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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 101 / 236
Excindogen DB18754
small molecule

Excindogen is an investigational immunotherapy.

Waktu Paruh-
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Exemestane Approved DB00990
small molecule | CAS: 107868-30-4

Exemestane is an oral steroidal aromatase inhibitor used in the adjuvant treatment of hormonally-responsive (also called hormone-receptor-positive, estrogen-responsive) breast cancer in postmenopausal women. It irreversibly binds to the active site of the enz…

Kategori:
AndrostanesAndrostenesAntineoplastic Agents +14
Target Protein:
Aromatase
Waktu Paruh24 hours
Vol. Distribusi-
Klirens-
Genetik -
Exenatide Approved DB01276
biotech | CAS: 141758-74-9

Exenatide is a glucagon-like peptide-1 (GLP-1) analog[L42690]. It activates the GLP-1 receptor and increases insulin secretion, decreases glucagon secretion, and slows gastric emptying to improve glycemic control[L42690]. Exenatide was given FDA approval on A…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnti-Obesity Agents +16
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh2.4 hours[Label]
Vol. Distribusi28.3L[Label].
Klirens9.1 L/hour[Label].
Genetik -
Exicorilant DB16162
small molecule | CAS: 1781244-77-6

Exicorilant is under investigation in clinical trial NCT03437941 (Study to Evaluate CORT125281 in Combination With Enzalutamide in Patients With Mcrpc).

Target Protein:
Glucocorticoid receptor
Waktu Paruh-
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Exidavnemab DB19452
biotech | CAS: 2438229-02-6

Exidavnemab is under investigation in clinical trial NCT06671938 (Safety, Tolerability, and Pharmacokinetics of Exidavnemab in Patients With Parkinson's Disease).

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Exisulind DB06246
small molecule | CAS: 59973-80-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +10
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseGlutathione S-transferase PAldo-keto reductase family 1 member B1 +4
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Exlinkibart DB17474
biotech | CAS: 2642171-64-8

Deskripsi belum tersedia.

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EXOB-001 DB18257
biotech

EXOB-001 consists of extracellular vesicles derived from cultured human umbilical cord mesenchymal stromal cells.

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biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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EXT608 DB18453
biotech

EXT608 is a long-acting PTH derivative under investigation for the treatment of hyperparathyroidism.[L48270]

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Ezabenlimab DB17483
biotech | CAS: 2249882-54-8

Deskripsi belum tersedia.

Waktu Paruh-
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biotech | CAS: 2226647-27-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Ezetimibe Approved DB00973
small molecule | CAS: 163222-33-1

Ezetimibe is a lipid-lowering compound that inhibits intestinal cholesterol and phytosterol absorption. The discovery and research of this drug began in the early 1990s, after the intravenous administration of radiolabelled ezetimibe in rats revealed that it …

Kategori:
Anticholesteremic AgentsAzetinesBCRP/ABCG2 Substrates +20
Target Protein:
NPC1-like intracellular cholesterol transporter 1Sterol O-acyltransferase 1Aminopeptidase N
Waktu ParuhBoth ezetimibe and …
Vol. DistribusiThe relative volume…
KlirensThere are no pharma…
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Ezogabine Approved DB04953
small molecule | CAS: 150812-12-7

Ezogabine (D23129) is a close structural analog of the centrally acting analgesic flupitrine. It is a neuronal potassium channel opener being developed as a first-in-class antiepileptic drug (AED) and is currently being studied in Phase 3 trials as an adjunct…

Kategori:
Acids, AcyclicAminesAniline Compounds +15
Target Protein:
Potassium voltage-gated channel subfamily KQT member 3Potassium voltage-gated channel subfamily KQT member 2Potassium voltage-gated channel subfamily KQT member 4 +1
Waktu ParuhTerminal half-life …
Vol. Distribusi8.7 L/kg
Klirens0.58 - 0.76 L/h·kg.…
Genetik -
Ezurpimtrostat DB16458
small molecule | CAS: 1914148-72-3

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
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Ezutromid DB12888
small molecule | CAS: 945531-77-1

Ezutromid has been investigated for the treatment of Muscular Dystrophy, Duchenne.

Kategori:
Heterocyclic Compounds, Fused-RingMuscular Dystrophy, Duchenne
Target Protein:
Utrophin
Waktu Paruh-
Vol. Distribusi-
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small molecule | CAS: 78-96-6

Deskripsi belum tersedia.

