Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 100 / 236
Etiracetam DB11868
small molecule | CAS: 33996-58-6

Etiracetam is under investigation in clinical trial NCT01137110 (Comparison of Short Duration Levetiracetam to Extended Course for Seizure Prophylaxis After Subarachnoid Hemorrhage (SAH)).

Kategori:
AcetamidesAcetatesAcids, Acyclic +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 848779-32-8

Etirinotecan pegol is under investigation in clinical trial NCT01663012 (Phase II NKTR-102 In Bevacizumab-Resistant High Grade Glioma).

Kategori:
AlcoholsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etodolac Approved DB00749
small molecule | CAS: 41340-25-4

Etodolac is a non-steroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic and antipyretic properties. Its therapeutic effects are due to its ability to inhibit prostaglandin synthesis. It is indicated for relief of signs and symptoms of rhe…

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +29
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Retinoic acid receptor RXR-alpha
Waktu ParuhTerminal t<sub>1/2<…
Vol. Distribusi* 390 mL/kg
Klirens* Oral cl=49.1 mL/h…
Genetik -
Etofamide Approved DB13258
small molecule | CAS: 25287-60-9

Etofamide is used as an antiamoebic agent. Etofamide, under the brand name Kitnos, was marketed in Brazil by Pfizer but has been discontinued [L5617].

Kategori:
AcetatesAcids, AcyclicAmebicides +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etofenamate DB08984
small molecule | CAS: 30544-47-9

Etofenamate is used to treat muscle and joint paint. It is a non-steroidal anti-inflammatory drug (NSAID).

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etofibrate DB08983
small molecule | CAS: 31637-97-5

Etofibrate is a fibrate produced by the combination of clofibrate ester linked to niacin. These components separate in the body slowly allowing for pharmacokinetics similar to controlled-release formulations.

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAnticholesteremic Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etomidate Approved DB00292
small molecule | CAS: 33125-97-2

Imidazole derivative anesthetic and hypnotic with little effect on blood gases, ventilation, or the cardiovascular system. It has been proposed as an induction anesthetic.

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +11
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-1Alpha-2B adrenergic receptor +1
Waktu Paruh75 minutes.
Vol. Distribusi-
Klirens-
Genetik -
Etonogestrel Approved DB00294
small molecule | CAS: 54048-10-1

Etonogestrel molecule is a 3-ketodesogestrel or 19-nortestosterone which is a synthetic biologically active metabolite of progestin desogestrel.[A37184] The first product including etonogestrel was developed by the Merck subsidiary Organon and FDA approved in…

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +18
Target Protein:
Progesterone receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe clearance rate …
Genetik -
Etoperidone DB09194
small molecule | CAS: 52942-31-1

Etoperidone is an atypical antidepressant introduced in Europe in 1977. It is a phenylpiperazine-substituted triazole derivative with a composition that classifies it as an analog of tradozone and presents a similar pharmacological profile.[T45] Etoperidone w…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsCombined Inhibitors of Serotonin/Norepinephrine Reuptake +12
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2CAlpha-1 adrenergic receptors +3
Waktu ParuhAfter oral administ…
Vol. DistribusiThe high protein bi…
KlirensThe apparent cleara…
Genetik -
Etoposide Approved DB00773
small molecule | CAS: 33419-42-0

A semisynthetic derivative of podophyllotoxin that exhibits antitumor activity. Etoposide inhibits DNA synthesis by forming a complex with topoisomerase II and DNA. This complex induces breaks in double stranded DNA and prevents repair by topoisomerase II bin…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicAntineoplastic and Immunomodulating Agents +38
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh4-11 hours
Vol. DistribusiThe disposition of …
Klirens* Total body cleara…
Genetik -
small molecule | CAS: 433304-61-1

Deskripsi belum tersedia.

Kategori:
Topoisomerase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etorphine DB01497
small molecule | CAS: 14521-96-1

A narcotic analgesic morphinan used as a sedative in veterinary practice. In certain countries, etorphine is classified as a Schedule 1 drug and hence, in these countries, it can be used legally only by health professionals and for research purposes. Etorphin…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +10
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etozoline DB08982
small molecule | CAS: 73-09-6

Etozoline is marketed in Europe under the names Diulozin, Elkapin, and Etopinil. Etozoline is a loop diuretic.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etranacogene dezaparvovec Approved DB16791
biotech | CAS: 2156583-26-3

Hemophilia B - also called factor IX deficiency or Christmas disease - is an X-linked genetic disorder resulting in an absence or deficiency of clotting factor IX.[L44176] Clotting factors, including factor IX, are necessary components of the signaling cascad…

Kategori:
Adeno-associated Viral Vector TherapiesBlood and Blood Forming OrgansBlood Coagulation Factors +2
Target Protein:
Coagulation factor IX
Waktu Paruh-
Vol. DistribusiIn a study to evalu…
KlirensIn a clinical study…
Genetik -
Etrasimod Approved DB14766
small molecule | CAS: 1206123-37-6

