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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 101 / 272
Denecimig DB18426
biotech | CAS: 2488745-86-2

Delpacibart is a humanized, bispecific, bivalent monoclonal antibody against coagulation factor 9.

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Denenicokin DB12908
biotech | CAS: 716840-32-3

Denenicokin is under investigation in clinical trial NCT01152788 (Phase II Study of Interleukin-21 (rIL-21) vs Dacarbazine (DTIC) in Patients With Metastatic or Recurrent Melanoma).

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Denfivontinib DB17159
small molecule | CAS: 1457983-28-6

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein kinase MerReceptor-type tyrosine-protein kinase FLT3
Waktu Paruh-
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Denibulin DB05932
small molecule | CAS: 284019-34-7

Denibulin is a novel small molecule Vascular Disrupting Agent under development by MediciNova for treatment of solid tumor cancers.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Vascular endothelial growth factor A, long formVascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 3
Waktu Paruh-
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Denifanstat DB17576
small molecule | CAS: 1399177-37-7

Denifanstat is an orally bioavailable fatty acid synthase (FASN) inhibitor. Due to its antineoplastic activities, it is being investigated for various cancers.

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Denileukin diftitox Approved DB00004
biotech | CAS: 173146-27-5

Denileukin diftitox is an IL2-receptor-directed cytotoxin, is a recombinant DNA-derived fusion protein composed of the amino acid sequences for diphtheria toxin fragments A and B (Met<sub>1</sub>-Thr<sub>387</sub>)-His and the sequence for human interleukin-2…

Kategori:
ADP Ribose TransferasesAmino Acids, Peptides, and ProteinsAntineoplastic Agents +15
Target Protein:
Interleukin-2 receptor subunit alphaInterleukin-2 receptor subunit beta
Waktu ParuhThe arithmetic mean…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Denosumab Approved DB06643
biotech | CAS: 615258-40-7

Denosumab is a novel, fully human IgG2 monoclonal antibody specific to receptor activator of nuclear factor kappa-B ligand (RANKL), suppresses bone resorption via inhibiting RANK-mediated activation of osteoclasts. It is the first and currently the only RANKL…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Tumor necrosis factor ligand superfamily member 11
Waktu ParuhAfter C<sub>max</su…
Vol. DistribusiThe central volume …
KlirensNo information is a…
Genetik -
biotech

Dental pulp is a soft, connective tissue present in the dental crown of both third molar and first premolar teeth. Dental pulp stem cells (DPSCs) exhibit fibro-blast like plasticity and adherent properties. They are harvested through surgical extraction of wi…

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Denufosol DB04983
small molecule | CAS: 211448-85-0

Denufosol was an inhaled drug used for the treatment of cystic fibrosis (CF), showing various improvements in lung function during a phase III clinical trial. A new drug application (NDA) was filed with the FDA in 2011, however, the second phase III clinical…

Kategori:
Cytosine NucleotidesDeoxyribonucleotidesNucleic Acids, Nucleotides, and Nucleosides +6
Target Protein:
P2Y purinoceptor 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Endoglucanase 5A
Waktu Paruh-
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Deoxycholic acid Approved DB03619
small molecule | CAS: 83-44-3

Deoxycholic acid is a a bile acid which emulsifies and solubilizes dietary fats in the intestine, and when injected subcutaneously, it disrupts cell membranes in adipocytes and destroys fat cells in that tissue. In April 2015, deoxycholic acid was approved by…

Kategori:
Bile Acids and SaltsBSEP/ABCB11 inducersCholagogues and Choleretics +9
Target Protein:
Proliferating cell nuclear antigenSteroid Delta-isomeraseCytochrome C +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 52474-59-6

Deskripsi belum tersedia.

Kategori:
Cytosine NucleotidesDeoxyribonucleotidesHeterocyclic Compounds, Fused-Ring +8
Target Protein:
Ribonuclease pancreatic
Waktu Paruh-
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Genetik -
small molecule | CAS: 501-15-5

Sympathomimetic, vasoconstrictor agent.

Kategori:
Agents that produce hypertensionAminesBenzene Derivatives +4
Waktu Paruh-
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Deoxyinosine DB02380
small molecule | CAS: 890-38-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Waktu Paruh-
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Genetik -
biotech

Deoxyribonuclease I (DNase I) is a human enzyme responsible for the digestion of extracellular DNA7[A227723]. It is normally found in saliva, urine, pancreatic secretions, and blood[A227723]. Because of the hypothesis that increased concentrations of high-mol…

Kategori:
Deoxyribonuclease I, antagonists & inhibitorsDeoxyribonucleasesEndodeoxyribonucleases +4
Waktu Paruh-
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Genetik -
small molecule | CAS: 964-26-1