Target Protein:
Glutamate mutase sigma subunit
Waktu Paruh-
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F6-734 DB17444
biotech

F6-734 is a bispecific monoclonal antibody with affinity for anticarcinoembryonic antigen (CEA) and anti-diethylenetriamine pentaacetic acid (DTPA) (hMN-14 × m734).[A255217,A255222]

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Fabomotizole DB13623
small molecule | CAS: 173352-21-1

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsNervous System +1
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Facinicline DB05586
small molecule | CAS: 677306-35-3

Deskripsi belum tersedia.

Kategori:
Bridged-Ring CompoundsHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
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Factor IX Complex (Human) Approved DB11330
biotech | CAS: 37224-63-8

Factor IX Complex is a sterile, lyophilized concentrate composed of a number of Vitamin K-dependent clotting factors found in functioning human plasma. Also known as prothrombin complex concentrate, products containing this complex often include Factor IX (an…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
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Fadrozole DB16832
small molecule | CAS: 102676-47-1

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, HormonalAromatase Inhibitors +7
Target Protein:
AromataseCytochrome P450 11B1, mitochondrial
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Fagrocorat DB14676
small molecule | CAS: 1044535-52-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
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Falimarev DB17333
biotech | CAS: 685563-14-8

Deskripsi belum tersedia.

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Fallypride DB15167
small molecule | CAS: 166173-78-0

Fallypride is under investigation in clinical trial NCT02310360 (Striatal and Extra-striatal Dopamine Release in Response to Food in Healthy Humans).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +5
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Fallypride F-18 DB19254
small molecule | CAS: 166173-82-6

Fallypride F-18 is under investigation in clinical trial NCT00846040 (Reduced Carbohydrate Versus Fat in Obese Subjects).

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Famciclovir Approved DB00426
small molecule | CAS: 104227-87-4

Famciclovir, marketed as Famvir by Novartis, is a guanine analogue used to treat herpes virus infections. It is most commonly used to treat herpes zoster (shingles). Famciclovir is a prodrug of penciclovir with higher oral bioavailability.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh10 hours
Vol. Distribusi* 1.08±0.17 L/kg [h…
Klirens* 36.6 +/- 6.3 L/hr…
Genetik -
Famitinib DB11741
small molecule | CAS: 1044040-56-3

Famitinib has been used in trials studying the treatment of Colorectal Cancer, Renal Cell Cancer, Colorectal Cancer Recurrent, Colorectal Cancer Metastatic, and Metastatic Renal Cell Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-RingReceptor Protein-Tyrosine Kinases, antagonists & inhibitors
Target Protein:
Platelet-derived growth factor receptor alphaReceptor-type tyrosine-protein kinase FLT3Mast/stem cell growth factor receptor Kit +4
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Famotidine Approved DB00927
small molecule | CAS: 76824-35-6

Famotidine is a competitive histamine-2 (H<sub>2</sub>) receptor antagonist that works to inhibit gastric acid secretion. It is commonly used in gastrointestinal conditions related to acid secretion, such as gastric ulcers and gastroesophageal reflux disease …

Kategori:
Acid ReducersAlimentary Tract and MetabolismAnti-Ulcer Agents +20
Target Protein:
Histamine H2 receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensRenal clearance is …
Genetik -
Famphur DB11408
small molecule | CAS: 52-85-7

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +8
Waktu Paruh-
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Famprofazone DB16702
small molecule | CAS: 22881-35-2

Famprofazone is a nonsteroidal anti-inflammatory agent found in combination products such as ‘Gewodin’ which is marketed in Taiwan.[L34724] It is important to note that the drug is metabolized to [methamphetamine] and [amphetamine] in the body and can lead to…

Kategori:
AminesAmphetaminesAnalgesics +7
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Famtozinameran Approved DB17088
biotech

The Omicron variant of SARS-CoV-2 is a variant of concern that was first reported in November 2021.[L43922] It tends to cause less severe disease but is significantly more virulent than both the original virus and earlier variants (e.g. Delta).[L43917] As of …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +12
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Fanapanel DB12393
small molecule | CAS: 161605-73-8

Fanapanel has been investigated for the treatment of Visual Acuity.

Kategori:
Heterocyclic Compounds, Fused-RingOrganophosphorus Compounds
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FAPi-46 GA-68 DB18827
small molecule | CAS: 2374784-98-0

Deskripsi belum tersedia.