Etrasimod is a synthetic next-generation selective Sphingosine 1-phosphate (S1P) receptor modulator that targets the S1P<sub>1,4,5</sub> with no detectable activity on S1P<sub>2</sub> and S1P<sub>3</sub> receptors. S1P receptors are membrane-derived lysophosp…

Kategori:
Acids, AcyclicAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +11
Target Protein:
Sphingosine 1-phosphate receptor 1Sphingosine 1-phosphate receptor 4Sphingosine 1-phosphate receptor 5
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe mean apparent v…
KlirensThe apparent steady…
Genetik -
Etravirine Approved DB06414
small molecule | CAS: 269055-15-4

Etravirine is an antiretroviral agent more specifically classified as a Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI). Etraverine is used clinically for the treatment of human immunodeficiency virus type 1 (HIV-1) infection. On January 18, 2007, the …

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiinfectives for Systemic Use +24
Target Protein:
Gag-Pol polyproteinGag-Pol polyproteinReverse transcriptase/RNaseH
Waktu ParuhHalf life of 9.05-4…
Vol. DistribusiDistribution of etr…
KlirensRenal clearance of …
Genetik -
Etripamil DB12605
small molecule | CAS: 1593673-23-4

Etripamil has been used in trials studying the treatment of Paroxysmal Supraventricular Tachycardia (PSVT).

Kategori:
Acids, CarbocyclicAntiarrhythmic agentsBenzene Derivatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etrolizumab DB12189
biotech | CAS: 1044758-60-2

Inflammatory bowel disease (IBD), including ulcerative colitis and Crohn's disease, is typified by a chronic gastrointestinal inflammatory microenvironment, driven in part by the excessive infiltration and retention of intestinal-homing lymphocytes.[A244564, …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Integrin beta-7
Waktu ParuhEtrolizumab adminis…
Vol. DistribusiModelling of etroli…
KlirensEtrolizumab has a m…
Genetik -
Etrumadenant DB17506
small molecule | CAS: 2239273-34-6

Deskripsi belum tersedia.

Target Protein:
Adenosine receptor A2aAdenosine receptor A2b
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etryptamine DB01546
small molecule | CAS: 2235-90-7

In the 1960's, alpha-ethyltryptamine (?ET), a non hydrazine reversible monoamine oxidase inhibitor, was developed in the United States by the Upjohn chemical company for use as an antidepressant. ?ET was an FDA approved antidepressant under the name Monase. H…

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ETX101 DB18579
biotech

ETX101 is a non-replicating recombinant adeno associated viral vector, serotype 9, designed to promote increased transcription of SCN1A gene.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etymemazine DB11517
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etynodiol DB13866
small molecule | CAS: 1231-93-2

Etynodiol (INN), or ethynodiol (BAN) is a steroidal progestin related to norethisterone which was never marketed. While etynodiol is sometimes used as a synonym for etynodiol diacetate, it usually refers to etynodiol diacetate (see [DB00823]), not etynodiol.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EU204 DB17438
biotech

EU204 (EBViNT) is an Epstein-Barr virus (EBV)-positive T-cell therapy currently undergoing phase 1 and 2a clinical trials in Korea for patients with EBV-positive lymphoma and solid cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eucalyptol DB03852
small molecule | CAS: 470-82-6

Eucalyptol is naturally produced cyclic ether and monoterpenoid. Eucalyptol is an ingredient in many brands of mouthwash and cough suppressant. It controls airway mucus hypersecretion and asthma via anti-inflammatory cytokine inhibition. Eucalyptol is an effe…

Kategori:
AgrochemicalsAlcoholsAnti-Infective Agents +29
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eucalyptus globulus pollen Approved DB10470
biotech

Eucalyptus globulus pollen is the pollen of the Eucalyptus globulus plant. Eucalyptus globulus pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eucalyptus gum Approved DB15537
biotech | CAS: 9000-20-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eugenol Approved DB09086
small molecule | CAS: 97-53-0

Eugenol is a naturally occurring phenolic molecule found in several plants such as cinnamon, clove, and bay leaves. It has been used as a topical antiseptic as a counter-irritant and in dental preparations with zinc oxide for root canal sealing and pain contr…

Kategori:
Acids, CarbocyclicAlkenesAllyl Compounds +11
Target Protein:
Amine oxidase [flavin-containing] BEstrogen receptorEstrogen receptor beta +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evalstotug DB19410
biotech | CAS: 2460399-39-5

Evalstotug is under investigation in clinical trial NCT05271604 (A Phase 2 Open Label Study of BA3021 in Patients With Recurrent or Metastatic Squamous Cell Carcinoma of the Head and Neck).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evatanepag DB12022
small molecule | CAS: 223488-57-1

Evatanepag has been used in trials studying the treatment of Tibial Fractures.