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleotidesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Target Protein:
Thymidylate synthaseDeoxyuridine 5'-triphosphate nucleotidohydrolaseThymidylate synthase +6
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Deoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrialDeoxyuridine 5'-triphosphate nucleotidohydrolaseDeoxyuridine 5'-triphosphate nucleotidohydrolase +2
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Septum formation protein MafPol polyproteinDeoxycytidine triphosphate deaminase +2
Waktu Paruh-
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biotech | CAS: 1585973-65-4

Depatuxizumab/Denintuzumab mafodotin has been used in trials studying the treatment of Lymphoma, Gliosarcoma, Glioblastoma, Malignant Glioma, Squamous Cell Tumors, and Glioblastoma Multiforme.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Tubulin beta chainEpidermal growth factor receptorB-lymphocyte antigen CD19
Waktu Paruh-
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Depelestat DB17873
biotech | CAS: 506433-25-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsLeukocyte Elastase, antagonists & inhibitors
Target Protein:
Neutrophil elastase
Waktu Paruh-
Vol. Distribusi-
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Depemokimab DB18846
biotech | CAS: 2243274-14-6

Depemokimab is under investigation in clinical trial NCT05274750 (Efficacy and Safety of Depemokimab (GSK3511294) in Participants With Chronic Rhinosinusitis With Nasal Polyps).

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Phosphopantetheine adenylyltransferase
Waktu Paruh-
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Depreotide DB11628
small molecule | CAS: 161982-62-3

Depreotide is an ingredient in the EMA-withdrawn product NeoSpect.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Deptropine DB13466
small molecule | CAS: 604-51-3

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntihistamines for Systemic UseAza Compounds +5
Waktu Paruh-
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Depulfavirine DB18890
small molecule | CAS: 867365-76-2

Depulfavirine is under investigation in clinical trial NCT05204394 (Study to Evaluate Efficacy and Safety of Switching to VM-1500A-LAI + 2nrtis From the 1st Line Standard of Care Therapy).

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Deracoxib DB11395
small molecule | CAS: 169590-41-4

Deracoxib is a non-steroidal anti-inflammatory drug of the coxib class, used in veterinary medicine to treat osteoarthritis in dogs. It is sold in tablets, which have added beefy flavour to increase palatability. Deramaxx received FDA approval in August 2002 …

Kategori:
AmidesAnalgesicsAnalgesics, Non-Narcotic +11
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Deramciclane DB06512
small molecule | CAS: 120444-71-5

Deramciclane (EGIS-3886) is used for the treatment of a number of anxiety disorders. Deramciclane differs from other anti anxiety medications in that it is not a benzodiazepine and so has a different structure and target. It antagonizes 5-HT2A receptors, agon…

Kategori:
Anti-Anxiety AgentsAnticonvulsantsAntidepressive Agents +17
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C
Waktu Paruh-
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Derazantinib DB14889
small molecule | CAS: 1234356-69-4

Derazantinib is under investigation in clinical trial NCT03230318 (Derazantinib in Subjects With FGFR2 Gene Fusion Positive Inoperable or Advanced Intrahepatic Cholangiocarcinoma).

Kategori:
AminesHeterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 1
Waktu Paruh-
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Derenofylline DB12446
small molecule | CAS: 251945-92-3

Derenofylline has been used in trials studying the treatment of Congestive Heart Failure and Acute Decompensated Heart Failure; Renal Dysfunction.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
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Dersalazine DB06251
small molecule | CAS: 188913-58-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +5
Target Protein:
Platelet-activating factor receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Dersimelagon DB18007
small molecule | CAS: 1835256-48-8

Deskripsi belum tersedia.

Target Protein:
Melanocyte-stimulating hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 130525-62-1

Deskripsi belum tersedia.

Target Protein:
Neuraminidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desaspidin DB13567
small molecule | CAS: 114-43-2

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnticestodalsAntiparasitic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Descartes-30 DB16361
biotech

Descartes-30 is an RNA-engineered off-the-shelf allogeneic mesenchymal stem cell (MSC) product developed by Cartesian Therapeutics.[L27531] The RNA-engineering is performed with Cartesian Therapeutics’ proprietary RNA Armory which is a platform that activates…

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Deserpidine Approved DB01089
small molecule | CAS: 131-01-1

Deserpidine is an ester alkaloid drug isolated from Rauwolfia canescens (family Apocynaceae) with antipsychotic and antihypertensive properties that has been used for the control of high blood pressure and for the relief of psychotic behavior.

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +8
Target Protein:
Synaptic vesicular amine transporterAngiotensin-converting enzyme
Waktu Paruh-
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Desflurane Approved DB01189
small molecule | CAS: 57041-67-5

Desflurane, or I-653, a a volatile anesthetic that is more rapidly cleared and less metabolized than previous inhaled anesthetics such as [methoxyflurane], [sevoflurane], [enflurane], or [isoflurane].[A226390,A39015,A226893]. It was developed in the late 1980…

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +14
Target Protein:
GABA(A) ReceptorGlycine receptor subunit alpha-1Glutamate receptor 1 +4
Waktu ParuhDesflurane has a te…
Vol. DistribusiDesflurane has a me…
KlirensA 26 g dose of desf…
Genetik -
Desidustat DB16135
small molecule | CAS: 1616690-16-4

Desidustat is under investigation in clinical trial NCT04012957 (Desidustat in the Treatment of Anemia in CKD).

