparationsAntirheumatic AgentsBCRP/ABCG2 Inhibitors +15
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu ParuhThe apparent mean t…
Vol. DistribusiThe apparent steady…
KlirensFollowing oral admi…
Genetik -
Fecal microbiota Approved DB17743
biotech

Fecal microbiota, given either as a rectal transplant or in an oral formulation of live spores, is an FDA-approved option to prevent the recurrence of _Clostridioides difficile_ infection (CDI) in patients given an antibacterial treatment for recurrent CDI.[A…

Kategori:
Miscellaneous Therapeutic Agents
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Fedovapagon DB11734
small molecule | CAS: 347887-36-9

Fedovapagon has been used in trials studying the treatment of Nocturia.

Target Protein:
Vasopressin V2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fedratinib Approved DB12500
small molecule | CAS: 936091-26-8

Fedratinib, also known as SAR302503 and TG101348, is a tyrosine kinase inhibitor used to treat intermediate-2 and high risk primary and secondary myelofibrosis.[A183176,L8090] It is an anilinopyrimidine derivative.[A183188] Fedratinib was granted FDA appro…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
Tyrosine-protein kinase JAK2Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase JAK1
Waktu ParuhThe half life of fe…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of fe…
Genetik -
Fedrilate DB13825
small molecule | CAS: 23271-74-1

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felbinac DB07477
small molecule | CAS: 5728-52-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +12
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Procathepsin L
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felcisetrag DB12725
small molecule | CAS: 916075-84-8

Felcisetrag (TD-8954) has been used in trials studying the treatment of Enteral Feeding Intolerance and Gastrointestinal Motility Disorder.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felodipine Approved DB01023
small molecule | CAS: 72509-76-3

Felodipine is a long-acting 1,4-dihydropyridine calcium channel blocker (CCB)b. It acts primarily on vascular smooth muscle cells by stabilizing voltage-gated L-type calcium channels in their inactive conformation. By inhibiting the influx of calcium in smoot…

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents causing hyperkalemiaAntiarrhythmic agents +31
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +10
Waktu Paruh17.5-31.5 hours in …
Vol. Distribusi* 10 L/kg
Klirens* 0.8 L/min [Young …
Genetik -
Felypressin DB00093
biotech | CAS: 56-59-7

A synthetic nonapeptide comprising cysteinyl, phenylalanyl, phenylalanyl, glutaminyl, asparaginyl, cysteinyl, prolyl, lysyl, and glycinamide residues in sequence, with a disulfide bridge joining the two cysteine residues. Its antidiuretic effects are less tha…

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsHormones +12
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felzartamab DB16375
biotech | CAS: 2197112-39-1

Felzartamab is under investigation in clinical trial NCT04145440 (Trial to Assess Safety and Efficacy of MOR202 in Anti-pla2r + Membranous Nephropathy (Amn)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenamole DB12506
small molecule | CAS: 5467-78-7

Fenamole has been investigated for the supportive care of Side Effects and Dental Plaque.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenbendazole DB11410
small molecule | CAS: 43210-67-9

Fenbendazole is a benzimidazole that presents a wide spectrum anthelmintic effect. It is used against a number of gastrointestinal parasites including giardia, roundworms, hookworms, whipworms, the Taenia genus of tapeworms, pinworms, aelurostrongylus, parago…

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenchone DB15918
small molecule | CAS: 1195-79-5

Deskripsi belum tersedia.

Kategori:
Bicyclic MonoterpenesBridged-Ring CompoundsMonoterpenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fendiline DB08980
small molecule | CAS: 13042-18-7

Fendiline is a coronary vasodilator which inhibits calcium function in muscle cells in excitation-contraction coupling. It has been proposed as an antiarrhythmic and antianginal agent. Fendiline is non-selective.