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Farampator DB15012
small molecule | CAS: 211735-76-1

Farampator is under investigation in clinical trial NCT00113022 (Org 24448 to Treat Major Depression).

Kategori:
Oxazoles
Target Protein:
Glutamate receptor 1
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Farglitazar DB19311
small molecule | CAS: 274687-78-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
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Faricimab Approved DB15303
biotech | CAS: 1607793-29-2

Retinal vascular diseases (RVDs) such as diabetic macular edema (DME), age-related macular degeneration (AMD), and retinal vein occlusion (RVO) are typically caused by retinal ischemia and subsequent neovascularization (NV).[A225985, A225990, A225995] Vascula…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Target Protein:
Vascular endothelial growth factor A, long formAngiopoietin-2
Waktu ParuhFaricimab has an es…
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Farletuzumab DB05595
biotech | CAS: 896723-44-7

Farletuzumab (MORAb-003) is a fully humanized monoclonal antibody against the folate receptor alpha, for the potential treatment of epithelial ovarian cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Folate receptor alpha
Waktu Paruh-
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biotech | CAS: 2407465-18-1

Farletuzumab ecteribulin is under investigation in clinical trial NCT04300556 (A Study to Evaluate the Safety, Tolerability, and Efficacy of Morab-202 (Herein Referred to as Farletuzumab Ecteribulin), a Folate Receptor Alpha (Fr?)-targeting Antibody-drug Conj…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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small molecule | CAS: 13058-04-3

Deskripsi belum tersedia.

Kategori:
OrganophosphatesOrganophosphorus CompoundsPotential QTc-Prolonging Agents +2
Target Protein:
Squalene synthaseProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaProtein farnesyltransferase subunit beta +9
Waktu Paruh-
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small molecule | CAS: 141702-36-5

Faropenem medoxomil is an ester prodrug derivative of the beta-lactam antibiotic [faropenem]. The prodrug form of faropenem offers dramatically improved oral bioavailability and leads to higher systemic concentrations of the drug. Faropenem medoxomil is a bro…

Kategori:
AmidesHeterocyclic Compounds, Fused-RingLactams +1
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 2BPeptidoglycan D,D-transpeptidase FtsI
Waktu Paruh-
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Fasentin DB16759
small molecule | CAS: 392721-37-8

Deskripsi belum tersedia.

Kategori:
AmidesAminesAniline Compounds
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Fasiglifam DB12491
small molecule | CAS: 1000413-72-8

Fasiglifam has been used in trials studying the treatment of Chronic Kidney Disease, Type 2 Diabetes Mellitus, and Diabetes Mellitus, Type 2.

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Free fatty acid receptor 1
Waktu Paruh-
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Fasinumab DB12157
biotech | CAS: 1190239-42-9

Fasinumab is a human IgG1k monoclonal antibody targeted against nerve growth factor (NGF). It is currently under investigation for the treatment osteoarthritic pain[A241045] and has demonstrated significantly greater pain relief and functional improvement as …

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Beta-nerve growth factor
Waktu Paruh-
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Fasudil DB08162
small molecule | CAS: 103745-39-7

Fasudil has been investigated in Carotid Stenosis.

Kategori:
Antiarrhythmic agentsCalcium Channel BlockersCalcium-Regulating Hormones and Agents +12
Target Protein:
Rho-associated protein kinase 1cAMP-dependent protein kinase inhibitor alphacAMP-dependent protein kinase catalytic subunit alpha +1
Waktu Paruh-
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Favezelimab DB16729
biotech | CAS: 2231068-83-8

Favezelimab is under investigation in clinical trial NCT04626479 (Substudy 03A: A Study of Immune and Targeted Combination Therapies in Participants With First Line (1L) Renal Cell Carcinoma (MK-3475-03A)).

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Favipiravir Approved DB12466
small molecule | CAS: 259793-96-9

Discovered by Toyama Chemical Co., Ltd. in Japan, favipiravir is a modified pyrazine analog that was initially approved for therapeutic use in resistant cases of influenza.[A191688,A191721] The antiviral targets RNA-dependent RNA polymerase (RdRp) enzymes, wh…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +11
Target Protein:
DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase subunit beta'RNA-directed RNA polymerase catalytic subunit
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe recommended ora…
Genetik -
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