Target Protein:
Prostaglandin E2 receptor EP2 subtype
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evenamide DB18775
small molecule | CAS: 1092977-61-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 308064-97-3

Evening primrose oil comes from the extraction from _Oenothera biennis_ seeds and it is commonly used as an alternative source for omega-6 essential fatty acids. In its composition it presents some fatty acids such as [DB00132] and [DB13854].[A33131] Evening …

Kategori:
Agents that reduce seizure thresholdAngiospermsAnti-Inflammatory Agents +26
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Evernia prunastri Approved DB14172
biotech

Evernia prunastri allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseStandardized Chemical Allergen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evexomostat DB19140
small molecule | CAS: 2416263-67-5

Evexomostat is under investigation in clinical trial NCT05570253 (A Study of SDX-7320 in Combination With Eribulin for People With Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evinacumab Approved DB15354
biotech | CAS: 1446419-85-7

Evinacumab is a recombinant human IgG4 monoclonal antibody targeted against angiopoietin-like protein 3 (ANGPTL3) and the first drug of its kind. The ANGPTL family of proteins serve a number of physiologic functions - including involvement in the regulation o…

Kategori:
Amino Acids, Peptides, and ProteinsAngiopoietin-like 3 InhibitorAngiopoietin-like 3 Inhibitors +8
Target Protein:
Angiopoietin-related protein 3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Evobrutinib DB15170
small molecule | CAS: 1415823-73-2

Evobrutinib is under investigation in clinical trial NCT03934502 (Effect of Meal Composition and Timing on Evobrutinib Bioavailability).

Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evocalcet DB12388
small molecule | CAS: 870964-67-3

Evocalcet has been used in trials studying the treatment of Hyperparathyroidism and Secondary Hyperparathyroidism.

Kategori:
Anti-Parathyroid AgentsCalcium HomeostasisSystemic Hormonal Preparations, Excl. Sex Hormones and Insulins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evodenoson DB12295
small molecule | CAS: 844873-47-8

Evodenoson has been used in trials studying the treatment of Open-angle Glaucoma and Ocular Hypertension.

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evofosfamide DB06091
small molecule | CAS: 918633-87-1

TH-302 is a novel cancer therapeutic specifically activated under the low oxygen or "hypoxic" conditions typical of solid tumor cancer cells. TH-302 is a nitroimidazole-linked prodrug of a brominated derivative of an isophosphoramide mustard previously used i…

Kategori:
Hydrocarbons, HalogenatedImidazolesMustard Compounds +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Evolocumab Approved DB09303
biotech | CAS: 1256937-27-5

Evolocumab is a monoclonal antibody designed for the treatment of hyperlipidemia by Amgen. It is a subcutaneous injection approved by the FDA for individuals on maximum statin therapy who still require additional LDL-cholesterol lowering. It is approved for b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu Paruh-
Vol. Distribusi-
KlirensEvolocumab showed n…
Genetik -
Evorpacept DB17573
biotech | CAS: 2484949-51-9

evorpacept is under investigation in clinical trial NCT04755244 (A Study of Evorpacept (ALX148) With Venetoclax and Azacitidine for Acute Myeloid Leukemia (ASPEN-05)).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EVT 201 DB05721
small molecule | CAS: 308239-86-3

EVT 201 is a novel partial positive allosteric modulator of the GABAA receptor complex which is being developed as a treatment for insomnia. It is being developed by Evotec Inc.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EVT 302 DB06057
small molecule

EVT 302 is an orally active, potent, highly selective and reversible inhibitor of MAO-B. It is in the development for smoking cessation, and potential for disease modification in Alzheimer's disease.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Holoclar (_ex vivo_ expanded autologous human corneal epithelial cells containing stem cells) is a stem cell therapy used to treat limbal stem cell deficiencies.[L48375]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exagamglogene autotemcel Approved DB15572
biotech

Sickle cell disease (SCD) is a genetic disorder characterized by the production of abnormal sickle-shaped red blood cells (called hemoglobin S, HbS) that initiate a pathophysiology resulting in severe pain, progressive multi-organ damage, and premature death.…

Kategori:
Autologous Cultured CellBlood and Blood Forming Organs
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exaluren DB17631
small molecule | CAS: 1375073-93-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exametazime Approved DB11179
small molecule | CAS: 105613-48-7

Exametazime is a diagnostic radiopharmaceutical agent commonly used for the preparation of Tc99m Exametazime injection. It acts as a chelating agent for the radioisotope technetium-99m to form a cationic complex. It is used in the detection of altered regiona…

Kategori:
Ketones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exarafenib DB17582
small molecule | CAS: 2639957-39-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exatecan DB12185
small molecule | CAS: 171335-80-1

Exatecan has been used in trials studying the treatment of Sarcoma, Leukemia, Lymphoma, Lung Cancer, and Liver Cancer, among others.

Kategori:
AlkaloidsAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exbivirumab DB17747
biotech | CAS: 569658-80-6

Exbivirumab is an investigational monoclonal antibody. It is one of the active ingredients in HepeX-B, a drug product containing two human monoclonal antibodies to the hepatitis B virus (HBV) surface antigen.[A259202]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4951–5000 dari 11778
Sebelumnya Halaman 100 / 236 Berikutnya