Kategori:
Agents causing hyperkalemiaAminesAntiarrhythmic agents +15
Target Protein:
5-hydroxytryptamine receptor 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenebrutinib DB14785
small molecule | CAS: 1434048-34-6

Fenebrutinib is under investigation in clinical trial NCT03174041 (A Drug-Drug Interaction Study Between GDC-0853 and Midazolam, Itraconazole, Rosuvastatin, and Simvastatin).

Kategori:
Pyridines
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenethylline DB01482
small molecule | CAS: 3736-08-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAminesCentral Nervous System Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenfluramine Approved DB00574
small molecule | CAS: 458-24-2

Dravet syndrome is a pediatric encephalopathy that typically manifests within the first year of life following exposure to elevated temperatures. It is characterized by recurrent pharmacoresistant seizures, which increase in frequency and severity with diseas…

Kategori:
Alimentary Tract and MetabolismAminesAnticonvulsants +27
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 2C +4
Waktu ParuhFenfluramine has an…
Vol. DistribusiFenfluramine has an…
KlirensFenfluramine has a …
Genetik -
Fenobam DB12931
small molecule | CAS: 57653-26-6

Fenobam is under investigation in clinical trial NCT00637221 (Open Label Study Investigating Safety and Efficacy of Fenobam anhydrous 50 mg - 150 mg on Prepulse Inhibition Tests and Continuous Performance Tasks, Adults With Fragile X Syndrome).

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenofibric acid Approved DB13873
small molecule | CAS: 42017-89-0

Fenofibric acid is a lipid-lowering agent that is used in severe hypertriglyceridemia, primary hyperlipidemia, and mixed dyslipidemia. It works to decrease elevated low-density lipoprotein cholesterol, total cholesterol, triglycerides, apolipoprotein B, while…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAnticholesteremic Agents +17
Target Protein:
Peroxisome proliferator-activated receptor alphaFatty acid-binding protein, liverMatrix metalloproteinase-25 +3
Waktu ParuhFollowing once dail…
Vol. DistribusiThe volume of distr…
KlirensIn five elderly vol…
Genetik -
Fenoldopam Approved DB00800
small molecule | CAS: 67227-56-9

A dopamine D1 receptor agonist that is used as an antihypertensive agent. It lowers blood pressure through arteriolar vasodilation.

Kategori:
Adrenergic and Dopaminergic AgentsAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +12
Target Protein:
D(1B) dopamine receptorD(1A) dopamine receptorAlpha-1B adrenergic receptor +5
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Fenoprofen Approved DB00573
small molecule | CAS: 29679-58-1

An anti-inflammatory analgesic and antipyretic highly bound to plasma proteins. It is pharmacologically similar to aspirin, but causes less gastrointestinal bleeding.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor alpha +1
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Fenoverine DB13042
small molecule | CAS: 37561-27-6

Fenoverine has been used in trials studying the treatment of Irritable Bowel Syndrome.

Kategori:
Alimentary Tract and MetabolismAutonomic AgentsDrugs for Functional Gastrointestinal Disorders +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenoxazoline DB13736
small molecule | CAS: 4846-91-7

Deskripsi belum tersedia.

Kategori:
Nasal PreparationsSympathomimetics, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenpiverinium DB13759
small molecule | CAS: 258329-46-3

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenpropidin Approved DB12728
small molecule | CAS: 67306-00-7

Fenpropidin has been investigated for the treatment of Hernia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingFungicides, Industrial +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenproporex DB01550
small molecule | CAS: 16397-28-7

Fenproporex is an orally active stimulant drug, which was developed in the 1960s. It is used as an appetite suppressant and a treatment for obesity. It is listed as an illicit substance in many countries due to addiction issues and listed as a prohibited subs…

Kategori:
AminesDrugs that are Mainly Renally ExcretedEthylamines +2
Waktu Paruh-
Vol. Distribusi-
KlirensThe amphetamine met…
Genetik -
Fenquizone DB13708
small molecule | CAS: 20287-37-0

Deskripsi belum tersedia.