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
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Desipramine Approved DB01151
small molecule | CAS: 50-47-5

Desipramine hydrochloride is a dibenzazepine-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individuals, de…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +52
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +14
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +4
Waktu Paruh7-60+ hours; 70% el…
Vol. Distribusi-
Klirens-
Genetik 7 Varian
Desirudin Approved DB11095
biotech | CAS: 120993-53-5

Desirudin is a direct inhibitor of human thrombin. It has a protein structure that is similar to that of hirudin, the naturally occurring anticoagulant present in the peripharyngeal glands in the medicinal leech, Hirudo medicinalis. Hirudin is a single polype…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Waktu Paruh~2 hours.
Vol. Distribusi0.25 L/kg.
Klirens1.5 to 2.7 mL/min/k…
Genetik -
Deslanoside Approved DB01078
small molecule | CAS: 17598-65-1

Deacetyllanatoside C. A cardiotonic glycoside from the leaves of Digitalis lanata.

Kategori:
Antiarrhythmic agentsCarbohydratesCardanolides +13
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh36 hours
Vol. Distribusi-
Klirens-
Genetik -
Desloratadine Approved DB00967
small molecule | CAS: 100643-71-8

Desloratadine is a second generation, tricyclic antihistamine that which has a selective and peripheral H1-antagonist action. It is the active descarboethoxy metabolite of loratidine (a second generation histamine). Desloratidine has a long-lasting effect and…

Kategori:
Anticholinergic AgentsAntihistamines for Systemic UseBenzocycloheptenes +13
Target Protein:
Histamine H1 receptor
Waktu ParuhDesloratadine has a…
Vol. Distribusi-
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Deslorelin DB11510
small molecule | CAS: 57773-65-6

Deslorelin acetate is an injectable gonadotropin releasing hormone super-agonist also known as an LHRH agonist. It stops the production of sex hormones.

Kategori:
Adrenal Cortex HormonesAlcohol Dehydrogenase, antagonists & inhibitorsAmino Acids, Peptides, and Proteins +12
Waktu Paruh-
Vol. Distribusi-
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Desmeninol DB15832
small molecule | CAS: 583-91-5

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13147-09-6

Desmethylprodine, a derivative of meperidine, is an opioid analgesic with the potency of morphine. It has been listed as a Schedule I controlled drug in the United States, and thus is not used clinically. It is known to be a designer drug, synthesized in 1977…

Kategori:
Isonipecotic AcidsPiperidines
Waktu Paruh-
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Genetik -
Desmopressin Approved DB00035
small molecule | CAS: 16679-58-6

Desmopressin (dDAVP), a synthetic analogue of 8-arginine vasopressin (ADH), is an antidiuretic peptide drug modified by deamination of 1-cysteine and substitution of 8-L-arginine by 8-D-arginine. ADH is an endogenous pituitary hormone that has a crucial role …

Kategori:
Agents that produce hypertensionAmino Acids, Peptides, and ProteinsAntidiuretic Agents +27
Target Protein:
Oxytocin receptorVasopressin V2 receptorVasopressin V1a receptor +1
Waktu ParuhFollowing an intran…
Vol. DistribusiThe distribution vo…
Klirens-
Genetik -
Desmoteplase DB04925
biotech | CAS: 145137-38-8

Desmoteplase is a chemical in the saliva of vampire bats. It activates plasminogen to the serine protease, plasmin. Plasmin acts by breaking down fibrin blood clots. When a vampire bat bites its victim, it secretes an enzyme that prevents the blood from clott…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBlood Proteins +13
Target Protein:
Plasminogen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desogestrel Approved DB00304
small molecule | CAS: 54024-22-5

Desogestrel, a prodrug, is a third generation progestogen[A176315] and hence, a member of the gonane family which was largely used in Europe before being approved in the US and Canada.[A176339] It was firstly generated from a study that showed that 11-beta an…

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +25
Target Protein:
Progesterone receptorEstrogen receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe apparent volume…
KlirensThe metabolic clear…
Genetik -
Desomorphine DB01531
small molecule | CAS: 427-00-9

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desonide Approved DB01260
small molecule | CAS: 638-94-8

A nonfluorinated corticosteroid anti-inflammatory agent used topically for dermatoses.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +18
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 94087-98-6

Deskripsi belum tersedia.

Waktu Paruh-
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Menampilkan 5001–5050 dari 13591
Sebelumnya Halaman 101 / 272 Berikutnya