Kategori:
DiureticsHeterocyclic Compounds, Fused-RingLow-Ceiling Diuretics, Excl. Thiazides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenretinide DB05076
small molecule | CAS: 65646-68-6

A synthetic retinoid that is used orally as a chemopreventive against prostate cancer and in women at risk of developing contralateral breast cancer. It is also effective as an antineoplastic agent.

Kategori:
AlkenesAnticarcinogenic AgentsAntineoplastic Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenspiride DB08979
small molecule | CAS: 5053-06-5

Fenspiride is an oxazolidinone spiro compound used as a drug in the treatment of certain respiratory diseases. It is approved for use in Russia for the treatment of acute and chronic inflammatory diseases of ENT organs and the respiratory tract (like rhinopha…

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fentanyl Approved DB00813
small molecule | CAS: 437-38-7

Fentanyl, a potent opioid agonist, was developed in the 1950s to fill a need for strong and rapid analgesia.[A179542] Because of these characteristics, fentanyl is commonly used to treat chronic cancer pain or in anesthesia.[Label,L6598,L6601,L6604,L6607,L922…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents that produce hypertension +32
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +1
Waktu ParuhThe half life of fe…
Vol. DistribusiThe intravenous vol…
KlirensTotal plasma cleara…
Genetik -
Fentiazac DB13217
small molecule | CAS: 18046-21-4

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAcids, AcyclicAgents causing hyperkalemia +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenticonazole DB13434
small molecule | CAS: 72479-26-6

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fentonium DB08978
small molecule | CAS: 34786-74-8

Fentonium is an atropine derivative.

Kategori:
Alimentary Tract and MetabolismAlkaloidsAza Compounds +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenvalerate DB18391
small molecule | CAS: 51630-58-1

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingCyclopentane Monoterpenes +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fepixnebart DB19079
biotech | CAS: 1799706-87-8

Fepixnebart is under investigation in clinical trial NCT04456686 (Chronic Pain Master Protocol (CPMP): A Study of LY3016859 in Participants With Osteoarthritis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Feprazone DB13364
small molecule | CAS: 30748-29-9

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferric ammonium citrate Approved DB09501
small molecule | CAS: 1185-57-5

Deskripsi belum tersedia.

Kategori:
AminesAmmonium CompoundsContrast Media +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferric carboxymaltose Approved DB08917
small molecule | CAS: 9007-72-1

Ferric carboxymaltose is an iron replacement product and, chemically, an iron-carbohydrate complex. It was FDA approved on July 25, 2013.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDisaccharides +5
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe estimated volum…
Klirens-
Genetik -
Ferric cation Approved DB13949
small molecule | CAS: 20074-52-6

Iron is a transition metal with a symbol Fe and atomic number 26. By mass, it is the most common element on Earth. Iron is an essential element involved in various metabolic processes, including oxygen transport, deoxyribonucleic acid (DNA) synthesis, and ene…

Kategori:
Iron CompoundsParenteral Iron ReplacementPhosphate Binder +2
Target Protein:
Transferrin receptor protein 1Iron(3+)-hydroxamate-binding protein FhuD
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiLess than 65% of ir…
KlirensThe rate of iron lo…
Genetik -
Ferric chloride Approved DB15536
small molecule | CAS: 7705-08-0

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAnions +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferric derisomaltose Approved DB15617
small molecule | CAS: 1345510-43-1

Iron deficiency is an extremely common condition and is the most frequent cause of anemia worldwide. Iron deficiency results when iron intake, iron stores, and loss of iron from the body do not adequately support production of erythrocytes, also known as red …

Kategori:
Anemia, Iron-DeficiencyAntianemia DrugsAntianemic Preparations +6
Target Protein:
Hemoglobin subunit alphaTransferrin receptor
Waktu ParuhThe plasma-half liv…
Vol. DistribusiFerric derisomaltos…
KlirensIntravenous iron is…
Genetik -
Ferric glycerophosphate Approved DB15934
small molecule | CAS: 1301-70-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1309-33-7

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansIron Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 5051–5100 dari 11778
Sebelumnya Halaman 102 / 236 Berikutnya